
Recettore adrenergico
I recettori adrenergici sono GPCR attivati dalle catecolamine, come l'adrenalina e la noradrenalina. Questi recettori sono classificati in sottotipi alfa e beta, ognuno dei quali svolge un ruolo chiave nella regolazione della frequenza cardiaca, della pressione sanguigna e della risposta di lotta o fuga. I modulatori dei recettori adrenergici sono essenziali nel trattamento delle malattie cardiovascolari, dell'asma e dei disturbi d'ansia. Presso CymitQuimica, offriamo una vasta gamma di modulatori dei recettori adrenergici di alta qualità per supportare la tua ricerca in endocrinologia, farmacologia cardiovascolare e risposta allo stress.
Sottocategorie di "Recettore adrenergico"
Trovati 728 prodotti di "Recettore adrenergico"
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Prenalterol hydrochloride
CAS:Prenalterol HCl: beta 1-specific agonist; treats acute cardiac failure, shock, low-output post-MI, Shy-Drager syndrome.Formula:C12H20ClNO3Colore e forma:SolidPeso molecolare:261.75Phentolamine Analogue 1
CAS:Phentolamine Analogue 1 is an analogue of phentolamine. Phentolamine is a nonselective antagonist of α-adrenergic.Formula:C17H19N3OPurezza:99.96%Colore e forma:SolidPeso molecolare:281.35L-796568 free base
CAS:L-796568 is a potent β3 agonist for obesity with 600x selectivity over β1/β2 receptors (EC50: 3.6 nM).Formula:C31H27F3N4O3S2Colore e forma:SolidPeso molecolare:624.7BU-E 75
CAS:BU-E 75 is an agonist of the histamine H2.Formula:C21H24F2N6Colore e forma:SolidPeso molecolare:398.45NGD9002
CAS:NGD9002 is a novel generation, topology 2 selective corticotropin releasing factor-1 (CRF-1) receptor antagonist agent.Formula:C20H31N5OPurezza:98%Colore e forma:SolidPeso molecolare:357.49LK 204-545
CAS:LK 204-545 is a highly selective antagonist of beta1-adrenoceptor.Formula:C25H32N4O6Colore e forma:SolidPeso molecolare:484.54SDZ-NVI-085
CAS:SDZ-NVI-085 is an α1 adrenergic receptor agonist and a competitive antagonist of 5-hydroxytryptamine.Formula:C15H21NO2SColore e forma:SolidPeso molecolare:279.4α1 adrenoceptor-MO-1
CAS:α1 adrenoceptor-MO-1 (S enantiomer) has affinity at alpha 1 adrenergic receptor with alphalytic activity and analgesic action.Formula:C20H24ClN5OPurezza:99.20% - 99.29%Colore e forma:SolidPeso molecolare:385.890990CL
CAS:0990CL is an effective heterotrimer Gαi subunit specific inhibitor, which can interact with purified Go± in GDP-bound state, and can block α2AR mediated cAMPFormula:C21H21N5Purezza:98.99%Colore e forma:SolidPeso molecolare:343.42CGP-20712
CAS:CGP-20712 is a selective β 1-adrenoceptor antagonist with an IC50 of 0.7 nM.Formula:C23H25F3N4O5Purezza:99.40% - 99.58%Colore e forma:SolidPeso molecolare:494.46OPC-28326
CAS:OPC-28326: an α2-adrenergic blocker; dilates blood vessels; inhibits α2A/B/C receptors with Ki 2040/285/55 nM.Formula:C26H35N3O2Purezza:99.79%Colore e forma:SolidPeso molecolare:421.58Deriglidole
CAS:Deriglidole (SL 86-0715), an alpha2 receptor inhibitor, blocks colistin/Idazoxan but not prazosin/α2-adrenergic receptors.Formula:C16H21N3Purezza:98.12% - 99.03%Colore e forma:SolidPeso molecolare:255.36(±)-Prenalterol
CAS:(±)-Prenalterol (H 80/62) is an agonist of beta-2- and beta-1-adrenergic receptors and is used to study chronic congestive heart failure.Formula:C12H19NO3Purezza:99.73%Colore e forma:SolidPeso molecolare:225.28Talibegron hydrochloride
CAS:Talibegron hydrochloride: β3 adrenoceptor agonist, pD2 3.72, relaxes rat arteries, reduces leptin in mice.Formula:C18H22ClNO4Purezza:99.82%Colore e forma:SolidPeso molecolare:351.83Teoprolol
CAS:Teoprolol is a blocker of β-adrenergic receptor.Formula:C23H30N6O4Purezza:98%Colore e forma:SolidPeso molecolare:454.52(±)-Penbutolol
CAS:(±)-Penbutolol ((Rac)-Penbutolol) is the racemic form of Penbutolol. It acts as an orally active β-adrenergic receptor antagonist. (±)-Penbutolol mitigates the tachycardia induced by exercise, reduces the increase in peak expiratory flow rate (PEFR) caused by physical activity, and decreases plasma renin activity (PRA) at rest. The peak plasma concentration of this compound is achieved one hour after oral administration, with a half-life of 4.5 hours, and it is metabolized into active metabolites in the body. This compound is utilized in research related to cardiovascular diseases.Formula:C18H29NO2Colore e forma:SolidPeso molecolare:291.43Nipradolol
CAS:Nipradolol blocks alpha-1-adrenergic receptors, lowers IOP in rabbits, and reduces NA-induced muscle contraction and dog artery vasodilation.Formula:C15H22N2O6Colore e forma:SolidPeso molecolare:326.35Sulfinalol hydrochloride
CAS:Sulfinalol hydrochloride is an orally active β-adrenoceptor (β-adrenoceptor) antagonist that exhibits direct vasodilatory activity. It is also classified as an antihypertensive agent.Formula:C20H28ClNO4SColore e forma:SolidPeso molecolare:413.96Butopamine hydrochloride
CAS:Butopamine hydrochloride is an orally active inotropic compound that is more effective at increasing heart rate compared to Dobutamine.Formula:C18H24ClNO3Colore e forma:SolidPeso molecolare:337.84BRL-37344
CAS:<p>BRL-37344 is a selective β3-adrenergic receptor agonist. It significantly reduces the body weight of obese mice.</p>Formula:C19H22ClNO4Colore e forma:SolidPeso molecolare:363.84
