
recettore 5-HT
I recettori 5-HT, noti anche come recettori della serotonina, sono un gruppo di recettori accoppiati alle proteine G (GPCR) che mediano gli effetti della serotonina, un neurotrasmettitore coinvolto nella regolazione dell'umore, dell'ansia, del sonno, dell'appetito e di altri processi fisiologici. Questi recettori sono suddivisi in diversi sottotipi, ciascuno con funzioni e proprietà farmacologiche distinte. I modulatori dei recettori 5-HT sono ampiamente studiati per il loro ruolo nel trattamento della depressione, dei disturbi d'ansia e di altre condizioni neuropsichiatriche. Presso CymitQuimica, offriamo una gamma di modulatori dei recettori 5-HT di alta qualità per supportare la tua ricerca in neurofarmacologia, disturbi dell'umore e segnalazione GPCR.
Trovati 1025 prodotti di "recettore 5-HT"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Agomelatine-d6
CAS:Agomelatine D6 (S-20098 D6) is a deuterium-labeled Agomelatine. Agomelatine is a specific agonist of MT1 and MT2 receptors.Formula:C15H17NO2Purezza:98%Colore e forma:SolidPeso molecolare:249.34Quetiapine-d4 hemifumarate
CAS:Quetiapine D4 hemifumarate is the deuterium labeled Quetiapine hemifumarate. Quetiapine hemifumarate is a agonist of 5-HT receptors and a antagonist of dopamine receptor,with ntidepressant and anxiolytic.Formula:C25H29N3O6SPurezza:98%Colore e forma:White SolidPeso molecolare:503.61Ziprasidone amino acid
CAS:Ziprasidone Impurity C is a byproduct of Ziprasidone, an antipsychotic that blocks 5-HT and dopamine receptors.Formula:C21H23ClN4O2SColore e forma:SolidPeso molecolare:430.95Paliperidone Palmitate
CAS:Paliperidone: atypical antipsychotic, dopamine & serotonin antagonist, affects α1/α2 adrenergic and H1 histamine receptors.Formula:C39H57FN4O4Purezza:98%Colore e forma:SolidPeso molecolare:664.89Quetiapine-d8 Fumarate
CAS:Quetiapine-d8 Fumarate is a deuterated compound of Quetiapine Fumarate. Quetiapine Fumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.Formula:C25H21D8N3O6SColore e forma:SolidPeso molecolare:507.63Spiroxatrine
CAS:Spiroxatrine (R 5188) is a 5-HT1α and α2-adrenergic dual antagonist with sedative activity for the study of diseases related to the cardiovascular system.Formula:C22H25N3O3Purezza:99.94%Colore e forma:SolidPeso molecolare:379.45Asenapine hydrochloride
CAS:Asenapine hydrochloride (Org 5222 hydrochloride) is an antagonist of 5-hydroxytryptamine, adrenergic, dopamine, and histamine receptors with antipsychotic effects.Formula:C17H17Cl2NOColore e forma:SolidPeso molecolare:322.23Levomepromazine
CAS:Levomepromazine (Methotrimeprazine) is a Ca2+ release inducer with antiviral, anti-inflammatory, neuroprotective, sedative, and anti-nociceptive activities.Formula:C19H24N2OSPurezza:99.15%Colore e forma:SolidPeso molecolare:328.47Clozapine-d8
CAS:Clozapine-d8 is a deuterium-labeled analog of Clozapine, used as an internal standard for mass spectrometric analysis of this atypical antipsychotic.Formula:C18H19ClN4Colore e forma:SolidPeso molecolare:334.87Nefazodone
CAS:Nefazodone (Nefadar) is an oral antidepressant that is an antagonist of postsynaptic 5-HT 2A receptors and 5-HT 2C receptors, and SNDRI.Formula:C25H32ClN5O2Purezza:99.85%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:470.01Ref: TM-T21451
2mg42,00€5mg60,00€10mg87,00€1mL*10mM (DMSO)95,00€25mg177,00€50mg276,00€100mg422,00€200mg604,00€WAY-100635
CAS:WAY-100635 is a potent 5-HT 1A receptor antagonist pyramidal neuron firing frequency during conditioned reflexes; a dopamine D4 receptor agonist .Formula:C25H34N4O2Purezza:98.972%Colore e forma:SolidPeso molecolare:422.56(Rac)-Rotigotine hydrochloride
CAS:(Rac)-Rotigotine hydrochloride is a racemate of Rotigotine. Rotigotine is a full agonist of dopamine receptor, a partial the 5-HT1A receptor agonist.Formula:C19H26ClNOSColore e forma:SolidPeso molecolare:351.93Alosetron D3 Hydrochloride
CAS:Alosetron D3 (GR 68755 D3) Hydrochloride is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.Formula:C17H19ClN4OPurezza:98%Colore e forma:SolidPeso molecolare:333.83Cariprazine D6
CAS:Cariprazine D6 (RGH-188 D6) is a deuterium-labeled Cariprazine. Cariprazine is an antipsychotic agent (D3 receptors, Ki: 0.085 nM; D2 receptors, Ki: 0.49 nM).Formula:C21H26D6Cl2N4OPurezza:98%Colore e forma:SolidPeso molecolare:433.45Vilazodone-d8
CAS:Vilazodone D8 is a deuterium-labeled vilazodone. Vilazodone is a combined inhibitor of serotonin specific reuptake (SSRI) and agonist of 5-HT1A receptor partial.Formula:C26H27N5O2Purezza:98%Colore e forma:SolidPeso molecolare:449.57Dehydroaripiprazole
CAS:Dehydroaripiprazole (DM-14857), aripiprazole's active metabolite, is formed by CYP3A4 and CYP2D6, with similar antipsychotic effects.Formula:C23H25Cl2N3O2Purezza:98.7%Colore e forma:SolidPeso molecolare:446.37Quetiapine-d8 Hemifumarate
CAS:Quetiapine-d8 Hemifumarate is a deuterated compound of Quetiapine Hemifumarate. Quetiapine Hemifumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.Formula:C25H21D8N3O6SColore e forma:SolidPeso molecolare:507.63Asenapine
CAS:Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, and histamine receptor antagonist with antipsychotic properties for the treatment of schizophreniaFormula:C17H16ClNOPurezza:99.64%Colore e forma:CoaPeso molecolare:285.775-HT3 antagonist 5
CAS:5-HT3 antagonist 5, a quinoxalin-2-carboxamide, blocks 5-HT3 receptors and has antidepressant effects in mice.Formula:C16H13N3O2Purezza:99.84%Colore e forma:SolidPeso molecolare:279.295-HT2B antagonist-1
CAS:Orally active 5-HT2B antagonist; IC50 = 33.4 nM; potential for hepatocellular, cardiovascular, GI disease research.Formula:C11H14BrN5Purezza:99.965%Colore e forma:SolidPeso molecolare:296.17
