
recettore 5-HT
I recettori 5-HT, noti anche come recettori della serotonina, sono un gruppo di recettori accoppiati alle proteine G (GPCR) che mediano gli effetti della serotonina, un neurotrasmettitore coinvolto nella regolazione dell'umore, dell'ansia, del sonno, dell'appetito e di altri processi fisiologici. Questi recettori sono suddivisi in diversi sottotipi, ciascuno con funzioni e proprietà farmacologiche distinte. I modulatori dei recettori 5-HT sono ampiamente studiati per il loro ruolo nel trattamento della depressione, dei disturbi d'ansia e di altre condizioni neuropsichiatriche. Presso CymitQuimica, offriamo una gamma di modulatori dei recettori 5-HT di alta qualità per supportare la tua ricerca in neurofarmacologia, disturbi dell'umore e segnalazione GPCR.
Trovati 1025 prodotti di "recettore 5-HT"
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Metoclopramide
CAS:Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.Formula:C14H22ClN3O2Purezza:99.75%Colore e forma:SolidPeso molecolare:299.80Harmine
CAS:Harmine (Telepathine) is an alkaloid isolated from seeds of Peganum harmala.Formula:C13H12N2OPurezza:98.29% - 99.92%Colore e forma:Off-White SolidPeso molecolare:212.25Ramosetron hydrochloride
CAS:Ramosetron hydrochloride (YM-060) is a serotonin 5-HT3 receptor antagonist. It is used to treat diarrhea-predominant irritable bowel syndrome and nausea.Formula:C17H18ClN3OPurezza:99.95%Colore e forma:SolidPeso molecolare:315.8Cilansetron Hydrochloride
CAS:Cilansetron Hydrochloride can be used for irritable Bowel Syndrome (IBS) with Diarrhea Predominance.Formula:C20H24ClN3O2Colore e forma:SolidPeso molecolare:373.88Amitriptyline
CAS:Amitriptyline: a tricyclic antidepressant used for depression and neuropathic pain.Formula:C20H23NPurezza:98.24% - 99.64%Colore e forma:Crystals SolidPeso molecolare:277.4Trazodone
CAS:Trazodone (AF-1161), a 5-HT 2A/2C receptor antagonist, is used as an antidepressant for treating major anxiety disorders and depressive disorder.Formula:C19H22ClN5OPurezza:99.79% - 99.92%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:371.861-(1-Naphthyl) piperazine hydrochloride
CAS:1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multipleFormula:C14H17ClN2Purezza:98.27%Colore e forma:SolidPeso molecolare:248.75A-582941 dihydrochloride
CAS:A-582941 dihydrochloride (A 582941) is a Selective agonist of α7 nAChR partialFormula:C17H22Cl2N4Purezza:99.55%Colore e forma:SolidPeso molecolare:353.29Ref: TM-T22016
1mg42,00€5mg88,00€10mg120,00€25mg235,00€50mg354,00€100mg533,00€200mg743,00€1mL*10mM (DMSO)87,00€Sertindole
CAS:Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).Formula:C24H26ClFN4OPurezza:99.87% - 99.92%Colore e forma:Off-White To Pale Yellow SolidPeso molecolare:440.94Rizatriptan benzoate
CAS:Rizatriptan benzoate (MK-462 Benzoate) selectively binds to and activates serotonin (5-HT) 1B receptors and 5-HT 1D receptors providing relief of migraineFormula:C22H25N5O2Purezza:99% - 99.79%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:391.47Ref: TM-T1512
10mg44,00€25mg74,00€50mg119,00€100mg173,00€200mg259,00€500mg437,00€1mL*10mM (DMSO)48,00€PU02
CAS:PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.Formula:C16H12N4SPurezza:99.35%Colore e forma:SolidPeso molecolare:292.36Pimavanserin tartrate
CAS:Pimavanserin tartrate is a potent 5-HT 2A receptor inverse agonist used to treat Parkinson's disease-related psychosis.Cost-effective and quality-assured.Formula:C50H68F2N6O4·C4H6O6Purezza:99.24% - 99.98%Colore e forma:SolidPeso molecolare:1005.27-Amino-4-(trifluoromethyl)coumarin
CAS:7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) is a 5-Hydroxytryptamine Receptor Subtype 1E (HTR1E) antagonist.Formula:C10H6F3NO2Purezza:97.31% - 97.84%Colore e forma:Yellow PowderPeso molecolare:229.16F-15599
CAS:F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).Formula:C19H21ClF2N4OPurezza:98.72%Colore e forma:SolidPeso molecolare:394.85Ref: TM-T7281
1mg49,00€5mg92,00€10mg152,00€25mg295,00€50mg477,00€100mg715,00€200mg982,00€1mL*10mM (DMSO)104,00€Pirenperone
CAS:Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.Formula:C23H24FN3O2Purezza:99.2%Colore e forma:SolidPeso molecolare:393.45Syk Inhibitor II dihydrochloride dihydrate
CAS:Potent, selective ATP-competitive Syk Inhibitor II (IC50: 41 nM), with anti-allergic properties, in dihydrochloride dihydrate form.Formula:C14H21Cl2F3N6O3Colore e forma:SolidPeso molecolare:449.265-HT1A modulator 2 hydrochloride
CAS:5-HT1A modulator 2 hydrochloride is a modulator of 5-HT1A showing an affinity of 53 nM for 5-HT1A binding.Formula:C11H16ClNOPurezza:98.5%Colore e forma:SolidPeso molecolare:213.7Pardoprunox hydrochloride
CAS:Pardoprunox hydrochloride (SLV-308 hydrochloride) is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1)Formula:C12H16ClN3O2Purezza:98.95% - 99.13%Colore e forma:SolidPeso molecolare:269.73Pimavanserin
CAS:Pimavanserin is a potent 5-HT2A inverse agonist, used to treat Parkinson's psychosis.Formula:C25H34FN3O2Purezza:97.84% - 99.69%Colore e forma:Pale Yellow To Pale Orange SolidPeso molecolare:427.55Olanzapine HCl
CAS:Olanzapine HCl, an FDA-approved atypical antipsychotic for schizophrenia and bipolar disorder, resembles clozapine and quetiapine.Formula:C17H21ClN4SColore e forma:SolidPeso molecolare:348.89
