CymitQuimica logo
Recettore adrenergico

Recettore adrenergico

I recettori adrenergici sono GPCR attivati dalle catecolamine, come l'adrenalina e la noradrenalina. Questi recettori sono classificati in sottotipi alfa e beta, ognuno dei quali svolge un ruolo chiave nella regolazione della frequenza cardiaca, della pressione sanguigna e della risposta di lotta o fuga. I modulatori dei recettori adrenergici sono essenziali nel trattamento delle malattie cardiovascolari, dell'asma e dei disturbi d'ansia. Presso CymitQuimica, offriamo una vasta gamma di modulatori dei recettori adrenergici di alta qualità per supportare la tua ricerca in endocrinologia, farmacologia cardiovascolare e risposta allo stress.

Sottocategorie di "Recettore adrenergico"

Trovati 728 prodotti di "Recettore adrenergico"

Ordinare per

Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
prodotti per pagina.
  • Prenalterol hydrochloride

    CAS:
    Prenalterol HCl: beta 1-specific agonist; treats acute cardiac failure, shock, low-output post-MI, Shy-Drager syndrome.
    Formula:C12H20ClNO3
    Colore e forma:Solid
    Peso molecolare:261.75
  • Phentolamine Analogue 1

    CAS:
    Phentolamine Analogue 1 is an analogue of phentolamine. Phentolamine is a nonselective antagonist of α-adrenergic.
    Formula:C17H19N3O
    Purezza:99.96%
    Colore e forma:Solid
    Peso molecolare:281.35
  • L-796568 free base

    CAS:
    L-796568 is a potent β3 agonist for obesity with 600x selectivity over β1/β2 receptors (EC50: 3.6 nM).
    Formula:C31H27F3N4O3S2
    Colore e forma:Solid
    Peso molecolare:624.7
  • BU-E 75

    CAS:
    BU-E 75 is an agonist of the histamine H2.
    Formula:C21H24F2N6
    Colore e forma:Solid
    Peso molecolare:398.45
  • NGD9002

    CAS:
    NGD9002 is a novel generation, topology 2 selective corticotropin releasing factor-1 (CRF-1) receptor antagonist agent.
    Formula:C20H31N5O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:357.49
  • LK 204-545

    CAS:
    LK 204-545 is a highly selective antagonist of beta1-adrenoceptor.
    Formula:C25H32N4O6
    Colore e forma:Solid
    Peso molecolare:484.54
  • SDZ-NVI-085

    CAS:
    SDZ-NVI-085 is an α1 adrenergic receptor agonist and a competitive antagonist of 5-hydroxytryptamine.
    Formula:C15H21NO2S
    Colore e forma:Solid
    Peso molecolare:279.4
  • α1 adrenoceptor-MO-1

    CAS:
    α1 adrenoceptor-MO-1 (S enantiomer) has affinity at alpha 1 adrenergic receptor with alphalytic activity and analgesic action.
    Formula:C20H24ClN5O
    Purezza:99.20% - 99.29%
    Colore e forma:Solid
    Peso molecolare:385.89
  • 0990CL

    CAS:
    0990CL is an effective heterotrimer Gαi subunit specific inhibitor, which can interact with purified Go± in GDP-bound state, and can block α2AR mediated cAMP
    Formula:C21H21N5
    Purezza:98.99%
    Colore e forma:Solid
    Peso molecolare:343.42
  • CGP-20712

    CAS:
    CGP-20712 is a selective β 1-adrenoceptor antagonist with an IC50 of 0.7 nM.
    Formula:C23H25F3N4O5
    Purezza:99.40% - 99.58%
    Colore e forma:Solid
    Peso molecolare:494.46
  • OPC-28326

    CAS:
    OPC-28326: an α2-adrenergic blocker; dilates blood vessels; inhibits α2A/B/C receptors with Ki 2040/285/55 nM.
    Formula:C26H35N3O2
    Purezza:99.79%
    Colore e forma:Solid
    Peso molecolare:421.58
  • Deriglidole

    CAS:
    Deriglidole (SL 86-0715), an alpha2 receptor inhibitor, blocks colistin/Idazoxan but not prazosin/α2-adrenergic receptors.
    Formula:C16H21N3
    Purezza:98.12% - 99.03%
    Colore e forma:Solid
    Peso molecolare:255.36
  • (±)-Prenalterol

    CAS:
    (±)-Prenalterol (H 80/62) is an agonist of beta-2- and beta-1-adrenergic receptors and is used to study chronic congestive heart failure.
    Formula:C12H19NO3
    Purezza:99.73%
    Colore e forma:Solid
    Peso molecolare:225.28
  • Talibegron hydrochloride

    CAS:
    Talibegron hydrochloride: β3 adrenoceptor agonist, pD2 3.72, relaxes rat arteries, reduces leptin in mice.
    Formula:C18H22ClNO4
    Purezza:99.82%
    Colore e forma:Solid
    Peso molecolare:351.83
  • Teoprolol

    CAS:
    Teoprolol is a blocker of β-adrenergic receptor.
    Formula:C23H30N6O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:454.52
  • (±)-Penbutolol

    CAS:
    (±)-Penbutolol ((Rac)-Penbutolol) is the racemic form of Penbutolol. It acts as an orally active β-adrenergic receptor antagonist. (±)-Penbutolol mitigates the tachycardia induced by exercise, reduces the increase in peak expiratory flow rate (PEFR) caused by physical activity, and decreases plasma renin activity (PRA) at rest. The peak plasma concentration of this compound is achieved one hour after oral administration, with a half-life of 4.5 hours, and it is metabolized into active metabolites in the body. This compound is utilized in research related to cardiovascular diseases.
    Formula:C18H29NO2
    Colore e forma:Solid
    Peso molecolare:291.43
  • Nipradolol

    CAS:
    Nipradolol blocks alpha-1-adrenergic receptors, lowers IOP in rabbits, and reduces NA-induced muscle contraction and dog artery vasodilation.
    Formula:C15H22N2O6
    Colore e forma:Solid
    Peso molecolare:326.35
  • Sulfinalol hydrochloride

    CAS:
    Sulfinalol hydrochloride is an orally active β-adrenoceptor (β-adrenoceptor) antagonist that exhibits direct vasodilatory activity. It is also classified as an antihypertensive agent.
    Formula:C20H28ClNO4S
    Colore e forma:Solid
    Peso molecolare:413.96
  • Butopamine hydrochloride

    CAS:
    Butopamine hydrochloride is an orally active inotropic compound that is more effective at increasing heart rate compared to Dobutamine.
    Formula:C18H24ClNO3
    Colore e forma:Solid
    Peso molecolare:337.84
  • BRL-37344

    CAS:
    <p>BRL-37344 is a selective β3-adrenergic receptor agonist. It significantly reduces the body weight of obese mice.</p>
    Formula:C19H22ClNO4
    Colore e forma:Solid
    Peso molecolare:363.84