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GluR

GluR

Gli inibitori dei recettori del glutammato sono composti che bloccano l'attività dei recettori del glutammato, i principali recettori dei neurotrasmettitori eccitatori nel cervello. Questi recettori svolgono un ruolo cruciale nella trasmissione sinaptica, nella plasticità, nell'apprendimento e nella memoria. La disregolazione della segnalazione del glutammato è associata a vari disturbi neurologici, come l'epilessia, l'ictus e le malattie neurodegenerative. Gli inibitori dei recettori del glutammato sono essenziali per studiare i meccanismi dell'eccitotossicità e sviluppare strategie neuroprotettive. Presso CymitQuimica, offriamo una gamma di inibitori dei recettori del glutammato per supportare la vostra ricerca sulla funzione sinaptica, la neuroprotezione e i disturbi cognitivi.

Trovati 263 prodotti di "GluR"

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  • (S)-HexylHIBO

    CAS:
    Group I mGlu receptor antagonist
    Formula:C12H20N2O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:256.3

    Ref: TM-T23299

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • LSP1-2111

    CAS:
    LSP1-2111 is a mGlu4 receptor subtype agonist.
    Formula:C12H17N2O9P
    Colore e forma:Solid
    Peso molecolare:364.25

    Ref: TM-T27856

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • Lu-AF11205

    CAS:
    Lu-AF11205 is a potent positive allosteric modulator (PAM) of mGlu5 receptor.
    Formula:C17H16N2OS
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:296.39

    Ref: TM-T27860

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • (RS)-4-Carboxyphenylglycine

    CAS:
    (RS)-4-Carboxyphenylglycine is a racemic mixture. (S)-4-Carboxyphenylglycine is a selective mGlu1α receptor antagonist.
    Formula:C9H9NO4
    Purezza:97.22% - >99.99%
    Colore e forma:Solid
    Peso molecolare:195.17

    Ref: TM-T23262

    5mg
    39,00€
    10mg
    55,00€
    25mg
    90,00€
    50mg
    123,00€
    100mg
    172,00€
    500mg
    410,00€
  • (R)-4-Carboxyphenylglycine

    CAS:
    (R)-4-Carboxyphenylglycine is a NMDA receptor antagonist.
    Formula:C9H9NO4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:195.17

    Ref: TM-T23217

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • VU0652835

    CAS:
    VU0652835 is a negative allosteric modulator of metabotropic glutamate receptor subtype 5 (mGlu5) (IC50: 81 nM).
    Formula:C16H19N3O3S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:333.41

    Ref: TM-T13319

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • VU0486321

    CAS:
    VU0486321: potent mGlu1 PAM, rat PK CLp 13.3 mL/min/kg, t1/2 54 min, human fu 0.05, rat fu 0.03, great CNS penetration Kp 1.02.
    Formula:C20H12ClFN2O4
    Colore e forma:Solid
    Peso molecolare:398.77

    Ref: TM-T35081

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • A-850002

    CAS:
    A-850002 is a bioactive chemical.
    Formula:C18H16N4OS
    Colore e forma:Solid
    Peso molecolare:336.41

    Ref: TM-T29513

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • JNJ-55511118

    CAS:
    <p>JNJ-55511118 is a TARP γ8 allosteric modulator with anticonvulsant activity, which can be used in research on chronic operant alcohol self-administration.</p>
    Formula:C14H8ClF3N2O2
    Colore e forma:Solid
    Peso molecolare:328.67

    Ref: TM-T25558

    1mg
    120,00€
    5mg
    347,00€
    10mg
    621,00€
    25mg
    1.397,00€
  • DCB

    CAS:
    <p>DCB is an mGluR5 allosteric ligand that blocks mGluR modulation, countering DMeOB and DFB effects.</p>
    Formula:C14H10Cl2N2
    Purezza:99.12% - 99.9%
    Colore e forma:Solid
    Peso molecolare:277.15

    Ref: TM-T22711

    10mg
    52,00€
    25mg
    87,00€
    50mg
    143,00€
    100mg
    225,00€
    200mg
    331,00€
  • N,N-Dipropyldopamine (hydrobromide)

    CAS:
    N,N-Dipropyldopamine is a dopamine agonist reducing DOPA and locomotion in rats and mice, reversible by spiroperidol.
    Formula:C14H24BrNO2
    Colore e forma:Solid
    Peso molecolare:318.255

    Ref: TM-T38221

    1mg
    170,00€
    5mg
    743,00€
    10mg
    1.301,00€
  • ML337

    CAS:
    ML337 is a negative allosteric modulator of mGlu3 with an IC50 of 593 nM.
    Formula:C21H20FNO3
    Purezza:99.83%
    Colore e forma:Solid
    Peso molecolare:353.39

    Ref: TM-T23003

    1mg
    35,00€
    5mg
    64,00€
    10mg
    97,00€
    25mg
    207,00€
    50mg
    309,00€
    100mg
    Prezzo su richiesta
    1mL*10mM (DMSO)
    75,00€
  • LY382884

    CAS:
    LY382884 is a selective and potent GluR5 kainate receptor antagonist with anxiolytic activity.LY382884 blocks blockade of mossy fibre LTP induction.
    Formula:C18H23NO4
    Purezza:98.32% - 98.71%
    Colore e forma:Solid
    Peso molecolare:317.38

    Ref: TM-T27949

    1mg
    710,00€
    5mg
    1.491,00€
    10mg
    1.882,00€
    25mg
    2.452,00€
    50mg
    3.022,00€
    100mg
    4.085,00€
  • TC-N 22A

    CAS:
    TC-N 22A is a strong, selective, oral active mGlu4 forward allosteric regulator (PAM) that can cross the blood-brain barrier.
    Formula:C14H13N5S
    Purezza:99.95%
    Colore e forma:Solid
    Peso molecolare:283.35

    Ref: TM-T23440

    1mg
    120,00€
    5mg
    250,00€
    10mg
    309,00€
    25mg
    520,00€
    50mg
    748,00€
    100mg
    1.026,00€
  • CPPHA

    CAS:
    <p>CPPHA, a positive allosteric modulator of glutamate receptors mGluR5 and mGluR1, is commonly used in development for central nervous system diseases.</p>
    Formula:C22H15ClN2O4
    Purezza:98.07%
    Colore e forma:Solid
    Peso molecolare:406.82

    Ref: TM-T10881

    5mg
    34,00€
    25mg
    Prezzo su richiesta
    50mg
    Prezzo su richiesta
  • ML289

    CAS:
    ML289 is a potent CNS-penetrant mGlu3 modulator with IC50 of 0.66 μM, >15-fold selectivity over mGlu2, and inactive against mGlu5.
    Formula:C22H23NO3
    Purezza:99.54%
    Colore e forma:Solid
    Peso molecolare:349.42

    Ref: TM-T23000

    5mg
    50,00€
    10mg
    80,00€
    25mg
    145,00€
    50mg
    225,00€
    100mg
    339,00€
    200mg
    470,00€
    1mL*10mM (DMSO)
    51,00€
  • Foliglurax

    CAS:
    Foliglurax is a highly selective brain-penetrant metabotropic glutamate receptor 4 positive allosteric modulator (mGluR4 PAM) (EC50: 79 nM).
    Formula:C23H23N3O3S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:421.51

    Ref: TM-T11311L

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • VU6001376

    CAS:
    VU6001376 is an effective and selective positive allosteric modulator of the metabotropic glutamate receptor 4 (EC50: 50.1 nM).
    Formula:C18H14F2N6OS
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:400.41

    Ref: TM-T17248

    25mg
    1.586,00€
    50mg
    2.072,00€
    100mg
    2.660,00€
  • Ro 67-4853

    CAS:
    Ro 67-4853 is a positive allosteric modulator of mGluR1, selectively enhancing the response to the agonist (S)-3,5-dihydroxy-phenylglycine (DHPG).
    Formula:C19H19NO4
    Purezza:98.57%
    Colore e forma:Solid
    Peso molecolare:325.36

    Ref: TM-T23248

    1mg
    65,00€
    5mg
    139,00€
    10mg
    197,00€
    25mg
    339,00€
    50mg
    500,00€
    100mg
    712,00€
    200mg
    938,00€
  • VU0155041 sodium

    CAS:
    VU0155041 sodium is a positive allosteric modulator of mGluR4 that promotes extinction in male rats.
    Formula:C14H14Cl2NNaO3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:338.16

    Ref: TM-T23507

    5mg
    106,00€
    10mg
    188,00€
    50mg
    540,00€