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Ricettore GABA

Ricettore GABA

I recettori GABA sono i principali recettori dei neurotrasmettitori inibitori nel sistema nervoso centrale, svolgendo un ruolo cruciale nella regolazione dell'eccitabilità neuronale e nel mantenimento dell'equilibrio tra eccitazione e inibizione. La disfunzione dei recettori GABA è implicata in vari disturbi neurologici e psichiatrici, tra cui epilessia, ansia e depressione. Presso CymitQuimica, offriamo una gamma completa di modulatori dei recettori GABA per supportare la tua ricerca in neurobiologia, salute mentale e sviluppo terapeutico.

Trovati 365 prodotti di "Ricettore GABA"

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  • Loreclezole hydrochloride

    CAS:
    Loreclezole hydrochloride is an antiepileptic, enhancing GABA A receptors with β2/β3 subunits.
    Formula:C10H7Cl4N3
    Colore e forma:Solid
    Peso molecolare:310.99
  • Kavain

    CAS:
    <p>Kavain, a compound extracted from the Kava plant, Piper methysticum, is found to be involved in TNF-α expression in human and mouse cells via regulation of</p>
    Formula:C14H14O3
    Purezza:99.93% - ≥95%
    Colore e forma:Solid
    Peso molecolare:230.26
  • Guvacine hydrochloride

    CAS:
    <p>Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)</p>
    Formula:C6H10ClNO2
    Purezza:98.42%
    Colore e forma:Solid
    Peso molecolare:163.602
  • Amentoflavone

    CAS:
    Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.
    Formula:C30H18O10
    Purezza:98.21% - 99.22%
    Colore e forma:Odourless Whitish Solid
    Peso molecolare:538.46
  • L-DABA

    CAS:
    <p>L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 &gt; 500 μM).</p>
    Formula:C4H10N2O2
    Purezza:99.32%
    Colore e forma:Solid
    Peso molecolare:118.13
  • Baclofen hydrochloride

    CAS:
    Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.
    Formula:C10H13Cl2NO2
    Purezza:99.55%
    Colore e forma:Solid
    Peso molecolare:250.122
  • Aminooxyacetic acid hemihydrochloride

    CAS:
    Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA
    Formula:C2H5NO3·5HCl
    Purezza:98.03%
    Colore e forma:Light Beige Crystalline Powder
    Peso molecolare:109.3
  • Tiagabine

    CAS:
    Tiagabine (NO050328) is an Anti-epileptic Agent.
    Formula:C20H25NO2S2
    Purezza:99.25% - 99.67%
    Colore e forma:White To Off-White Crystalline Solid
    Peso molecolare:375.55
  • SSD114 HCl

    CAS:
    <p>SSD114 is a novel GABAB receptor positive allosteric modulator.</p>
    Formula:C18H21ClF3N3O
    Purezza:99.03% - 99.95%
    Colore e forma:Solid
    Peso molecolare:387.83
  • p-Hydroxybenzaldehyde

    CAS:
    1.
    Formula:C7H6O2
    Purezza:99.05% - 99.86%
    Colore e forma:Solid
    Peso molecolare:122.12
  • Miltirone

    CAS:
    Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.
    Formula:C19H22O2
    Purezza:99.22% - 99.66%
    Colore e forma:Solid
    Peso molecolare:282.38
  • Acamprosate calcium

    CAS:
    Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.
    Formula:C10H20CaN2O8S2
    Purezza:98% - 99.93%
    Colore e forma:White Odorless Or Nearly Odorless Powder
    Peso molecolare:400.48
  • Lorediplon

    CAS:
    Lorediplon is a novel hypnotic drug acting as a GABAA receptor modulator, differentially active at the α1-subunit, associated with promoting sleep.
    Formula:C20H15FN4O2S
    Purezza:99.12% - 99.19%
    Colore e forma:Solid
    Peso molecolare:394.42
  • Cyclothiazide

    CAS:
    <p>Cyclothiazide enhances AMPA receptors, prevents desensitization, and boosts glutamic acid response (EC50 = 3.8µM).</p>
    Formula:C14H16ClN3O4S2
    Purezza:98.23% - 99.49%
    Colore e forma:Crystals From Dilute Alcohol Solid
    Peso molecolare:389.88
  • Darigabat

    CAS:
    Darigabat (PF-06372865) is a GABAA receptor modulator with anxiolytic activity that inhibits α2, α1 PAM, and α2 PAM.
    Formula:C22H21FN4O3S
    Purezza:98.42% - 99.29%
    Colore e forma:Solid
    Peso molecolare:440.49
  • Riluzole

    CAS:
    <p>Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.</p>
    Formula:C8H5F3N2OS
    Purezza:99.71% - 99.88%
    Colore e forma:Powder
    Peso molecolare:234.2
  • CGP 36216 hydrochloride

    CAS:
    CGP 36216 hydrochloride is a potent and selective antagonist of GABAB receptors (IC50: 43 μM).
    Formula:C5H14NO2P
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:151.14
  • 17-PA

    CAS:
    17-PA is a GABAA receptor antagonist.
    Formula:C25H34O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:350.54
  • CGP11952

    CAS:
    CGP11952 is same the benzodiazepines in its pharmacological action and it also is an experimental benzodiazepine derivative.
    Formula:C21H21Cl2N5O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:446.33
  • GABA-AT-IN-1

    CAS:
    GABA-AT-IN-1 (Compound 6) is an inhibitor of γ-aminobutyric acid transaminase (GABA-AT) that crosses the blood-brain barrier.
    Formula:C23H18N2O6
    Colore e forma:Solid
    Peso molecolare:418.4