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Ricettore GABA

Ricettore GABA

I recettori GABA sono i principali recettori dei neurotrasmettitori inibitori nel sistema nervoso centrale, svolgendo un ruolo cruciale nella regolazione dell'eccitabilità neuronale e nel mantenimento dell'equilibrio tra eccitazione e inibizione. La disfunzione dei recettori GABA è implicata in vari disturbi neurologici e psichiatrici, tra cui epilessia, ansia e depressione. Presso CymitQuimica, offriamo una gamma completa di modulatori dei recettori GABA per supportare la tua ricerca in neurobiologia, salute mentale e sviluppo terapeutico.

Trovati 365 prodotti di "Ricettore GABA"

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  • Ro 15-1310

    CAS:
    Ro 15-3505, a benzodiazepine receptor partial inverse agonist, has shown the ability to improve impaired recent memory of aged mice.
    Formula:C15H14ClN3O3
    Colore e forma:Solid
    Peso molecolare:319.74
  • NO 711

    CAS:
    NO 711(NNC-711 free acid) is a selective inhibitor of GAT-1, which enhances non-rapid eye movement sleep, and prevents paclitaxel-induced neuropathic pain.
    Formula:C21H22N2O3
    Purezza:99.70%
    Colore e forma:Solid
    Peso molecolare:350.41
  • trans-4-Hydroxycrotonic acid

    CAS:
    ligand of γ-hydroxybutyric acid (GHB) receptor
    Formula:C4H6O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:102.09
  • (±)-Homoproline Hydrochloride

    CAS:
    (±)-Homoproline Hydrochloride. Affordable Excellence: Reliable Quality You Can Trust
    Formula:C6H12ClNO2
    Purezza:99.69%
    Colore e forma:Solid
    Peso molecolare:165.62
  • CP-409092 hydrochloride

    CAS:
    CP-409092 hydrochloride is a partial agonist of the GABAA receptor with anti-anxiety activity.
    Formula:C17H20ClN3O2
    Colore e forma:Solid
    Peso molecolare:333.81
  • Arbaclofen placarbil

    CAS:
    Arbaclofen placarbil is a GABA(B) receptor agonist with better ADMET than R-baclofen, reducing postprandial reflux in GERD.
    Formula:C19H26ClNO6
    Colore e forma:Solid
    Peso molecolare:399.87
  • LY 81067

    CAS:
    LY 81067, a new anticonvulsant, prevents PTZ- and picrotoxin-induced seizures in mice via picrotoxin site interaction.
    Formula:C22H24N4O
    Colore e forma:Solid
    Peso molecolare:360.45
  • Ethyl dirazepate

    CAS:
    Ethyl dirazepate has anxiolytic and hypnotic and possibly other characteristic benzodiazepine properties,is a drug which is a benzodiazepine derivative.
    Formula:C18H14Cl2N2O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:377.22
  • U-7524

    CAS:
    U-7524 (AOAA), an inhibitor of GABA-T and other PLP-dependent enzymes, disrupts the Schiff base linkage, forming oxime complexes.
    Formula:C2H5NO3
    Colore e forma:Solid
    Peso molecolare:91.07
  • Y 23684

    CAS:
    Y-23684 is an anxiolytic drug with a novel chemical structure. It has similar effects to benzodiazepine drugs and is classed as a nonbenzodiazepine anxiolytic.
    Formula:C18H13ClN2O2S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:356.83
  • Cyprodenate

    CAS:
    Cyprodenate (Actebral) is a potent orally active brain-activating agent with appetite-suppressing properties, useful in studying metabolic.
    Formula:C13H25NO2
    Colore e forma:Solid
    Peso molecolare:227.34
  • SCH 50911 hydrochloride

    CAS:
    SCH 50911 hydrochloride is a selective, orally-active and competitive antagonist of γ-Aminobutyric acid B GABA(B) receptor(IC50 : 1.1 μM).
    Formula:C8H16ClNO3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:209.67
  • DS1

    CAS:
    DS1 is a GABAA receptor agonist which can stimulate gonadotropin subunit gene expression in mouse.
    Formula:C18H10Br2ClN3OS
    Colore e forma:Solid
    Peso molecolare:511.62
  • CP-457920

    CAS:
    CP-457920 is a selective α5 GABAA receptor inverse agonist that is suitable for investigating dementia in Alzheimer's disease.
    Formula:C18H17N3O3
    Purezza:99.06% - 99.74%
    Colore e forma:Solid
    Peso molecolare:323.35
  • 3-Methyl-GABA

    CAS:
    3-Methyl-GABA activates GABA aminotransferase, fits GABAaR, stimulates GAD, and acts as an anticonvulsant.
    Formula:C20H30N2O10S2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:522.59
  • U 90042

    CAS:
    GABAA receptor ligand
    Formula:C17H13ClN6O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:352.78
  • Ro15-4513

    CAS:
    Ro15-4513 is imidazobenzodiazepinone derivative and is a partial inverse agonist of benzodiazepine receptors. Ro15-4513 is an effective ethanol antagonist.
    Formula:C15H14N6O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:326.31
  • Bifenazate

    CAS:
    Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.
    Formula:C17H20N2O3
    Purezza:99.62%
    Colore e forma:Solid Crystalline
    Peso molecolare:300.35
  • COR627

    CAS:
    COR627 is the GABA receptor positive allosteric modulator.
    Formula:C20H27NO3S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:361.5
  • 2-Hydroxysaclofen

    CAS:
    2-Hydroxysaclofen is a GABAB receptor antagonist.
    Formula:C9H12ClNO4S
    Purezza:98%
    Colore e forma:White Solid
    Peso molecolare:265.71