
Deidrogenasi
Le deidrogenasi sono enzimi coinvolti nelle reazioni di ossidoriduzione delle vie metaboliche, svolgendo un ruolo centrale nella produzione di energia e nella respirazione cellulare. Questi enzimi sono cruciali per processi come il ciclo dell'acido citrico, la glicolisi e l'ossidazione degli acidi grassi. Gli inibitori delle deidrogenasi sono strumenti importanti nello studio delle malattie metaboliche, del cancro e dello stress ossidativo. Presso CymitQuimica, offriamo una selezione completa di inibitori delle deidrogenasi per supportare la tua ricerca in metabolismo, biologia del cancro e biochimica.
Trovati 300 prodotti di "Deidrogenasi"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Brequinar sodium
CAS:Bipenquinate is a potent and selective inhibitor of dihydroorotate dehydrogenase (DHODH) with IC50 of 20 nM, blocking de novo pyrimidine biosynthesis.Formula:C23H14F2NNaO2Purezza:98.16%Colore e forma:SolidPeso molecolare:397.36WIN 18446
CAS:inhibitor of aldehyde dehydrogenase 1a2 (ALDH1a2)Formula:C12H20Cl4N2O2Purezza:99.69%Colore e forma:SolidPeso molecolare:366.11DS-1001b
CAS:DS-1001b is an inhibitor of mutant IDH-1 (Isocitrate Dehydrogenase-1)Formula:C29H29Cl3FN3O4Purezza:99.81%Colore e forma:SolidPeso molecolare:608.92BAY-1436032
CAS:BAY-1436032 is a novel, selective and orally available inhibitor of pan-mutant isocitrate dehydrogenase 1 (IDH1).Formula:C26H30F3N3O3Purezza:99.65% - 99.71%Colore e forma:SolidPeso molecolare:489.53DS44960156
CAS:DS44960156 is an inhibitor of methylenetetrahydrofolate dehydrogenase 2 (MTHFD2) that inhibits both MTHFD2 and MTHFD1 and can be used in cancer research.Formula:C20H15NO5Purezza:99.13%Colore e forma:SolidPeso molecolare:349.34Enasidenib mesylate
CAS:Enasidenib mesylate (AG-221 mesylate) is a IDH2 inhibitor that promotes differentiation of leukemia myeloid cells for the treatment of acute myeloid leukemia.Formula:C20H21F6N7O4SPurezza:99.85%Colore e forma:SolidPeso molecolare:569.48GSK1940029
CAS:GSK1940029 (SCD inhibitor 1) is a stearoyl-coa desaturase (SCD) inhibitor.Formula:C18H16Cl2N4O2Purezza:99.48% - 99.49%Colore e forma:SolidPeso molecolare:391.25Triflupromazine
CAS:Triflupromazine is a dopamine receptor D1/D2 antagonist and LHDA inhibitor that suppresses dopamine activity in (CNS)mental disorders, sedation, and antiemesis.Formula:C18H19F3N2SColore e forma:SolidPeso molecolare:352.42Nitrophenide
CAS:Nitrophenide, a 3,3'-Dinitrodiphenyl disulfide, blocks M1PDH in the mannitol cycle, serving as an anticoccidial.Formula:C12H8N2O4S2Purezza:99.78%Colore e forma:SolidPeso molecolare:308.33hDHODH-IN-2
CAS:<p>hDHODH-IN-2: Leflunomide metabolite analog, inhibits human dihydroorotate dehydrogenase, anti-inflammatory.</p>Formula:C19H16N2O2Purezza:98%Colore e forma:SolidPeso molecolare:304.349SCH-451659
CAS:SCH-451659 is an 17β-hydroxysteroid dehydrogenases (17β-HSDs) inhibitor.Formula:C30H39Cl2N3O2Purezza:98%Colore e forma:SolidPeso molecolare:544.56673-A
CAS:673-A inhibits ALDH1A, depletes ovarian CSCs, induces necroptosis, and reverses chemo resistance.Formula:C15H13NOColore e forma:SolidPeso molecolare:223.27DHODH-IN-12
CAS:DHODH-IN-12 is a leflunomide derivative and a weak dihydrorotate dehydrogenase (DHODH) inhibitor with a pKa of 5.07.Formula:C10H9N3O2Purezza:99.53%Colore e forma:SolidPeso molecolare:203.2CM39
CAS:CM39 inhibits ALDH, linked to cancer stem-like cells & chemoresistance.Formula:C19H15FN4OSColore e forma:SolidPeso molecolare:366.41Nitrefazole
CAS:Nitrefazole: a 4-nitroimidazole, inhibits ALDH enzyme crucial for alcohol metabolism, has potent, durable effects.Formula:C10H8N4O4Colore e forma:SolidPeso molecolare:248.1911β-HSD1-IN-6
CAS:11β-HSD1-IN-6 is a potent inhibitor of 11β hydroxysteroid dehydrogenase enzymes (11β-HSDs).Formula:C21H19ClN4OColore e forma:SolidPeso molecolare:378.86MEDS433
CAS:MEDS433 inhibits dihydroorotate dehydrogenase (IC50 1.2 nM) and blocks replication of hCoV-OC43, hCoV-229E, SARS-CoV-2 at nanomolar levels.Formula:C20H11F4N3O2Colore e forma:SolidPeso molecolare:401.31hDHODH-IN-11
CAS:hDHODH-IN-11: potent hDHODH inhibitor, IC50 7.2 nM, low cytotoxicity, for AML research.Formula:C24H23N3O3Colore e forma:SolidPeso molecolare:401.46RS6212
CAS:<p>RS6212 is a specific lactate dehydrogenase (LDH) inhibitor (IC50=12.03 μ M)。 RS6212 shows strong anticancer activity in a variety of cancer cell lines.</p>Formula:C20H22N4O3SColore e forma:SolidPeso molecolare:398.48AMG-221
CAS:AMG-221: potent 11β-HSD1 inhibitor, lowers glucose & insulin, reduces obesity in mice.Formula:C14H22N2OSPurezza:98%Colore e forma:SolidPeso molecolare:266.4
