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AChR

AChR

Gli inibitori del recettore dell'acetilcolina (AChR) sono composti che bloccano l'attività dei recettori dell'acetilcolina, fondamentali per la neurotrasmissione nei sistemi nervoso centrale e periferico. Gli AChR svolgono un ruolo cruciale nella contrazione muscolare, nella memoria e nelle funzioni cognitive. Gli inibitori degli AChR vengono utilizzati per studiare condizioni come la miastenia grave, l'Alzheimer e altri disturbi neurologici. Modulando l'attività degli AChR, questi inibitori possono aiutare a svelare le complessità della segnalazione colinergica nel cervello. Presso CymitQuimica, offriamo una gamma di inibitori degli AChR per supportare la tua ricerca in neuroscienze, farmacologia e malattie neurodegenerative.

Trovati 617 prodotti di "AChR"

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  • Glycerophosphoinositol choline

    CAS:
    Glycerophosphoinositol choline is the salt of choline and glycerophosphoinositol.
    Formula:C14H32NO12P
    Colore e forma:Solid
    Peso molecolare:437.38
  • Clorprenaline

    CAS:
    Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.
    Formula:C11H16ClNO
    Purezza:98.9%
    Colore e forma:Solid
    Peso molecolare:213.7
  • NKH477

    CAS:
    NKH477 (Colforsin dapropate hydrochloride) is a derivative of forskolin with antidepressant activity.
    Formula:C27H44ClNO8
    Purezza:98% - 98%
    Colore e forma:Solid
    Peso molecolare:546.09
  • Biperiden

    CAS:
    Biperiden is a muscarinic antagonist for Parkinson's and drug-induced extrapyramidal symptoms.
    Formula:C21H29NO
    Purezza:99.65%
    Colore e forma:Crystals Solid
    Peso molecolare:311.46
  • SSR180711 hydrochloride

    CAS:
    SSR180711 hydrochloride (SSR-180711A HCl) is an Alpha7 nicotinic acetylcholine partial agonist that can be used to study neurolysis.
    Formula:C14H18BrClN2O2
    Purezza:99.22%
    Colore e forma:Solid
    Peso molecolare:361.66
  • NBTGR

    CAS:
    NBTGR is a potent nucleoside transport inhibitor(adenosine uptake ,Ki of 70 nM).
    Formula:C17H18N6O6S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:434.43
  • Dexetimide

    CAS:
    Dexetimide, a muscarinic receptor antagonist, treats neuroleptic-induced parkinsonism.
    Formula:C23H26N2O2
    Colore e forma:Solid
    Peso molecolare:362.46
  • Metixene hydrochloride hydrate

    CAS:
    Metixene HCl hydrate is a potential anticholinergic for Parkinson's with IC50 of 55 nM and Ki of 15 nM against muscarine receptors.
    Formula:C20H26ClNOS
    Purezza:99.99%
    Colore e forma:Solid
    Peso molecolare:363.95
  • N6-Methyladenosine 5'-monophosphate disodium salt

    CAS:
    N6-Methyladenosine 5'-monophosphate disodium salt is a glycogen phosphorylase b activator and an inhibitor of adenylate kinase II.
    Formula:C11H14N5Na2O7P
    Purezza:99.36% - 99.36%
    Colore e forma:Solid
    Peso molecolare:405.21
  • Varenicline Hydrochloride

    CAS:
    Varenicline Hydrochloride (CP 526555) is an orally active partial agonist of the α4β2 nicotinic acetylcholine receptor (α4β2 nAChR, IC50 = 250 nM).
    Formula:C13H14ClN3
    Purezza:99.854%
    Colore e forma:Solid
    Peso molecolare:247.72
  • Tolterodine

    CAS:
    Tolterodine ((R)-(+)-Tolterodine) is an mACh antagonist used in the treatment of detrusor instability and overactive bladder syndrome.
    Formula:C22H31NO
    Purezza:99.71%
    Colore e forma:White Like Or Light Brown Crystalline Powder
    Peso molecolare:325.49
  • Ispronicline

    CAS:
    Ispronicline (TC-1734) An orally active, selective, and potent α4β2 nAChR partial agonist with antidepressant, neuroprotective, and long-lasting cognitive
    Formula:C14H22N2O
    Purezza:97.70% - 99.16%
    Colore e forma:Solid
    Peso molecolare:234.34
  • Cevimeline

    CAS:
    Cevimeline: muscarinic agonist, treats dry mouth & Sjögren's, boosts saliva post-cancer radiotherapy.
    Formula:C10H17NOS
    Colore e forma:Off-White Solid
    Peso molecolare:199.31
  • Fesoterodine L-mandelate

    CAS:
    Fesoterodine L-mandelate is a efficacious antimuscarinic agent for the overactive bladder (OAB).
    Formula:C34H45NO6
    Colore e forma:Solid
    Peso molecolare:563.735
  • Tebanicline dihydrochloride

    CAS:
    Tebanicline dihydrochloride: oral analgesic, nAChR modulator, Ki=37 pM at α4β2 receptors, inhibits cytisine binding.
    Formula:C9H13Cl3N2O
    Colore e forma:Solid
    Peso molecolare:271.57
  • YM-58790 hydrochloride

    CAS:
    YM-58790 is a potent M3 muscarinic receptor antagonist(Ki of 15 nM).
    Formula:C27H32ClN3O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:466.02
  • Fipexide hydrochloride

    CAS:
    Fipexide (hydrochloride) is a kind of psychoactive drug of the piperazine class.
    Formula:C20H22Cl2N2O4
    Colore e forma:Solid
    Peso molecolare:425.31
  • Telenzepine dihydrochloride

    CAS:
    muscarinic M1 receptor antagonist
    Formula:C19H23ClN4O2S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:406.93
  • NS3861 fumarate

    CAS:
    NS3861 fumarate, a partial α3β4 nAChR agonist, binds α3β2, α4β4, α4β2 with Ki values of 0.62, 25, 7.8, 55 nM.
    Formula:C16H18BrNO4S
    Colore e forma:Solid
    Peso molecolare:400.29
  • Sabcomeline hydrochloride

    CAS:
    Sabcomeline is a selective M1 receptor partial agonist.
    Formula:C10H16ClN3O
    Colore e forma:Solid
    Peso molecolare:229.71
  • Clothianidin

    CAS:
    Clothianidin (TI 435), an insecticide, stimulates nAChR as acetylcholine agonist, not AChE inhibitor.
    Formula:C6H8ClN5O2S
    Purezza:99.71% - 99.87%
    Colore e forma:Solid Powder
    Peso molecolare:249.68
  • VU0152099

    CAS:
    VU0152099 is a potent and selective M4 mAChR allosteric potentiator(EC50 = 380 ± 93 nM).
    Formula:C18H17N3O3S
    Purezza:98.46%
    Colore e forma:Solid
    Peso molecolare:355.41
  • TBPB

    CAS:
    <p>TBPB is an allosteric M1 mAChR agonist.</p>
    Formula:C25H32N4O
    Purezza:97.87% - 99.9%
    Colore e forma:Solid
    Peso molecolare:404.55
  • Nitrobenzylthioinosine

    CAS:
    <p>Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.</p>
    Formula:C17H17N5O6S
    Purezza:99.69% - 99.74%
    Colore e forma:Off-White Solid
    Peso molecolare:419.41
  • Umeclidinium bromide

    CAS:
    Umeclidinium bromide (GSK573719A) is a novel mAChR antagonist.
    Formula:C29H34BrNO2
    Purezza:98.4% - 99.89%
    Colore e forma:Solid
    Peso molecolare:508.49
  • Pempidine

    CAS:
    Pempidine (1,2,2,6,6-Pentamethylpiperidine) is a nicotinic antagonist, has been used as a ganglionic blocker in the treatment of hypertension.
    Formula:C10H21N
    Purezza:98.18% - 99.28%
    Colore e forma:Colorless - Light Yellow Clear Liquid
    Peso molecolare:155.28
  • Methylbenactyzium Bromide

    CAS:
    Methylbenactyzium Bromide (Semulgin) is an anticonvulsant that is the active metabolite of trimethadione.
    Formula:C21H28BrNO3
    Purezza:99.29%
    Colore e forma:Solid
    Peso molecolare:422.36
  • Rivanicline hemioxalate


    <p>Rivanicline hemioxalate is a selective α4β2 nicotinic receptor agonist (K i =26 nM), over 1,000x preference to α7 (K i =3.6 μM), with limited side effects.</p>
    Formula:C12H16N2O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:207.23
  • PSEM 89S TFA

    CAS:
    <p>PSEM 89S TFA is a brain-penetrant and selective ion channels agonist, and is orthogonally selective for Q79G and L141F, respectively.</p>
    Formula:C18H23F3N2O5
    Purezza:99.9%
    Colore e forma:Solid
    Peso molecolare:404.38
  • Prifinium bromide

    CAS:
    <p>Prifinium bromide is a quaternary ammon antimuscarinic. It inhibits hyperkinesia of the digestive organs and urinary tract and has a spasmolytic action.</p>
    Formula:C22H28BrN
    Purezza:97.99%
    Colore e forma:Solid
    Peso molecolare:386.37
  • (S)-UFR2709

    CAS:
    (S)-UFR2709, a nAChR competitive antagonist, favors α4β2 over α7, reduces anxiety and alcohol use in rats.
    Formula:C13H17NO2
    Colore e forma:Solid
    Peso molecolare:219.284
  • Oxotremorine sesquifumarate

    CAS:
    <p>Oxotremorine sesquifumarate is a muscarinic agonist.</p>
    Formula:C12H18N2OC4H4O4
    Purezza:97.94%
    Colore e forma:Solid
    Peso molecolare:380.39
  • (-)-(S)-B-973B

    CAS:
    <p>(-)-(S)-B-973B is an effective allosteric agonist and a positive allosteric modulator of α7 nAChR.</p>
    Formula:C24H26F2N6O
    Purezza:99.52%
    Colore e forma:Solid
    Peso molecolare:452.5
  • Mecamylamine hydrochloride

    CAS:
    Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.
    Formula:C11H22ClN
    Purezza:99.76% - >99.99%
    Colore e forma:White Solid
    Peso molecolare:203.75
  • VU0152100

    CAS:
    <p>VU0152100 is an effective and selective allosteric potentiator of M4 mAChR (EC50: 380 ± 93 nM).</p>
    Formula:C18H19N3O2S
    Purezza:99.56%
    Colore e forma:Solid
    Peso molecolare:341.43
  • OXOMEMAZINE

    CAS:
    Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in cough research.
    Formula:C18H22N2O2S
    Purezza:99.58%
    Colore e forma:Solid
    Peso molecolare:330.44
  • Darifenacin

    CAS:
    Darifenacin (UK-88525) is a muscarinic receptor M3 antagonist with anticonvulsant activity and can be used to study urinary incontinence and overactive bladder.
    Formula:C28H30N2O2
    Purezza:99.78%
    Colore e forma:Solid
    Peso molecolare:426.55
  • Dicyclomine

    CAS:
    Dicyclomine: oral muscarinic antagonist, eases GI muscle spasms, high affinity for M1/M2 receptors, Ki of 5.1 nM/54.6 nM.
    Formula:C19H35NO2
    Colore e forma:Solid
    Peso molecolare:309.49
  • JHU37160

    CAS:
    JHU37160 is a DREADD agonist with Ki of 1.9 nM for hM3Dq, 3.6 nM for hM4Di, and EC50 of 18.5 nM (hM3Dq), 0.2 nM (hM4Di) in HEK-293 cell assays.
    Formula:C19H20ClFN4
    Purezza:99.87%
    Colore e forma:Solid
    Peso molecolare:358.84
  • Dronedarone

    CAS:
    <p>Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.</p>
    Formula:C31H44N2O5S
    Purezza:98.85% - 99.58%
    Colore e forma:Solid
    Peso molecolare:556.76
  • Nor-benzetimide

    CAS:
    Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.
    Formula:C16H20N2O2
    Purezza:98.63%
    Colore e forma:Solid
    Peso molecolare:272.34
  • Isopropamide Iodide

    CAS:
    <p>Isopropamide iodide: long-acting anticholinergic, treats peptic ulcers, GI disorders, Alzheimer's.</p>
    Formula:C23H33IN2O
    Purezza:99.67%
    Colore e forma:Solid
    Peso molecolare:480.43
  • W-84 dibromide

    CAS:
    <p>W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.</p>
    Formula:C32H44Br2N4O4
    Purezza:95.56%
    Colore e forma:Solid
    Peso molecolare:708.52
  • CCMI

    CAS:
    <p>CCMI (AVL-3288) is a potent and selective modulator of α7 nAChR-positive allosteric.</p>
    Formula:C19H15Cl2N3O2
    Purezza:>99.99%
    Colore e forma:Solid
    Peso molecolare:388.25
  • Glycopyrrolate

    CAS:
    Glycopyrrolate: muscarinic antagonist, antispasmodic for GI issues, reduces salivation with anesthesia.
    Formula:C19H28BrNO3
    Purezza:99.41% - 99.64%
    Colore e forma:Solid
    Peso molecolare:398.33
  • Ursulcholic acid

    CAS:
    Ursulcholic acid (Ursulcholic) is a water-soluble anticholinergic compound.
    Formula:C24H40O10S2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:552.7
  • VU0357017 hydrochloride

    CAS:
    VU0357017 hydrochloride (ML071 hydrochloride) is highly selective M1 agonists act at an allosteric site to activate the receptor (EC50: 477 ± 172 nM; Pec50: 6.
    Formula:C18H28ClN3O3
    Purezza:99% - 99.97%
    Colore e forma:Solid
    Peso molecolare:369.89
  • Revefenacin

    CAS:
    Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.
    Formula:C35H43N5O4
    Purezza:98.12%
    Colore e forma:Solid
    Peso molecolare:597.75
  • BNC210

    CAS:
    BNC210 (IW-2143) is a α7 nAChR negative allosteric modulator. BNC210 has potent activity in animal models of anxiety and depression.
    Formula:C17H23N3O3
    Purezza:97.05% - >99.99%
    Colore e forma:Solid
    Peso molecolare:317.38
  • PNU-282987 S enantiomer free base

    CAS:
    PNU-282987 S enantiomer free base is an agonist of α7 nicotinic acetylcholine receptor (α7 nAChR).
    Formula:C14H17ClN2O
    Purezza:99.74%
    Colore e forma:Solid
    Peso molecolare:264.75
  • Piperidolate

    CAS:
    Piperidolate inhibits intestinal cramp induced by acetylcholine
    Formula:C21H25NO2
    Purezza:98.45%
    Colore e forma:Solid
    Peso molecolare:323.43
  • BQCA

    CAS:
    <p>BQCA (benzylquinolone carboxylic acid) a highly selective allosteric M1 mAChR modulator.</p>
    Formula:C18H15NO4
    Purezza:97.22%
    Colore e forma:Solid
    Peso molecolare:309.32
  • Varenicline dihydrochloride

    CAS:
    Varenicline dihydrochloride is a Selective α4β2 nicotinic acetylcholine receptor partial agonist.
    Formula:C13H15Cl2N3
    Purezza:99.88% - 99.97%
    Colore e forma:Solid
    Peso molecolare:284.18
  • Harman hydrochloride

    CAS:
    Harman hydrochloride triggers CYP1A1 gene via AhR, potentially causing mutations and cancer.
    Formula:C12H11ClN2
    Purezza:99.35%
    Colore e forma:Solid
    Peso molecolare:218.68
  • Imidafenacin

    CAS:
    Imidafenacin (KRP-197)(KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM.
    Formula:C20H21N3O
    Purezza:99.17%
    Colore e forma:Solid
    Peso molecolare:319.4
  • EB-3D

    CAS:
    EB-3D is a potent and selective choline kinase alpha 1 (ChoKα1) inhibitor(IC50 : 1 μM).with anti-cancer activity.
    Formula:C30H36Br2N4O2
    Purezza:99.48%
    Colore e forma:Solid
    Peso molecolare:644.4
  • JHU37152

    CAS:
    JHU37152 is a DREADD agonist; Ki: 1.8 nM at hM3Dq, 8.7 nM at hM4Di; EC50: 5 nM (hM3Dq), 0.5 nM (hM4Di) in HEK-293 cell assays.
    Formula:C19H20ClFN4
    Purezza:99.72%
    Colore e forma:Solid
    Peso molecolare:358.84
  • SEN12333

    CAS:
    <p>SEN12333 is an α7 nicotinic acetylcholine receptor (nAChR) agonist</p>
    Formula:C20H25N3O2
    Purezza:99.02%
    Colore e forma:Solid
    Peso molecolare:339.43
  • mAChR-IN-1 hydrochloride

    CAS:
    mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 Nm.
    Formula:C23H26ClIN2O2
    Purezza:99.87%
    Colore e forma:Solid
    Peso molecolare:524.82
  • 4BP-TQS

    CAS:
    4BP-TQS is an allosteric agonist of α7 nAChRs.
    Formula:C18H17BrN2O2S
    Purezza:99.96%
    Colore e forma:Solid
    Peso molecolare:405.31
  • Tebanicline hydrochloride

    CAS:
    Tebanicline hydrochloride (Ebanicline hydrochloride) , is an effective synthetic nicotinic (non-opioid) analgesic drug.
    Formula:C9H12Cl2N2O
    Purezza:91.74% - 98.78%
    Colore e forma:Solid
    Peso molecolare:235.11
  • PHA 543613 hydrochloride

    CAS:
    PHA-543613 hydrochloride, a potent α7 nicotinic receptor agonist, may treat schizophrenia-related cognitive deficits.
    Formula:C15H18ClN3O2
    Colore e forma:Solid
    Peso molecolare:307.78
  • Pozanicline dihydrochloride

    CAS:
    Pozanicline dihydrochloride (ABT-089 dihydrochloride) is an orally bioavailable agonist of nicotinic acetylcholine receptor (nAChR) (Ki = 16.7 nM)
    Formula:C11H18Cl2N2O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:265.18
  • VU0467154

    CAS:
    VU0467154 is a positive allosteric modulator of the M4 muscarinic acetylcholine receptor.
    Formula:C17H15F3N4O3S2
    Purezza:99.51% - 99.53%
    Colore e forma:Solid
    Peso molecolare:444.45
  • Pempidine HCl

    CAS:
    Pempidine HCl, a nicotinic antagonist and former hypertension treatment, now mainly serves as a lab tool.
    Formula:C10H22ClN
    Colore e forma:Solid
    Peso molecolare:191.74
  • Atracurium besylate

    CAS:
    Atracurium besylate (51W89) is a short-acting, non-depolarizing muscle relaxant, not affecting the heart or reliant on kidneys.
    Formula:C65H82N2O18S2
    Purezza:98.94% - 99.71%
    Colore e forma:Solid
    Peso molecolare:1243.49
  • VU0119498

    CAS:
    VU0119498 is a M1 muscarinic receptor agonist (EC50 = 3.1 μM) and pan mAChR M3, M5 positive allosteric modulator (PAM),and is a neuroprotective agent.
    Formula:C15H10BrNO2
    Purezza:97.56%
    Colore e forma:Solid
    Peso molecolare:316.15
  • Batefenterol Succinate

    CAS:
    Batefenterol Succinate is a first-in-class inhaled bifunctional bronchodilator possessing muscarinic receptor antagonist and β2-adrenoceptor agonist properties.
    Formula:C44H48ClN5O11
    Colore e forma:Solid
    Peso molecolare:858.34
  • Varenicline Tartrate

    CAS:
    <p>Varenicline Tartrate (CP 526555-18) is a benzazepine derivative that functions as an ALPHA4/BETA2 NICOTINIC RECEPTOR partial agonist.</p>
    Formula:C13H13N3·C4H6O6
    Purezza:98.23% - 98.32%
    Colore e forma:Tan Solid
    Peso molecolare:361.35
  • VU0238441

    CAS:
    VU0238441 is agonist of Muscarinic acetylcholine receptor M5 (human) with EC50 of 2.1μM.
    Formula:C16H9ClF3NO2
    Purezza:100%
    Colore e forma:Solid
    Peso molecolare:339.7
  • Encenicline hydrochloride

    CAS:
    Encenicline hydrochloride (EVP-6124 hydrochloride) is a new-type partial agonist of α7 neuronal nicotinic acetylcholine receptors (nAChRs).
    Formula:C16H17ClN2OS·HCl
    Purezza:98.34% - 99.85%
    Colore e forma:Solid
    Peso molecolare:357.3
  • 9-Ethyladenine

    CAS:
    9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].
    Formula:C7H9N5
    Purezza:99.35% - 99.37%
    Colore e forma:Solid
    Peso molecolare:163.18
  • VU 0238429

    CAS:
    <p>VU 0238429 (SCR-1481B1) is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5)( EC50 : 1.16 μM).</p>
    Formula:C17H12F3NO4
    Purezza:>99.99%
    Colore e forma:Solid
    Peso molecolare:351.28
  • MC-Val-Cit-PAB

    CAS:
    <p>MC-Val-Cit-PAB: cathepsin-cleavable ADC linker used in FDA-approved brentuximab vedotin.</p>
    Formula:C28H40N6O7
    Purezza:98.24%
    Colore e forma:Solid
    Peso molecolare:572.65
  • NS3861

    CAS:
    NS3861 is a selective agonist for α3β4/α4β2 nAChRs, preferring β-subunits, with no effect on α4-based receptors.
    Formula:C12H14BrNS
    Purezza:99.853%
    Colore e forma:Solid
    Peso molecolare:284.22
  • Dinotefuran

    CAS:
    Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.
    Formula:C7H14N4O3
    Purezza:99.89%
    Colore e forma:White Crystalline Powder
    Peso molecolare:202.21
  • Thiacloprid

    CAS:
    Thiacloprid: insecticide targeting insect nAChRs, IC50 - Drosophila: 2.7 nM, Mouse α4β2 nAChRs: 860 nM.
    Formula:C10H9ClN4S
    Purezza:98.66% - 99.95%
    Colore e forma:Yellowish Crystalline Powder
    Peso molecolare:252.72
  • Ipratropium Bromide

    CAS:
    Ipratropium Bromide (Sch 1000) is an antagonist of muscarinic receptors and is used in COPD and asthma studies.
    Formula:C20H30BrNO3
    Purezza:99.92%
    Colore e forma:Solid
    Peso molecolare:412.37
  • Encenicline

    CAS:
    Encenicline (EVP-6124), a selective α7 nAChRs agonist, targets cognitive impairment in schizophrenia and Alzheimer's.
    Formula:C16H17ClN2OS
    Purezza:99.20%
    Colore e forma:Solid
    Peso molecolare:320.84
  • Oxyphencyclimine Hydrochloride

    CAS:
    <p>Oxyphencyclimine Hydrochloride (Ulcociclinina) is a synthetic tertiary amine and antimuscarinic agent with antispasmodic and antisecretory activities.</p>
    Formula:C20H29ClN2O3
    Purezza:99.55%
    Colore e forma:Solid
    Peso molecolare:380.91
  • Oxyphenonium bromide

    CAS:
    <p>Oxyphenonium bromide is an anticholinergic used to study and treat ulcers and relieve visceral spasms.</p>
    Formula:C21H34BrNO3
    Purezza:98.96%
    Colore e forma:Solid
    Peso molecolare:428.404
  • Propiverine

    CAS:
    Propiverine reduces muscle spasms by limiting calcium influx, targeting bladder smooth muscles, aiding OAB research.
    Formula:C23H29NO3
    Colore e forma:Solid
    Peso molecolare:367.48
  • Cyclopentolate Hydrochloride

    CAS:
    Cyclopentolate Hydrochloride is a muscarinic acetylcholine receptors antagonist with Kis of 1.62, 27.5, and 2.63 nM for M1, M2, and M3 receptors, respectively.
    Formula:C17H26ClNO3
    Purezza:99.91%
    Colore e forma:Solid
    Peso molecolare:327.85
  • A-867744

    CAS:
    <p>A-867744 is an effective and selective type II positive allosteric modulator of the α7 nAChR (EC50: 1.0 μM).</p>
    Formula:C20H19ClN2O3S
    Purezza:95.66%
    Colore e forma:Solid
    Peso molecolare:402.89
  • VU10010

    CAS:
    <p>VU10010 (VU 10010) is allosteric potentiator of M4 acetylcholine receptors.</p>
    Formula:C17H16ClN3OS
    Purezza:99.36%
    Colore e forma:Solid
    Peso molecolare:345.85
  • Pirmenol

    CAS:
    Pirmenol is a new antiarrhythmic drug
    Formula:C22H30N2O
    Purezza:97.24%
    Colore e forma:Solid
    Peso molecolare:338.49
  • Mivacurium dichloride

    CAS:
    Mivacurium dichloride: non-depolarizing, quick-acting muscle relaxant for minor surgeries and tracheal intubation.
    Formula:C58H80Cl2N2O14
    Purezza:99.2% - 99.48%
    Colore e forma:Off-White Solid
    Peso molecolare:1100.17
  • SQ22536

    CAS:
    SQ22536, a tetrahydrofuryl adenosine analogue, inhibits adenylate cyclase in catfish and rat hepatocytes non-competitively.
    Formula:C9H11N5O
    Purezza:99.18%
    Colore e forma:Off-White Solid
    Peso molecolare:205.22
  • Coluracetam

    CAS:
    Coluracetam (MKC-231)(MKC-231) is a Choline Uptake Enhancer.
    Formula:C19H23N3O3
    Purezza:99.96%
    Colore e forma:Solid
    Peso molecolare:341.4
  • Mecamylamine

    CAS:
    <p>Mecamylamine: oral, noncompetitive nAChR blocker, crosses blood-brain barrier, for neuropsychiatric and hypertension research.</p>
    Formula:C11H21N
    Colore e forma:Solid
    Peso molecolare:167.29
  • Bestim

    CAS:
    Bestim is an immunomodulatory dipeptide that is synthetic.
    Formula:C16H19N3O5
    Purezza:99.76%
    Colore e forma:Solid
    Peso molecolare:333.34
  • Aclidinium bromide

    CAS:
    <p>Aclidinium bromide (LAS-W 330) is a synthetic anticholinergic agent that is used as an inhalant for treatment of acute bronchospasm due to chronic bronchitis.</p>
    Formula:C26H30NO4S2·Br
    Purezza:99.53% - 99.69%
    Colore e forma:Solid
    Peso molecolare:564.55
  • Ilmetropium iodide

    CAS:
    Ilmetropium iodide is a bronchodilator.
    Formula:C20H30INO3
    Purezza:98.45%
    Colore e forma:Solid
    Peso molecolare:459.36
  • Fesoterodine

    CAS:
    Fesoterodine is an oral mAChR blocker (pKi: 7.3-8.0) for M1-M5, used to treat OAB.
    Formula:C26H37NO3
    Purezza:97.1%
    Colore e forma:Solid
    Peso molecolare:411.58
  • DMAB-anabaseine dihydrochloride

    CAS:
    <p>DMAB-anabaseine dihydrochloride (N,N-dimethyl-4-[(E)-(6-pyridin-3-yl-3,4-dihydro-2H-pyridin-5-ylidene)methyl]aniline;dihydrochloride) is an α7-containing</p>
    Formula:C19H23Cl2N3
    Purezza:99.91%
    Colore e forma:Solid
    Peso molecolare:364.31
  • Ethyl (triphenylphosphoranylidene) acetate

    CAS:
    <p>Ethyl (triphenylphosphoranylidene) acetate ((Carbethoxymethylene)triphenylphosphorane) may act as an cholinesterase inhibitor that inhibits AChE and BChE.</p>
    Formula:C22H21O2P
    Purezza:97.985%
    Colore e forma:White Or Slight Yellow Powder
    Peso molecolare:348.37
  • Brompheniramine

    CAS:
    Brompheniramine, an alkylamine antihistamine, targets H1 receptors (Kd=6.06nM) and has anticholinergic/depressant qualities. Blocks Ca/Na/hERG channels.
    Formula:C16H19BrN2
    Colore e forma:Solid
    Peso molecolare:319.24
  • Solifenacin hydrochloride

    CAS:
    Solifenacin Hcl is a muscarinic receptor antagonist.
    Formula:C23H27ClN2O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:398.93
  • Benzetimide hydrochloride

    CAS:
    Benzetimide hydrochloride (R4929) is an antagonist of muscarinic acetylcholine receptor.treatment neuroleptic-induced parkinsonism.
    Formula:C23H27ClN2O2
    Purezza:99.32%
    Colore e forma:Off-White Powder
    Peso molecolare:398.93
  • LY2119620

    CAS:
    LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.
    Formula:C19H24ClN5O3S
    Purezza:99.7%
    Colore e forma:Solid
    Peso molecolare:437.94
  • α-Conotoxin MII acetate


    α-Conotoxin MII acetate is a 16-amino acid peptide from the venom of the marine snail Conus magus.
    Formula:C69H107N23O24S4
    Purezza:94.82% - 97.79%
    Colore e forma:Solid
    Peso molecolare:1770.99
  • Anisotropine Methylbromide

    CAS:
    Anisotropine Methylbromide is an anticholinergic agent and has been used for relief of gastrointestinal spasm and for the suppression of gastric acid secretion.
    Formula:C17H32BrNO2
    Purezza:99.73%
    Colore e forma:Crystals From Acetone Solid
    Peso molecolare:362.35
  • ST034307

    CAS:
    ST034307 is an effective and selective inhibitor of adenylyl cyclase 1 (IC50: 2.3 μM).
    Formula:C10H4Cl4O2
    Purezza:99.28%
    Colore e forma:Solid
    Peso molecolare:297.95
  • Adiphenine

    CAS:
    Adiphenine is an inhibitor of nicotinic receptors.
    Formula:C20H25NO2
    Colore e forma:Solid
    Peso molecolare:311.42
  • Cyclodrine hydrochloride

    CAS:
    Cyclodrine hydrochloride is a dual cholinergic muscarinic receptor (mAChR) and nicotinic receptor (nAChR) antagonist that can be used in the study of
    Formula:C19H30ClNO3
    Purezza:98.59%
    Colore e forma:Solid
    Peso molecolare:355.9
  • PHA 568487

    CAS:
    PHA 568487: α-7 nAChR agonist, rapid brain uptake, lessens oxidative stress & neuroinflammation.
    Formula:C20H24N2O7
    Colore e forma:Solid
    Peso molecolare:404.419
  • PHA 568487 free base

    CAS:
    <p>PHA 568487 free base, an α7 nicotinic receptor agonist, designed to reduce bioactivation and improve in vivo tolerability.</p>
    Formula:C16H20N2O3
    Purezza:99.74%
    Colore e forma:Solid
    Peso molecolare:288.34
  • Mc-​Val-​Ala-​PAB

    CAS:
    <p>Mc-Val-Ala-PAB, an effective linker, is utilized in antibody-drug-conjugate (ADC).</p>
    Formula:C25H34N4O6
    Purezza:98.34% - 99.24%
    Colore e forma:Solid
    Peso molecolare:486.56
  • Oxyphencyclimine

    CAS:
    Oxyphencyclimine is a muscarinic receptor antagonist (MRA) anticholinergic drug used to treat peptic ulcers.
    Formula:C20H28N2O3
    Colore e forma:Solid
    Peso molecolare:344.45
  • suvn-911

    CAS:
    suvn-911 is a potent and selective antagonist of neuronal nicotinic acetylcholine α4β2 receptor (Ki = 1.5 nM) with antidepressant activity.
    Formula:C11H14Cl2N2O
    Purezza:98.88%
    Colore e forma:Solid
    Peso molecolare:261.15
  • Propantheline

    CAS:
    Propantheline: oral muscarinic receptor blocker for smooth muscle issues, hyperhidrosis, and bladder control.
    Formula:C23H30NO3
    Colore e forma:Solid
    Peso molecolare:368.49
  • Piperidolate hydrochloride

    CAS:
    Piperidolate hydrochloride, an antimuscarinic, reduces acetylcholine-induced intestinal spasms in rats and dogs.
    Formula:C21H26ClNO2
    Purezza:99.5%
    Colore e forma:Solid
    Peso molecolare:359.89
  • TQS

    CAS:
    TQS (4-Naphthalen-1-yl-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-8-sulfonamide) is a positive allosteric modulator of α7 nACh receptors.
    Formula:C22H20N2O2S
    Purezza:98.56%
    Colore e forma:Solid
    Peso molecolare:376.47
  • KH7

    CAS:
    KH7 is a soluble inhibitor of adenylyl cyclase (sAC)-specific.
    Formula:C17H15BrN4O2S
    Purezza:98.43%
    Colore e forma:Solid
    Peso molecolare:419.3
  • Succinylcholine Chloride Dihydrate

    CAS:
    <p>Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.</p>
    Formula:C14H30N2O4·2Cl·2H2O
    Purezza:99.87%
    Colore e forma:White Solid
    Peso molecolare:397.34
  • Nitenpyram

    CAS:
    <p>Nitenpyram (Capstar) is a nicotinic acetylcholine receptor (AchR) agonist, used as veterinary medicine to treat parasites of livestock and pets.</p>
    Formula:C11H15ClN4O2
    Purezza:99.03%
    Colore e forma:Light-Yellow Crystal
    Peso molecolare:270.72
  • Procyclidine hydrochloride

    CAS:
    <p>Procyclidine hydrochloride ((±)-Procyclidine hydrochlorid) is a potent anticholinergic agent and also have NMDA antagonist properties.</p>
    Formula:C19H30ClNO
    Purezza:99.24% - 99.88%
    Colore e forma:Crystals From Petroleum Ether White Powder
    Peso molecolare:323.9
  • NS9283

    CAS:
    <p>NS9283, a positive allosteric modulator selective for the α4β2 form, reduces ethanol consumption.</p>
    Formula:C14H8N4O
    Purezza:99.12%
    Colore e forma:Solid
    Peso molecolare:248.24
  • Sofpironium bromide

    CAS:
    <p>Sofpironium bromide (BBI4000) belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.</p>
    Formula:C22H32BrNO5
    Purezza:98.85%
    Colore e forma:Solid
    Peso molecolare:470.4
  • Batefenterol

    CAS:
    <p>Batefenterol (GSK961081) is a muscarinic antagonist and β2-agonist with high affinity (Ki: 1.4/1.3/3.7 nM).</p>
    Formula:C40H42ClN5O7
    Purezza:97.94% - 98.4%
    Colore e forma:Solid
    Peso molecolare:740.24
  • Nanofin

    CAS:
    <p>Nanofin (Lupetidine) is a neuropathic blocker, with antihypertensive effect.</p>
    Formula:C7H15N
    Purezza:97.38% - 99.818%
    Colore e forma:Clear Colorless To Slightly Yellow Liquid
    Peso molecolare:113.2
  • MC-Val-Cit-PABC-PNP

    CAS:
    MC-Val-Cit-PABC-PNP, also known as Mc-Val-Cit-PABC-PNP, is a cathepsin cleavable ADC peptide linker.
    Formula:C35H43N7O11
    Purezza:97.2% - 98.055%
    Colore e forma:Solid
    Peso molecolare:737.76
  • Blarcamesine

    CAS:
    <p>Blarcamesine (AVex-73) is a muscarinic M1 agonist potentially for the treatment of Alzheimer's disease.</p>
    Formula:C19H23NO
    Purezza:99.87%
    Colore e forma:Solid
    Peso molecolare:281.39
  • ML380

    CAS:
    <p>ML380 is a highly potent and the first CNS penetrant M5 positive allosteric modulator (PAM).</p>
    Formula:C23H25F3N4O3S
    Purezza:99.69%
    Colore e forma:Solid
    Peso molecolare:494.53
  • PNU-120596

    CAS:
    <p>PNU-120596 (NSC-216666) is a positive allosteric modulator of α7 nAChR with EC50 of 216 nM.</p>
    Formula:C13H14ClN3O4
    Purezza:99.82%
    Colore e forma:Solid
    Peso molecolare:311.72
  • NS 1738

    CAS:
    NS 1738 (NSC-213859) is a positive allosteric modulator of the α7-containing neuronal nicotinic acetylcholine receptors (nAChRs)
    Formula:C14H9Cl2F3N2O2
    Purezza:99.11%
    Colore e forma:Solid
    Peso molecolare:365.13
  • Nitrocaramiphen hydrochloride

    CAS:
    Nitrocaramiphen hydrochloride is a selective M1 muscarinic antagonist and inhibits binding to sigma sites in brain.
    Formula:C18H27ClN2O4
    Purezza:99.74%
    Colore e forma:Solid
    Peso molecolare:370.87
  • A 582941 HCl (848591-90-2(free base))


    <p>A-582941 is a alpha7 neuronal nicotinic receptor agonist with broad spectrum cognition-enhancing properties</p>
    Formula:C17H21ClN4
    Purezza:99.83%
    Colore e forma:Solid
    Peso molecolare:316.83
  • Solifenacin

    CAS:
    Solifenacin (YM905 free base) (YM905 free base) is a novel muscarinic receptor antagonist, its pKis for M1, M2 and M3 receptors is of 7.6, 6.9 and 8.0,
    Formula:C23H26N2O2
    Purezza:99.87%
    Colore e forma:Solid
    Peso molecolare:362.46
  • Syn-Ake acetate

    CAS:
    Syn-Ake acetate (Dipeptide diaminobutyroyl benzylamide) is a muscarinic acetylcholine receptor antagonist.
    Formula:C19H29N5O3·2(C2H4O2)
    Purezza:99.60%
    Colore e forma:Solid
    Peso molecolare:495.58
  • Velufenacin

    CAS:
    Velufenacin is an antagonist of muscarinic receptor[1].
    Formula:C19H20ClFN2O2
    Purezza:99.65%
    Colore e forma:Solid
    Peso molecolare:362.83
  • Mepenzolate Bromide

    CAS:
    <p>Mepenzolate Bromide (Colibantil) is a muscarinic antagonist used to treat gastrointestinal conditions.</p>
    Formula:C21H26BrNO3
    Purezza:95.73% - 99.21%
    Colore e forma:Solid
    Peso molecolare:420.34
  • AF-710B

    CAS:
    <p>AF710B is an enantiomer of AF710. AF-710B is also a sigma and M1 muscarinic receptors agonist.</p>
    Formula:C20H27N3OS
    Purezza:98.62% - 99.89%
    Colore e forma:Solid
    Peso molecolare:357.51
  • Pentoxyverine

    CAS:
    Pentoxyverine (Carbetapentan) is an orally available cough suppressant, an antagonist of muscarinic receptor M1 and an agonist of the σ1 receptor.
    Formula:C20H31NO3
    Purezza:97.11%
    Colore e forma:Solid
    Peso molecolare:333.47
  • Xanomeline tartrate

    CAS:
    Xanomeline tartrate (LY 246708 tartrate) 是 M1和 M4 mAChR 激动剂,具有抗精神病样活性,可改善认知,可用于研究精神分裂症和阿尔茨海默病。
    Formula:C18H29N3O7S
    Purezza:99.19% - 99.99%
    Colore e forma:Solid
    Peso molecolare:431.5
  • Pipecuronium bromide

    CAS:
    Pipecuronium bromide (RGH-1106) is an nAChR antagonist that also acts as a non-depolarising steroidal neuromuscular blocker that causes muscle relaxation.
    Formula:C35H62Br2N4O4
    Purezza:>99.99%
    Colore e forma:Powder
    Peso molecolare:762.7
  • Monepantel

    CAS:
    Monepantel (AAD1566) is an organic anthelmintic and an antagonist of nAChRs from roundworms and esophageostomy.
    Formula:C20H13F6N3O2S
    Purezza:99.83%
    Colore e forma:White Powder
    Peso molecolare:473.39
  • Varenicline

    CAS:
    Varenicline (CP 526555) is a selective partial agonist of the α4β2 nAChR and a full agonist of the α3β4 nAChR and α7 nAChR.
    Formula:C13H13N3
    Purezza:99.76%
    Colore e forma:Solid
    Peso molecolare:211.26
  • Atropine hydrobromide

    CAS:
    Atropine hydrobromide is a biochemical.
    Formula:C17H24BrNO3
    Colore e forma:Solid
    Peso molecolare:370.28
  • Pyrantel

    CAS:
    Pyrantel: Nicotinic agonist; causes spastic paralysis in nematodes by depolarizing block.
    Formula:C11H14N2S
    Purezza:98%
    Colore e forma:Crystals From Methanol Yellowish Crystalline Powder
    Peso molecolare:206.31
  • Anatabine dicitrate


    Anatabine dicitrate is a tobacco alkaloid that can cross the blood-brain barrier.
    Formula:C22H28N2O14
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:544.46
  • Flavoxate

    CAS:
    <p>Flavoxate is an anticholinergic with antimuscarinic effects.</p>
    Formula:C24H25NO4
    Colore e forma:Solid
    Peso molecolare:391.46
  • (±)-Atropine-d3 (N-methyl-d3)

    CAS:
    (±)-Atropine-d3 (N-methyl-d3) is a deuterated compound of (±)-Atropine. (±)-Atropine has a CAS number of 51-55-8. Atropine Sulfate is the sulfate salt of atropine, a naturally-occurring alkaloid isolated from the plant Atropa belladonna. Atropine functions as a sympathetic, competitive antagonist of muscarinic cholinergic receptors, thereby abolishing the effects of parasympathetic stimulation.
    Formula:C17H20D3NO3
    Peso molecolare:292.39
  • Diphenidol

    CAS:
    <p>Diphenidol, a muscarinic antagonist, is employed as an antivertigo and antiemetic agent.</p>
    Formula:C21H27NO
    Colore e forma:Needles From Petroleum Ether Solid
    Peso molecolare:309.45
  • VU0029767

    CAS:
    <p>VU0029767 is an allosteric enhancer of the M1 muscarinic receptor, capable of modulating the receptor's activity. This compound enhances M1 receptor activity by increasing agonist affinity. However, VU0029767 demonstrates distinct characteristics from other compounds, particularly under varying experimental conditions such as its interaction with mutated M1 receptors and its effects on downstream signaling pathways.</p>
    Formula:C21H21N3O3
    Colore e forma:Solid
    Peso molecolare:363.41
  • Catestatin

    CAS:
    Non-competitive inhibitor of nicotinic receptors; blocks cationic signalling and catecholamine release; stimulates histamine release. IC50 ~200-250nM.
    Formula:C107H173N37O26S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:2425.84
  • N-Biotinyl p-aminophenyl arsenic acid

    CAS:
    N-Biotinyl p-aminophenyl arsenic acid is a bifunctional reagent that binds to streptavidin and disulfide compounds. It diminishes the binding sites of rbungarotoxin on reduced nicotinic receptors with an IC50 ranging from 10-300 nM, thus shielding the receptors from irreversible alkylation by bromoacetylcholine.
    Formula:C16H22AsN3O4S
    Colore e forma:Solid
    Peso molecolare:427.35
  • Phenglutarimide hydrochloride

    CAS:
    Phenglutarimide hydrochloride is an anticholinergic. It is used as an antiparkinsonian agent.
    Formula:C17H25ClN2O2
    Colore e forma:Solid
    Peso molecolare:324.85
  • Aprofene

    CAS:
    <p>Aprofene blocks acetylcholine receptors, used for peptic ulcers, endarteritis, cholecystitis, and colitis.</p>
    Formula:C21H27NO2
    Colore e forma:Solid
    Peso molecolare:325.44
  • Dianicline dihydrochloride

    CAS:
    Dianicline dihydrochloride is a partial agonist of α4β2 nicotinic acetylcholine receptor. It increases cessation rates in a dose-dependent manner.
    Formula:C13H16N2O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:216.28
  • Biperiden lactate

    CAS:
    <p>Biperiden lactate is a biochemical.</p>
    Formula:C24H35NO4
    Colore e forma:Solid
    Peso molecolare:401.54
  • AN317

    CAS:
    AN317 is a selective agonist for the nicotinic acetylcholine receptor (nAChR) containing α6β2, with dissociation constants (Ki) of 6.2 nM and 4.1 nM for the α6/α3β2β3 and α4β2 receptor subtypes, respectively. It induces dopamine release in rat striatal synaptosomes, enhances the activity of dopaminergic neurons in the substantia nigra, and exhibits protective effects against the dopaminergic neurotoxin MPP+ in rat neurons. AN317 also demonstrates favorable pharmacokinetic properties in rats and permeability across the blood-brain barrier (BB).
    Formula:C13H19N3
    Colore e forma:Solid
    Peso molecolare:217.31
  • Azacyclonol hydrochloride

    CAS:
    Azacyclonol hydrochloride can be used in the treatment of chronic schizophrenia.
    Formula:C18H22ClNO
    Colore e forma:Off White Crystalline Powder
    Peso molecolare:303.83
  • Oxantel

    CAS:
    <p>Oxantel is a fumarate reductase inhibitor with anthelmintic activity.</p>
    Formula:C13H16N2O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:216.28
  • Sulindac sulfide

    CAS:
    Sulindac sulfide: NSAID targeting COX-1, inhibits Ras-Raf-1 and gamma-secretase (IC50: 20.2 μM), active sulinic acid metabolite.
    Formula:C20H17FO2S
    Purezza:99.35%
    Colore e forma:Solid
    Peso molecolare:340.41
  • BTM-1086

    CAS:
    BTM-1086 is a potent gastric secretory inhibitor and an anti-ulcer agent.
    Formula:C21H25N3OS
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:367.51
  • CP-601932

    CAS:
    CP-601932 (free base) is a selective base α( 4) β( 2) Nicotinic acetylcholine receptor agonist.
    Formula:C12H12F3N
    Colore e forma:Solid
    Peso molecolare:227.23
  • Eucatropine

    CAS:
    Eucatropine, an anticholinergic agent, acts as a potent inhibitor of the muscarinic acetylcholine receptor (mAChR) with an IC 50 value of 0.583 μM.
    Formula:C17H25NO3
    Colore e forma:Solid
    Peso molecolare:291.39
  • Thiochrome

    CAS:
    Thiochrome is a selective enhancer of M4 muscarinic receptor of acetylcholine (ACh) affinity.
    Formula:C12H14N4OS
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:262.33
  • GAT107

    CAS:
    GAT107, a strong α7 nicotinic receptor modulator, aids inflammation and neuropathic pain in mice.
    Formula:C18H17BrN2O2S
    Purezza:99.33%
    Colore e forma:Solid
    Peso molecolare:405.31
  • VU0090157

    CAS:
    VU0090157, a novel allosteric potentiators of M1 muscarinic receptor, may provide novel treatments for schizophrenia and Alzheimer's disease.
    Formula:C19H21N3O7
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:403.39
  • S-(+)-Mecamylamine hydrochloride

    CAS:
    Dexmecamylamine( TC-5214, NIH-11008) is used as a nicotinic channel modulator with antidepressant activity.
    Formula:C11H22ClN
    Colore e forma:Solid
    Peso molecolare:203.75
  • T761-0184

    CAS:
    T761-0184 is a potent antagonist of α7 nicotinic receptor (nAChR) [1].
    Formula:C16H20FN3O
    Colore e forma:Solid
    Peso molecolare:289.35
  • Revatropate

    CAS:
    Revatropate, a selective muscarinic antagonist, is an antimuscarinic drug.
    Formula:C19H27NO4S
    Colore e forma:Solid
    Peso molecolare:365.49
  • Rispenzepine

    CAS:
    Rispenzepine, a novel mAChRs M1/M3 antagonist, treats immune, infections, and respiratory issues.
    Formula:C19H20N4O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:336.39
  • SCH 57790

    CAS:
    SCH 57790: selective muscarinic M2 blocker, boosts acetylcholine & cognition, may treat Alzheimer's.
    Formula:C25H31N3O2S
    Purezza:99.12% - 99.69%
    Colore e forma:Solid
    Peso molecolare:437.6
  • Tarafenacin

    CAS:
    Tarafenacin is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over the M2 receptor.
    Formula:C21H20F4N2O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:408.39
  • Milameline

    CAS:
    Milameline is a muscarinic receptor agonist that improves cognition.
    Formula:C8H14N2O
    Colore e forma:Solid
    Peso molecolare:154.21
  • Biricodar dicitrate

    CAS:
    Biricodar dicitrate (VX-710) is a potent MDR inhibitor with no anticancer activity and can be used to study prostate cancer.
    Formula:C46H57N3O21
    Purezza:97.78% - 99.78%
    Colore e forma:Solid
    Peso molecolare:987.95
  • Sofiniclin

    CAS:
    Sofiniclin (ABT 894) is an agonist of nicotinic acetylcholine receptor (nAChR). It is used for the research for attention-deficit/hyperactivity disorder (ADHD).
    Formula:C10H11Cl2N3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:244.12
  • SR 16584

    CAS:
    α3β4 nAChR antagonist
    Formula:C17H22N2O
    Purezza:99.84%
    Colore e forma:Solid
    Peso molecolare:270.37
  • Bibn 99

    CAS:
    <p>Bibn 99, a lipophilic and selective muscarinic M2 receptor antagonist, has applications in cognitive performance and Alzheimer's Disease.</p>
    Formula:C31H42ClN5O3
    Colore e forma:Solid
    Peso molecolare:568.15
  • VU 6008667

    CAS:
    VU 6008667 is a selective negative allosteric M5 NAM modulator (IC50s: 1.2 μM and 1.6 μM for human M5 and rat M5, respectively).
    Formula:C24H17ClF2N2O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:438.85
  • Rivanicline

    CAS:
    Rivanicline is a selective α4β2 nicotinic receptor agonist (Ki=26 nM), with >1,000x less affinity for α7 receptors.
    Formula:C10H14N2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:162.23
  • Rapacuronium bromide

    CAS:
    Rapacuronium bromide is an allosteric muscarinic acetylcholine receptor (mAChR) modulator.
    Formula:C37H61BrN2O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:677.8
  • ML375

    CAS:
    ML375 is a potent, selective and CNS penetrant M5 negative allosteric modulator (NAM).
    Formula:C23H15ClF2N2O2
    Colore e forma:Solid
    Peso molecolare:424.83
  • Sch412348

    CAS:
    Sch412348: potent A2A receptor antagonist, Ki=0.6 nM, >1000-fold selectivity vs. other adenosine receptors.
    Formula:C22H21F2N9O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:465.46
  • CP-601927

    CAS:
    CP-601927 is a nicotinic acetylcholine receptor (NACHR) agonist with permeability, high affinity, and selectivity.
    Formula:C12H12F3N
    Colore e forma:Solid
    Peso molecolare:227.23
  • Arecaidine propargyl ester tosylate

    CAS:
    Arecaidine propargyl ester tosylate is a muscarinic receptor agonist.
    Formula:C17H21NO5S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:351.42
  • VMY-2-95

    CAS:
    VMY-2-95 is an α4β2 nicotinic acetylcholine receptors (nAChRs) selective desensitizer.
    Formula:C17H16N2O
    Colore e forma:Solid
    Peso molecolare:264.32
  • RJR 2429 dihydrochloride

    CAS:
    nAChR agonist that displays selectivity for α4β2
    Formula:C12H18Cl2N2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:261.19
  • J 104129 fumarate

    CAS:
    M3 muscarinic receptor antagonist
    Formula:C24H36N2O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:384.55
  • Alvameline maleate

    CAS:
    Alvameline maleate is used as a Partial M1 Agonist and M2/M3 Antagonist.
    Formula:C13H19N5O4
    Colore e forma:Solid
    Peso molecolare:309.32
  • Vinconate

    CAS:
    Vinconate is an indolonaphthyridine derivative and can stimulate the muscarinic acetylcholine receptor.
    Formula:C18H20N2O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:296.36
  • AT-1001

    CAS:
    AT-1001 is an α3β4 nAChR partial agonist reducing nicotine relapse and withdrawal with negligible impact on food response and dopamine release.
    Formula:C15H21BrN2
    Colore e forma:Solid
    Peso molecolare:309.24
  • PD-102807

    CAS:
    PD-102807 is a selective and competitive M4 muscarinic receptor antagonist for Parkinson's disease research, inhibit airway smooth muscle (ASM) contraction.
    Formula:C23H24N2O4
    Purezza:98.90%
    Colore e forma:Solid
    Peso molecolare:392.45
  • Rivanicline oxalate

    CAS:
    Rivanicline oxalate is an agonist of neuronal nicotinic receptor, showing high selectivity for the α4β2 subtype (Ki=26 nM).
    Formula:C12H16N2O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:252.27
  • Bradanicline HCl

    CAS:
    Bradanicline(TC-5619) is the agonist of Alpha-7 Nicotinic Receptor.
    Formula:C22H24ClN3O2
    Colore e forma:Solid
    Peso molecolare:397.9
  • S 24795

    CAS:
    S 24795 (Catestatin acetate(142211-96-9 free base)) is an α7 nAChR partial agonist.
    Formula:C14H13BrINO
    Purezza:99.934%
    Colore e forma:Solid
    Peso molecolare:418.07
  • DREADD agonist 21 dihydrochloride

    CAS:
    DREADD agonist 21 dihydrochloride is a potent human muscarinic acetylcholine M3 receptors ( hM3Dq ) agonist with EC 50 of 1.7 nM [1].
    Formula:C17H20Cl2N4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:351.27
  • BPIPP

    CAS:
    guanylyl cyclase (GC) and adenylyl cyclase (AC) inhibitor
    Formula:C22H16BrN3O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:450.28
  • Procyclidine

    CAS:
    Procyclidine is an anticholinergic, muscarinic and NMDA antagonist used in Parkinson's and psychiatric disorder studies.
    Formula:C19H29NO
    Colore e forma:Solid
    Peso molecolare:287.44
  • Oxybutynin R-isomer HCl

    CAS:
    Aroxybutynin, R-isomer of oxybutynin, is a muscarinic antagonist with antispasmodic effects on bladder muscle, weaker than atropine.
    Formula:C22H32ClNO3
    Colore e forma:Solid
    Peso molecolare:393.95
  • VU0455691

    CAS:
    VU0455691 is a selective M1 Muscarinic Receptor Allosteric Modulators.
    Formula:C24H25N5O3S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:463.55
  • Ambutonium bromide

    CAS:
    Ambutonium bromide is an antagonist of acetylcholine.
    Formula:C20H27BrN2O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:391.35
  • (±)-Muscarine chloride

    CAS:
    (±)-Muscarine chloride is the racemate of Muscarine chloride. Muscarine is a prototypical agonist for the muscarinic acetylcholine receptor [1] [2].
    Formula:C9H20ClNO2
    Colore e forma:Solid
    Peso molecolare:209.71
  • Methapyrilene

    CAS:
    Methapyrilene is a histamine H1 antagonist with sedative action.
    Formula:C14H19N3S
    Colore e forma:Liquid Physical Description Clear Colorless Liquid (Ntp 1992)
    Peso molecolare:261.39
  • Milameline hydrochloride

    CAS:
    Milameline hydrochloride is a Muscarinic receptor agonist.
    Formula:C8H15ClN2O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:190.67
  • Cycrimine

    CAS:
    Cycrimine: oral M1 mAChR blocker, lowers acetylcholine, antispasmodic, for Parkinson's and mental disorder studies.
    Formula:C19H29NO
    Colore e forma:Solid
    Peso molecolare:287.44
  • Parapenzolate bromide

    CAS:
    Parapenzolate bromide is an orally active mAChR antagonist. parapenzolate bromide is an anticholinergic and antitussive agent.
    Formula:C21H26BrNO3
    Colore e forma:Solid
    Peso molecolare:420.347