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Recettore adrenergico

Recettore adrenergico

I recettori adrenergici sono GPCR attivati dalle catecolamine, come l'adrenalina e la noradrenalina. Questi recettori sono classificati in sottotipi alfa e beta, ognuno dei quali svolge un ruolo chiave nella regolazione della frequenza cardiaca, della pressione sanguigna e della risposta di lotta o fuga. I modulatori dei recettori adrenergici sono essenziali nel trattamento delle malattie cardiovascolari, dell'asma e dei disturbi d'ansia. Presso CymitQuimica, offriamo una vasta gamma di modulatori dei recettori adrenergici di alta qualità per supportare la tua ricerca in endocrinologia, farmacologia cardiovascolare e risposta allo stress.

Sottocategorie di "Recettore adrenergico"

Trovati 717 prodotti di "Recettore adrenergico"

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  • Iobenguane sulfate

    CAS:
    Iobenguane sulfate is used in radioiodinated form to diagnose and treat adrenergic tumors.
    Formula:C8H10IN3H2O4S
    Purezza:99.04%
    Colore e forma:Solid
    Peso molecolare:324.12
  • Phentolamine mesylate

    CAS:
    Phentolamine mesylate: nonselective alpha-blocker for hypertension, pheochromocytoma, Raynaud's, frostbite, impotence, and vascular issues.
    Formula:C17H19N3O·CH4O3S
    Purezza:99.87% - >99.99%
    Colore e forma:By The Metabolic Processes Of Bacillus Subtilis And Licheniformis
    Peso molecolare:377.46
  • Salmeterol

    CAS:
    Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.
    Formula:C25H37NO4
    Purezza:99.2% - 99.9%
    Colore e forma:Solid
    Peso molecolare:415.57
  • Moxonidine

    CAS:
    Moxonidine (BDF5895) is a selective agonist at the imidazoline receptor subtype 1, acting as an antihypertensive drug.
    Formula:C9H12ClN5O
    Purezza:99.81% - 99.94%
    Colore e forma:Crystal
    Peso molecolare:241.68
  • CXCR7 antagonist-1

    CAS:
    <p>CXCR7 antagonist-1 is a specific antagonist of the binding of the SDF-1 chemokine or I-TAC to the chemokine receptor CXCR7.</p>
    Formula:C21H19FN6O
    Purezza:99.93%
    Colore e forma:Solid
    Peso molecolare:390.41
  • 2-(1-Piperazinyl)pyrimidine

    CAS:
    2-(1-Piperazinyl)pyrimidine is used as an anti-anxiety drug.
    Formula:C8H12N4
    Purezza:98.46%
    Colore e forma:Liquid - Crystal - Lump
    Peso molecolare:164.21
  • Brefonalol HCl


    Brefonalol HCl, ADRA blocker for neurological/cardiovascular issues, treats angina, arrhythmias, hypertension.
    Formula:C22H29ClN2O2
    Purezza:99.98%
    Colore e forma:Solid
    Peso molecolare:388.93
  • Naftopidil

    CAS:
    Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-
    Formula:C24H28N2O3
    Purezza:99.60% - 99.97%
    Colore e forma:White Crystalline Powder
    Peso molecolare:392.49
  • Bambuterol hydrochloride

    CAS:
    Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.
    Formula:C18H30ClN3O5
    Purezza:99.53% - 99.61%
    Colore e forma:White Solid
    Peso molecolare:403.91
  • Fenspiride hydrochloride

    CAS:
    Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.
    Formula:C15H20N2O2·HCl
    Purezza:99.64% - 99.92%
    Colore e forma:Solid
    Peso molecolare:296.79
  • Terazosin hydrochloride

    CAS:
    <p>Terazosin HCl (Hytrin) treats BPH and hypertension by blocking alpha1, affecting bladder and vessel muscles.</p>
    Formula:C19H26ClN5O4
    Purezza:99.69% - 99.91%
    Colore e forma:Solid
    Peso molecolare:423.89
  • Dabuzalgron

    CAS:
    Dabuzalgron (Ro 115-1240) is an orally active selective alpha-1A adrenergic receptor agonist used to treat urinary incontinence.
    Formula:C12H16ClN3O3S
    Purezza:98.35%
    Colore e forma:Solid
    Peso molecolare:317.79
  • Methyldopa

    CAS:
    Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or
    Formula:C10H13NO4
    Purezza:98.95% - 99.86%
    Colore e forma:Less Or Almost Colorless Crystals Or White To Yellowish-White Fine
    Peso molecolare:211.21
  • Terbutaline Sulfate

    CAS:
    Terbutaline Sulfate (Terbutaline hemisulfate) is a selective beta-2 adrenergic agonist used as a bronchodilator and tocolytic.
    Formula:C12H19NO3H2SO4
    Purezza:99.47% - 99.94%
    Colore e forma:Crystalline Powder
    Peso molecolare:274.32
  • Tamsulosin hydrochloride

    CAS:
    <p>Tamsulosin hydrochloride (Flomax hydrochloride) is the hydrochloride salt of tamsulosin, a sulfonamide derivative with α1 adrenergic antagonist activity.</p>
    Formula:C20H29ClN2O5S
    Purezza:95.45% - 99.95%
    Colore e forma:White To Off-White Solid
    Peso molecolare:444.97
  • Perphenazine

    CAS:
    <p>Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.</p>
    Formula:C21H26ClN3OS
    Purezza:99.3% - 99.99%
    Colore e forma:Solid
    Peso molecolare:403.97
  • Urapidil hydrochloride

    CAS:
    Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.
    Formula:C20H29N5O3·HCl
    Purezza:99.58%
    Colore e forma:White Or Off-White Crystalline Powder
    Peso molecolare:423.94
  • Isoprenaline hydrochloride

    CAS:
    Isoprenaline hydrochloride (NCI-c55630) is a potent beta-adrenergic agonist with the peripheral vasodilator, bronchodilator, and cardiac stimulating properties.
    Formula:C11H18ClNO3
    Purezza:98% - 99.65%
    Colore e forma:Turn Brownish-Pink Upon Prolonged Exposure To Air (Ntp 1992)
    Peso molecolare:247.719
  • Blonanserin

    CAS:
    Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.
    Formula:C23H30FN3
    Purezza:99.85%
    Colore e forma:Solid
    Peso molecolare:367.5
  • Olanzapine

    CAS:
    Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.
    Formula:C17H20N4S
    Purezza:99.86% - ≥95%
    Colore e forma:Yellowish Crystalline Powder
    Peso molecolare:312.43
  • PF-610355 HCl


    <p>PF-610355 HCl is a selective and potent β2-adrenergic receptor agonist, a bronchodilator, and for asthma and chronic obstructive pulmonary disease.</p>
    Formula:C19H22ClN7O6
    Purezza:97.97%
    Colore e forma:Solid
    Peso molecolare:479.87
  • Acebutolol hydrochloride

    CAS:
    <p>Acebutolol HCl: cardioselective beta-blocker, minimal bronchial impact, intrinsic sympathomimetic, treats hypertension &amp; ventricular arrhythmias.</p>
    Formula:C18H29ClN2O4
    Purezza:99.92% - >99.99%
    Colore e forma:White Or Slightly Off-White Crystalline Powder Solid
    Peso molecolare:372.89
  • Heptaminol hydrochloride

    CAS:
    Heptaminol hydrochloride (RP-2831 hydrochloride), a vasoconstrictor, is used in the therapy of hypotension, especially orthostatic hypotension.
    Formula:C8H20ClNO
    Purezza:98.61%
    Colore e forma:White Crystalline Powder
    Peso molecolare:181.71
  • DSP-4 hydrochloride

    CAS:
    <p>DSP-4 hydrochloride is a neurotoxin that degrades noradrenergic neurons in rats and crosses the blood-brain barrier.</p>
    Formula:C11H16BrCl2N
    Purezza:99.9%
    Colore e forma:Solid
    Peso molecolare:313.06
  • Ifenprodil Tartrate

    CAS:
    Ifenprodil is a selective NMDA receptor (glutamate) antagonist.
    Formula:C21H27NO2C4H6O6
    Purezza:99.02% - 99.55%
    Colore e forma:Solid
    Peso molecolare:400.49
  • Synephrine

    CAS:
    Synephrine (Oxedrine) is sympathetic alpha-adrenergic agonist used as a vasoconstrictor in circulatory failure, asthma, nasal congestion, and glaucoma.
    Formula:C9H13NO2
    Purezza:99.274% - >99.99%
    Colore e forma:Solid
    Peso molecolare:167.21
  • Mirabegron

    CAS:
    <p>Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.</p>
    Formula:C21H24N4O2S
    Purezza:99.64%
    Colore e forma:Light Yellow To Yellow Solid
    Peso molecolare:396.51
  • Noradrenaline bitartrate

    CAS:
    <p>Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors.</p>
    Formula:C12H19NO10
    Purezza:99.53% - >99.99%
    Colore e forma:Solid
    Peso molecolare:337.28
  • Ifenprodil

    CAS:
    Ifenprodil (RC61-91) inhibits NMDA receptor subunits GluN1 & GluN2B, GIRK channels, and affects alpha1, serotonin, sigma receptors.
    Formula:C21H27NO2
    Purezza:99.58%
    Colore e forma:White Crystalline Powder
    Peso molecolare:325.44
  • Dopexamine hydrochloride

    CAS:
    Dopexamine hydrochloride (FPL60278AR) is a β2-adrenoceptor agonist that modulates inflammation and protects organs without affecting hemodynamics.
    Formula:C22H34Cl2N2O2
    Purezza:98.55%
    Colore e forma:Solid
    Peso molecolare:429.42
  • Nylidrin hydrochloride

    CAS:
    Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells & human basophils.
    Formula:C19H26ClNO2
    Purezza:99.35%
    Colore e forma:Solid
    Peso molecolare:335.87
  • Trifluoperazine dihydrochloride

    CAS:
    Trifluoperazine dihydrochloride (SKF5019) is a potent dopamine D2 receptor inhibitor used as an antipsychotic and an antiemetic.
    Formula:C21H26Cl2F3N3S
    Purezza:99.57% - 99.96%
    Colore e forma:Cream Fine Powder
    Peso molecolare:480.43
  • (3aR,9aR)-Fluparoxan

    CAS:
    <p>(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Formula:C10H10FNO2
    Purezza:97.82%
    Colore e forma:Soild
    Peso molecolare:195.19
  • DL-Norepinephrine hydrochloride

    CAS:
    DL-Norepinephrine hydrochloride (DL-lysine) is a high-affinity basic amino acid substrate of amino acid transporter b0 + with a Km value in the range of 100-400
    Formula:C8H12ClNO3
    Purezza:98.45% - 98.82%
    Colore e forma:Solid
    Peso molecolare:205.639
  • Labetalol hydrochloride

    CAS:
    Labetalol hydrochloride (Sch-15719W), a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.
    Formula:C19H25ClN2O3
    Purezza:99.54% - 99.85%
    Colore e forma:Solid
    Peso molecolare:364.87
  • Alfuzosin hydrochloride

    CAS:
    <p>Alfuzosin hydrochloride (Alfuzosin HCl) is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).</p>
    Formula:C19H27N5O4·HCl
    Purezza:99.78%
    Colore e forma:White To Off-White Solid
    Peso molecolare:425.91
  • Indacaterol maleate

    CAS:
    Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.
    Formula:C28H32N2O7
    Purezza:99.03% - 99.67%
    Colore e forma:Solid
    Peso molecolare:508.56
  • Clonidine hydrochloride

    CAS:
    Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.
    Formula:C9H10Cl3N3
    Purezza:99.16% - 99.86%
    Colore e forma:Solid
    Peso molecolare:266.55
  • Silodosin

    CAS:
    Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.
    Formula:C25H32F3N3O4
    Purezza:99.282% - 99.76%
    Colore e forma:Colorless To Pink Solid
    Peso molecolare:495.53
  • Carvedilol phosphate hemihydrate

    CAS:
    Carvedilol phosphate hemihydrate (BM 14190 phosphate hemihydrate) is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent.
    Formula:C24H26N2O4·5H2O·H3O4P
    Purezza:99.24% - 99.98%
    Colore e forma:Solid
    Peso molecolare:513.49
  • Octopamine hydrochloride

    CAS:
    Octopamine hydrochloride is akin to noradrenaline and acts as a neurohormone, neurotransmitter, and neuromodulator in invertebrates.
    Formula:C8H12ClNO2
    Purezza:98.87% - 99.85%
    Colore e forma:White Or Off-White Solid
    Peso molecolare:189.64
  • 2',5'-Dideoxyadenosine

    CAS:
    2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).
    Formula:C10H13N5O2
    Purezza:99.55%
    Colore e forma:White Solid
    Peso molecolare:235.24
  • Metaproterenol hemisulfate

    CAS:
    Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.
    Formula:C11H17NO3·5H2O4S
    Purezza:98.53% - 99.74%
    Colore e forma:Solid
    Peso molecolare:260.3
  • Tizanidine hydrochloride

    CAS:
    <p>Tizanidine hydrochloride (Tizanidine HCl), an α2-adrenergic receptor agonist, inhibits neurotransmitter release from CNS noradrenergic neurons.</p>
    Formula:C9H9Cl2N5S
    Purezza:99.96%
    Colore e forma:Solid White
    Peso molecolare:290.17
  • Moxisylyte hydrochloride

    CAS:
    Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.
    Formula:C16H26ClNO3
    Purezza:99.94% - ≥95%
    Colore e forma:Solid
    Peso molecolare:315.84
  • Adrenalone hydrochloride

    CAS:
    Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.
    Formula:C9H11NO3·HCl
    Purezza:99.94%
    Colore e forma:Solid
    Peso molecolare:217.65
  • Fluparoxan hydrochloride

    CAS:
    <p>Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Formula:C10H11ClFNO2
    Purezza:99.98%
    Colore e forma:Soild
    Peso molecolare:231.65
  • Isoxsuprine hydrochloride

    CAS:
    Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.
    Formula:C18H24ClNO3
    Purezza:99.38%
    Colore e forma:Crystals From Water Solid
    Peso molecolare:337.84
  • Nicergoline

    CAS:
    Nicergoline (Nicergolinum) is an ergot derivative used to treat senile dementia and other disorders with vascular origins.
    Formula:C24H26BrN3O3
    Purezza:98% - 99.80%
    Colore e forma:Solid
    Peso molecolare:484.39
  • Nebivolol hydrochloride

    CAS:
    <p>Nebivolol hydrochloride is a beta-1 blocker and vasodilator treating hypertension and heart failure in the elderly.</p>
    Formula:C22H25F2NO4·HCl
    Purezza:99.77% - >99.99%
    Colore e forma:White To Off-White Powder
    Peso molecolare:441.90