
Recettore adrenergico
I recettori adrenergici sono GPCR attivati dalle catecolamine, come l'adrenalina e la noradrenalina. Questi recettori sono classificati in sottotipi alfa e beta, ognuno dei quali svolge un ruolo chiave nella regolazione della frequenza cardiaca, della pressione sanguigna e della risposta di lotta o fuga. I modulatori dei recettori adrenergici sono essenziali nel trattamento delle malattie cardiovascolari, dell'asma e dei disturbi d'ansia. Presso CymitQuimica, offriamo una vasta gamma di modulatori dei recettori adrenergici di alta qualità per supportare la tua ricerca in endocrinologia, farmacologia cardiovascolare e risposta allo stress.
Sottocategorie di "Recettore adrenergico"
Trovati 736 prodotti per "Recettore adrenergico".
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Iobenguane sulfate
CAS:Iobenguane sulfate is used in radioiodinated form to diagnose and treat adrenergic tumors.Formula:C8H10IN3H2O4SPurezza:99.04%Colore e forma:SolidPeso molecolare:324.12Ref: TM-T15588
5mg66,00€1mL*10mM (DMSO)73,00€10mg96,00€25mg197,00€50mg354,00€100mg530,00€500mg1.153,00€Propafenone
CAS:Propafenone: a drug for ventricular arrhythmias with mild beta-blocker activity, prolongs refractory period, and reduces heart automaticity.Formula:C21H27NO3Purezza:99.02%Colore e forma:SolidPeso molecolare:341.44Naftopidil
CAS:Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-Formula:C24H28N2O3Purezza:99.60% - 99.97%Colore e forma:SolidPeso molecolare:392.49Moxonidine
CAS:Moxonidine (BDF5895) is a selective agonist at the imidazoline receptor subtype 1, acting as an antihypertensive drug.Formula:C9H12ClN5OPurezza:99.81% - 99.94%Colore e forma:White SolidPeso molecolare:241.68Dabuzalgron
CAS:Dabuzalgron (Ro 115-1240) is an orally active selective alpha-1A adrenergic receptor agonist used to treat urinary incontinence.Formula:C12H16ClN3O3SPurezza:98.35%Colore e forma:SolidPeso molecolare:317.79Ref: TM-T10952
1mg35,00€5mg79,00€1mL*10mM (DMSO)86,00€10mg128,00€25mg200,00€50mg299,00€100mg432,00€200mg602,00€Nebivolol hydrochloride
CAS:Nebivolol hydrochloride is a beta-1 blocker and vasodilator treating hypertension and heart failure in the elderly.Formula:C22H25F2NO4·HClPurezza:99.77% - >99.99%Colore e forma:White SolidPeso molecolare:441.90Brefonalol HCl
Brefonalol HCl, ADRA blocker for neurological/cardiovascular issues, treats angina, arrhythmias, hypertension.Formula:C22H29ClN2O2Purezza:99.98%Colore e forma:SolidPeso molecolare:388.93Urapidil hydrochloride
CAS:Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.Formula:C20H29N5O3·HClPurezza:99.58%Colore e forma:SolidPeso molecolare:423.94Olanzapine
CAS:Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.Formula:C17H20N4SPurezza:99.86% - ≥95%Colore e forma:SolidPeso molecolare:312.43Fenspiride hydrochloride
CAS:Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.Formula:C15H20N2O2·HClPurezza:99.64% - 99.92%Colore e forma:SolidPeso molecolare:296.79Heptaminol hydrochloride
CAS:Heptaminol hydrochloride (RP-2831 hydrochloride), a vasoconstrictor, is used in the therapy of hypotension, especially orthostatic hypotension.Formula:C8H20ClNOPurezza:98.61%Colore e forma:SolidPeso molecolare:181.71Terazosin hydrochloride
CAS:Terazosin HCl (Hytrin) treats BPH and hypertension by blocking alpha1, affecting bladder and vessel muscles.Formula:C19H26ClN5O4Purezza:99.68% - 99.91%Colore e forma:SolidPeso molecolare:423.89Ifenprodil
CAS:Ifenprodil (RC61-91) inhibits NMDA receptor subunits GluN1 & GluN2B, GIRK channels, and affects alpha1, serotonin, sigma receptors.Formula:C21H27NO2Purezza:99.58%Colore e forma:White Crystalline PowderPeso molecolare:325.44Ref: TM-T1186L
1mg63,00€5mg135,00€1mL*10mM (DMSO)141,00€10mg197,00€25mg323,00€50mg462,00€100mg640,00€Phentolamine mesylate
CAS:Phentolamine mesylate: nonselective alpha-blocker for hypertension, pheochromocytoma, Raynaud's, frostbite, impotence, and vascular issues.Formula:C17H19N3O·CH4O3SPurezza:99.87% - >99.99%Colore e forma:By The Metabolic Processes Of Bacillus Subtilis And LicheniformisPeso molecolare:377.46Methyldopa
CAS:Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive orFormula:C10H13NO4Purezza:98.95% - 99.86%Colore e forma:SolidPeso molecolare:211.21Tamsulosin hydrochloride
CAS:Tamsulosin hydrochloride (Flomax hydrochloride) is the hydrochloride salt of tamsulosin, a sulfonamide derivative with α1 adrenergic antagonist activity.Formula:C20H29ClN2O5SPurezza:97.16% - 99.98%Colore e forma:White SolidPeso molecolare:444.97Alfuzosin hydrochloride
CAS:Alfuzosin hydrochloride (Alfuzosin HCl) is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).Formula:C19H27N5O4·HClPurezza:99.78%Colore e forma:White To Off-White SolidPeso molecolare:425.91PF-610355 HCl
PF-610355 HCl is a selective and potent β2-adrenergic receptor agonist, a bronchodilator, and for asthma and chronic obstructive pulmonary disease.Formula:C19H22ClN7O6Purezza:97.97%Colore e forma:SolidPeso molecolare:479.87Blonanserin
CAS:Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.Formula:C23H30FN3Purezza:99.85% - 99.99%Colore e forma:SolidPeso molecolare:367.50Synephrine
CAS:Synephrine (Oxedrine) is sympathetic alpha-adrenergic agonist used as a vasoconstrictor in circulatory failure, asthma, nasal congestion, and glaucoma.Formula:C9H13NO2Purezza:99.27% - >99.99%Colore e forma:SolidPeso molecolare:167.21Bambuterol hydrochloride
CAS:Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.Formula:C18H30ClN3O5Purezza:99.53% - 99.61%Colore e forma:SolidPeso molecolare:403.91Acebutolol hydrochloride
CAS:Acebutolol HCl: cardioselective beta-blocker, minimal bronchial impact, intrinsic sympathomimetic, treats hypertension & ventricular arrhythmias.Formula:C18H29ClN2O4Purezza:99.92% - >99.99%Colore e forma:SolidPeso molecolare:372.89Isoprenaline hydrochloride
CAS:Isoprenaline hydrochloride (NCI-c55630) is a potent beta-adrenergic agonist with the peripheral vasodilator, bronchodilator, and cardiac stimulating properties.Formula:C11H18ClNO3Purezza:98% - 99.65%Colore e forma:Turn Brownish-Pink Upon Prolonged Exposure To Air (Ntp 1992)Peso molecolare:247.719Tizanidine hydrochloride
CAS:Tizanidine hydrochloride (Tizanidine HCl), an α2-adrenergic receptor agonist, inhibits neurotransmitter release from CNS noradrenergic neurons.Formula:C9H9Cl2N5SPurezza:99.96%Colore e forma:SolidPeso molecolare:290.17Ref: TM-T0290
1mL*10mM (DMSO)35,00€10mg49,00€25mg60,00€50mg90,00€100mg100,00€200mg126,00€500mg200,00€Labetalol hydrochloride
CAS:Labetalol hydrochloride (Sch-15719W), a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.Formula:C19H25ClN2O3Purezza:99.54% - 99.81%Colore e forma:SolidPeso molecolare:364.87DSP-4 hydrochloride
CAS:DSP-4 hydrochloride is a neurotoxin that degrades noradrenergic neurons in rats and crosses the blood-brain barrier.Formula:C11H16BrCl2NPurezza:99.9%Colore e forma:White SolidPeso molecolare:313.06CXCR7 antagonist-1
CAS:CXCR7 antagonist-1 is a specific antagonist of the binding of the SDF-1 chemokine or I-TAC to the chemokine receptor CXCR7.Formula:C21H19FN6OPurezza:99.93%Colore e forma:Red SolidPeso molecolare:390.41Carvedilol phosphate hemihydrate
CAS:Carvedilol phosphate hemihydrate (BM 14190 phosphate hemihydrate) is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent.Formula:C24H26N2O4·5H2O·H3O4PPurezza:99.24% - 99.98%Colore e forma:White SolidPeso molecolare:513.49Mirabegron
CAS:Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.Formula:C21H24N4O2SPurezza:99.64%Colore e forma:SolidPeso molecolare:396.51Terbutaline Sulfate
CAS:Terbutaline Sulfate (Terbutaline hemisulfate) is a selective beta-2 adrenergic agonist used as a bronchodilator and tocolytic.Formula:C12H19NO3H2SO4Purezza:99.47% - 99.94%Colore e forma:Crystalline PowderPeso molecolare:274.32(3aR,9aR)-Fluparoxan
CAS:(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmentalFormula:C10H10FNO2Purezza:97.82%Colore e forma:SolidPeso molecolare:195.19Dopexamine hydrochloride
CAS:Dopexamine hydrochloride (FPL60278AR) is a β2-adrenoceptor agonist that modulates inflammation and protects organs without affecting hemodynamics.Formula:C22H34Cl2N2O2Purezza:98.55%Colore e forma:SolidPeso molecolare:429.42Trifluoperazine dihydrochloride
CAS:Trifluoperazine dihydrochloride (SKF5019) is a potent dopamine D2 receptor inhibitor used as an antipsychotic and an antiemetic.Formula:C21H26Cl2F3N3SPurezza:99.57% - 99.96%Colore e forma:SolidPeso molecolare:480.43Isoxsuprine hydrochloride
CAS:Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.Formula:C18H24ClNO3Purezza:99.38%Colore e forma:Crystals From Water SolidPeso molecolare:337.84Nylidrin hydrochloride
CAS:Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells & human basophils.Formula:C19H26ClNO2Purezza:99.35%Colore e forma:White SolidPeso molecolare:335.872',5'-Dideoxyadenosine
CAS:2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).Formula:C10H13N5O2Purezza:99.55%Colore e forma:SolidPeso molecolare:235.24Upidosin
CAS:Upidosin (SB-216469), a uroselective α1 blocker: Ki α1a=0.34 nM, α1b=3.9 nM, α1d=1.5 nM, α2=33.3 nM.Formula:C31H33N3O4Purezza:99.66%Colore e forma:SolidPeso molecolare:511.61DL-Norepinephrine hydrochloride
CAS:DL-Norepinephrine hydrochloride (DL-lysine) is a high-affinity basic amino acid substrate of amino acid transporter b0 + with a Km value in the range of 100-400Formula:C8H12ClNO3Purezza:98.45% - 98.82%Colore e forma:Yellow SolidPeso molecolare:205.64Moxisylyte hydrochloride
CAS:Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.Formula:C16H26ClNO3Purezza:99.94% - ≥95%Colore e forma:SolidPeso molecolare:315.84Salmeterol
CAS:Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.Formula:C25H37NO4Purezza:99.2% - 99.9%Colore e forma:SolidPeso molecolare:415.57Indacaterol maleate
CAS:Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.Formula:C28H32N2O7Purezza:99.03% - 99.67%Colore e forma:SolidPeso molecolare:508.56Clonidine hydrochloride
CAS:Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.Formula:C9H10Cl3N3Purezza:99.16% - 99.86%Colore e forma:SolidPeso molecolare:266.55Silodosin
CAS:Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.Formula:C25H32F3N3O4Purezza:99.28% - 99.76%Colore e forma:White SolidPeso molecolare:495.53Ref: TM-T1504
5mg34,00€1mL*10mM (DMSO)35,00€10mg50,00€25mg73,00€50mg92,00€100mg99,00€200mg126,00€1500mg267,00€Perphenazine
CAS:Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.Formula:C21H26ClN3OSPurezza:99.3% - 99.99%Colore e forma:White SolidPeso molecolare:403.97Octopamine hydrochloride
CAS:Octopamine hydrochloride is akin to noradrenaline and acts as a neurohormone, neurotransmitter, and neuromodulator in invertebrates.Formula:C8H12ClNO2Purezza:98.87% - 99.85%Colore e forma:Yellow SolidPeso molecolare:189.64Adrenalone hydrochloride
CAS:Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.Formula:C9H11NO3·HClPurezza:99.94%Colore e forma:SolidPeso molecolare:217.65Metaproterenol hemisulfate
CAS:Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.Formula:C11H17NO3·5H2O4SPurezza:98.53% - 99.74%Colore e forma:White SolidPeso molecolare:260.3Nicergoline
CAS:Nicergoline (Nicergolinum) is an ergot derivative used to treat senile dementia and other disorders with vascular origins.Formula:C24H26BrN3O3Purezza:98% - 99.80%Colore e forma:White SolidPeso molecolare:484.39Fluparoxan hydrochloride
CAS:Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmentalFormula:C10H11ClFNO2Purezza:99.98%Colore e forma:SolidPeso molecolare:231.65Clozapine
CAS:Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.Formula:C18H19ClN4Purezza:99.91% - 99.93%Colore e forma:Yellow SolidPeso molecolare:326.82
