
Recettore adrenergico
I recettori adrenergici sono GPCR attivati dalle catecolamine, come l'adrenalina e la noradrenalina. Questi recettori sono classificati in sottotipi alfa e beta, ognuno dei quali svolge un ruolo chiave nella regolazione della frequenza cardiaca, della pressione sanguigna e della risposta di lotta o fuga. I modulatori dei recettori adrenergici sono essenziali nel trattamento delle malattie cardiovascolari, dell'asma e dei disturbi d'ansia. Presso CymitQuimica, offriamo una vasta gamma di modulatori dei recettori adrenergici di alta qualità per supportare la tua ricerca in endocrinologia, farmacologia cardiovascolare e risposta allo stress.
Sottocategorie di "Recettore adrenergico"
Trovati 728 prodotti di "Recettore adrenergico"
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Nolomirole HCl
CAS:<p>Nolomirole HCl (CHF 1035) is a novel selective dopamine agonist with oral activity and inhibitory effects on norepinephrine release, which can be used to study</p>Formula:C19H28ClNO4Purezza:99.03% - >99.99%Colore e forma:SolidPeso molecolare:369.88Bunazosin Hydrochloride
CAS:Bunazosin Hydrochloride (E 1015) is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an ocular hypotensive drug.Formula:C19H28ClN5O3Purezza:99.12%Colore e forma:SolidPeso molecolare:409.91GW-597901
CAS:GW-597901, an β2 adrenergic receptor agonist, is used potentially for the treatment of asthma and chronic obstructive.Formula:C25H38N2O6SColore e forma:SolidPeso molecolare:494.64Abediterol
CAS:Abediterol (LAS100977): potent, long-acting beta-2 agonist for asthma and COPD treatment.Formula:C25H30F2N2O4Colore e forma:SolidPeso molecolare:460.51Fiduxosin
CAS:Fiduxosin is a selective and potent α1-adrenoceptor antagonist with inhibitory effects on α1a-adrenoceptor, α1b-adrenoceptor and α1d-adrenoceptor, with KiFormula:C30H29N5O4SPurezza:99.73%Colore e forma:SolidPeso molecolare:555.65Mefenidil
CAS:Mefenidil (McN-2378), a selective cerebral vasodilator, was shown to increase CBF in healthy brains without stimulating O2 uptake in a dog anesthesia model.Formula:C12H11N3Purezza:98.27%Colore e forma:SolidPeso molecolare:197.24Fiduxosin hydrochloride
CAS:Fiduxosin hydrochloride is an alpha 1a-adrenoceptor antagonist that may be useful in the treatment of Benign Prostatic Hyperplasia.Formula:C30H30ClN5O4SColore e forma:SolidPeso molecolare:592.11Epinephrine HCl
CAS:Epinephrine HCl is a hormone and neurotransmitter secreted by the adrenal medulla, agonist of α-adrenergic and β-adrenergic receptor.Formula:C9H14ClNO3Purezza:99.48%Colore e forma:SolidPeso molecolare:219.67L-796568 dihydrochloride
CAS:L-796568: potent β3 agonist (EC50 = 3.6 nM), >600-fold selectivity vs β1/β2, good oral bioavailability, long action.Formula:C31H29Cl2F3N4O3S2Colore e forma:SolidPeso molecolare:697.62β3-AR agonist 2
CAS:β3-AR agonist 2 is a potent and selective agonist of β3-adrenergic receptor (β3-AR with an EC50 of 8 nM).Formula:C27H38N4O7SPurezza:98%Colore e forma:SolidPeso molecolare:562.68BMS-194449
CAS:BMS-194449 is a full beta 3 agonist.Formula:C24H24F4N2O6SColore e forma:SolidPeso molecolare:544.52Ro-70-0004
CAS:Ro-70-0004 is a selective antagonist of alpha1A-adrenoceptor.Formula:C20H24F4N4O3Colore e forma:SolidPeso molecolare:444.42N-5984
CAS:<p>N-5984, a β3-adrenergic receptor agonist, is used potentially for the treatment of obesity, overactive bladder and type 2 diabetes.</p>Formula:C20H22ClNO5Purezza:98%Colore e forma:SolidPeso molecolare:391.85Indacaterol acetate
CAS:Indacaterol acetate is an ultra-long-acting beta-adrenoceptor agonist.Formula:C26H32N2O5Colore e forma:SolidPeso molecolare:452.54BI-167107
CAS:BI-167107 is a high affinity, full agonist that binds to the β2 adrenergic receptor (β2AR, Kd of 84 pM).Formula:C21H26N2O4Colore e forma:SolidPeso molecolare:370.444-hydroxy Nebivolol hydrochloride
CAS:4-Hydroxy Nebivolol, a primary metabolite of Nebivolol, results from the enzymatic hydroxylation of Nebivolol by the cytochrome P450 (CYP) isoform CYP2D6.Formula:C22H25F2NO5HClColore e forma:SolidPeso molecolare:457.9Vemtoberant
CAS:Vemtoberant is a β3 adrenergic antagonist used in β3-related disorder research like heart failure.Formula:C29H37N3O8S2Colore e forma:SolidPeso molecolare:619.75AGN 192836
CAS:AGN 192836 is a potent and selective α2 adrenergic agonist (EC50s: 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor).Formula:C12H13N3O2Colore e forma:SolidPeso molecolare:231.25AR-08
CAS:<p>AR-08 is a potent α2-adrenergic receptor agonist for the study of ADHD and attention deficit.</p>Formula:C12H12N6Purezza:99.7%Colore e forma:SolidPeso molecolare:240.26N-5984 Hydrochloride
CAS:N-5984 Hydrochloride is a beta3-AR agonist.Formula:C20H23Cl2NO5Colore e forma:SolidPeso molecolare:428.31
