
Ricettore GABA
I recettori GABA sono i principali recettori dei neurotrasmettitori inibitori nel sistema nervoso centrale, svolgendo un ruolo cruciale nella regolazione dell'eccitabilità neuronale e nel mantenimento dell'equilibrio tra eccitazione e inibizione. La disfunzione dei recettori GABA è implicata in vari disturbi neurologici e psichiatrici, tra cui epilessia, ansia e depressione. Presso CymitQuimica, offriamo una gamma completa di modulatori dei recettori GABA per supportare la tua ricerca in neurobiologia, salute mentale e sviluppo terapeutico.
Trovati 365 prodotti di "Ricettore GABA"
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Ro 15-1310
CAS:Ro 15-3505, a benzodiazepine receptor partial inverse agonist, has shown the ability to improve impaired recent memory of aged mice.Formula:C15H14ClN3O3Colore e forma:SolidPeso molecolare:319.74NO 711
CAS:NO 711(NNC-711 free acid) is a selective inhibitor of GAT-1, which enhances non-rapid eye movement sleep, and prevents paclitaxel-induced neuropathic pain.Formula:C21H22N2O3Purezza:99.70%Colore e forma:SolidPeso molecolare:350.41trans-4-Hydroxycrotonic acid
CAS:ligand of γ-hydroxybutyric acid (GHB) receptorFormula:C4H6O3Purezza:98%Colore e forma:SolidPeso molecolare:102.09(±)-Homoproline Hydrochloride
CAS:(±)-Homoproline Hydrochloride. Affordable Excellence: Reliable Quality You Can TrustFormula:C6H12ClNO2Purezza:99.69%Colore e forma:SolidPeso molecolare:165.62CP-409092 hydrochloride
CAS:CP-409092 hydrochloride is a partial agonist of the GABAA receptor with anti-anxiety activity.Formula:C17H20ClN3O2Colore e forma:SolidPeso molecolare:333.81Arbaclofen placarbil
CAS:Arbaclofen placarbil is a GABA(B) receptor agonist with better ADMET than R-baclofen, reducing postprandial reflux in GERD.Formula:C19H26ClNO6Colore e forma:SolidPeso molecolare:399.87LY 81067
CAS:LY 81067, a new anticonvulsant, prevents PTZ- and picrotoxin-induced seizures in mice via picrotoxin site interaction.Formula:C22H24N4OColore e forma:SolidPeso molecolare:360.45Ethyl dirazepate
CAS:Ethyl dirazepate has anxiolytic and hypnotic and possibly other characteristic benzodiazepine properties,is a drug which is a benzodiazepine derivative.Formula:C18H14Cl2N2O3Purezza:98%Colore e forma:SolidPeso molecolare:377.22U-7524
CAS:U-7524 (AOAA), an inhibitor of GABA-T and other PLP-dependent enzymes, disrupts the Schiff base linkage, forming oxime complexes.Formula:C2H5NO3Colore e forma:SolidPeso molecolare:91.07Y 23684
CAS:Y-23684 is an anxiolytic drug with a novel chemical structure. It has similar effects to benzodiazepine drugs and is classed as a nonbenzodiazepine anxiolytic.Formula:C18H13ClN2O2SPurezza:98%Colore e forma:SolidPeso molecolare:356.83Cyprodenate
CAS:Cyprodenate (Actebral) is a potent orally active brain-activating agent with appetite-suppressing properties, useful in studying metabolic.Formula:C13H25NO2Colore e forma:SolidPeso molecolare:227.34SCH 50911 hydrochloride
CAS:SCH 50911 hydrochloride is a selective, orally-active and competitive antagonist of γ-Aminobutyric acid B GABA(B) receptor(IC50 : 1.1 μM).Formula:C8H16ClNO3Purezza:98%Colore e forma:SolidPeso molecolare:209.67DS1
CAS:DS1 is a GABAA receptor agonist which can stimulate gonadotropin subunit gene expression in mouse.Formula:C18H10Br2ClN3OSColore e forma:SolidPeso molecolare:511.62CP-457920
CAS:CP-457920 is a selective α5 GABAA receptor inverse agonist that is suitable for investigating dementia in Alzheimer's disease.Formula:C18H17N3O3Purezza:99.06% - 99.74%Colore e forma:SolidPeso molecolare:323.353-Methyl-GABA
CAS:3-Methyl-GABA activates GABA aminotransferase, fits GABAaR, stimulates GAD, and acts as an anticonvulsant.Formula:C20H30N2O10S2Purezza:98%Colore e forma:SolidPeso molecolare:522.59U 90042
CAS:GABAA receptor ligandFormula:C17H13ClN6OPurezza:98%Colore e forma:SolidPeso molecolare:352.78Ro15-4513
CAS:Ro15-4513 is imidazobenzodiazepinone derivative and is a partial inverse agonist of benzodiazepine receptors. Ro15-4513 is an effective ethanol antagonist.Formula:C15H14N6O3Purezza:98%Colore e forma:SolidPeso molecolare:326.31Bifenazate
CAS:Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.Formula:C17H20N2O3Purezza:99.62%Colore e forma:Solid CrystallinePeso molecolare:300.35COR627
CAS:COR627 is the GABA receptor positive allosteric modulator.Formula:C20H27NO3SPurezza:98%Colore e forma:SolidPeso molecolare:361.52-Hydroxysaclofen
CAS:2-Hydroxysaclofen is a GABAB receptor antagonist.Formula:C9H12ClNO4SPurezza:98%Colore e forma:White SolidPeso molecolare:265.71
