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Src

Src

Gli inibitori di Src sono composti che prendono di mira le chinasi della famiglia Src, coinvolte in vari processi cellulari, tra cui crescita, differenziazione e angiogenesi. Le chinasi Src svolgono un ruolo critico nelle vie di segnalazione che promuovono la formazione di nuovi vasi sanguigni nei tumori. Inibendo Src, è possibile interrompere queste vie, riducendo così l'angiogenesi e la crescita tumorale. Gli inibitori di Src sono ampiamente utilizzati nella ricerca sul cancro e nello sviluppo terapeutico. Presso CymitQuimica, offriamo una selezione completa di inibitori di Src di alta qualità per supportare la tua ricerca in oncologia, segnalazione cellulare e angiogenesi.

Trovati 79 prodotti di "Src"

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  • Tetramethylcurcumin

    CAS:
    <p>Tetramethylcurcumin is a novel curcumin analog, is an effective inhibitors of STAT3 phosphorylation, DNA binding activity, and transactivation in vitro.it also</p>
    Formula:C25H28O6
    Purezza:97.69% - 99.94%
    Colore e forma:Solid
    Peso molecolare:424.49
  • Bafetinib

    CAS:
    <p>Bafetinib (INNO-406): Dual Bcr-Abl/Lyn inhibitor; IC50: 5.8/19 nM; ineffective against T315I mutant, less on c-Kit/PDGFR.</p>
    Formula:C30H31F3N8O
    Purezza:94.16% - 99.68%
    Colore e forma:Solid
    Peso molecolare:576.62
  • 7-Hydroxy-4H-chromen-4-one

    CAS:
    <p>7-Hydroxy-4H-chromen-4-one (7-hydroxy-4-benzopyrone) is a Src kinase inhibitor (IC50 of &lt;300 μM).</p>
    Formula:C9H6O3
    Purezza:97.65%
    Colore e forma:Solid
    Peso molecolare:162.14
  • XL228

    CAS:
    <p>XL228 is an inhibitor of multi-targeted tyrosine kinase (IC50s: 5, 3.1, 1.6, 6.1, 2 nM for Bcr-Abl, Aurora A, IGF-1R, Src, and Lyn, respectively).</p>
    Formula:C22H31N9O
    Purezza:99.07%
    Colore e forma:Solid
    Peso molecolare:437.54
  • Pelitinib

    CAS:
    <p>Pelitinib (EKB-569) (EKB-569) is an effective irreversible EGFR inhibitor (IC50: 38.5 nM).</p>
    Formula:C24H23ClFN5O2
    Purezza:98.37% - 99.84%
    Colore e forma:Off-White Solid
    Peso molecolare:467.92
  • Tirbanibulin

    CAS:
    <p>Tirbanibulin (KX2-391) is a highly selective Src kinase inhibitor that has demonstrated efficacy in pre-Clinicalal animal models of a variety of cancers.</p>
    Formula:C26H29N3O3
    Purezza:99.43% - 99.67%
    Colore e forma:Solid
    Peso molecolare:431.53
  • PD-089828

    CAS:
    <p>PD 089828 inhibits FGFR1, PDGFRβ, EGFR (IC50s: 0.15-5.47 μM), and c-Src (IC50: 0.18 μM).</p>
    Formula:C18H18Cl2N6O
    Purezza:97.39%
    Colore e forma:Solid
    Peso molecolare:405.28
  • PD173955

    CAS:
    <p>PD173955 is src family-selective tyrosine kinase inhibitor with IC50 of ~22 nM for Src, Yes and Abl kinase; less potent for FGFRα and no activity on InsR and</p>
    Formula:C21H16Cl2N4OS
    Purezza:98.52% - 98.99%
    Colore e forma:Solid
    Peso molecolare:443.35
  • Spebrutinib

    CAS:
    <p>Spebrutinib (LMK-435) is an orally bioavailable, selective inhibitor of Bruton's agammaglobulinemia tyrosine kinase (BTK), with potential antineoplastic</p>
    Formula:C22H22FN5O3
    Purezza:97.02% - >99.99%
    Colore e forma:Solid
    Peso molecolare:423.44
  • OXSI-2

    CAS:
    <p>OXSI-2 (Syk Inhibitor) is an inhibitor of Syk with an EC50 of 313 nM and an IC50 of 14 nM.</p>
    Formula:C18H15N3O3S
    Purezza:98%
    Colore e forma:Dark Orange Solid
    Peso molecolare:353.39
  • TC-S 7003

    CAS:
    TC-S 7003 (Lck Inhibitor) is a Lck inhibitor with anti-inflammatory activity that inhibits T-cell proliferation and can be used to study arthritis.
    Formula:C31H30N8O
    Purezza:99.74%
    Colore e forma:Solid
    Peso molecolare:530.62
  • A 419259 trihydrochloride

    CAS:
    A 419259 trihydrochloride (RK 20449 trihydrochloride) is an Src family kinases inhibitor (IC50s: 9 nM, 3 nM and 3 nM for Src, Lck and Lyn).
    Formula:C29H37Cl3N6O
    Purezza:99.75% - 99.96%
    Colore e forma:Solid
    Peso molecolare:592
  • BT424

    CAS:
    BT424, a specific HCK inhibitor, modulates macrophage activation and autophagy in vitro, and mitigates inflammation and renal fibrosis in the UUO model [1].
    Formula:C22H15BCl2N2O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:421.08
  • TG 100572 Hydrochloride

    CAS:
    <p>TG 100572 Hydrochloride is a inhibitor of multi-targeted kinase which inhibits receptor tyrosine kinases and Src kinases(IC50s of 2, 7, 2, 16, 13, 5, 0.5, 6, 0.</p>
    Formula:C26H27Cl2N5O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:512.43
  • TL02-59

    CAS:
    <p>TL02-59: Fgr inhibitor (IC50=0.03nM), also targets Lyn (0.1nM), Hck (160nM), halts acute myelogenous leukemia growth.</p>
    Formula:C32H34F3N5O4
    Purezza:98.77%
    Colore e forma:Solid
    Peso molecolare:609.64
  • KB SRC 4

    CAS:
    <p>KB SRC 4 is a selective and potent c-Src inhibitor with antitumour activity that inhibits the growth of cancer cells.CAS 번호13460-73-83-4</p>
    Formula:C32H23ClN8
    Purezza:98.83% - 99.34%
    Colore e forma:Solid
    Peso molecolare:555.03
  • CH6953755

    CAS:
    <p>CH6953755: oral YES1 kinase inhibitor, IC50 1.8 nM, potent, selective, anticancer, halts cell proliferation.</p>
    Formula:C26H22F2N6O4S
    Purezza:98.03%
    Colore e forma:Solid
    Peso molecolare:552.55
  • Src Inhibitor 3

    CAS:
    <p>Src Inhibitor 3 blocks c-Src kinase (IC50 &lt;3 nM CSK HTRF, &lt;4 nM Caliper), boosting T cell growth from receptor signals.</p>
    Formula:C34H32ClFN8O4
    Purezza:98.35%
    Colore e forma:Solid
    Peso molecolare:671.12
  • CGP062464

    CAS:
    <p>CGP062464 is an inhibitor of the tyrosine kinase c-Src, with an IC50 of less than 50 nM. It is utilized in research related to osteoporosis and tumor-induced hypercalcemia.</p>
    Formula:C18H14N4
    Colore e forma:Solid
    Peso molecolare:286.331