CymitQuimica logo
Ricettore GABA

Ricettore GABA

I recettori GABA sono i principali recettori dei neurotrasmettitori inibitori nel sistema nervoso centrale, svolgendo un ruolo cruciale nella regolazione dell'eccitabilità neuronale e nel mantenimento dell'equilibrio tra eccitazione e inibizione. La disfunzione dei recettori GABA è implicata in vari disturbi neurologici e psichiatrici, tra cui epilessia, ansia e depressione. Presso CymitQuimica, offriamo una gamma completa di modulatori dei recettori GABA per supportare la tua ricerca in neurobiologia, salute mentale e sviluppo terapeutico.

Trovati 364 prodotti di "Ricettore GABA"

Ordinare per

Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
prodotti per pagina.
  • Flufiprole

    CAS:
    Flufiprole is used as a phenylpyrazole pesticide. It has enantioselective metabolism in human and rat liver microsomes.
    Formula:C16H10Cl2F6N4OS
    Colore e forma:Solid
    Peso molecolare:491.24
  • AHN-683

    CAS:
    AHN-683 is a fluorescent ligand. It was used for peripheral-type benzodiazepine receptors.
    Formula:C42H32FN3O7
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:709.72
  • LU-32-176B

    CAS:
    LU32-176B is a bioactive chemical.
    Formula:C23H24F2N2O2
    Colore e forma:Solid
    Peso molecolare:398.45
  • Imagabalin

    CAS:
    Imagabalin is an active compound used in the study of neurological diseases.
    Formula:C9H19NO2
    Colore e forma:Solid
    Peso molecolare:173.25
  • Riluzole-13C,15N2

    CAS:
    <p>Riluzole-13C,15N2 (PK 26124-13C,15N2) is a 13C and 15N labeled form of Riluzole, a glutamate antagonist with anticonvulsant activity, inhibiting GABA uptake.</p>
    Formula:CC7H5F3OS15N2
    Colore e forma:Solid
    Peso molecolare:237.18
  • Fipronil sulfone

    CAS:
    Fipronil sulfone is an insecticide fipronil. Its metabolite fipronil sulphone is an inhibitor of rat ɑ1β2γ2L GABA(A) receptor.
    Formula:C12H4Cl2F6N4O2S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:453.14
  • Nitrazolam

    CAS:
    Nitrazolam is a benzodiazepine compound that may exhibit central nervous system depressant properties similar to traditional benzodiazepine drugs by acting on the GABA receptors (GABA receptor). These effects include sedation, hypnosis, anxiolytic, and anticonvulsant activities.
    Formula:C17H13N5O2
    Colore e forma:Solid
    Peso molecolare:319.32
  • Azocarnil


    <p>Azocarnil is a GABAergic agonist-enhancer used in neurological system research.</p>
    Colore e forma:Odour Solid
  • Furosemide sodium

    CAS:
    <p>Furosemide sodium: potent NKCC inhibitor, loop diuretic, treats heart failure, hypertension, edema, selective GABAA antagonist.</p>
    Formula:C12H10ClN2NaO5S
    Purezza:99.52% - >99.99%
    Colore e forma:Solid
    Peso molecolare:352.73
  • 12,14-Dichlorodehydroabietic acid

    CAS:
    12,14-Dichlorodehydroabietic acid activates BK channels, blocks GABA A receptors, and increases calcium and neurotransmitter release.
    Formula:C20H26Cl2O2
    Colore e forma:Solid
    Peso molecolare:369.33
  • DAA-1106

    CAS:
    DAA-1106 is a potent and selective ligand for PBR, acting as a potent and selective agonist at the peripheral benzodiazepine receptor.
    Formula:C23H22FNO4
    Purezza:99.54%
    Colore e forma:Solid
    Peso molecolare:395.42
  • RuBi-GABA

    CAS:
    Ruthenium-bipyridine-triphenylphosphine caged GABA
    Formula:C42H39F6N5O2P2Ru
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:922.8
  • Neurotransmitter Receptor Compound Library


    <p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening;</p>
    Colore e forma:Odour Solid
  • Anticonvulsant agent 8


    Anticonvulsant agent 8 (compound D4) is a chemical used in treating epilepsy by inhibiting GABAA currents. In mouse models, its ED50 values are 2.23 mg/kg for the maximal electroshock (MES) test and 24.60 mg/kg for the pentylenetetrazol (PTZ) test.
    Formula:C15H11N5O
    Colore e forma:Solid
    Peso molecolare:277.28
  • CGP 35348

    CAS:
    CGP 35348 是 GABAB 受体的选择性拮抗剂 (EC50 = 34 μM)。 CGP 35348 可用于研究白化新生小鼠脑损伤后的神经肌肉协调和空间学习。
    Formula:C8H20NO4P
    Purezza:≥98%
    Colore e forma:Solid
    Peso molecolare:225.22
  • Anisatin


    <p>Anisatin is a useful organic compound for research related to life sciences and the catalog number is T124719.</p>
    Formula:C15H20O8
    Colore e forma:Solid
    Peso molecolare:328.317
  • Atagabalin

    CAS:
    Atagabalin (PD 0200390), a gabamimetic for insomnia treatment and related to gabapentin, was halted due to poor trial outcomes.
    Formula:C10H19NO2
    Colore e forma:Solid
    Peso molecolare:185.26
  • (1S,3R)-3-Aminocyclopentane carboxylic acid

    CAS:
    <p>(1S,3R)-3-Aminocyclopentane carboxylic acid exhibits activity on GABAA receptors.</p>
    Formula:C6H11NO2
    Colore e forma:Solid
    Peso molecolare:129.16
  • Nipecotic acid

    CAS:
    <p>Compound PDK0243, with CAS No. 498-95-3, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0243 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>
    Formula:C6H11NO2
    Colore e forma:Off-White To Pale Yellow-Beige Powder
    Peso molecolare:129.16
  • Ion Channel Targeted Library


    <p>A unique collection of 931 compounds targeting ion channels for research in ion channels-related diseases and ion channel drug discovery;</p>
    Colore e forma:Odour Solid