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Ricettore GABA

Ricettore GABA

I recettori GABA sono i principali recettori dei neurotrasmettitori inibitori nel sistema nervoso centrale, svolgendo un ruolo cruciale nella regolazione dell'eccitabilità neuronale e nel mantenimento dell'equilibrio tra eccitazione e inibizione. La disfunzione dei recettori GABA è implicata in vari disturbi neurologici e psichiatrici, tra cui epilessia, ansia e depressione. Presso CymitQuimica, offriamo una gamma completa di modulatori dei recettori GABA per supportare la tua ricerca in neurobiologia, salute mentale e sviluppo terapeutico.

Trovati 365 prodotti di "Ricettore GABA"

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  • (1S,3R)-3-Aminocyclopentane carboxylic acid

    CAS:
    <p>(1S,3R)-3-Aminocyclopentane carboxylic acid exhibits activity on GABAA receptors.</p>
    Formula:C6H11NO2
    Colore e forma:Solid
    Peso molecolare:129.16
  • Ion Channel Targeted Library


    <p>A unique collection of 931 compounds targeting ion channels for research in ion channels-related diseases and ion channel drug discovery;</p>
    Colore e forma:Odour Solid
  • S-8510 free base

    CAS:
    S-8510 is a GABA-A receptor inverse agonist enhancing memory, LTP, and neurotransmitters in rats.
    Formula:C12H10N4O2
    Colore e forma:Solid
    Peso molecolare:242.23
  • Imagabalin

    CAS:
    Imagabalin is an active compound used in the study of neurological diseases.
    Formula:C9H19NO2
    Colore e forma:Solid
    Peso molecolare:173.25
  • FGIN-1-43

    CAS:
    FGIN-1-43 is a potent and specific ligand for the mitochondrial DBI receptor.
    Formula:C28H36Cl2N2O
    Purezza:99.57%
    Colore e forma:Solid
    Peso molecolare:487.5
  • (Iso)-Atagabalin HCl

    CAS:
    <p>(Iso)-Atagabalin HCl(isomer-Atagabalin HCl) is an alpha -2- delta ligand that can be used to treat non-restorative sleep.</p>
    Formula:C10H20ClNO2
    Purezza:99.26% - >99.99%
    Colore e forma:Soild
    Peso molecolare:221.72
  • MIDD0301

    CAS:
    <p>MIDD0301 is a potent positive allosteric α5β3γ selective GABAA receptor (GABAAR) ligand with EC50 of 17 nM.</p>
    Formula:C19H13BrFN3O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:414.23
  • 12,14-Dichlorodehydroabietic acid

    CAS:
    12,14-Dichlorodehydroabietic acid activates BK channels, blocks GABA A receptors, and increases calcium and neurotransmitter release.
    Formula:C20H26Cl2O2
    Colore e forma:Solid
    Peso molecolare:369.33
  • 3-Aminopropylphosphonic Acid

    CAS:
    <p>3-aminopropylphosphonic acid (3-APPA) is a phosphonic analog of GABA that acts as a partial agonist of GABAB receptors (IC50 = 1.5 μM in a radioligand binding</p>
    Formula:C3H10NO3P
    Purezza:99.84%
    Colore e forma:Light Yellow Liquid
    Peso molecolare:139.09
  • Endosulfan I

    CAS:
    <p>Endosulfan I is one of the two major stereoisomers of the broad-spectrum insecticide Endosulfan inhibi the GABA/benzodiazepine/picrotoxin complex</p>
    Formula:C9H6Cl6O3S
    Purezza:99.86%
    Colore e forma:Solid
    Peso molecolare:406.93
  • DAA-1106

    CAS:
    DAA-1106 is a potent and selective ligand for PBR, acting as a potent and selective agonist at the peripheral benzodiazepine receptor.
    Formula:C23H22FNO4
    Purezza:99.54%
    Colore e forma:Solid
    Peso molecolare:395.42
  • Atagabalin

    CAS:
    Atagabalin (PD 0200390), a gabamimetic for insomnia treatment and related to gabapentin, was halted due to poor trial outcomes.
    Formula:C10H19NO2
    Colore e forma:Solid
    Peso molecolare:185.26
  • Fipronil sulfone

    CAS:
    Fipronil sulfone is an insecticide fipronil. Its metabolite fipronil sulphone is an inhibitor of rat ɑ1β2γ2L GABA(A) receptor.
    Formula:C12H4Cl2F6N4O2S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:453.14
  • Chrodrimanin B

    CAS:
    Chrodrimanin B is a useful organic compound for research related to life sciences. The catalog number is T126052 and the CAS number is 132196-54-4.
    Formula:C27H32O8
    Colore e forma:Solid
    Peso molecolare:484.545
  • Emamectin B1a

    CAS:
    <p>Emamectin B1a can be used in relevant research in the life sciences. Its product number is T37663 and CAS number is 121124-29-6.</p>
    Formula:C49H75NO13
    Colore e forma:Solid
    Peso molecolare:886.133
  • Flufiprole

    CAS:
    Flufiprole is used as a phenylpyrazole pesticide. It has enantioselective metabolism in human and rat liver microsomes.
    Formula:C16H10Cl2F6N4OS
    Colore e forma:Solid
    Peso molecolare:491.24
  • 3-Aminopropylphosphinic acid

    CAS:
    <p>3-Aminopropylphosphinic acid (3-APPA) is a phosphonic analog of gamma-aminobutyric acid (GABA).</p>
    Formula:C3H10NO2P
    Colore e forma:Solid
    Peso molecolare:123.092
  • Anticonvulsant agent 9


    <p>Anticonvulsant agent 9 (compound 4f) is an activator of the α1β2γ2GABA_A receptor, with an EC50 value of 1.24 μM. It inhibits the inactivation of Nav1.2 channels and exhibits significant anticonvulsant activity.</p>
    Formula:C22H24N4O2
    Colore e forma:Solid
    Peso molecolare:376.45
  • AHN-683

    CAS:
    AHN-683 is a fluorescent ligand. It was used for peripheral-type benzodiazepine receptors.
    Formula:C42H32FN3O7
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:709.72
  • LU-32-176B

    CAS:
    LU32-176B is a bioactive chemical.
    Formula:C23H24F2N2O2
    Colore e forma:Solid
    Peso molecolare:398.45