CymitQuimica logo
Recettore dell'istamina

Recettore dell'istamina

I recettori dell'istamina sono GPCR che mediano gli effetti dell'istamina, un'ammina biogena coinvolta nelle risposte immunitarie, nella secrezione acida gastrica e nella neurotrasmissione. Esistono quattro sottotipi di recettori dell'istamina (H1, H2, H3 e H4), ognuno dei quali svolge ruoli distinti nelle reazioni allergiche, nella funzione gastrica e nell'attività del sistema nervoso centrale. Gli antagonisti dei recettori dell'istamina sono ampiamente utilizzati nel trattamento delle allergie, delle ulcere peptiche e della cinetosi. Presso CymitQuimica, offriamo una selezione completa di modulatori dei recettori dell'istamina di alta qualità per supportare la tua ricerca in immunologia, gastroenterologia e neurofarmacologia.

Trovati 382 prodotti di "Recettore dell'istamina"

Ordinare per

Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
prodotti per pagina.
  • Lafutidine

    CAS:
    Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.
    Formula:C22H29N3O4S
    Purezza:98.55%
    Colore e forma:Yellowish White Crystalline Powder
    Peso molecolare:431.55
  • Mepyramine maleate

    CAS:
    Mepyramine maleate is a mild hypnotic, local anesthetic, and H1 histamine antagonist for allergies and colds.
    Formula:C21H27N3O5
    Purezza:99.51% - 99.7%
    Colore e forma:White Crystalline Powder
    Peso molecolare:401.47
  • Tripelennamine hydrochloride

    CAS:
    Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.
    Formula:C16H21N3·HCl
    Purezza:99.54% - 99.81%
    Colore e forma:White Solid
    Peso molecolare:291.82
  • Pimethixene

    CAS:
    <p>Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 &amp; muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.</p>
    Formula:C19H19NS
    Purezza:97.50%
    Colore e forma:Solid
    Peso molecolare:293.43
  • Terfenadine

    CAS:
    Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.
    Formula:C32H41NO2
    Purezza:98.76% - 99.75%
    Colore e forma:Solid
    Peso molecolare:471.67
  • Chloropyramine hydrochloride

    CAS:
    Chloropyramine hydrochloride (Alergosan) is a histamine receptor H1 antagonist.
    Formula:C16H20ClN3·HCl
    Purezza:99.45% - 99.8%
    Colore e forma:Solid
    Peso molecolare:326.26
  • Fenspiride hydrochloride

    CAS:
    Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.
    Formula:C15H20N2O2·HCl
    Purezza:99.64% - 99.92%
    Colore e forma:Solid
    Peso molecolare:296.79
  • Clemastine fumarate

    CAS:
    Clemastine fumarate (Meclastine (fumarate)) is a synthetic ethanolamine with anticholinergic, sedative, and histamine H1 antagonistic properties.
    Formula:C25H30ClNO5
    Purezza:99.52% - >99.99%
    Colore e forma:Colorless To Faintly Yellow Crystalline Powder Appearance White Or Almost White Crystalline Powder
    Peso molecolare:459.97
  • Promethazine hydrochloride

    CAS:
    Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.
    Formula:C17H20N2S·HCl
    Purezza:99.85%
    Colore e forma:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)
    Peso molecolare:320.88
  • Astemizole

    CAS:
    <p>Astemizole (Laridal) is a long-acting antihistamine for allergies like rhinitis and asthma, with fewer anticholinergic effects.</p>
    Formula:C28H31FN4O
    Purezza:98.24% - 99.67%
    Colore e forma:White Crystals Solid
    Peso molecolare:458.57
  • Pemirolast potassium

    CAS:
    Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.
    Formula:C10H7KN6O
    Purezza:98.91% - 99.63%
    Colore e forma:Crystals From Dimethylformamide Crystalline Solid
    Peso molecolare:266.31
  • MK-0249 FA


    MK-0249 FA is an H3 inverse agonist that can be used to study attention-deficit, hyperactivity disorder and cognitive disorders in adults.
    Formula:C24H26F3N3O4
    Purezza:99.98%
    Colore e forma:Solid
    Peso molecolare:477.48
  • Histamine

    CAS:
    Histamine (Ergamine) is an amine derived by the enzymatic decarboxylation of histamine. Histamine is a potent stimulant of gastric secretion of central action. High-Quality, Low-Cost!
    Formula:C5H9N3
    Purezza:96.63% - >99.99%
    Colore e forma:Needles From Chloroform Solid
    Peso molecolare:111.15
  • Triprolidine hydrochloride monohydrate

    CAS:
    Triprolidine hydrochloride monohydrate is a histamine H1 antagonist used in allergic rhinitis, asthma.
    Formula:C19H25ClN2O
    Purezza:99.68% - 99.81%
    Colore e forma:White Crystalline Powder
    Peso molecolare:332.87
  • Fexofenadine hydrochloride

    CAS:
    Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor antagonist, with
    Formula:C32H40ClNO4
    Purezza:>99.99%
    Colore e forma:White Crystalline Powder
    Peso molecolare:538.12
  • Dimenhydrinate

    CAS:
    Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.
    Formula:C24H28ClN5O3
    Purezza:99.57% - 99.77%
    Colore e forma:Crystals Physical Description Crystalline White Powder (Ntp 1992)
    Peso molecolare:469.96
  • Levodropropizine

    CAS:
    Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.
    Formula:C13H20N2O2
    Purezza:99.87% - 99.93%
    Colore e forma:White Or Off White Crystalline Powder
    Peso molecolare:236.31
  • Cyproheptadine hydrochloride sesquihydrate

    CAS:
    Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.
    Formula:C21H24ClNO
    Purezza:99.77% - >99.99%
    Colore e forma:White To Slightly Yellowish Crystalline Solid
    Peso molecolare:341.88
  • Brompheniramine maleate

    CAS:
    Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.
    Formula:C16H19BrN2·C4H4O4
    Purezza:99.80%
    Colore e forma:Crystal Powder
    Peso molecolare:435.31
  • Doxylamine succinate

    CAS:
    <p>Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.</p>
    Formula:C21H28N2O5
    Purezza:99.61%
    Colore e forma:5 1 (Ntp 1992)
    Peso molecolare:388.46
  • Antazoline hydrochloride

    CAS:
    Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenous
    Formula:C17H19N3·HCl
    Purezza:98% - 99.53%
    Colore e forma:White Or Almost White Crystalline Powder
    Peso molecolare:301.82
  • Mizolastine

    CAS:
    Mizolastine (SL 850324), an antihistamine with IC50 of 47 nM, treats allergies like hay fever and hives.
    Formula:C24H25FN6O
    Purezza:98% - 99.75%
    Colore e forma:Solid
    Peso molecolare:432.49
  • Azatadine dimaleate

    CAS:
    <p>Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).</p>
    Formula:C28H30N2O8
    Purezza:99.7% - >99.99%
    Colore e forma:Powder
    Peso molecolare:522.55
  • Ranitidine Hydrochloride

    CAS:
    Ranitidine Hydrochloride (AH19065) is a competitive and reversible inhibitor of histamine H2-receptor antagonists with antacid activity.
    Formula:C13H23ClN4O3S
    Purezza:99.30% - 99.49%
    Colore e forma:Solid
    Peso molecolare:350.86
  • Orphenadrine hydrochloride

    CAS:
    Orphenadrine hydrochloride (Mephenamin) is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.
    Formula:C18H23NO·HCl
    Purezza:99.88%
    Colore e forma:Liquid About 5 5 Bitter Numbing Taste (Ntp 1992)
    Peso molecolare:305.85
  • Diphenylpyraline hydrochloride

    CAS:
    Diphenylpyraline hydrochloride treats Parkinsonism. It's an antihistamine with anticholinergic properties and inhibits dopamine reuptake.
    Formula:C19H23NO·HCl
    Purezza:98.72%
    Colore e forma:Solid
    Peso molecolare:317.85
  • Amodiaquine dihydrochloride dihydrate

    CAS:
    <p>Amodiaquine dihydrochloride dihydrate (Amodiaquin hydrochloride) is an orally active 4-aminoquinoline derivative with antimalarial and anti-inflammatory effects</p>
    Formula:C20H28Cl3N3O3
    Purezza:99.97%
    Colore e forma:Solid
    Peso molecolare:464.82
  • Chlorprothixene hydrochloride

    CAS:
    Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.
    Formula:C18H18ClNS·HCl
    Purezza:99.76%
    Colore e forma:White Powder
    Peso molecolare:352.32
  • Meclizine dihydrochloride

    CAS:
    Meclizine dihydrochloride (NSC28728) is a histamine H1 antagonist used in the treatment of motion sickness, vertigo, and nausea during pregnancy and radiation
    Formula:C25H27ClN2·2HCl
    Purezza:98.05% - 99.79%
    Colore e forma:White Slightly Yellowish Crystalline Powder
    Peso molecolare:463.87
  • Rupatadine Fumarate

    CAS:
    Rupatadine Fumarate (Rinialer) (UR-12592 Fumarate) is a potent dual PAF/H1 antagonist with Ki of 0.55/0.1 uM.
    Formula:C26H26ClN3·C4H4O4
    Purezza:99.86%
    Colore e forma:White Or Almost-White Powder
    Peso molecolare:532.03
  • Mifentidine

    CAS:
    Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.
    Formula:C13H16N4
    Purezza:98.34% - 99.73%
    Colore e forma:Solid
    Peso molecolare:228.29
  • Ketotifen fumarate

    CAS:
    Ketotifen fumarate (HC 20511 fumarate) is a cycloheptathiophene blocker of histamine H1 receptors and release of inflammatory mediators.
    Formula:C23H23NO5S
    Purezza:99.25% - 99.73%
    Colore e forma:Solid
    Peso molecolare:425.50
  • Perphenazine

    CAS:
    <p>Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.</p>
    Formula:C21H26ClN3OS
    Purezza:99.3% - 99.99%
    Colore e forma:Solid
    Peso molecolare:403.97
  • Dexchlorpheniramine Maleate

    CAS:
    Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active isomer of chlorpheniramine.
    Formula:C20H23ClN2O4
    Purezza:99.58%
    Colore e forma:White Or Almost White Crystalline Powder
    Peso molecolare:390.86
  • Hydroxyzine Pamoate

    CAS:
    Hydroxyzine Pamoate (Bobsule) is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria and histamine-mediated pruritus.
    Formula:C44H43ClN2O8
    Purezza:99.49%
    Colore e forma:Solid
    Peso molecolare:763.27
  • Traxanox

    CAS:
    Traxanox: oral diuretic, boosts phagocytosis in mice/rats, reverses antibody production inhibition in BALB/c mice.
    Formula:C13H6ClN5O2
    Purezza:98.37%
    Colore e forma:Solid
    Peso molecolare:299.67
  • BMY 25368 HCl

    CAS:
    BMY 25368 HCl is a competitive histamine H2 receptor antagonist that antagonizes gastric secretion stimulated by pentagastrin, ethacrynic choline, and food.
    Formula:C19H26ClN3O3
    Purezza:98.73% - 99.81%
    Colore e forma:Soild
    Peso molecolare:379.88
  • Azelastine hydrochloride

    CAS:
    Azelastine hydrochloride (Astelin) is a phthalazinone derivative with antihistaminergic activity.
    Formula:C22H24ClN3O·HCl
    Purezza:98% - >99.99%
    Colore e forma:White Crystalline Powder
    Peso molecolare:418.36
  • Azacyclonol

    CAS:
    Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.
    Formula:C18H21NO
    Purezza:99.46%
    Colore e forma:Solid Powder
    Peso molecolare:267.37
  • Cimetidine

    CAS:
    <p>Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS.</p>
    Formula:C10H16N6S
    Purezza:99.82%
    Colore e forma:Crystals Physical Description White Crystals With A Slight Sulfur-Mercaptan Odor (Ntp 1992)
    Peso molecolare:252.34
  • Mebhydrolin napadisylate

    CAS:
    Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergic
    Formula:C19H20N2C10H8O6S2
    Purezza:99.35% - 99.96%
    Colore e forma:White Or Almost White Crystalline
    Peso molecolare:420.52
  • Cinnarizine

    CAS:
    Cinnarizine is a piperazine, blocks H1-receptor & Ca-channels, has vasodilating & antiemetic effects, may cause Parkinson-like symptoms.
    Formula:C26H28N2
    Purezza:99.94%
    Colore e forma:Solid
    Peso molecolare:368.51
  • Carbinoxamine Maleate Salt

    CAS:
    Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.
    Formula:C20H23ClN2O5
    Purezza:99.97%
    Colore e forma:Off-White Solid
    Peso molecolare:406.86
  • Levocetirizine

    CAS:
    Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a Histamine H1 Receptor Antagonist.
    Formula:C21H25ClN2O3
    Purezza:98% - 99.94%
    Colore e forma:White Powder
    Peso molecolare:388.89
  • Famotidine

    CAS:
    Famotidine, a histamine H2-blocker, curbs gastric acid production, lowering volume and acidity.
    Formula:C8H15N7O2S3
    Purezza:98.93% - 99.91%
    Colore e forma:White To Off-White Crystalline Powder
    Peso molecolare:337.45
  • JNJ-39758979

    CAS:
    <p>JNJ-39758979: selective H4 receptor antagonist, Kis 12.5/5.3/25 nM (human/mouse/monkey), blocks histamine cAMP inhibition (pA2 7.9).</p>
    Formula:C11H19N5
    Purezza:98.33% - 99.62%
    Colore e forma:Solid
    Peso molecolare:221.3
  • Mianserin hydrochloride

    CAS:
    Mianserin HCl (Org GB 94): a tetracyclic antidepressant; blocks alpha-adrenergic, H1, serotonin receptors; may induce drowsiness, hematological issues.
    Formula:C18H21ClN2
    Purezza:99.63% - 99.82%
    Colore e forma:White And Film Coated Tablet And Seem To Be White Or White-Like After Removing It'S Film Coated
    Peso molecolare:300.83
  • Olopatadine hydrochloride

    CAS:
    Olopatadine hydrochloride (ALO4943A) is an antihistamine with mast-cell stabilizing properties used as eye drops in the treatment of ALLERGIC CONJUNCTIVITIS.
    Formula:C21H23NO3·HCl
    Purezza:99.62% - 99.64%
    Colore e forma:White Solid
    Peso molecolare:373.87
  • Talastine

    CAS:
    Talastine is an antihistamine compound that can induce an allergic rash.
    Formula:C19H21N3O
    Purezza:99.44% - 99.84%
    Colore e forma:Solid
    Peso molecolare:307.39
  • Benztropine mesylate

    CAS:
    <p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>
    Formula:C21H25NO·CH4SO3
    Purezza:98.41% - 99.96%
    Colore e forma:White Crystalline Powder; Odourless Or Almost Odourless
    Peso molecolare:403.53
  • Doxepin hydrochloride

    CAS:
    Doxepin hydrochloride, a dibenzoxepin tricyclic, blocks monoamine reuptake and has anticholinergic and antihistaminic effects. Mechanism partly unknown.
    Formula:C19H22ClNO
    Purezza:99.65% - 99.91%
    Colore e forma:White To Off-White Powder
    Peso molecolare:315.84
  • Fenclozine Maleate

    CAS:
    <p>Fenclozine Maleate (S 1429) is a potential histamine H1 receptor antagonist , which can be used to study fever, inflammation and pain.</p>
    Formula:C45H47ClN2O12
    Purezza:98.47%
    Colore e forma:Soild
    Peso molecolare:843.314
  • Carebastine

    CAS:
    Carebastine, the active metabolite of Ebastine, is an antagonist of the histamine H1 receptor.
    Formula:C32H37NO4
    Purezza:99.16%
    Colore e forma:Off-White Solid
    Peso molecolare:499.64
  • Mirtazapine

    CAS:
    Mirtazapine is a unique tetracyclic antidepressant, may cause temporary liver enzyme elevation, and is linked to rare liver injury.
    Formula:C17H19N3
    Purezza:99.98%
    Colore e forma:Solid
    Peso molecolare:265.35
  • Amitriptyline hydrochloride

    CAS:
    Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive
    Formula:C20H24ClN
    Purezza:97% - 99.94%
    Colore e forma:Crystals White To Off-White Powder
    Peso molecolare:313.86
  • Pheniramine maleate

    CAS:
    Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors.
    Formula:C16H20N2·C4H4O4
    Purezza:99.85%
    Colore e forma:Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°C
    Peso molecolare:356.42
  • Cetirizine dihydrochloride

    CAS:
    Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.
    Formula:C21H27Cl3N2O3
    Purezza:99.4% - 99.97%
    Colore e forma:Solid
    Peso molecolare:461.81
  • Roxatidine Acetate hydrochloride

    CAS:
    Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.
    Formula:C19H29ClN2O4
    Purezza:99.49%
    Colore e forma:Solid
    Peso molecolare:384.9
  • Chlorpheniramine maleate

    CAS:
    <p>Chlorpheniramine maleate (NCI-C55265) is a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, urticaria, and asthma.</p>
    Formula:C20H23ClN2O4
    Purezza:99.64% - 99.98%
    Colore e forma:Odorless White Crystalline Solid Or White Powder With A Bitter Taste
    Peso molecolare:390.87
  • Loratadine

    CAS:
    <p>Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria.</p>
    Formula:C22H23ClN2O2
    Purezza:99.71% - 99.98%
    Colore e forma:White Powder
    Peso molecolare:382.88
  • Betahistine mesylate

    CAS:
    <p>Betahistine mesylate (Extovyl), an H1 agonist and vasodilator, treats Meniere's disease and vascular headaches; risks with asthma/ulcers.</p>
    Formula:C8H12N2·2(CH4O3S)
    Purezza:98% - 99.85%
    Colore e forma:Coa
    Peso molecolare:328.4
  • (S)-Azelastine hydrochloride

    CAS:
    (S)-Azelastine HCl, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.
    Formula:C22H25Cl2N3O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:418.36
  • Histamine H4 receptor antagonist-1

    CAS:
    Histamine H4 receptor antagonist-1 is a potent antagonist of the histamine H4 receptor.
    Formula:C30H38N8O2
    Colore e forma:Solid
    Peso molecolare:542.68
  • Dalcotidine

    CAS:
    <p>Dalcotidine (KU 1257), a histamine H2/H9 blocker, inhibits acid secretion; Ki=0.040, KB=0.041, aids ulcer healing, may lower relapse.</p>
    Formula:C18H29N3O2
    Purezza:99.11%
    Colore e forma:Solid
    Peso molecolare:319.44
  • (+)-Dropropizine

    CAS:
    (+)-Dropropizine can inhibit histamine receptor, anti-allergic, and reduce a cough by modulation of neuropeptides involved in the cough reflex.
    Formula:C13H20N2O2
    Purezza:>99.99%
    Colore e forma:White Or Off White Crystalline Powder
    Peso molecolare:236.31
  • Tecastemizole

    CAS:
    Tecastemizole (R 43512) is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects.
    Formula:C19H21FN4
    Purezza:99.70%
    Colore e forma:Solid
    Peso molecolare:324.4
  • Sufotidine

    CAS:
    Sufotidine (AH 25352X) is a highly selective competitive H2 receptor antagonist.
    Formula:C20H31N5O3S
    Purezza:99.03% - 99.92%
    Colore e forma:Solid
    Peso molecolare:421.56
  • Cetirizine methyl ester

    CAS:
    Cetirizine methyl ester is a Cetirizine impurity, a long-acting, oral H1-antihistamine and hydroxyzine metabolite.
    Formula:C22H27ClN2O3
    Colore e forma:Solid
    Peso molecolare:402.91
  • Cetirizine Impurity C

    CAS:
    Cetirizine Impurity C - a metabolite of hydroxyzine, is a long-acting, oral H1-antihistamine.
    Formula:C21H25ClN2O3
    Colore e forma:Solid
    Peso molecolare:388.89
  • Cetirizine Impurity C dihydrochloride

    CAS:
    Cetirizine Impurity C dihydrochloride is a Cetirizine metabolite and long-acting H1-antihistamine.
    Formula:C21H27Cl3N2O3
    Colore e forma:Solid
    Peso molecolare:461.81
  • Conessine hydrobromide

    CAS:
    Conessine hydrobromide is a naturally occurring steroid alkaloid and has been used in traditional herbal medicine as a treatment for amoebic dysentery.
    Formula:C24H41BrN2
    Colore e forma:Solid
    Peso molecolare:437.51
  • Bodilisant

    CAS:
    Bodilisant: nanomolar-affinity hH3R ligand, derived from piperidine, with BODIPY fluorophore.
    Formula:C27H34BF2N3O
    Colore e forma:Solid
    Peso molecolare:465.4
  • Donetidine

    CAS:
    Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.
    Formula:C20H25N5O3S
    Purezza:99.32%
    Colore e forma:Solid
    Peso molecolare:415.51
  • 4-Methylhistamine

    CAS:
    <p>4-Methylhistamine serves as a potent agonist for the histamine 4 receptor (H4R), holding promise for research into immune-related diseases, including cancer and</p>
    Formula:C6H11N3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:125.17
  • Vapitadine

    CAS:
    Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.
    Formula:C17H20N4O
    Purezza:99.77% - 99.86%
    Colore e forma:Soild
    Peso molecolare:296.37
  • Nizatidine

    CAS:
    Nizatidine (Acinon) is a competitive and reversible histamine H2-receptor antagonist with antacid activity.
    Formula:C12H21N5O2S2
    Purezza:99.43%
    Colore e forma:White To Off-White Crystalline Powder
    Peso molecolare:331.46
  • Neurotransmitter Receptor Compound Library


    <p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening;</p>
    Colore e forma:Odour Solid
  • Levocarnitine propionate hydrochloride

    CAS:
    Levocarnitine propionate hydrochloride (ST-261) is used for the treatment of the deterioration of renal function, congestive heart failure, and other diseases.
    Formula:C10H20ClNO4
    Purezza:90% - 99.77%
    Colore e forma:Solid
    Peso molecolare:253.72
  • H4R antagonist 3

    CAS:
    <p>H4R antagonist 3 is a novel histamine-4 receptor (H4R) antagonist with an EC50 &lt;10 mM.H4R antagonist 3 has potential inflammatory activity for the study of</p>
    Formula:C19H21ClN4S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:372.92
  • Oxmetidine

    CAS:
    Oxmetidine (SKF 92994) is an H2R antagonist that inhibits transmembrane calcium flux in the cardiovascular system and is used in the study of duodenal ulcers.
    Formula:C19H21N5O3S
    Purezza:99.67%
    Colore e forma:Solid
    Peso molecolare:399.47
  • Methapyrilene hydrochloride

    CAS:
    <p>Methapyrilene hydrochloride is a biochemical.</p>
    Formula:C14H20ClN3S
    Colore e forma:Liquid Solution) 5 5 (Ntp 1992)
    Peso molecolare:297.85
  • KSK94 FA


    KSK94 FA is a potent histamine H3 receptor antagonist that inhibits H3 receptors and is used in the study of neuropathic pain and obesity.
    Formula:C26H28N4O3
    Purezza:97.51%
    Colore e forma:Soild
    Peso molecolare:444.53
  • KSK67

    CAS:
    <p>KSK67 is a selective dual antagonist of sigma-2 and histamine H3 receptors with inhibitory effects on H3 receptors, sigma-1, and sigma-2 receptors, with Ki</p>
    Formula:C22H27N3O2
    Purezza:99.11%
    Colore e forma:Soild
    Peso molecolare:365.47
  • Samelisant

    CAS:
    Samelisant (SUVN-G3031), a selective H3 inverse agonist, Ki=8.7/9.8 nM in humans/rats, has anti-narcoleptic properties.
    Formula:C21H31N3O3
    Purezza:99.59%
    Colore e forma:Solid
    Peso molecolare:373.49
  • Cetirizine Impurity D

    CAS:
    Cetirizine Impurity D, an antihistamine derivative, acts as a long-lasting H1-receptor antagonist with antiallergic effects.
    Formula:C30H28Cl2N2
    Colore e forma:Solid
    Peso molecolare:487.46
  • JNJ-10181457 (hydrochloride)

    CAS:
    JNJ-10181457 (hydrochloride) is a non-imidazole H3 receptor antagonist that is brain-penetrating and selective, increasing NE and acetylcholine concentrations
    Formula:C20H30Cl2N2O
    Colore e forma:Solid
    Peso molecolare:385.37
  • Dexchlorpheniramine free base

    CAS:
    <p>Dexchlorpheniramine Maleate, a histamine receptor antagonist, is used to treat urticaria, allergic rhinitis, allergic conjunctivitis and pruritus.</p>
    Formula:C16H19ClN2
    Purezza:98%
    Colore e forma:Oily Liquid Solid
    Peso molecolare:274.79
  • Thioperamide maleate

    CAS:
    <p>Thioperamide maleate (MR-12842 maleate) is an effective and selective antagonist of H3 receptor (Ki = 4.3 nM) for inhibition of [3H]histamine synthesis (Ki = 31</p>
    Formula:C19H28N4O4S
    Purezza:98.48%
    Colore e forma:Solid
    Peso molecolare:408.52
  • Histamine & Melatonin Receptor-Targeted Compound Library


    <p>A unique collection of xnum compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCS</p>
    Colore e forma:Odour Solid
  • Diphenhydramine hydrochloride

    CAS:
    <p>DPH: antihistamine for cough, nausea, itching, allergy, Parkinson's, sleep aid, cold remedy.</p>
    Formula:C17H22ClNO
    Purezza:99.84%
    Colore e forma:Taste Ph (5% Aqueous Solution) 4-6 (Ntp 1992)
    Peso molecolare:291.82
  • Nα-Methylhistamine FA


    Nα-Methylhistamine FA is a histamine H3 receptor agonist
    Formula:C7H13N3O2
    Purezza:>99.99%
    Colore e forma:Solid
    Peso molecolare:171.2
  • Sigma-1 receptor antagonist 5


    Sigma-1 receptor antagonist 5 (compound 12), a 4-pyridylpiperidine derivative, exhibits analgesic properties through its antagonistic action on sigma receptors
    Formula:C26H27N3O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:397.51
  • Cetirizine D8 dihydrochloride

    CAS:
    <p>Cetirizine D8 dihydrochloride is a deuterated H1-antihistamine with long-acting effects.</p>
    Formula:C21H26Cl2N2O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:433.4
  • AM-0466

    CAS:
    AM-0466 has a wide range of applications in life science related research.
    Formula:C27H19F3N4O4S
    Colore e forma:Solid
    Peso molecolare:552.52
  • 3-hydroxy Desloratidine

    CAS:
    3-hydroxy Desloratidine is a major metabolite of desloratadine , a tricyclic antagonist of the histamine H1 receptor.
    Formula:C19H19ClN2O
    Colore e forma:Solid
    Peso molecolare:326.82
  • Methimepip dihydrobromide

    CAS:
    Methimepip dihydrobromide is a selective H3R agonist.
    Formula:C10H19Br2N3
    Colore e forma:Solid
    Peso molecolare:341.091
  • Oxmetidine FA


    <p>Oxmetidine FA is an orally available specific histamine H2 receptor antagonist with antiulcerogenic properties.</p>
    Formula:C20H23N5O5S
    Purezza:97.34%
    Colore e forma:Soild
    Peso molecolare:445.49
  • Alcaftadine carboxylic acid

    CAS:
    Alcaftadine is a novel antihistamine for preventing allergic conjunctivitis.
    Formula:C19H21N3O2
    Colore e forma:Solid
    Peso molecolare:323.39
  • Acrivastine D7

    CAS:
    Acrivastine D7 is a deuterium labeled Acrivastine. Acrivastine is a short acting antagonist of histamine 1 receptor.
    Formula:C22H24N2O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:355.48
  • Hydroxyzine D8

    CAS:
    Hydroxyzine D8, a deuterium-labeled version of Hydroxyzine, acts as a histamine H1-receptor antagonist.
    Formula:C21H27ClN2O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:382.95
  • 1-Methyl-4-imidazoleacetic Acid (hydrochloride)

    CAS:
    MIMA, a stable histamine byproduct from N-methylhistamine oxidation, indicates systemic mastocytosis via urinary levels.
    Formula:C6H9ClN2O2
    Colore e forma:Solid
    Peso molecolare:176.601
  • Fexofenadine-d6

    CAS:
    Fexofenadine D6 is an antihistamine pharmaceutical drug.Fexofenadine D6 is deuterium labeled is Fexofenadine.
    Formula:C32H39NO4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:507.69
  • Cetirizine D4

    CAS:
    Cetirizine D4 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
    Formula:C21H25ClN2O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:392.91
  • Tiotidine

    CAS:
    Tiotidine is a selective histamine H2-receptor antagonist (pA2=7.3-7.8 for guinea-pig right atrium).
    Formula:C10H16N8S2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:312.42
  • Gizzerosine

    CAS:
    Gizzerosine, a biogenic amine formed during feed processing, is a toxicant that induces mortality in livestock.
    Formula:C11H20N4O2
    Colore e forma:Solid
    Peso molecolare:240.3
  • Cetirizine D8

    CAS:
    Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
    Formula:C21H25ClN2O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:396.94
  • WZ4141

    CAS:
    WZ4141 is an intermediate in compound synthesis.
    Formula:C16H13N3O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:279.29
  • Diphenylpyraline

    CAS:
    Diphenylpyridine is the first generation antihistamine, which has the anticholinergic effect of diphenylpiperidine.
    Formula:C19H23NO
    Colore e forma:Solid
    Peso molecolare:281.39
  • Doxepin D3 Hydrochloride

    CAS:
    Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin hydrochloride is also an effective CYP450 inhibitor, significantly inhibiting CYP450 2C19 and
    Formula:C19H22ClNO
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:318.86
  • Alimemazine D6

    CAS:
    Alimemazine D6 is a deuterium-labeled Alimemazine. Alimemazine is an antihistamine.
    Formula:C18H22N2S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:304.48
  • Antazoline phosphate

    CAS:
    Antazoline phosphate: H1 histamine receptor antagonist with anticholinergic effects, eases allergies.
    Formula:C17H22N3O4P
    Purezza:98%
    Colore e forma:Coa
    Peso molecolare:363.35
  • Emedastine Difumarate

    CAS:
    Emedastine Difumarate, an H1 receptor blocker for allergic conjunctivitis, reduces histamine-induced eye inflammation.
    Formula:C25H34N4O9
    Colore e forma:Solid
    Peso molecolare:534.56
  • Hydroxyzine dihydrochloride-d4

    CAS:
    Hydroxyzine dihydrochloride-d4 is a deuterated compound of Hydroxyzine dihydrochloride.
    Formula:C21H25D4Cl3N2O2
    Colore e forma:Solid
    Peso molecolare:451.85
  • Buclizine

    CAS:
    Buclizine is an orally active antihistamine, antiallergic compound. buclizine is also a strong teratogen in rats and exhibits antitumour effects.
    Formula:C28H33ClN2
    Colore e forma:Solid
    Peso molecolare:433.03
  • H4 Receptor antagonist 1

    CAS:
    H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.
    Formula:C16H17ClN4O
    Purezza:98.81%
    Colore e forma:Solid
    Peso molecolare:316.79
  • Mebhydrolin

    CAS:
    Mebhydrolin (Mebhydroline) is a specific histamine H1 receptor antagonist.
    Formula:C19H20N2
    Purezza:99.3% - ≥98%
    Colore e forma:Solid
    Peso molecolare:276.38
  • Fexofenadine

    CAS:
    Fexofenadine, a non-sedating antihistamine, treats allergies like hay fever and urticaria.
    Formula:C32H39NO4
    Purezza:99.35%
    Colore e forma:White To Off-White Solid
    Peso molecolare:501.66
  • Conessine

    CAS:
    <p>Conessine (Conessinum), a steroidal alkaloid isolated from Holarrhena floribunda, interacts with the histamine H3 receptor and has anti-malarial activity.</p>
    Formula:C24H40N2
    Purezza:99.65%
    Colore e forma:Solid
    Peso molecolare:356.59
  • Fexofenadine hydrochloride

    CAS:
    <p>Fexofenadine hydrochloride (Terfenidine carboxylate hydrochloride) is a second generation antihistamine that is used for the treatment of allergic rhinitis,</p>
    Formula:C32H39NO4·HCl
    Purezza:99.39% - ≥95%
    Colore e forma:Solid
    Peso molecolare:538.13
  • Acrivastine

    CAS:
    Acrivastine (Acrivastin) is a short-acting histamine 1 receptor antagonist.
    Formula:C22H24N2O2
    Purezza:99.73% - >99.99%
    Colore e forma:Solid
    Peso molecolare:348.44
  • Chlorphenoxamine

    CAS:
    <p>Chlorphenoxamine (Contristamine) is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.</p>
    Formula:C18H22ClNO
    Purezza:99.44% - 99.85%
    Colore e forma:Solid
    Peso molecolare:303.83
  • Epinastine

    CAS:
    Epinastine (WAL801) is an antihistamine, mast cell stabilizer, and H1 antagonist with anti-allergic properties.
    Formula:C16H15N3
    Purezza:99.94%
    Colore e forma:Solid
    Peso molecolare:249.31
  • Alcaftadine

    CAS:
    Alcaftadine (Lastacaft) is an H1 histamine receptor antagonist indicated for the prevention of itching associated with allergic conjunctivitis.
    Formula:C19H21N3O
    Purezza:98% - 98.65%
    Colore e forma:Solid
    Peso molecolare:307.39
  • Bepotastine Besilate

    CAS:
    Bepotastine Besilate (TAU 284) is a non-sedating and selective H1 receptor antagonist (pIC50: 5.7).
    Formula:C21H25ClN2O3·C6H6O3S
    Purezza:99.83% - 99.9%
    Colore e forma:Brown Viscous Liquid
    Peso molecolare:547.06
  • Desloratadine

    CAS:
    Desloratadine (Sch34117) is a long-acting piperidine derivate with selective H1 antihistaminergic and non-sedating properties.
    Formula:C19H19ClN2
    Purezza:99.79% - >99.99%
    Colore e forma:Solid
    Peso molecolare:310.82
  • Lodoxamide

    CAS:
    <p>Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.</p>
    Formula:C11H6ClN3O6
    Purezza:99.13% - 99.81%
    Colore e forma:Solid
    Peso molecolare:311.63
  • Niaprazine

    CAS:
    <p>Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.</p>
    Formula:C20H25FN4O
    Purezza:99.56%
    Colore e forma:Solid
    Peso molecolare:356.44
  • Ritanserin

    CAS:
    Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.
    Formula:C27H25F2N3OS
    Purezza:99.77% - 99.89%
    Colore e forma:Solid
    Peso molecolare:477.57
  • Emedastine

    CAS:
    <p>Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity.</p>
    Formula:C17H26N4O
    Purezza:97.1% - 97.76%
    Colore e forma:Oil
    Peso molecolare:302.41
  • Tesmilifene fumarate

    CAS:
    Tesmilifene fumarate (DPPE fumarate) (DPPE fumarate) is an H1C receptor antagonist。
    Formula:C23H29NO5
    Purezza:99.86%
    Colore e forma:Solid
    Peso molecolare:399.48
  • Diphenhydramine

    CAS:
    Diphenhydramine (Syntedril): first-gen antihistamine for allergies, antiemetic, antitussive, anticholinergic, sedative, treats drug-induced parkinsonism.
    Formula:C17H21NO
    Purezza:98.07%
    Colore e forma:Solid
    Peso molecolare:255.35
  • Ebastine

    CAS:
    Ebastine (Kestine) (trade names Evastin, Kestine, Ebastel, Aleva) is a non-sedating H1 antihistamine.
    Formula:C32H39NO2
    Purezza:99.65% - 99.99%
    Colore e forma:White To Off-White Powder
    Peso molecolare:469.66
  • Pitolisant hydrochloride

    CAS:
    Pitolisant hydrochloride (Ciproxidine) is a potent and selective inverse agonist of the histamine H3 receptor(Ki : 0.16 nM).
    Formula:C17H27Cl2NO
    Purezza:99.72% - 99.91%
    Colore e forma:Solid
    Peso molecolare:332.31
  • Clemizole

    CAS:
    Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.
    Formula:C19H20ClN3
    Purezza:98% - 99.65%
    Colore e forma:Solid
    Peso molecolare:325.84
  • HTMT dimaleate

    CAS:
    <p>HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.</p>
    Formula:C27H33F3N4O9
    Purezza:99.51%
    Colore e forma:Solid
    Peso molecolare:614.57
  • Hydroxyzine

    CAS:
    Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.
    Formula:C21H27ClN2O2
    Purezza:99.54% - ≥95%
    Colore e forma:Oil Solid
    Peso molecolare:374.9
  • Samelisant dihydrochloride

    CAS:
    SUVN-G3031: H3 receptor antagonist; may treat cognitive issues, ADHD, epilepsy, sleep, obesity, schizophrenia, eating disorders, pain.
    Formula:C21H33Cl2N3O3
    Colore e forma:Solid
    Peso molecolare:446.41
  • Bromodiphenhydramine hydrochloride

    CAS:
    <p>Bromodiphenhydramine hydrochloride is a new antihistaminic in the control of cutaneous.</p>
    Formula:C17H21BrClNO
    Purezza:97.29%
    Colore e forma:Solid
    Peso molecolare:370.71
  • BMY-25368

    CAS:
    BMY-25368 is a long-acting antagonist of the H2-receptor.
    Formula:C19H25N3O3
    Colore e forma:Solid
    Peso molecolare:343.42
  • JNJ-5207852 dihydrochloride

    CAS:
    JNJ-5207852 dihydrochloride is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor
    Formula:C20H34Cl2N2O
    Purezza:99.51%
    Colore e forma:Solid
    Peso molecolare:389.4
  • Clobenpropit 2HBr

    CAS:
    Clobenpropit 2HBr is a histamine H3 receptor antagonist. It has neuroprotective effects via stimulation of GABA release in the brain.
    Formula:C14H17ClN4S
    Colore e forma:Solid
    Peso molecolare:308.83
  • Bilastine

    CAS:
    Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration of
    Formula:C28H37N3O3
    Purezza:99.86% - >99.99%
    Colore e forma:Solid
    Peso molecolare:463.61
  • SCH-37370

    CAS:
    SCH-37370 is an effective and orally active dual antagonist of platelet-activating factor and histamine.
    Formula:C21H21ClN2O
    Purezza:99.07%
    Colore e forma:Solid
    Peso molecolare:352.86
  • Chlorpheniramine

    CAS:
    Chlorpheniramine is an H1 anti-histamine agent for IgE-mediated inflammation that is commonly used for allergic diseases.
    Formula:C16H19ClN2
    Colore e forma:Solid
    Peso molecolare:274.79
  • Fenspiride

    CAS:
    Fenspiride: oral non-steroidal anti-inflammatory, treats respiratory infections/otitis, inhibits H1-histamine receptors and PDE 3, 4, 5.
    Formula:C15H20N2O2
    Colore e forma:Solid
    Peso molecolare:260.33
  • Clobenpropit dihydrobromide

    CAS:
    Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07)
    Formula:C14H19Br2ClN4S
    Purezza:99.86%
    Colore e forma:Solid
    Peso molecolare:470.7
  • Bavisant dihydrochloride hydrate

    CAS:
    Bavisant dihydrochloride (JNJ31001074AAC) is an oral H3 receptor antagonist for ADHD treatment. Phase 2 trials show no significant benefits at 10 mg/day.
    Formula:C19H31Cl2N3O3
    Colore e forma:Solid
    Peso molecolare:420.38
  • Metiamide

    CAS:
    Metiamide (SK&F 92058) is a histamine H2-receptor antagonist .
    Formula:C9H16N4S2
    Purezza:97.41%
    Colore e forma:Solid
    Peso molecolare:244.38
  • 4-Methylhistamine hydrochloride

    CAS:
    <p>Compound with imidazole ring &amp; amine group; inhibits copper enzymes, affects gene expression.</p>
    Formula:C6H12ClN3
    Purezza:95%
    Colore e forma:Solid
    Peso molecolare:161.633
  • Irdabisant hydrochloride

    CAS:
    <p>Irdabisant (CEP-26401) is a selective H3R inverse agonist, BBB-penetrable, with cognition-enhancing effects.</p>
    Formula:C18H24ClN3O2
    Colore e forma:Solid
    Peso molecolare:349.86
  • Triprolidine hydrochloride

    CAS:
    Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.
    Formula:C19H23ClN2
    Colore e forma:Solid
    Peso molecolare:314.852
  • Triprolidine

    CAS:
    Triprolidine: oral H1 receptor blocker with motor/sensory spinal effects, for allergy research.
    Formula:C19H22N2
    Colore e forma:Solid
    Peso molecolare:278.39
  • GSK189254A

    CAS:
    GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).
    Formula:C21H25N3O2
    Purezza:98.71% - 99.858%
    Colore e forma:Solid
    Peso molecolare:351.44
  • Osthole

    CAS:
    Osthole (Osthol), a potential inhibitor of histamine H1 receptor, has been shown to stimulate osteoblast proliferation and differentiation.
    Formula:C15H16O3
    Purezza:99.93% - 99.96%
    Colore e forma:Fine White Powder
    Peso molecolare:244.29
  • Betazole

    CAS:
    Betazole, an oral H2 receptor agonist, stimulates gastric acid and raises bile duct pressure, used for gastric secretory testing.
    Formula:C5H9N3
    Colore e forma:Solid
    Peso molecolare:111.15
  • Betazole dihydrochloride

    CAS:
    <p>Betazole dihydrochloride (Betazole hydrochloride) is an agonist of H2 receptor.</p>
    Formula:C5H11Cl2N3
    Purezza:99.12%
    Colore e forma:Solid
    Peso molecolare:184.067
  • Mequitazine

    CAS:
    Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.
    Formula:C20H22N2S
    Purezza:99.98%
    Colore e forma:Solid
    Peso molecolare:322.47
  • Ciproxifan maleate

    CAS:
    <p>Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity</p>
    Formula:C20H22N2O6
    Purezza:99.39%
    Colore e forma:Solid
    Peso molecolare:386.4
  • Epinastine hydrochloride

    CAS:
    Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.
    Formula:C16H15N3·HCl
    Purezza:99.26% - 99.62%
    Colore e forma:White Solid
    Peso molecolare:285.77
  • Mecamylamine hydrochloride

    CAS:
    Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.
    Formula:C11H22ClN
    Purezza:99.76% - >99.99%
    Colore e forma:White Solid
    Peso molecolare:203.75
  • JNJ-7777120

    CAS:
    JNJ-7777120 is the first potent and selective non-imidazole histamine H4 receptor antagonist, exhibits >1000-fold selectivity over the other histamin receptors.
    Formula:C14H16ClN3O
    Purezza:99.83% - 99.96%
    Colore e forma:Solid
    Peso molecolare:277.75
  • Chlorcyclizine

    CAS:
    CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.
    Formula:C18H21ClN2
    Purezza:98.75%
    Colore e forma:Solid
    Peso molecolare:300.83
  • Chlorprothixene

    CAS:
    Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.
    Formula:C18H18ClNS
    Purezza:98.77% - 99.756%
    Colore e forma:Pale Yellow Crystals Solid
    Peso molecolare:315.86
  • VUF10460

    CAS:
    VUF10460 is a non-imidazole histamine H4 receptor agonist.
    Formula:C15H19N5
    Purezza:99.44% - 99.57%
    Colore e forma:Solid
    Peso molecolare:269.34
  • Dimaprit dihydrochloride

    CAS:
    Dimaprit dihydrochloride: selective H2 agonist, inhibits nNOS (IC50: 49 μM), boosts gastric acid.
    Formula:C6H15N3S·2HCl
    Purezza:99.79%
    Colore e forma:Solid
    Peso molecolare:234.19
  • Talastine HCl

    CAS:
    Talastine is an antihistamine drug.
    Formula:C19H22ClN3O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:343.86
  • C-Type Natriuretic Peptide (CNP) (1-22), human

    CAS:
    C-Type Natriuretic Peptide (CNP) (1-22), human is the 1-22 fragment of C-Type Natriuretic Peptide.
    Formula:C93H157N27O28S3
    Purezza:>99.99%
    Colore e forma:Solid
    Peso molecolare:2197.6
  • Tiaramide hydrochloride

    CAS:
    <p>Tiaramide hydrochloride (FK-1160) is an anti-inflammatory that blocks mast cell mediators and relaxes smooth muscles.</p>
    Formula:C15H19Cl2N3O3S
    Purezza:98.48%
    Colore e forma:Solid
    Peso molecolare:392.3
  • Tribenoside

    CAS:
    Tribenoside (BG-356) is a vasoprotectant with mild anti-inflammatory, analgesic, and wound healing properties.
    Formula:C29H34O6
    Purezza:≥98%
    Colore e forma:Liquid
    Peso molecolare:478.58
  • cicloprofen

    CAS:
    cicloprofen is Cell division cycle 7-related protein kinase (human) inhibitor.
    Formula:C16H14O2
    Purezza:98.15%
    Colore e forma:Solid
    Peso molecolare:238.2812
  • Acitazanolast

    CAS:
    <p>Acitazanolast (WP-871) is an anti-allergic drug candidate.</p>
    Formula:C9H7N5O3
    Purezza:98.25%
    Colore e forma:Solid
    Peso molecolare:233.18
  • 2-Pyridylethylamine dihydrochloride

    CAS:
    2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.
    Formula:C7H12Cl2N2
    Purezza:99.42%
    Colore e forma:Solid
    Peso molecolare:195.09
  • Decloxizine

    CAS:
    Decloxizine is a H1 receptor antagonist
    Formula:C21H28N2O2
    Purezza:99.53%
    Colore e forma:White Or Similar To White Powder
    Peso molecolare:340.46
  • Zotepine

    CAS:
    Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,
    Formula:C18H18ClNOS
    Purezza:99.78%
    Colore e forma:Solid
    Peso molecolare:331.86
  • Pemirolast

    CAS:
    Pemirolast: oral antiallergic, reduces paclitaxel reactions, inhibits neuropeptides, for asthma and conjunctivitis study.
    Formula:C10H8N6O
    Colore e forma:Solid
    Peso molecolare:228.21
  • Clemizole hydrochloride

    CAS:
    Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.
    Formula:C19H21Cl2N3
    Purezza:>99.99%
    Colore e forma:Solid
    Peso molecolare:362.3
  • Antazoline

    CAS:
    Antazoline has antihistamine and anticholinergic effects.It used to treat a variety of arrhythmias.
    Formula:C17H19N3
    Purezza:≥95%
    Colore e forma:White Crystalline Powder Solid
    Peso molecolare:265.35
  • Psoralenoside

    CAS:
    Psoralenoside: a compound from Psoralea fruit; has estrogenic, osteoblastic, antitumor, and antibacterial properties.
    Formula:C17H18O9
    Purezza:99.03% - 99.49%
    Colore e forma:Solid
    Peso molecolare:366.32
  • Betahistine EP Impurity C

    CAS:
    Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.
    Formula:C15H19N3
    Purezza:≥95%
    Colore e forma:Solid
    Peso molecolare:241.33
  • Dioxopromethazine hydrochloride

    CAS:
    Dioxopromethazine is a target-based classification of drug and available in a number of countries worldwide.
    Formula:C17H20N2O2S·HCl
    Purezza:99.58%
    Colore e forma:Solid
    Peso molecolare:352.88
  • Betahistine

    CAS:
    <p>Betahistine treats vertigo and balance issues in Ménière's disease; it's a histamine analog and H1 receptor agonist.</p>
    Formula:C8H12N2
    Purezza:99.87% - 99.87%
    Colore e forma:Yellowish Liquid Liquid Liquid
    Peso molecolare:136.19
  • Buclizine dihydrochloride

    CAS:
    Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic and
    Formula:C28H33ClN2·2HCl
    Purezza:98.05%
    Colore e forma:Off-White Powder
    Peso molecolare:505.95
  • S 38093

    CAS:
    S 38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).
    Formula:C17H24N2O2
    Purezza:99.95%
    Colore e forma:Solid
    Peso molecolare:288.38
  • Dioxopromethazine

    CAS:
    Dioxopromethazine (Dioxoprothazine) is a drug for the treatment of a cough and expectoration. It also can be used in local anesthesia.
    Formula:C17H20N2O2S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:316.42
  • Carcinine ditrifluoroacetate Acetate


    Carcinine ditrifluoroacetate Acetate (β-Alanylhistamine dihydrochloride) is an H3 receptor antagonist.
    Formula:C14H20F6N4O7
    Purezza:98.18%
    Colore e forma:Solid
    Peso molecolare:470.32
  • Decloxizine dihydrochloride

    CAS:
    <p>Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.</p>
    Formula:C21H28N2O2·2ClH
    Purezza:99.73%
    Colore e forma:Solid
    Peso molecolare:413.39
  • Histamine Phosphate

    CAS:
    Histamine Phosphate (Histamine acid phosphate) acts directly on the blood vessels to dilate arteries and capillaries mediated by both H 1- and H 2-receptors.
    Formula:C5H9N·2H3O4P
    Purezza:>99.99%
    Colore e forma:White Crystal Powder
    Peso molecolare:307.14
  • Alginic acid

    CAS:
    Alginic acid, a polysaccharide from brown seaweed, has anti-anaphylactic and anti-inflammatory properties and is used in food industry.
    Formula:C14H22O13
    Purezza:≥98%
    Colore e forma:Solid
    Peso molecolare:398.317
  • Betahistine dihydrochloride

    CAS:
    Betahistine dihydrochloride (Betahistine 2HCl) is a histamine analog and H1 receptor agonist that serves as a vasodilator.
    Formula:C8H14Cl2N2
    Purezza:99.22% - 99.88%
    Colore e forma:White To Light Yellow Crystalline Powder
    Peso molecolare:209.12
  • Thonzylamine

    CAS:
    Thonzylamine is an antihistamine/anticholinergic, combined with Clofedanol or Phenylephrine for cold, hay fever, or allergy relief.
    Formula:C16H22N4O
    Purezza:99.45%
    Colore e forma:Solid
    Peso molecolare:286.37
  • Alimemazine hemitartrate

    CAS:
    Alimemazine hemitartrate (Trimeprazine hemitartrate) is aphenothiazine derivative that is used as an antipruritic.
    Formula:C18H22N2SC4H6O6
    Purezza:98.16% - 99.69%
    Colore e forma:Solid
    Peso molecolare:448.53
  • JNJ-5207852

    CAS:
    JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.
    Formula:C20H32N2O
    Purezza:97.19%
    Colore e forma:Solid
    Peso molecolare:316.48
  • LML134

    CAS:
    LML134 (LML-134) is an inverse agonist of Histamine 3 receptor (H3R)(hH3R cAMP and hH3R bdg with Kis of 0.3 nM and 12 nM).
    Formula:C19H29N5O3
    Purezza:99.36%
    Colore e forma:Solid
    Peso molecolare:375.47
  • S 38093 HCl

    CAS:
    S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors.
    Formula:C17H25ClN2O2
    Purezza:97.91%
    Colore e forma:Solid
    Peso molecolare:324.85
  • Hydroxyzine dihydrochloride

    CAS:
    <p>Hydroxyzine dihydrochloride treats allergies, pruritus, anxiety; causes drowsiness; also an antiemetic and sedative.</p>
    Formula:C21H27ClN2O2·2HCl
    Purezza:99.46% - 99.79%
    Colore e forma:Oil Powder
    Peso molecolare:447.83
  • OXOMEMAZINE

    CAS:
    Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in cough research.
    Formula:C18H22N2O2S
    Purezza:99.58%
    Colore e forma:Solid
    Peso molecolare:330.44
  • Ranitidine

    CAS:
    Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors).
    Formula:C13H22N4O3S
    Purezza:99.52%
    Colore e forma:Solid Solid
    Peso molecolare:314.40
  • Bepotastine

    CAS:
    Bepotastine (Bepotastine free base) free base is a histamine 1 (H1) receptor antagonis.
    Formula:C21H25ClN2O3
    Purezza:99.75%
    Colore e forma:Solid
    Peso molecolare:388.89
  • Latrepirdine dihydrochloride

    CAS:
    Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.
    Formula:C21H25N3·2HCl
    Purezza:98.45%
    Colore e forma:Solid
    Peso molecolare:392.37
  • Levocetirizine Dihydrochloride

    CAS:
    <p>Levocetirizine Dihydrochloride is a third-gen antihistamine targeting H1-receptors, treating allergies and urticaria.</p>
    Formula:C21H27Cl3N2O3
    Purezza:99.89%
    Colore e forma:White Or Off-White Crystalline Powder
    Peso molecolare:461.81