
Ricettore GABA
I recettori GABA sono i principali recettori dei neurotrasmettitori inibitori nel sistema nervoso centrale, svolgendo un ruolo cruciale nella regolazione dell'eccitabilità neuronale e nel mantenimento dell'equilibrio tra eccitazione e inibizione. La disfunzione dei recettori GABA è implicata in vari disturbi neurologici e psichiatrici, tra cui epilessia, ansia e depressione. Presso CymitQuimica, offriamo una gamma completa di modulatori dei recettori GABA per supportare la tua ricerca in neurobiologia, salute mentale e sviluppo terapeutico.
Trovati 365 prodotti di "Ricettore GABA"
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Loreclezole hydrochloride
CAS:Loreclezole hydrochloride is an antiepileptic, enhancing GABA A receptors with β2/β3 subunits.Formula:C10H7Cl4N3Colore e forma:SolidPeso molecolare:310.99Kavain
CAS:<p>Kavain, a compound extracted from the Kava plant, Piper methysticum, is found to be involved in TNF-α expression in human and mouse cells via regulation of</p>Formula:C14H14O3Purezza:99.93% - ≥95%Colore e forma:SolidPeso molecolare:230.26Guvacine hydrochloride
CAS:<p>Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)</p>Formula:C6H10ClNO2Purezza:98.42%Colore e forma:SolidPeso molecolare:163.602Amentoflavone
CAS:Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.Formula:C30H18O10Purezza:98.21% - 99.22%Colore e forma:Odourless Whitish SolidPeso molecolare:538.46L-DABA
CAS:<p>L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 > 500 μM).</p>Formula:C4H10N2O2Purezza:99.32%Colore e forma:SolidPeso molecolare:118.13Baclofen hydrochloride
CAS:Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.Formula:C10H13Cl2NO2Purezza:99.55%Colore e forma:SolidPeso molecolare:250.122Aminooxyacetic acid hemihydrochloride
CAS:Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABAFormula:C2H5NO3·5HClPurezza:98.03%Colore e forma:Light Beige Crystalline PowderPeso molecolare:109.3Tiagabine
CAS:Tiagabine (NO050328) is an Anti-epileptic Agent.Formula:C20H25NO2S2Purezza:99.25% - 99.67%Colore e forma:White To Off-White Crystalline SolidPeso molecolare:375.55SSD114 HCl
CAS:<p>SSD114 is a novel GABAB receptor positive allosteric modulator.</p>Formula:C18H21ClF3N3OPurezza:99.03% - 99.95%Colore e forma:SolidPeso molecolare:387.83p-Hydroxybenzaldehyde
CAS:1.Formula:C7H6O2Purezza:99.05% - 99.86%Colore e forma:SolidPeso molecolare:122.12Miltirone
CAS:Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.Formula:C19H22O2Purezza:99.22% - 99.66%Colore e forma:SolidPeso molecolare:282.38Acamprosate calcium
CAS:Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.Formula:C10H20CaN2O8S2Purezza:98% - 99.93%Colore e forma:White Odorless Or Nearly Odorless PowderPeso molecolare:400.48Lorediplon
CAS:Lorediplon is a novel hypnotic drug acting as a GABAA receptor modulator, differentially active at the α1-subunit, associated with promoting sleep.Formula:C20H15FN4O2SPurezza:99.12% - 99.19%Colore e forma:SolidPeso molecolare:394.42Cyclothiazide
CAS:<p>Cyclothiazide enhances AMPA receptors, prevents desensitization, and boosts glutamic acid response (EC50 = 3.8µM).</p>Formula:C14H16ClN3O4S2Purezza:98.23% - 99.49%Colore e forma:Crystals From Dilute Alcohol SolidPeso molecolare:389.88Darigabat
CAS:Darigabat (PF-06372865) is a GABAA receptor modulator with anxiolytic activity that inhibits α2, α1 PAM, and α2 PAM.Formula:C22H21FN4O3SPurezza:98.42% - 99.29%Colore e forma:SolidPeso molecolare:440.49Riluzole
CAS:<p>Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.</p>Formula:C8H5F3N2OSPurezza:99.71% - 99.88%Colore e forma:PowderPeso molecolare:234.2CGP 36216 hydrochloride
CAS:CGP 36216 hydrochloride is a potent and selective antagonist of GABAB receptors (IC50: 43 μM).Formula:C5H14NO2PPurezza:98%Colore e forma:SolidPeso molecolare:151.1417-PA
CAS:17-PA is a GABAA receptor antagonist.Formula:C25H34OPurezza:98%Colore e forma:SolidPeso molecolare:350.54CGP11952
CAS:CGP11952 is same the benzodiazepines in its pharmacological action and it also is an experimental benzodiazepine derivative.Formula:C21H21Cl2N5O2Purezza:98%Colore e forma:SolidPeso molecolare:446.33GABA-AT-IN-1
CAS:GABA-AT-IN-1 (Compound 6) is an inhibitor of γ-aminobutyric acid transaminase (GABA-AT) that crosses the blood-brain barrier.Formula:C23H18N2O6Colore e forma:SolidPeso molecolare:418.4
