
recettore 5-HT
I recettori 5-HT, noti anche come recettori della serotonina, sono un gruppo di recettori accoppiati alle proteine G (GPCR) che mediano gli effetti della serotonina, un neurotrasmettitore coinvolto nella regolazione dell'umore, dell'ansia, del sonno, dell'appetito e di altri processi fisiologici. Questi recettori sono suddivisi in diversi sottotipi, ciascuno con funzioni e proprietà farmacologiche distinte. I modulatori dei recettori 5-HT sono ampiamente studiati per il loro ruolo nel trattamento della depressione, dei disturbi d'ansia e di altre condizioni neuropsichiatriche. Presso CymitQuimica, offriamo una gamma di modulatori dei recettori 5-HT di alta qualità per supportare la tua ricerca in neurofarmacologia, disturbi dell'umore e segnalazione GPCR.
Trovati 1025 prodotti di "recettore 5-HT"
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Quetiapine-d4 fumarate
CAS:Deuterium-labeled Quetiapine fumarate; an antidepressant and anxiolytic 5-HT agonist, dopamine antagonist.Formula:C25H29N3O6SPurezza:98%Colore e forma:SolidPeso molecolare:503.611,8-Cineole
CAS:Eucalyptol, a natural monoterpenoid and cyclic ether found in eucalyptus species, effectively controls excessive airway mucus secretion and asthma by inhibiting pro-inflammatory cytokines. It serves as an efficacious treatment for non-purulent sinusitis, reducing inflammation and pain when applied topically, and demonstrating leukemic cell-killing capabilities in vitro.Formula:C10H18OPurezza:97.44% - 97.44%Colore e forma:SolidPeso molecolare:154.25Desmethyl Mirtazapine (hydrochloride)
CAS:Desmethyl mirtazapine is a metabolite of the antidepressant mirtazapine.1It is formed from mirtazapine by the cytochrome P450 (CYP) isoform CYP3A4.Formula:C16H18ClN3Colore e forma:SolidPeso molecolare:287.79SB 699551
CAS:SB 699551 is a selective 5-HT5A antagonist (Ki=6.31 nM) that enhances 5-HT neuronal function. It inhibits SERT (Ki=25.12 nM),inhibit breast cancer.Formula:C34H45N3OPurezza:99.83%Colore e forma:SoildPeso molecolare:511.74Ref: TM-T23325L
1mg190,00€5mg471,00€10mg662,00€25mg1.036,00€50mg1.429,00€100mg1.821,00€200mg2.489,00€LEK 8804
CAS:LEK 8804 is a 5-HT(2) receptor antagonist and 5-HT(1A) receptor agonist.Formula:C19H19N3OColore e forma:SolidPeso molecolare:305.37Alosetron
CAS:Alosetron, a 5-HT3 antagonist, is used for the management of severe diarrhea-predominant irritable bowel syndrome (IBS) in women only.Formula:C17H18N4OPurezza:98%Colore e forma:Crystalline PowderPeso molecolare:294.36Triazolomethylindole-3-acetic acid
CAS:Triazolomethylindole-3-acetic acid is a metabolite of Rizatriptan, which acts as an agonist for the serotonin (5-HT) receptor subtypes 5-HT1B and 5-HT1D.Formula:C13H12N4O2Colore e forma:SolidPeso molecolare:256.26Isobutyryl-L-carnitine
CAS:Isobutyryl-L-carnitine is a member of the class of compounds known as acylcarnitines. Isobutyryl-L-carnitine is a product of the acyl-CoA dehydrogenases.Formula:C11H21NO4Purezza:98%Colore e forma:SolidPeso molecolare:231.29MR33317
MR33317 is an inhibitor of acetylcholinesterase with an IC50 value of 41 nM. Additionally, it acts as an agonist for brain 5-HT4 receptors.Formula:C22H28ClN3O2Peso molecolare:401.187Cianopramine hydrochloride
CAS:Cianopramine hydrochloride is a bio-active chemical.Formula:C20H24ClN3Colore e forma:SolidPeso molecolare:341.88(R,R)-Palonosetron Hydrochloride
CAS:(R,R)-Palonosetron Hydrochloride is the active enantiomer of PalonosetronFormula:C19H25ClN2OPurezza:98%Colore e forma:SolidPeso molecolare:332.87R 50595
CAS:R 50595 is a selective non-competitive cisapride antagonist.Formula:C30H35Cl2F2N3O3Purezza:98%Colore e forma:SolidPeso molecolare:594.52Cinanserin hydrochloride
CAS:Cinanserin hydrochloride (SQ 10643) is a 5-HT2 receptor blocker (Ki: 41 nM) and SARS-CoV 3C-like protease inhibitor.Formula:C20H25ClN2OSPurezza:99.57%Colore e forma:SolidPeso molecolare:376.94Zalospirone
CAS:Zalospirone is a 5-HT1A receptor agonist that can be used to study anxiety disorders and major depressive disorder.Formula:C24H29N5O2Purezza:98.24% - 99.82%Colore e forma:SolidPeso molecolare:419.52Peptide 401
CAS:Peptide 401: AMP from bee/wasp venom, triggers histamine release, reduces paw swelling.Formula:C110H192N40O24S4Purezza:98%Colore e forma:SolidPeso molecolare:2587.22Asenapine citrate
CAS:Asenapine citrate: atypical antipsychotic for schizophrenia, bipolar disorder; targets serotonin, adrenoceptors, dopamine, histamine (pKi: 8.2-10.5).Formula:C23H24ClNO8Colore e forma:SolidPeso molecolare:477.89Alverine hydrochloride
CAS:Alverine hydrochloride is a parasympatholytic.Formula:C20H28ClNColore e forma:SolidPeso molecolare:317.9Vortioxetine D8
CAS:Vortioxetine D8 is a deuterium-labeled antidepressant inhibiting 5-HT1A/B, 5-HT3A, 5-HT7 receptors & SERT (Ki: 15-1.6 nM).Formula:C18H22N2SPurezza:98%Colore e forma:SolidPeso molecolare:306.5Serazapine
CAS:Serazapine is a highly specific serotonin (5-HT2) binding inhibitor with anxiolytic activity for the treatment of anxiety disorders.
Formula:C22H23N3O2Purezza:98.71% - 99.57%Colore e forma:SolidPeso molecolare:361.44Donitriptan hydrochloride
CAS:Donitriptan hydrochloride (Donitriptan monohydrochloride) is a potent, high efficacy agonist of 5-HT1B/1D receptors with pKis of 9.4 and 9.3, respectivelyFormula:C23H26ClN5O2Purezza:99.8% - 99.86%Colore e forma:SolidPeso molecolare:439.94Ref: TM-T21666
2mg40,00€5mg49,00€10mg64,00€25mg135,00€50mg240,00€100mg339,00€200mg439,00€500mgPrezzo su richiesta

