
Caseina chinasi
Le caseina chinasi sono una famiglia di proteine chinasi serina/treonina che regolano vari processi cellulari, tra cui la riparazione del DNA, i ritmi circadiani e la trasduzione del segnale. Queste chinasi sono coinvolte nella fosforilazione di numerose proteine e sono implicate in malattie come il cancro, i disturbi neurodegenerativi e le sindromi metaboliche. Presso CymitQuimica, offriamo una selezione di inibitori della caseina chinasi per supportare la tua ricerca nella trasduzione del segnale, nella regolazione del ciclo cellulare e nello sviluppo terapeutico.
Trovati 150 prodotti per "Caseina chinasi".
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p38α inhibitor 8
CAS:p38α inhibitor8 (Compound 1) demonstrates inhibitory activity against p38αMAPK and CK1δ, with IC50 values of 0.21 µM and 0.202 µM, respectively.Formula:C17H13FN6Colore e forma:SolidPeso molecolare:320.324Casein kinase 1δ-IN-18
CAS:Casein kinase1δ-IN-18 (compound 660) is an inhibitor of casein kinase 1δ (CK1δ), which can be utilized for research in neurodegenerative diseases.Formula:C16H12ClN3O2S2Colore e forma:SolidPeso molecolare:377.868p38α MAPK/CK1δ inhibitor-1
CAS:p38αMAPK/CK1δ inhibitor-1 (Compound 3) exhibits inhibitory activity against p38αMAPK and CK1δ, with IC50 values of 0.185 µM and 0.089 µM, respectively.Formula:C24H17FN6O2Colore e forma:SolidPeso molecolare:440.429Casein kinase 1δ-IN-30
CAS:Casein kinase1δ-IN-30 (Compound 581) is an inhibitor of casein kinase 1δ (CK1δ). It can be utilized in research related to neurodegenerative diseases.Formula:C18H15BrN6O2SColore e forma:SolidPeso molecolare:459.32dCK1α-2
dCK1α-2 is an orally effective CK1α molecular glue (Molecular Glue) degrader that targets p53 pathway-related targets. It demonstrates antitumor efficacy in mouse models by enhancing the expression of p53-related genes.Formula:C24H24ClN5O4Colore e forma:SolidPeso molecolare:481.93CK1δ-IN-8
CAS:CK1δ-IN-8 (Compound 429) is a CK1δ inhibitor suitable for Alzheimer's disease research.Formula:C14H9N3O2S2Colore e forma:SolidPeso molecolare:315.37Casein kinase 1δ-IN-16
CAS:Casein kinase1δ-IN-16 (compound 506) is an inhibitor of casein kinase 1δ (CK1δ). This compound is applicable in research related to neurodegenerative diseases.Formula:C17H12N4S2Colore e forma:SolidPeso molecolare:336.434CK2 inhibitor 2
CAS:CK2 Inhibitor 2, characterized as a potent, selective, and orally active inhibitor of CK2, demonstrates an impressive IC50 value of 0.66 nM.Formula:C21H17ClN4O2Purezza:99.02%Colore e forma:SolidPeso molecolare:392.84Ref: TM-T35557
1mg62,00€5mg138,00€1mL*10mM (DMSO)152,00€10mg215,00€25mg425,00€50mg637,00€100mg853,00€200mg1.153,00€AMG-548 dihydrochloride
AMG-548 dihydrochloride, an oral p38α inhibitor (Ki: 0.5 nM), selectively targets p38β, γ, δ, inhibits TNFα (IC50: 3 nM), and suppresses Wnt signaling.Formula:C29H29Cl2N5OColore e forma:SolidPeso molecolare:534.48Ref: TM-T63762
Prodotto fuori produzioneAMG-548 hydrochloride
AMG-548 hydrochloride: orally active, p38α inhibitor (Ki=0.5 nM), 1000x less for p38γ/δ, also blocks TNFα (IC50=3 nM) & inhibits casein kinase 1 δ/ε.Formula:C29H28ClN5OColore e forma:SolidPeso molecolare:498.02Ref: TM-T63371
Prodotto fuori produzione

