AChR
Gli inibitori del recettore dell'acetilcolina (AChR) sono composti che bloccano l'attività dei recettori dell'acetilcolina, fondamentali per la neurotrasmissione nei sistemi nervoso centrale e periferico. Gli AChR svolgono un ruolo cruciale nella contrazione muscolare, nella memoria e nelle funzioni cognitive. Gli inibitori degli AChR vengono utilizzati per studiare condizioni come la miastenia grave, l'Alzheimer e altri disturbi neurologici. Modulando l'attività degli AChR, questi inibitori possono aiutare a svelare le complessità della segnalazione colinergica nel cervello. Presso CymitQuimica, offriamo una gamma di inibitori degli AChR per supportare la tua ricerca in neuroscienze, farmacologia e malattie neurodegenerative.
Trovati 619 prodotti di "AChR"
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Benzamide Derivative 1
CAS:Benzamide Derivative 1 Benzamide derivative with gastrokinetic activity.Benzamide Derivative 1 can be used in the study of gastrointestinal diseases.Formula:C22H34ClN3O3Purezza:>99.99%Colore e forma:SolidPeso molecolare:423.98Tebanicline tosylate
CAS:Tebanicline: synthetic, potent, non-opioid analgesic, less toxic than epibatidine; relieves neuropathic pain, acts on α3β4 and α4β2 nicotinic receptors.Formula:C16H19ClN2O4SPurezza:98%Colore e forma:SolidPeso molecolare:370.85WIN 62,577
CAS:WIN 62,577 is a allosteric antagonist of mAChR.Formula:C29H31N3OPurezza:98%Colore e forma:SolidPeso molecolare:437.58Beperidium iodide
CAS:Beperidium iodide is a competitive antagonist of the acetylcholine receptor (pA2: 7.93).Formula:C23H34IN3O3Colore e forma:SolidPeso molecolare:527.44TC 1698 dihydrochloride
CAS:nicotinic α7 receptor agonistFormula:C13H18N2Purezza:98%Colore e forma:SolidPeso molecolare:202.3SM-21 maleate
CAS:Increases release of acetylcholine,σ2 antagonistFormula:C22H28ClNO7Purezza:98%Colore e forma:SolidPeso molecolare:453.91TC-T 6000
CAS:TC-T 6000 (hENT4-IN-1) is an ENT4 inhibitor with vasodilator activity that inhibits hENT1 and hENT2 for the study of cancer and cardiovascular damage.Formula:C26H48N8O2Purezza:98.14%Colore e forma:SolidPeso molecolare:504.71Terodiline hydrochloride
CAS:<p>Terodiline hydrochloride is an antagonist of M1-selective muscarinic receptor (mAChR)(Kbs of 15, 160, 280, and 198 nM in rabbit vas deferens (M1), atria (M2),</p>Formula:C20H28ClNPurezza:98%Colore e forma:SolidPeso molecolare:317.9YM-46303
CAS:YM-46303 is a selective and potent muscarinic receptor antagonist that exhibits high affinity for the M3 receptor.YM-46303 can be used to study bradycardia inFormula:C20H23ClN2O2Purezza:>99.99%Colore e forma:SolidPeso molecolare:358.86CHF5407
CAS:CHF5407（SVT-47060） is a potent and selective muscarinic M3 receptor antagonist with prolonged action at muscarinic receptors.CHF5407 has an effect onFormula:C27H25BrF4N2O3SPurezza:99.54% - >99.99%Colore e forma:SolidPeso molecolare:613.46TC299423
CAS:TC299423 is a novel agonist for nicotinic acetylcholine receptors (nAChRs). TC299423 modestly selectively targets α6β2 subtype.Formula:C11H15N3Colore e forma:SolidPeso molecolare:189.26TC 2559 difumarate
CAS:partial agonist of α4β2 nicotinic acetylcholine receptorFormula:C12H18N2OC4H404Purezza:98%Colore e forma:SolidPeso molecolare:380.39Tridihexethyl chloride
CAS:Tridihexethyl is an anticholinergic, antimuscarinic, and antispasmolytic drug, which can be used to treat acquired nystagmus or peptic ulcer disease.Formula:C21H36ClNOColore e forma:SolidPeso molecolare:353.97KL8604166
CAS:KL8604166 (UCB-11056) is a potential puzzle compound.UCB-11056 amplifies the formation of inducible cyclic AMP in rat brain tissue.Formula:C12H21N5O2Purezza:99.21%Colore e forma:SolidPeso molecolare:267.33PF-06767832
CAS:PF-06767832: selective M1 PAM (EC50=60 nM), no M2-M5 activity, good CNS penetration, but has GI and cardiovascular risks.Formula:C22H23N3O3SColore e forma:SolidPeso molecolare:409.5Hadacidin
CAS:Hadacidin is an inhibitor of AMP synthesis. Hadacidin and hadacidin analogues have anticancer activity and activity against adenylosuccinate synthetase.Formula:C3H5NO4Colore e forma:SolidPeso molecolare:119.08Glucagon Receptor Antagonist I
CAS:Glucagon antagonist I blocks the GCGR (IC50=181 nM), stops glucagon-induced glycogenolysis, and lowers glucose in glucagon-treated humanized mice.Formula:C20H30N2OSColore e forma:SolidPeso molecolare:346.53S16961
CAS:S16961 (S169611) is an agonist of nicotinic receptor.Formula:C41H71NO6Purezza:99.69%Colore e forma:SolidPeso molecolare:674.01RJR-2429
CAS:RJR-2429 is a potent AChR agonist.Formula:C12H16N2Colore e forma:SolidPeso molecolare:188.27CC4
CAS:Selective α6β2/α4β2 partial agonist; Ki: 12/26nM (rat); poor α3β4/α7 affinity; stimulates dopamine release; reduces nicotine self-admin in rats.Formula:C24H30N4O2Colore e forma:SolidPeso molecolare:406.52
