CymitQuimica logo
FAAH

FAAH

La Fatty Acid Amide Hydrolase (FAAH) è un enzima che degrada gli amidi degli acidi grassi, inclusi gli endocannabinoidi come l'anandamide. Questi composti sono coinvolti nella regolazione del dolore, dell'umore, dell'appetito e della memoria. L'inibizione della FAAH può aumentare i livelli di queste molecole di segnalazione, offrendo potenziali benefici terapeutici per il dolore, l'ansia e le malattie neurodegenerative. Presso CymitQuimica, offriamo una selezione di inibitori della FAAH per supportare la tua ricerca in neuroscienze, gestione del dolore e segnalazione endocannabinoide.

Trovati 65 prodotti di "FAAH"

Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
prodotti per pagina.
  • CAY10435
    Targetmol
    + Info

    CAY10435

    CAS:
    <p>CAY10435, a β-ketooxazapyridine and selective FAAH inhibitor, exhibits antimicrobial properties. It binds non-competitively to the FAAH of Dictyostelium discoideum, demonstrating a Kd value of 0.57 nM [1] [2].</p>
    Formula:C18H26N2O2
    Colore e forma:Solid
    Peso molecolare:302.41

    Ref: TM-T84554

  • FAAH/cPLA2α-IN-1
    Targetmol
    + Info

    FAAH/cPLA2α-IN-1

    CAS:
    FAAH/cPLA2α-IN-1 is a compound that simultaneously inhibits both FAAH and cPLA2α, demonstrating potent activity with half-maximal inhibitory concentrations (
    Formula:C19H26N4O5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:390.43

    Ref: TM-T82421

  • OMDM-5
    Targetmol
    + Info

    OMDM-5

    CAS:
    OMDM-5 is a potent vanilloid receptor type 1 (TRPV1, EC50 = 75 nM) agonist, showing weak ligand activity at cannabinoid type 1 receptor (CB1, Ki=4.9 μM).
    Formula:C26H44N2O3
    Purezza:99.73%
    Colore e forma:Solid
    Peso molecolare:432.64

    Ref: TM-T12306

  • JP104
    Targetmol
    + Info

    JP104

    CAS:
    JP104 is an aryl carbamate that irreversibly inhibits fatty acid amide hydrolase (FAAH) with a pIC50 value of approximately 8 [1].
    Formula:C25H30N2O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:406.52

    Ref: TM-T78593

  • PDP-EA
    Targetmol
    + Info

    PDP-EA

    CAS:
    <p>PDP-EA is an activator of fatty acid amide hydrolase(FAAH) and enhances the amidohydrolase activity of FAAH.</p>
    Formula:C25H43NO3
    Purezza:99.59%
    Colore e forma:Solid
    Peso molecolare:405.61

    Ref: TM-T28353

  • FAAH inhibitor 2
    Targetmol
    + Info

    FAAH inhibitor 2

    CAS:
    FAAH Inhibitor 2 (Compound 17b) is an irreversible inhibitor of fatty acid amide hydrolase (FAAH), demonstrating an IC50 value of 0.153 μM [1].
    Formula:C24H40N2O2
    Colore e forma:Solid
    Peso molecolare:388.59

    Ref: TM-T84404

  • MK-3168 (12C)
    Targetmol
    + Info

    MK-3168 (12C)

    CAS:
    <p>MK-3168 (12C) functions as a FAAH inhibitor, exhibiting IC50 values of 1.0 nM, 5.5 nM, and 1.7 nM for human, rhesus, and rat respectively. It demonstrates effective brain uptake and FAAH-specific signaling. Additionally, 11 C MK-3168 is applicable as a FAAH PET tracer.</p>
    Formula:C21H21ClN4OS
    Colore e forma:Solid
    Peso molecolare:412.94

    Ref: TM-T200270

  • Logo CymitQuimica
    Targetmol
    + Info

    FAAH/MAGL-IN-1

    <p>FAAH/MAGL-IN-1 (SIH 3) inhibits FAAH &amp; MAGL with IC50 of 31 &amp; 29 nM, useful in neuropathic pain research.</p>
    Formula:C15H9Cl2N3O3
    Colore e forma:Solid
    Peso molecolare:350.16

    Ref: TM-T61198

  • Irafamdastat
    Targetmol
    + Info

    Irafamdastat

    CAS:
    Irafamdastat (BMS-986368) [Example 74] is an inhibitor of FAAH and MAGL, with IC50 values of ≤ 100 nM for human FAAH and 100 nM-1 μM for human MAGL. It exhibits anticonvulsant properties.
    Formula:C20H21F3N4O4
    Colore e forma:Solid
    Peso molecolare:438.40

    Ref: TM-T211809

  • AZ513
    Targetmol
    + Info

    AZ513

    CAS:
    <p>AZ513 is a reversible FAAH inhibitor, exhibiting an IC50 of 551 nM for human FAAH and 27 nM for rat FAAH. It inhibits the hydrolysis of arachidonoyl ethanolamide in HEK293 cells transfected with human FAAH, with an IC50 of 360 nM.</p>
    Formula:C14H9Cl2N3O
    Colore e forma:Solid
    Peso molecolare:306.147

    Ref: TM-T204429

  • Sob-AM2
    Targetmol
    + Info

    Sob-AM2

    CAS:
    Sob-AM2 is an effective substrate targeting the fatty acid amide hydrolase (FAAH) expressed in the brain, with a Km of 1.3 μM. It delivers higher concentrations of Sobetirome to the central nervous system at minimal peripheral systemic doses, thereby activating the central thyroid hormone receptor β (TRβ).
    Formula:C21H27NO3
    Colore e forma:Solid
    Peso molecolare:341.44

    Ref: TM-T200594

  • FAAH/MAGL-IN-2
    Targetmol
    + Info

    FAAH/MAGL-IN-2

    CAS:
    FAAH/MAGL-IN-2: potent, reversible, oral FAAH & MAGL inhibitor, IC50: 11/36 nM, may research neuropathic pain, no locomotion issue.
    Formula:C15H13Cl2N3O3S
    Colore e forma:Solid
    Peso molecolare:386.25

    Ref: TM-T61707

  • Logo CymitQuimica
    Targetmol
    + Info

    FAAH/MAGL-IN-3

    <p>FAAH/MAGL-IN-3 irreversibly inhibits FAAH (IC50: 179 nM) &amp; MAGL (IC50: 759 nM) with low PAMPA permeability.</p>
    Formula:C21H25N3O6S
    Colore e forma:Solid
    Peso molecolare:447.5

    Ref: TM-T62671

  • Dual FAAH/sEH-IN-1
    Targetmol
    + Info

    Dual FAAH/sEH-IN-1

    CAS:
    <p>Dual FAAH/sEH-IN-1 inhibits both sEH (IC50: 9.6 nM) and FAAH (IC50: 7 nM), offering potent anti-inflammatory effects.</p>
    Formula:C25H22ClN3O3S2
    Purezza:99.89%
    Colore e forma:Solid
    Peso molecolare:512.04

    Ref: TM-T63536

  • TC-F 2
    Targetmol
    + Info

    TC-F 2

    CAS:
    TC-F 2 is a FAAH inhibitor.
    Formula:C26H25N5O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:439.51

    Ref: TM-T23432

    1mg
    Fuori produzione
    Prodotto fuori produzione