Recettore dell'istamina
I recettori dell'istamina sono GPCR che mediano gli effetti dell'istamina, un'ammina biogena coinvolta nelle risposte immunitarie, nella secrezione acida gastrica e nella neurotrasmissione. Esistono quattro sottotipi di recettori dell'istamina (H1, H2, H3 e H4), ognuno dei quali svolge ruoli distinti nelle reazioni allergiche, nella funzione gastrica e nell'attività del sistema nervoso centrale. Gli antagonisti dei recettori dell'istamina sono ampiamente utilizzati nel trattamento delle allergie, delle ulcere peptiche e della cinetosi. Presso CymitQuimica, offriamo una selezione completa di modulatori dei recettori dell'istamina di alta qualità per supportare la tua ricerca in immunologia, gastroenterologia e neurofarmacologia.
Trovati 382 prodotti di "Recettore dell'istamina"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Dimenhydrinate
CAS:Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.Formula:C24H28ClN5O3Purezza:99.57% - 99.77%Colore e forma:Crystals Physical Description Crystalline White Powder (Ntp 1992)Peso molecolare:469.96Chloropyramine hydrochloride
CAS:Chloropyramine hydrochloride (Alergosan) is a histamine receptor H1 antagonist.Formula:C16H20ClN3·HClPurezza:99.45% - 99.8%Colore e forma:SolidPeso molecolare:326.26Lafutidine
CAS:Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.Formula:C22H29N3O4SPurezza:98.55%Colore e forma:Yellowish White Crystalline PowderPeso molecolare:431.55Levodropropizine
CAS:Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.Formula:C13H20N2O2Purezza:99.87% - 99.93%Colore e forma:White Or Off White Crystalline PowderPeso molecolare:236.31Fexofenadine hydrochloride
CAS:Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor antagonist, withFormula:C32H40ClNO4Purezza:>99.99%Colore e forma:White Crystalline PowderPeso molecolare:538.12Fenspiride hydrochloride
CAS:Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.Formula:C15H20N2O2·HClPurezza:99.64% - 99.92%Colore e forma:SolidPeso molecolare:296.79Benztropine mesylate
CAS:<p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>Formula:C21H25NO·CH4SO3Purezza:98.41% - 99.96%Colore e forma:White Crystalline Powder; Odourless Or Almost OdourlessPeso molecolare:403.53Traxanox
CAS:Traxanox: oral diuretic, boosts phagocytosis in mice/rats, reverses antibody production inhibition in BALB/c mice.Formula:C13H6ClN5O2Purezza:98.37%Colore e forma:SolidPeso molecolare:299.67Amodiaquine dihydrochloride dihydrate
CAS:<p>Amodiaquine dihydrochloride dihydrate (Amodiaquin hydrochloride) is an orally active 4-aminoquinoline derivative with antimalarial and anti-inflammatory effects</p>Formula:C20H28Cl3N3O3Purezza:99.97%Colore e forma:SolidPeso molecolare:464.82Antazoline hydrochloride
CAS:Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenousFormula:C17H19N3·HClPurezza:98% - 99.53%Colore e forma:White Or Almost White Crystalline PowderPeso molecolare:301.82Brompheniramine maleate
CAS:Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.Formula:C16H19BrN2·C4H4O4Purezza:99.80%Colore e forma:Crystal PowderPeso molecolare:435.31Triprolidine hydrochloride monohydrate
CAS:Triprolidine hydrochloride monohydrate is a histamine H1 antagonist used in allergic rhinitis, asthma.Formula:C19H25ClN2OPurezza:99.68% - 99.81%Colore e forma:White Crystalline PowderPeso molecolare:332.87Mepyramine maleate
CAS:Mepyramine maleate is a mild hypnotic, local anesthetic, and H1 histamine antagonist for allergies and colds.Formula:C21H27N3O5Purezza:99.51% - 99.7%Colore e forma:White Crystalline PowderPeso molecolare:401.47Astemizole
CAS:<p>Astemizole (Laridal) is a long-acting antihistamine for allergies like rhinitis and asthma, with fewer anticholinergic effects.</p>Formula:C28H31FN4OPurezza:98.24% - 99.67%Colore e forma:White Crystals SolidPeso molecolare:458.57Tripelennamine hydrochloride
CAS:Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.Formula:C16H21N3·HClPurezza:99.54% - 99.81%Colore e forma:White SolidPeso molecolare:291.82Cimetidine
CAS:<p>Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS.</p>Formula:C10H16N6SPurezza:99.82%Colore e forma:Crystals Physical Description White Crystals With A Slight Sulfur-Mercaptan Odor (Ntp 1992)Peso molecolare:252.34Famotidine
CAS:Famotidine, a histamine H2-blocker, curbs gastric acid production, lowering volume and acidity.Formula:C8H15N7O2S3Purezza:98.93% - 99.91%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:337.45Rupatadine Fumarate
CAS:Rupatadine Fumarate (Rinialer) (UR-12592 Fumarate) is a potent dual PAF/H1 antagonist with Ki of 0.55/0.1 uM.Formula:C26H26ClN3·C4H4O4Purezza:99.86%Colore e forma:White Or Almost-White PowderPeso molecolare:532.03Ketotifen fumarate
CAS:Ketotifen fumarate (HC 20511 fumarate) is a cycloheptathiophene blocker of histamine H1 receptors and release of inflammatory mediators.Formula:C23H23NO5SPurezza:99.25% - 99.73%Colore e forma:SolidPeso molecolare:425.50Chlorprothixene hydrochloride
CAS:Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.Formula:C18H18ClNS·HClPurezza:99.76%Colore e forma:White PowderPeso molecolare:352.32Diphenylpyraline hydrochloride
CAS:Diphenylpyraline hydrochloride treats Parkinsonism. It's an antihistamine with anticholinergic properties and inhibits dopamine reuptake.Formula:C19H23NO·HClPurezza:98.72%Colore e forma:SolidPeso molecolare:317.85Azatadine dimaleate
CAS:<p>Azatadine dimaleate (SCH10649) is an inhibitor for histamine（IC50=6.5 nM） and cholinergic（IC50=10 nM）.</p>Formula:C28H30N2O8Purezza:99.7% - >99.99%Colore e forma:PowderPeso molecolare:522.55Dexchlorpheniramine Maleate
CAS:Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active isomer of chlorpheniramine.Formula:C20H23ClN2O4Purezza:99.58%Colore e forma:White Or Almost White Crystalline PowderPeso molecolare:390.86Cetirizine dihydrochloride
CAS:Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.Formula:C21H27Cl3N2O3Purezza:99.4% - 99.97%Colore e forma:SolidPeso molecolare:461.81Cyproheptadine hydrochloride sesquihydrate
CAS:Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.Formula:C21H24ClNOPurezza:99.77% - >99.99%Colore e forma:White To Slightly Yellowish Crystalline SolidPeso molecolare:341.88Perphenazine
CAS:<p>Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.</p>Formula:C21H26ClN3OSPurezza:99.3% - 99.99%Colore e forma:SolidPeso molecolare:403.97Mifentidine
CAS:Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.Formula:C13H16N4Purezza:98.34% - 99.73%Colore e forma:SolidPeso molecolare:228.29Doxylamine succinate
CAS:<p>Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.</p>Formula:C21H28N2O5Purezza:99.61%Colore e forma:5 1 (Ntp 1992)Peso molecolare:388.46Promethazine hydrochloride
CAS:Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.Formula:C17H20N2S·HClPurezza:99.85%Colore e forma:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Peso molecolare:320.88Mebhydrolin napadisylate
CAS:Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergicFormula:C19H20N2C10H8O6S2Purezza:99.35% - 99.96%Colore e forma:White Or Almost White CrystallinePeso molecolare:420.52Mizolastine
CAS:Mizolastine (SL 850324), an antihistamine with IC50 of 47 nM, treats allergies like hay fever and hives.Formula:C24H25FN6OPurezza:98% - 99.75%Colore e forma:SolidPeso molecolare:432.49Terfenadine
CAS:Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.Formula:C32H41NO2Purezza:98.76% - 99.75%Colore e forma:SolidPeso molecolare:471.67Doxepin hydrochloride
CAS:Doxepin hydrochloride, a dibenzoxepin tricyclic, blocks monoamine reuptake and has anticholinergic and antihistaminic effects. Mechanism partly unknown.Formula:C19H22ClNOPurezza:99.65% - 99.91%Colore e forma:White To Off-White PowderPeso molecolare:315.84JNJ-39758979
CAS:<p>JNJ-39758979: selective H4 receptor antagonist, Kis 12.5/5.3/25 nM (human/mouse/monkey), blocks histamine cAMP inhibition (pA2 7.9).</p>Formula:C11H19N5Purezza:98.33% - 99.62%Colore e forma:SolidPeso molecolare:221.3Talastine
CAS:Talastine is an antihistamine compound that can induce an allergic rash.Formula:C19H21N3OPurezza:99.44% - 99.84%Colore e forma:SolidPeso molecolare:307.39Azacyclonol
CAS:Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.Formula:C18H21NOPurezza:99.46%Colore e forma:Solid PowderPeso molecolare:267.37Pheniramine maleate
CAS:Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors.Formula:C16H20N2·C4H4O4Purezza:99.85%Colore e forma:Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°CPeso molecolare:356.42Hydroxyzine Pamoate
CAS:Hydroxyzine Pamoate (Bobsule) is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria and histamine-mediated pruritus.Formula:C44H43ClN2O8Purezza:99.49%Colore e forma:SolidPeso molecolare:763.27Ranitidine Hydrochloride
CAS:Ranitidine Hydrochloride (AH19065) is a competitive and reversible inhibitor of histamine H2-receptor antagonists with antacid activity.Formula:C13H23ClN4O3SPurezza:99.30% - 99.49%Colore e forma:SolidPeso molecolare:350.86Histamine
CAS:Histamine (Ergamine) is an amine derived by the enzymatic decarboxylation of histamine. Histamine is a potent stimulant of gastric secretion of central action. High-Quality, Low-Cost!Formula:C5H9N3Purezza:96.63% - >99.99%Colore e forma:Needles From Chloroform SolidPeso molecolare:111.15Cinnarizine
CAS:Cinnarizine is a piperazine, blocks H1-receptor & Ca-channels, has vasodilating & antiemetic effects, may cause Parkinson-like symptoms.Formula:C26H28N2Purezza:99.94%Colore e forma:SolidPeso molecolare:368.51Meclizine dihydrochloride
CAS:Meclizine dihydrochloride (NSC28728) is a histamine H1 antagonist used in the treatment of motion sickness, vertigo, and nausea during pregnancy and radiationFormula:C25H27ClN2·2HClPurezza:98.05% - 99.79%Colore e forma:White Slightly Yellowish Crystalline PowderPeso molecolare:463.87Levocetirizine
CAS:Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a Histamine H1 Receptor Antagonist.Formula:C21H25ClN2O3Purezza:98% - 99.94%Colore e forma:White PowderPeso molecolare:388.89Carbinoxamine Maleate Salt
CAS:Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.Formula:C20H23ClN2O5Purezza:99.97%Colore e forma:Off-White SolidPeso molecolare:406.86Orphenadrine hydrochloride
CAS:Orphenadrine hydrochloride (Mephenamin) is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.Formula:C18H23NO·HClPurezza:99.88%Colore e forma:Liquid About 5 5 Bitter Numbing Taste (Ntp 1992)Peso molecolare:305.85MK-0249 FA
MK-0249 FA is an H3 inverse agonist that can be used to study attention-deficit, hyperactivity disorder and cognitive disorders in adults.Formula:C24H26F3N3O4Purezza:99.98%Colore e forma:SolidPeso molecolare:477.48Pemirolast potassium
CAS:Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.Formula:C10H7KN6OPurezza:98.91% - 99.63%Colore e forma:Crystals From Dimethylformamide Crystalline SolidPeso molecolare:266.31Clemastine fumarate
CAS:Clemastine fumarate (Meclastine (fumarate)) is a synthetic ethanolamine with anticholinergic, sedative, and histamine H1 antagonistic properties.Formula:C25H30ClNO5Purezza:99.52% - >99.99%Colore e forma:Colorless To Faintly Yellow Crystalline Powder Appearance White Or Almost White Crystalline PowderPeso molecolare:459.97Roxatidine Acetate hydrochloride
CAS:Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.Formula:C19H29ClN2O4Purezza:99.49%Colore e forma:SolidPeso molecolare:384.9Pimethixene
CAS:<p>Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.</p>Formula:C19H19NSPurezza:97.50%Colore e forma:SolidPeso molecolare:293.43
