
AChR
Gli inibitori del recettore dell'acetilcolina (AChR) sono composti che bloccano l'attività dei recettori dell'acetilcolina, fondamentali per la neurotrasmissione nei sistemi nervoso centrale e periferico. Gli AChR svolgono un ruolo cruciale nella contrazione muscolare, nella memoria e nelle funzioni cognitive. Gli inibitori degli AChR vengono utilizzati per studiare condizioni come la miastenia grave, l'Alzheimer e altri disturbi neurologici. Modulando l'attività degli AChR, questi inibitori possono aiutare a svelare le complessità della segnalazione colinergica nel cervello. Presso CymitQuimica, offriamo una gamma di inibitori degli AChR per supportare la tua ricerca in neuroscienze, farmacologia e malattie neurodegenerative.
Trovati 617 prodotti di "AChR"
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Glycerophosphoinositol choline
CAS:Glycerophosphoinositol choline is the salt of choline and glycerophosphoinositol.Formula:C14H32NO12PColore e forma:SolidPeso molecolare:437.38Clorprenaline
CAS:Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.Formula:C11H16ClNOPurezza:98.9%Colore e forma:SolidPeso molecolare:213.7NKH477
CAS:NKH477 (Colforsin dapropate hydrochloride) is a derivative of forskolin with antidepressant activity.Formula:C27H44ClNO8Purezza:98% - 98%Colore e forma:SolidPeso molecolare:546.09Biperiden
CAS:Biperiden is a muscarinic antagonist for Parkinson's and drug-induced extrapyramidal symptoms.Formula:C21H29NOPurezza:99.65%Colore e forma:Crystals SolidPeso molecolare:311.46SSR180711 hydrochloride
CAS:SSR180711 hydrochloride (SSR-180711A HCl) is an Alpha7 nicotinic acetylcholine partial agonist that can be used to study neurolysis.Formula:C14H18BrClN2O2Purezza:99.22%Colore e forma:SolidPeso molecolare:361.66NBTGR
CAS:NBTGR is a potent nucleoside transport inhibitor(adenosine uptake ,Ki of 70 nM).Formula:C17H18N6O6SPurezza:98%Colore e forma:SolidPeso molecolare:434.43Dexetimide
CAS:Dexetimide, a muscarinic receptor antagonist, treats neuroleptic-induced parkinsonism.Formula:C23H26N2O2Colore e forma:SolidPeso molecolare:362.46Metixene hydrochloride hydrate
CAS:Metixene HCl hydrate is a potential anticholinergic for Parkinson's with IC50 of 55 nM and Ki of 15 nM against muscarine receptors.Formula:C20H26ClNOSPurezza:99.99%Colore e forma:SolidPeso molecolare:363.95N6-Methyladenosine 5'-monophosphate disodium salt
CAS:N6-Methyladenosine 5'-monophosphate disodium salt is a glycogen phosphorylase b activator and an inhibitor of adenylate kinase II.Formula:C11H14N5Na2O7PPurezza:99.36% - 99.36%Colore e forma:SolidPeso molecolare:405.21Varenicline Hydrochloride
CAS:Varenicline Hydrochloride (CP 526555) is an orally active partial agonist of the α4β2 nicotinic acetylcholine receptor (α4β2 nAChR, IC50 = 250 nM).Formula:C13H14ClN3Purezza:99.854%Colore e forma:SolidPeso molecolare:247.72Tolterodine
CAS:Tolterodine ((R)-(+)-Tolterodine) is an mACh antagonist used in the treatment of detrusor instability and overactive bladder syndrome.Formula:C22H31NOPurezza:99.71%Colore e forma:White Like Or Light Brown Crystalline PowderPeso molecolare:325.49Ispronicline
CAS:Ispronicline (TC-1734) An orally active, selective, and potent α4β2 nAChR partial agonist with antidepressant, neuroprotective, and long-lasting cognitiveFormula:C14H22N2OPurezza:97.70% - 99.16%Colore e forma:SolidPeso molecolare:234.34Cevimeline
CAS:Cevimeline: muscarinic agonist, treats dry mouth & Sjögren's, boosts saliva post-cancer radiotherapy.Formula:C10H17NOSColore e forma:Off-White SolidPeso molecolare:199.31Fesoterodine L-mandelate
CAS:Fesoterodine L-mandelate is a efficacious antimuscarinic agent for the overactive bladder (OAB).Formula:C34H45NO6Colore e forma:SolidPeso molecolare:563.735Tebanicline dihydrochloride
CAS:Tebanicline dihydrochloride: oral analgesic, nAChR modulator, Ki=37 pM at α4β2 receptors, inhibits cytisine binding.Formula:C9H13Cl3N2OColore e forma:SolidPeso molecolare:271.57YM-58790 hydrochloride
CAS:YM-58790 is a potent M3 muscarinic receptor antagonist(Ki of 15 nM).Formula:C27H32ClN3O2Purezza:98%Colore e forma:SolidPeso molecolare:466.02Fipexide hydrochloride
CAS:Fipexide (hydrochloride) is a kind of psychoactive drug of the piperazine class.Formula:C20H22Cl2N2O4Colore e forma:SolidPeso molecolare:425.31Telenzepine dihydrochloride
CAS:muscarinic M1 receptor antagonistFormula:C19H23ClN4O2SPurezza:98%Colore e forma:SolidPeso molecolare:406.93NS3861 fumarate
CAS:NS3861 fumarate, a partial α3β4 nAChR agonist, binds α3β2, α4β4, α4β2 with Ki values of 0.62, 25, 7.8, 55 nM.Formula:C16H18BrNO4SColore e forma:SolidPeso molecolare:400.29Sabcomeline hydrochloride
CAS:Sabcomeline is a selective M1 receptor partial agonist.Formula:C10H16ClN3OColore e forma:SolidPeso molecolare:229.71Clothianidin
CAS:Clothianidin (TI 435), an insecticide, stimulates nAChR as acetylcholine agonist, not AChE inhibitor.Formula:C6H8ClN5O2SPurezza:99.71% - 99.87%Colore e forma:Solid PowderPeso molecolare:249.68VU0152099
CAS:VU0152099 is a potent and selective M4 mAChR allosteric potentiator(EC50 = 380 ± 93 nM).Formula:C18H17N3O3SPurezza:98.46%Colore e forma:SolidPeso molecolare:355.41TBPB
CAS:<p>TBPB is an allosteric M1 mAChR agonist.</p>Formula:C25H32N4OPurezza:97.87% - 99.9%Colore e forma:SolidPeso molecolare:404.55Nitrobenzylthioinosine
CAS:<p>Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.</p>Formula:C17H17N5O6SPurezza:99.69% - 99.74%Colore e forma:Off-White SolidPeso molecolare:419.41Umeclidinium bromide
CAS:Umeclidinium bromide (GSK573719A) is a novel mAChR antagonist.Formula:C29H34BrNO2Purezza:98.4% - 99.89%Colore e forma:SolidPeso molecolare:508.49Pempidine
CAS:Pempidine (1,2,2,6,6-Pentamethylpiperidine) is a nicotinic antagonist, has been used as a ganglionic blocker in the treatment of hypertension.Formula:C10H21NPurezza:98.18% - 99.28%Colore e forma:Colorless - Light Yellow Clear LiquidPeso molecolare:155.28Methylbenactyzium Bromide
CAS:Methylbenactyzium Bromide (Semulgin) is an anticonvulsant that is the active metabolite of trimethadione.Formula:C21H28BrNO3Purezza:99.29%Colore e forma:SolidPeso molecolare:422.36Rivanicline hemioxalate
<p>Rivanicline hemioxalate is a selective α4β2 nicotinic receptor agonist (K i =26 nM), over 1,000x preference to α7 (K i =3.6 μM), with limited side effects.</p>Formula:C12H16N2O4Purezza:98%Colore e forma:SolidPeso molecolare:207.23PSEM 89S TFA
CAS:<p>PSEM 89S TFA is a brain-penetrant and selective ion channels agonist, and is orthogonally selective for Q79G and L141F, respectively.</p>Formula:C18H23F3N2O5Purezza:99.9%Colore e forma:SolidPeso molecolare:404.38Prifinium bromide
CAS:<p>Prifinium bromide is a quaternary ammon antimuscarinic. It inhibits hyperkinesia of the digestive organs and urinary tract and has a spasmolytic action.</p>Formula:C22H28BrNPurezza:97.99%Colore e forma:SolidPeso molecolare:386.37(S)-UFR2709
CAS:(S)-UFR2709, a nAChR competitive antagonist, favors α4β2 over α7, reduces anxiety and alcohol use in rats.Formula:C13H17NO2Colore e forma:SolidPeso molecolare:219.284Oxotremorine sesquifumarate
CAS:<p>Oxotremorine sesquifumarate is a muscarinic agonist.</p>Formula:C12H18N2OC4H4O4Purezza:97.94%Colore e forma:SolidPeso molecolare:380.39(-)-(S)-B-973B
CAS:<p>(-)-(S)-B-973B is an effective allosteric agonist and a positive allosteric modulator of α7 nAChR.</p>Formula:C24H26F2N6OPurezza:99.52%Colore e forma:SolidPeso molecolare:452.5Mecamylamine hydrochloride
CAS:Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.Formula:C11H22ClNPurezza:99.76% - >99.99%Colore e forma:White SolidPeso molecolare:203.75VU0152100
CAS:<p>VU0152100 is an effective and selective allosteric potentiator of M4 mAChR (EC50: 380 ± 93 nM).</p>Formula:C18H19N3O2SPurezza:99.56%Colore e forma:SolidPeso molecolare:341.43OXOMEMAZINE
CAS:Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in cough research.Formula:C18H22N2O2SPurezza:99.58%Colore e forma:SolidPeso molecolare:330.44Darifenacin
CAS:Darifenacin (UK-88525) is a muscarinic receptor M3 antagonist with anticonvulsant activity and can be used to study urinary incontinence and overactive bladder.Formula:C28H30N2O2Purezza:99.78%Colore e forma:SolidPeso molecolare:426.55Dicyclomine
CAS:Dicyclomine: oral muscarinic antagonist, eases GI muscle spasms, high affinity for M1/M2 receptors, Ki of 5.1 nM/54.6 nM.Formula:C19H35NO2Colore e forma:SolidPeso molecolare:309.49JHU37160
CAS:JHU37160 is a DREADD agonist with Ki of 1.9 nM for hM3Dq, 3.6 nM for hM4Di, and EC50 of 18.5 nM (hM3Dq), 0.2 nM (hM4Di) in HEK-293 cell assays.Formula:C19H20ClFN4Purezza:99.87%Colore e forma:SolidPeso molecolare:358.84Dronedarone
CAS:<p>Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.</p>Formula:C31H44N2O5SPurezza:98.85% - 99.58%Colore e forma:SolidPeso molecolare:556.76Nor-benzetimide
CAS:Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.Formula:C16H20N2O2Purezza:98.63%Colore e forma:SolidPeso molecolare:272.34Isopropamide Iodide
CAS:<p>Isopropamide iodide: long-acting anticholinergic, treats peptic ulcers, GI disorders, Alzheimer's.</p>Formula:C23H33IN2OPurezza:99.67%Colore e forma:SolidPeso molecolare:480.43W-84 dibromide
CAS:<p>W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.</p>Formula:C32H44Br2N4O4Purezza:95.56%Colore e forma:SolidPeso molecolare:708.52CCMI
CAS:<p>CCMI (AVL-3288) is a potent and selective modulator of α7 nAChR-positive allosteric.</p>Formula:C19H15Cl2N3O2Purezza:>99.99%Colore e forma:SolidPeso molecolare:388.25Glycopyrrolate
CAS:Glycopyrrolate: muscarinic antagonist, antispasmodic for GI issues, reduces salivation with anesthesia.Formula:C19H28BrNO3Purezza:99.41% - 99.64%Colore e forma:SolidPeso molecolare:398.33Ursulcholic acid
CAS:Ursulcholic acid (Ursulcholic) is a water-soluble anticholinergic compound.Formula:C24H40O10S2Purezza:98%Colore e forma:SolidPeso molecolare:552.7VU0357017 hydrochloride
CAS:VU0357017 hydrochloride (ML071 hydrochloride) is highly selective M1 agonists act at an allosteric site to activate the receptor (EC50: 477 ± 172 nM; Pec50: 6.Formula:C18H28ClN3O3Purezza:99% - 99.97%Colore e forma:SolidPeso molecolare:369.89Revefenacin
CAS:Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.Formula:C35H43N5O4Purezza:98.12%Colore e forma:SolidPeso molecolare:597.75BNC210
CAS:BNC210 (IW-2143) is a α7 nAChR negative allosteric modulator. BNC210 has potent activity in animal models of anxiety and depression.Formula:C17H23N3O3Purezza:97.05% - >99.99%Colore e forma:SolidPeso molecolare:317.38PNU-282987 S enantiomer free base
CAS:PNU-282987 S enantiomer free base is an agonist of α7 nicotinic acetylcholine receptor (α7 nAChR).Formula:C14H17ClN2OPurezza:99.74%Colore e forma:SolidPeso molecolare:264.75Piperidolate
CAS:Piperidolate inhibits intestinal cramp induced by acetylcholineFormula:C21H25NO2Purezza:98.45%Colore e forma:SolidPeso molecolare:323.43BQCA
CAS:<p>BQCA (benzylquinolone carboxylic acid) a highly selective allosteric M1 mAChR modulator.</p>Formula:C18H15NO4Purezza:97.22%Colore e forma:SolidPeso molecolare:309.32Varenicline dihydrochloride
CAS:Varenicline dihydrochloride is a Selective α4β2 nicotinic acetylcholine receptor partial agonist.Formula:C13H15Cl2N3Purezza:99.88% - 99.97%Colore e forma:SolidPeso molecolare:284.18Harman hydrochloride
CAS:Harman hydrochloride triggers CYP1A1 gene via AhR, potentially causing mutations and cancer.Formula:C12H11ClN2Purezza:99.35%Colore e forma:SolidPeso molecolare:218.68Imidafenacin
CAS:Imidafenacin (KRP-197)(KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM.Formula:C20H21N3OPurezza:99.17%Colore e forma:SolidPeso molecolare:319.4EB-3D
CAS:EB-3D is a potent and selective choline kinase alpha 1 (ChoKα1) inhibitor(IC50 : 1 μM).with anti-cancer activity.Formula:C30H36Br2N4O2Purezza:99.48%Colore e forma:SolidPeso molecolare:644.4JHU37152
CAS:JHU37152 is a DREADD agonist; Ki: 1.8 nM at hM3Dq, 8.7 nM at hM4Di; EC50: 5 nM (hM3Dq), 0.5 nM (hM4Di) in HEK-293 cell assays.Formula:C19H20ClFN4Purezza:99.72%Colore e forma:SolidPeso molecolare:358.84SEN12333
CAS:<p>SEN12333 is an α7 nicotinic acetylcholine receptor (nAChR) agonist</p>Formula:C20H25N3O2Purezza:99.02%Colore e forma:SolidPeso molecolare:339.43mAChR-IN-1 hydrochloride
CAS:mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 Nm.Formula:C23H26ClIN2O2Purezza:99.87%Colore e forma:SolidPeso molecolare:524.824BP-TQS
CAS:4BP-TQS is an allosteric agonist of α7 nAChRs.Formula:C18H17BrN2O2SPurezza:99.96%Colore e forma:SolidPeso molecolare:405.31Tebanicline hydrochloride
CAS:Tebanicline hydrochloride (Ebanicline hydrochloride) , is an effective synthetic nicotinic (non-opioid) analgesic drug.Formula:C9H12Cl2N2OPurezza:91.74% - 98.78%Colore e forma:SolidPeso molecolare:235.11PHA 543613 hydrochloride
CAS:PHA-543613 hydrochloride, a potent α7 nicotinic receptor agonist, may treat schizophrenia-related cognitive deficits.Formula:C15H18ClN3O2Colore e forma:SolidPeso molecolare:307.78Pozanicline dihydrochloride
CAS:Pozanicline dihydrochloride (ABT-089 dihydrochloride) is an orally bioavailable agonist of nicotinic acetylcholine receptor (nAChR) (Ki = 16.7 nM)Formula:C11H18Cl2N2OPurezza:98%Colore e forma:SolidPeso molecolare:265.18VU0467154
CAS:VU0467154 is a positive allosteric modulator of the M4 muscarinic acetylcholine receptor.Formula:C17H15F3N4O3S2Purezza:99.51% - 99.53%Colore e forma:SolidPeso molecolare:444.45Pempidine HCl
CAS:Pempidine HCl, a nicotinic antagonist and former hypertension treatment, now mainly serves as a lab tool.Formula:C10H22ClNColore e forma:SolidPeso molecolare:191.74Atracurium besylate
CAS:Atracurium besylate (51W89) is a short-acting, non-depolarizing muscle relaxant, not affecting the heart or reliant on kidneys.Formula:C65H82N2O18S2Purezza:98.94% - 99.71%Colore e forma:SolidPeso molecolare:1243.49VU0119498
CAS:VU0119498 is a M1 muscarinic receptor agonist (EC50 = 3.1 μM) and pan mAChR M3, M5 positive allosteric modulator (PAM),and is a neuroprotective agent.Formula:C15H10BrNO2Purezza:97.56%Colore e forma:SolidPeso molecolare:316.15Batefenterol Succinate
CAS:Batefenterol Succinate is a first-in-class inhaled bifunctional bronchodilator possessing muscarinic receptor antagonist and β2-adrenoceptor agonist properties.Formula:C44H48ClN5O11Colore e forma:SolidPeso molecolare:858.34Varenicline Tartrate
CAS:<p>Varenicline Tartrate (CP 526555-18) is a benzazepine derivative that functions as an ALPHA4/BETA2 NICOTINIC RECEPTOR partial agonist.</p>Formula:C13H13N3·C4H6O6Purezza:98.23% - 98.32%Colore e forma:Tan SolidPeso molecolare:361.35VU0238441
CAS:VU0238441 is agonist of Muscarinic acetylcholine receptor M5 (human) with EC50 of 2.1μM.Formula:C16H9ClF3NO2Purezza:100%Colore e forma:SolidPeso molecolare:339.7Encenicline hydrochloride
CAS:Encenicline hydrochloride (EVP-6124 hydrochloride) is a new-type partial agonist of α7 neuronal nicotinic acetylcholine receptors (nAChRs).Formula:C16H17ClN2OS·HClPurezza:98.34% - 99.85%Colore e forma:SolidPeso molecolare:357.39-Ethyladenine
CAS:9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].Formula:C7H9N5Purezza:99.35% - 99.37%Colore e forma:SolidPeso molecolare:163.18VU 0238429
CAS:<p>VU 0238429 (SCR-1481B1) is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5)( EC50 : 1.16 μM).</p>Formula:C17H12F3NO4Purezza:>99.99%Colore e forma:SolidPeso molecolare:351.28MC-Val-Cit-PAB
CAS:<p>MC-Val-Cit-PAB: cathepsin-cleavable ADC linker used in FDA-approved brentuximab vedotin.</p>Formula:C28H40N6O7Purezza:98.24%Colore e forma:SolidPeso molecolare:572.65NS3861
CAS:NS3861 is a selective agonist for α3β4/α4β2 nAChRs, preferring β-subunits, with no effect on α4-based receptors.Formula:C12H14BrNSPurezza:99.853%Colore e forma:SolidPeso molecolare:284.22Dinotefuran
CAS:Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.Formula:C7H14N4O3Purezza:99.89%Colore e forma:White Crystalline PowderPeso molecolare:202.21Thiacloprid
CAS:Thiacloprid: insecticide targeting insect nAChRs, IC50 - Drosophila: 2.7 nM, Mouse α4β2 nAChRs: 860 nM.Formula:C10H9ClN4SPurezza:98.66% - 99.95%Colore e forma:Yellowish Crystalline PowderPeso molecolare:252.72Ipratropium Bromide
CAS:Ipratropium Bromide (Sch 1000) is an antagonist of muscarinic receptors and is used in COPD and asthma studies.Formula:C20H30BrNO3Purezza:99.92%Colore e forma:SolidPeso molecolare:412.37Encenicline
CAS:Encenicline (EVP-6124), a selective α7 nAChRs agonist, targets cognitive impairment in schizophrenia and Alzheimer's.Formula:C16H17ClN2OSPurezza:99.20%Colore e forma:SolidPeso molecolare:320.84Oxyphencyclimine Hydrochloride
CAS:<p>Oxyphencyclimine Hydrochloride (Ulcociclinina) is a synthetic tertiary amine and antimuscarinic agent with antispasmodic and antisecretory activities.</p>Formula:C20H29ClN2O3Purezza:99.55%Colore e forma:SolidPeso molecolare:380.91Oxyphenonium bromide
CAS:<p>Oxyphenonium bromide is an anticholinergic used to study and treat ulcers and relieve visceral spasms.</p>Formula:C21H34BrNO3Purezza:98.96%Colore e forma:SolidPeso molecolare:428.404Propiverine
CAS:Propiverine reduces muscle spasms by limiting calcium influx, targeting bladder smooth muscles, aiding OAB research.Formula:C23H29NO3Colore e forma:SolidPeso molecolare:367.48Cyclopentolate Hydrochloride
CAS:Cyclopentolate Hydrochloride is a muscarinic acetylcholine receptors antagonist with Kis of 1.62, 27.5, and 2.63 nM for M1, M2, and M3 receptors, respectively.Formula:C17H26ClNO3Purezza:99.91%Colore e forma:SolidPeso molecolare:327.85A-867744
CAS:<p>A-867744 is an effective and selective type II positive allosteric modulator of the α7 nAChR (EC50: 1.0 μM).</p>Formula:C20H19ClN2O3SPurezza:95.66%Colore e forma:SolidPeso molecolare:402.89VU10010
CAS:<p>VU10010 (VU 10010) is allosteric potentiator of M4 acetylcholine receptors.</p>Formula:C17H16ClN3OSPurezza:99.36%Colore e forma:SolidPeso molecolare:345.85Pirmenol
CAS:Pirmenol is a new antiarrhythmic drugFormula:C22H30N2OPurezza:97.24%Colore e forma:SolidPeso molecolare:338.49Mivacurium dichloride
CAS:Mivacurium dichloride: non-depolarizing, quick-acting muscle relaxant for minor surgeries and tracheal intubation.Formula:C58H80Cl2N2O14Purezza:99.2% - 99.48%Colore e forma:Off-White SolidPeso molecolare:1100.17SQ22536
CAS:SQ22536, a tetrahydrofuryl adenosine analogue, inhibits adenylate cyclase in catfish and rat hepatocytes non-competitively.Formula:C9H11N5OPurezza:99.18%Colore e forma:Off-White SolidPeso molecolare:205.22Coluracetam
CAS:Coluracetam (MKC-231)(MKC-231) is a Choline Uptake Enhancer.Formula:C19H23N3O3Purezza:99.96%Colore e forma:SolidPeso molecolare:341.4Mecamylamine
CAS:<p>Mecamylamine: oral, noncompetitive nAChR blocker, crosses blood-brain barrier, for neuropsychiatric and hypertension research.</p>Formula:C11H21NColore e forma:SolidPeso molecolare:167.29Bestim
CAS:Bestim is an immunomodulatory dipeptide that is synthetic.Formula:C16H19N3O5Purezza:99.76%Colore e forma:SolidPeso molecolare:333.34Aclidinium bromide
CAS:<p>Aclidinium bromide (LAS-W 330) is a synthetic anticholinergic agent that is used as an inhalant for treatment of acute bronchospasm due to chronic bronchitis.</p>Formula:C26H30NO4S2·BrPurezza:99.53% - 99.69%Colore e forma:SolidPeso molecolare:564.55Ilmetropium iodide
CAS:Ilmetropium iodide is a bronchodilator.Formula:C20H30INO3Purezza:98.45%Colore e forma:SolidPeso molecolare:459.36Fesoterodine
CAS:Fesoterodine is an oral mAChR blocker (pKi: 7.3-8.0) for M1-M5, used to treat OAB.Formula:C26H37NO3Purezza:97.1%Colore e forma:SolidPeso molecolare:411.58DMAB-anabaseine dihydrochloride
CAS:<p>DMAB-anabaseine dihydrochloride (N,N-dimethyl-4-[(E)-(6-pyridin-3-yl-3,4-dihydro-2H-pyridin-5-ylidene)methyl]aniline;dihydrochloride) is an α7-containing</p>Formula:C19H23Cl2N3Purezza:99.91%Colore e forma:SolidPeso molecolare:364.31Ethyl (triphenylphosphoranylidene) acetate
CAS:<p>Ethyl (triphenylphosphoranylidene) acetate ((Carbethoxymethylene)triphenylphosphorane) may act as an cholinesterase inhibitor that inhibits AChE and BChE.</p>Formula:C22H21O2PPurezza:97.985%Colore e forma:White Or Slight Yellow PowderPeso molecolare:348.37Brompheniramine
CAS:Brompheniramine, an alkylamine antihistamine, targets H1 receptors (Kd=6.06nM) and has anticholinergic/depressant qualities. Blocks Ca/Na/hERG channels.Formula:C16H19BrN2Colore e forma:SolidPeso molecolare:319.24Solifenacin hydrochloride
CAS:Solifenacin Hcl is a muscarinic receptor antagonist.Formula:C23H27ClN2O2Purezza:98%Colore e forma:SolidPeso molecolare:398.93Benzetimide hydrochloride
CAS:Benzetimide hydrochloride (R4929) is an antagonist of muscarinic acetylcholine receptor.treatment neuroleptic-induced parkinsonism.Formula:C23H27ClN2O2Purezza:99.32%Colore e forma:Off-White PowderPeso molecolare:398.93LY2119620
CAS:LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.Formula:C19H24ClN5O3SPurezza:99.7%Colore e forma:SolidPeso molecolare:437.94α-Conotoxin MII acetate
α-Conotoxin MII acetate is a 16-amino acid peptide from the venom of the marine snail Conus magus.Formula:C69H107N23O24S4Purezza:94.82% - 97.79%Colore e forma:SolidPeso molecolare:1770.99Anisotropine Methylbromide
CAS:Anisotropine Methylbromide is an anticholinergic agent and has been used for relief of gastrointestinal spasm and for the suppression of gastric acid secretion.Formula:C17H32BrNO2Purezza:99.73%Colore e forma:Crystals From Acetone SolidPeso molecolare:362.35ST034307
CAS:ST034307 is an effective and selective inhibitor of adenylyl cyclase 1 (IC50: 2.3 μM).Formula:C10H4Cl4O2Purezza:99.28%Colore e forma:SolidPeso molecolare:297.95Adiphenine
CAS:Adiphenine is an inhibitor of nicotinic receptors.Formula:C20H25NO2Colore e forma:SolidPeso molecolare:311.42Cyclodrine hydrochloride
CAS:Cyclodrine hydrochloride is a dual cholinergic muscarinic receptor (mAChR) and nicotinic receptor (nAChR) antagonist that can be used in the study ofFormula:C19H30ClNO3Purezza:98.59%Colore e forma:SolidPeso molecolare:355.9PHA 568487
CAS:PHA 568487: α-7 nAChR agonist, rapid brain uptake, lessens oxidative stress & neuroinflammation.Formula:C20H24N2O7Colore e forma:SolidPeso molecolare:404.419PHA 568487 free base
CAS:<p>PHA 568487 free base, an α7 nicotinic receptor agonist, designed to reduce bioactivation and improve in vivo tolerability.</p>Formula:C16H20N2O3Purezza:99.74%Colore e forma:SolidPeso molecolare:288.34Mc-Val-Ala-PAB
CAS:<p>Mc-Val-Ala-PAB, an effective linker, is utilized in antibody-drug-conjugate (ADC).</p>Formula:C25H34N4O6Purezza:98.34% - 99.24%Colore e forma:SolidPeso molecolare:486.56Oxyphencyclimine
CAS:Oxyphencyclimine is a muscarinic receptor antagonist (MRA) anticholinergic drug used to treat peptic ulcers.Formula:C20H28N2O3Colore e forma:SolidPeso molecolare:344.45suvn-911
CAS:suvn-911 is a potent and selective antagonist of neuronal nicotinic acetylcholine α4β2 receptor (Ki = 1.5 nM) with antidepressant activity.Formula:C11H14Cl2N2OPurezza:98.88%Colore e forma:SolidPeso molecolare:261.15Propantheline
CAS:Propantheline: oral muscarinic receptor blocker for smooth muscle issues, hyperhidrosis, and bladder control.Formula:C23H30NO3Colore e forma:SolidPeso molecolare:368.49Piperidolate hydrochloride
CAS:Piperidolate hydrochloride, an antimuscarinic, reduces acetylcholine-induced intestinal spasms in rats and dogs.Formula:C21H26ClNO2Purezza:99.5%Colore e forma:SolidPeso molecolare:359.89TQS
CAS:TQS (4-Naphthalen-1-yl-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-8-sulfonamide) is a positive allosteric modulator of α7 nACh receptors.Formula:C22H20N2O2SPurezza:98.56%Colore e forma:SolidPeso molecolare:376.47KH7
CAS:KH7 is a soluble inhibitor of adenylyl cyclase (sAC)-specific.Formula:C17H15BrN4O2SPurezza:98.43%Colore e forma:SolidPeso molecolare:419.3Succinylcholine Chloride Dihydrate
CAS:<p>Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.</p>Formula:C14H30N2O4·2Cl·2H2OPurezza:99.87%Colore e forma:White SolidPeso molecolare:397.34Nitenpyram
CAS:<p>Nitenpyram (Capstar) is a nicotinic acetylcholine receptor (AchR) agonist, used as veterinary medicine to treat parasites of livestock and pets.</p>Formula:C11H15ClN4O2Purezza:99.03%Colore e forma:Light-Yellow CrystalPeso molecolare:270.72Procyclidine hydrochloride
CAS:<p>Procyclidine hydrochloride ((±)-Procyclidine hydrochlorid) is a potent anticholinergic agent and also have NMDA antagonist properties.</p>Formula:C19H30ClNOPurezza:99.24% - 99.88%Colore e forma:Crystals From Petroleum Ether White PowderPeso molecolare:323.9NS9283
CAS:<p>NS9283, a positive allosteric modulator selective for the α4β2 form, reduces ethanol consumption.</p>Formula:C14H8N4OPurezza:99.12%Colore e forma:SolidPeso molecolare:248.24Sofpironium bromide
CAS:<p>Sofpironium bromide (BBI4000) belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.</p>Formula:C22H32BrNO5Purezza:98.85%Colore e forma:SolidPeso molecolare:470.4Batefenterol
CAS:<p>Batefenterol (GSK961081) is a muscarinic antagonist and β2-agonist with high affinity (Ki: 1.4/1.3/3.7 nM).</p>Formula:C40H42ClN5O7Purezza:97.94% - 98.4%Colore e forma:SolidPeso molecolare:740.24Nanofin
CAS:<p>Nanofin (Lupetidine) is a neuropathic blocker, with antihypertensive effect.</p>Formula:C7H15NPurezza:97.38% - 99.818%Colore e forma:Clear Colorless To Slightly Yellow LiquidPeso molecolare:113.2MC-Val-Cit-PABC-PNP
CAS:MC-Val-Cit-PABC-PNP, also known as Mc-Val-Cit-PABC-PNP, is a cathepsin cleavable ADC peptide linker.Formula:C35H43N7O11Purezza:97.2% - 98.055%Colore e forma:SolidPeso molecolare:737.76Blarcamesine
CAS:<p>Blarcamesine (AVex-73) is a muscarinic M1 agonist potentially for the treatment of Alzheimer's disease.</p>Formula:C19H23NOPurezza:99.87%Colore e forma:SolidPeso molecolare:281.39ML380
CAS:<p>ML380 is a highly potent and the first CNS penetrant M5 positive allosteric modulator (PAM).</p>Formula:C23H25F3N4O3SPurezza:99.69%Colore e forma:SolidPeso molecolare:494.53PNU-120596
CAS:<p>PNU-120596 (NSC-216666) is a positive allosteric modulator of α7 nAChR with EC50 of 216 nM.</p>Formula:C13H14ClN3O4Purezza:99.82%Colore e forma:SolidPeso molecolare:311.72NS 1738
CAS:NS 1738 (NSC-213859) is a positive allosteric modulator of the α7-containing neuronal nicotinic acetylcholine receptors (nAChRs)Formula:C14H9Cl2F3N2O2Purezza:99.11%Colore e forma:SolidPeso molecolare:365.13Nitrocaramiphen hydrochloride
CAS:Nitrocaramiphen hydrochloride is a selective M1 muscarinic antagonist and inhibits binding to sigma sites in brain.Formula:C18H27ClN2O4Purezza:99.74%Colore e forma:SolidPeso molecolare:370.87A 582941 HCl (848591-90-2(free base))
<p>A-582941 is a alpha7 neuronal nicotinic receptor agonist with broad spectrum cognition-enhancing properties</p>Formula:C17H21ClN4Purezza:99.83%Colore e forma:SolidPeso molecolare:316.83Solifenacin
CAS:Solifenacin (YM905 free base) (YM905 free base) is a novel muscarinic receptor antagonist, its pKis for M1, M2 and M3 receptors is of 7.6, 6.9 and 8.0,Formula:C23H26N2O2Purezza:99.87%Colore e forma:SolidPeso molecolare:362.46Syn-Ake acetate
CAS:Syn-Ake acetate (Dipeptide diaminobutyroyl benzylamide) is a muscarinic acetylcholine receptor antagonist.Formula:C19H29N5O3·2(C2H4O2)Purezza:99.60%Colore e forma:SolidPeso molecolare:495.58Velufenacin
CAS:Velufenacin is an antagonist of muscarinic receptor[1].Formula:C19H20ClFN2O2Purezza:99.65%Colore e forma:SolidPeso molecolare:362.83Mepenzolate Bromide
CAS:<p>Mepenzolate Bromide (Colibantil) is a muscarinic antagonist used to treat gastrointestinal conditions.</p>Formula:C21H26BrNO3Purezza:95.73% - 99.21%Colore e forma:SolidPeso molecolare:420.34AF-710B
CAS:<p>AF710B is an enantiomer of AF710. AF-710B is also a sigma and M1 muscarinic receptors agonist.</p>Formula:C20H27N3OSPurezza:98.62% - 99.89%Colore e forma:SolidPeso molecolare:357.51Pentoxyverine
CAS:Pentoxyverine (Carbetapentan) is an orally available cough suppressant, an antagonist of muscarinic receptor M1 and an agonist of the σ1 receptor.Formula:C20H31NO3Purezza:97.11%Colore e forma:SolidPeso molecolare:333.47Xanomeline tartrate
CAS:Xanomeline tartrate (LY 246708 tartrate) 是 M1和 M4 mAChR 激动剂,具有抗精神病样活性,可改善认知,可用于研究精神分裂症和阿尔茨海默病。Formula:C18H29N3O7SPurezza:99.19% - 99.99%Colore e forma:SolidPeso molecolare:431.5Pipecuronium bromide
CAS:Pipecuronium bromide (RGH-1106) is an nAChR antagonist that also acts as a non-depolarising steroidal neuromuscular blocker that causes muscle relaxation.Formula:C35H62Br2N4O4Purezza:>99.99%Colore e forma:PowderPeso molecolare:762.7Monepantel
CAS:Monepantel (AAD1566) is an organic anthelmintic and an antagonist of nAChRs from roundworms and esophageostomy.Formula:C20H13F6N3O2SPurezza:99.83%Colore e forma:White PowderPeso molecolare:473.39Varenicline
CAS:Varenicline (CP 526555) is a selective partial agonist of the α4β2 nAChR and a full agonist of the α3β4 nAChR and α7 nAChR.Formula:C13H13N3Purezza:99.76%Colore e forma:SolidPeso molecolare:211.26Atropine hydrobromide
CAS:Atropine hydrobromide is a biochemical.Formula:C17H24BrNO3Colore e forma:SolidPeso molecolare:370.28Pyrantel
CAS:Pyrantel: Nicotinic agonist; causes spastic paralysis in nematodes by depolarizing block.Formula:C11H14N2SPurezza:98%Colore e forma:Crystals From Methanol Yellowish Crystalline PowderPeso molecolare:206.31Anatabine dicitrate
Anatabine dicitrate is a tobacco alkaloid that can cross the blood-brain barrier.Formula:C22H28N2O14Purezza:98%Colore e forma:SolidPeso molecolare:544.46Flavoxate
CAS:<p>Flavoxate is an anticholinergic with antimuscarinic effects.</p>Formula:C24H25NO4Colore e forma:SolidPeso molecolare:391.46(±)-Atropine-d3 (N-methyl-d3)
CAS:(±)-Atropine-d3 (N-methyl-d3) is a deuterated compound of (±)-Atropine. (±)-Atropine has a CAS number of 51-55-8. Atropine Sulfate is the sulfate salt of atropine, a naturally-occurring alkaloid isolated from the plant Atropa belladonna. Atropine functions as a sympathetic, competitive antagonist of muscarinic cholinergic receptors, thereby abolishing the effects of parasympathetic stimulation.Formula:C17H20D3NO3Peso molecolare:292.39Diphenidol
CAS:<p>Diphenidol, a muscarinic antagonist, is employed as an antivertigo and antiemetic agent.</p>Formula:C21H27NOColore e forma:Needles From Petroleum Ether SolidPeso molecolare:309.45VU0029767
CAS:<p>VU0029767 is an allosteric enhancer of the M1 muscarinic receptor, capable of modulating the receptor's activity. This compound enhances M1 receptor activity by increasing agonist affinity. However, VU0029767 demonstrates distinct characteristics from other compounds, particularly under varying experimental conditions such as its interaction with mutated M1 receptors and its effects on downstream signaling pathways.</p>Formula:C21H21N3O3Colore e forma:SolidPeso molecolare:363.41Catestatin
CAS:Non-competitive inhibitor of nicotinic receptors; blocks cationic signalling and catecholamine release; stimulates histamine release. IC50 ~200-250nM.Formula:C107H173N37O26SPurezza:98%Colore e forma:SolidPeso molecolare:2425.84N-Biotinyl p-aminophenyl arsenic acid
CAS:N-Biotinyl p-aminophenyl arsenic acid is a bifunctional reagent that binds to streptavidin and disulfide compounds. It diminishes the binding sites of rbungarotoxin on reduced nicotinic receptors with an IC50 ranging from 10-300 nM, thus shielding the receptors from irreversible alkylation by bromoacetylcholine.Formula:C16H22AsN3O4SColore e forma:SolidPeso molecolare:427.35Phenglutarimide hydrochloride
CAS:Phenglutarimide hydrochloride is an anticholinergic. It is used as an antiparkinsonian agent.Formula:C17H25ClN2O2Colore e forma:SolidPeso molecolare:324.85Aprofene
CAS:<p>Aprofene blocks acetylcholine receptors, used for peptic ulcers, endarteritis, cholecystitis, and colitis.</p>Formula:C21H27NO2Colore e forma:SolidPeso molecolare:325.44Dianicline dihydrochloride
CAS:Dianicline dihydrochloride is a partial agonist of α4β2 nicotinic acetylcholine receptor. It increases cessation rates in a dose-dependent manner.Formula:C13H16N2OPurezza:98%Colore e forma:SolidPeso molecolare:216.28Biperiden lactate
CAS:<p>Biperiden lactate is a biochemical.</p>Formula:C24H35NO4Colore e forma:SolidPeso molecolare:401.54AN317
CAS:AN317 is a selective agonist for the nicotinic acetylcholine receptor (nAChR) containing α6β2, with dissociation constants (Ki) of 6.2 nM and 4.1 nM for the α6/α3β2β3 and α4β2 receptor subtypes, respectively. It induces dopamine release in rat striatal synaptosomes, enhances the activity of dopaminergic neurons in the substantia nigra, and exhibits protective effects against the dopaminergic neurotoxin MPP+ in rat neurons. AN317 also demonstrates favorable pharmacokinetic properties in rats and permeability across the blood-brain barrier (BB).Formula:C13H19N3Colore e forma:SolidPeso molecolare:217.31Azacyclonol hydrochloride
CAS:Azacyclonol hydrochloride can be used in the treatment of chronic schizophrenia.Formula:C18H22ClNOColore e forma:Off White Crystalline PowderPeso molecolare:303.83Oxantel
CAS:<p>Oxantel is a fumarate reductase inhibitor with anthelmintic activity.</p>Formula:C13H16N2OPurezza:98%Colore e forma:SolidPeso molecolare:216.28Sulindac sulfide
CAS:Sulindac sulfide: NSAID targeting COX-1, inhibits Ras-Raf-1 and gamma-secretase (IC50: 20.2 μM), active sulinic acid metabolite.Formula:C20H17FO2SPurezza:99.35%Colore e forma:SolidPeso molecolare:340.41BTM-1086
CAS:BTM-1086 is a potent gastric secretory inhibitor and an anti-ulcer agent.Formula:C21H25N3OSPurezza:98%Colore e forma:SolidPeso molecolare:367.51CP-601932
CAS:CP-601932 (free base) is a selective base α( 4) β( 2) Nicotinic acetylcholine receptor agonist.Formula:C12H12F3NColore e forma:SolidPeso molecolare:227.23Eucatropine
CAS:Eucatropine, an anticholinergic agent, acts as a potent inhibitor of the muscarinic acetylcholine receptor (mAChR) with an IC 50 value of 0.583 μM.Formula:C17H25NO3Colore e forma:SolidPeso molecolare:291.39Thiochrome
CAS:Thiochrome is a selective enhancer of M4 muscarinic receptor of acetylcholine (ACh) affinity.Formula:C12H14N4OSPurezza:98%Colore e forma:SolidPeso molecolare:262.33GAT107
CAS:GAT107, a strong α7 nicotinic receptor modulator, aids inflammation and neuropathic pain in mice.Formula:C18H17BrN2O2SPurezza:99.33%Colore e forma:SolidPeso molecolare:405.31VU0090157
CAS:VU0090157, a novel allosteric potentiators of M1 muscarinic receptor, may provide novel treatments for schizophrenia and Alzheimer's disease.Formula:C19H21N3O7Purezza:98%Colore e forma:SolidPeso molecolare:403.39S-(+)-Mecamylamine hydrochloride
CAS:Dexmecamylamine( TC-5214, NIH-11008) is used as a nicotinic channel modulator with antidepressant activity.Formula:C11H22ClNColore e forma:SolidPeso molecolare:203.75T761-0184
CAS:T761-0184 is a potent antagonist of α7 nicotinic receptor (nAChR) [1].Formula:C16H20FN3OColore e forma:SolidPeso molecolare:289.35Revatropate
CAS:Revatropate, a selective muscarinic antagonist, is an antimuscarinic drug.Formula:C19H27NO4SColore e forma:SolidPeso molecolare:365.49Rispenzepine
CAS:Rispenzepine, a novel mAChRs M1/M3 antagonist, treats immune, infections, and respiratory issues.Formula:C19H20N4O2Purezza:98%Colore e forma:SolidPeso molecolare:336.39SCH 57790
CAS:SCH 57790: selective muscarinic M2 blocker, boosts acetylcholine & cognition, may treat Alzheimer's.Formula:C25H31N3O2SPurezza:99.12% - 99.69%Colore e forma:SolidPeso molecolare:437.6Tarafenacin
CAS:Tarafenacin is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over the M2 receptor.Formula:C21H20F4N2O2Purezza:98%Colore e forma:SolidPeso molecolare:408.39Milameline
CAS:Milameline is a muscarinic receptor agonist that improves cognition.Formula:C8H14N2OColore e forma:SolidPeso molecolare:154.21Biricodar dicitrate
CAS:Biricodar dicitrate (VX-710) is a potent MDR inhibitor with no anticancer activity and can be used to study prostate cancer.Formula:C46H57N3O21Purezza:97.78% - 99.78%Colore e forma:SolidPeso molecolare:987.95Sofiniclin
CAS:Sofiniclin (ABT 894) is an agonist of nicotinic acetylcholine receptor (nAChR). It is used for the research for attention-deficit/hyperactivity disorder (ADHD).Formula:C10H11Cl2N3Purezza:98%Colore e forma:SolidPeso molecolare:244.12SR 16584
CAS:α3β4 nAChR antagonistFormula:C17H22N2OPurezza:99.84%Colore e forma:SolidPeso molecolare:270.37Bibn 99
CAS:<p>Bibn 99, a lipophilic and selective muscarinic M2 receptor antagonist, has applications in cognitive performance and Alzheimer's Disease.</p>Formula:C31H42ClN5O3Colore e forma:SolidPeso molecolare:568.15VU 6008667
CAS:VU 6008667 is a selective negative allosteric M5 NAM modulator (IC50s: 1.2 μM and 1.6 μM for human M5 and rat M5, respectively).Formula:C24H17ClF2N2O2Purezza:98%Colore e forma:SolidPeso molecolare:438.85Rivanicline
CAS:Rivanicline is a selective α4β2 nicotinic receptor agonist (Ki=26 nM), with >1,000x less affinity for α7 receptors.Formula:C10H14N2Purezza:98%Colore e forma:SolidPeso molecolare:162.23Rapacuronium bromide
CAS:Rapacuronium bromide is an allosteric muscarinic acetylcholine receptor (mAChR) modulator.Formula:C37H61BrN2O4Purezza:98%Colore e forma:SolidPeso molecolare:677.8ML375
CAS:ML375 is a potent, selective and CNS penetrant M5 negative allosteric modulator (NAM).Formula:C23H15ClF2N2O2Colore e forma:SolidPeso molecolare:424.83Sch412348
CAS:Sch412348: potent A2A receptor antagonist, Ki=0.6 nM, >1000-fold selectivity vs. other adenosine receptors.Formula:C22H21F2N9OPurezza:98%Colore e forma:SolidPeso molecolare:465.46CP-601927
CAS:CP-601927 is a nicotinic acetylcholine receptor (NACHR) agonist with permeability, high affinity, and selectivity.Formula:C12H12F3NColore e forma:SolidPeso molecolare:227.23Arecaidine propargyl ester tosylate
CAS:Arecaidine propargyl ester tosylate is a muscarinic receptor agonist.Formula:C17H21NO5SPurezza:98%Colore e forma:SolidPeso molecolare:351.42VMY-2-95
CAS:VMY-2-95 is an α4β2 nicotinic acetylcholine receptors (nAChRs) selective desensitizer.Formula:C17H16N2OColore e forma:SolidPeso molecolare:264.32RJR 2429 dihydrochloride
CAS:nAChR agonist that displays selectivity for α4β2Formula:C12H18Cl2N2Purezza:98%Colore e forma:SolidPeso molecolare:261.19J 104129 fumarate
CAS:M3 muscarinic receptor antagonistFormula:C24H36N2O2Purezza:98%Colore e forma:SolidPeso molecolare:384.55Alvameline maleate
CAS:Alvameline maleate is used as a Partial M1 Agonist and M2/M3 Antagonist.Formula:C13H19N5O4Colore e forma:SolidPeso molecolare:309.32Vinconate
CAS:Vinconate is an indolonaphthyridine derivative and can stimulate the muscarinic acetylcholine receptor.Formula:C18H20N2O2Purezza:98%Colore e forma:SolidPeso molecolare:296.36AT-1001
CAS:AT-1001 is an α3β4 nAChR partial agonist reducing nicotine relapse and withdrawal with negligible impact on food response and dopamine release.Formula:C15H21BrN2Colore e forma:SolidPeso molecolare:309.24PD-102807
CAS:PD-102807 is a selective and competitive M4 muscarinic receptor antagonist for Parkinson's disease research, inhibit airway smooth muscle (ASM) contraction.Formula:C23H24N2O4Purezza:98.90%Colore e forma:SolidPeso molecolare:392.45Rivanicline oxalate
CAS:Rivanicline oxalate is an agonist of neuronal nicotinic receptor, showing high selectivity for the α4β2 subtype (Ki=26 nM).Formula:C12H16N2O4Purezza:98%Colore e forma:SolidPeso molecolare:252.27Bradanicline HCl
CAS:Bradanicline(TC-5619) is the agonist of Alpha-7 Nicotinic Receptor.Formula:C22H24ClN3O2Colore e forma:SolidPeso molecolare:397.9S 24795
CAS:S 24795 (Catestatin acetate(142211-96-9 free base)) is an α7 nAChR partial agonist.Formula:C14H13BrINOPurezza:99.934%Colore e forma:SolidPeso molecolare:418.07DREADD agonist 21 dihydrochloride
CAS:DREADD agonist 21 dihydrochloride is a potent human muscarinic acetylcholine M3 receptors ( hM3Dq ) agonist with EC 50 of 1.7 nM [1].Formula:C17H20Cl2N4Purezza:98%Colore e forma:SolidPeso molecolare:351.27BPIPP
CAS:guanylyl cyclase (GC) and adenylyl cyclase (AC) inhibitorFormula:C22H16BrN3O3Purezza:98%Colore e forma:SolidPeso molecolare:450.28Procyclidine
CAS:Procyclidine is an anticholinergic, muscarinic and NMDA antagonist used in Parkinson's and psychiatric disorder studies.Formula:C19H29NOColore e forma:SolidPeso molecolare:287.44Oxybutynin R-isomer HCl
CAS:Aroxybutynin, R-isomer of oxybutynin, is a muscarinic antagonist with antispasmodic effects on bladder muscle, weaker than atropine.Formula:C22H32ClNO3Colore e forma:SolidPeso molecolare:393.95VU0455691
CAS:VU0455691 is a selective M1 Muscarinic Receptor Allosteric Modulators.Formula:C24H25N5O3SPurezza:98%Colore e forma:SolidPeso molecolare:463.55Ambutonium bromide
CAS:Ambutonium bromide is an antagonist of acetylcholine.Formula:C20H27BrN2OPurezza:98%Colore e forma:SolidPeso molecolare:391.35(±)-Muscarine chloride
CAS:(±)-Muscarine chloride is the racemate of Muscarine chloride. Muscarine is a prototypical agonist for the muscarinic acetylcholine receptor [1] [2].Formula:C9H20ClNO2Colore e forma:SolidPeso molecolare:209.71Methapyrilene
CAS:Methapyrilene is a histamine H1 antagonist with sedative action.Formula:C14H19N3SColore e forma:Liquid Physical Description Clear Colorless Liquid (Ntp 1992)Peso molecolare:261.39Milameline hydrochloride
CAS:Milameline hydrochloride is a Muscarinic receptor agonist.Formula:C8H15ClN2OPurezza:98%Colore e forma:SolidPeso molecolare:190.67Cycrimine
CAS:Cycrimine: oral M1 mAChR blocker, lowers acetylcholine, antispasmodic, for Parkinson's and mental disorder studies.Formula:C19H29NOColore e forma:SolidPeso molecolare:287.44Parapenzolate bromide
CAS:Parapenzolate bromide is an orally active mAChR antagonist. parapenzolate bromide is an anticholinergic and antitussive agent.Formula:C21H26BrNO3Colore e forma:SolidPeso molecolare:420.347

