Recettore dell'istamina
I recettori dell'istamina sono GPCR che mediano gli effetti dell'istamina, un'ammina biogena coinvolta nelle risposte immunitarie, nella secrezione acida gastrica e nella neurotrasmissione. Esistono quattro sottotipi di recettori dell'istamina (H1, H2, H3 e H4), ognuno dei quali svolge ruoli distinti nelle reazioni allergiche, nella funzione gastrica e nell'attività del sistema nervoso centrale. Gli antagonisti dei recettori dell'istamina sono ampiamente utilizzati nel trattamento delle allergie, delle ulcere peptiche e della cinetosi. Presso CymitQuimica, offriamo una selezione completa di modulatori dei recettori dell'istamina di alta qualità per supportare la tua ricerca in immunologia, gastroenterologia e neurofarmacologia.
Trovati 385 prodotti di "Recettore dell'istamina"
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Triprolidine hydrochloride
CAS:Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.Formula:C19H23ClN2Colore e forma:SolidPeso molecolare:314.852Triprolidine
CAS:Triprolidine: oral H1 receptor blocker with motor/sensory spinal effects, for allergy research.Formula:C19H22N2Colore e forma:SolidPeso molecolare:278.39GSK189254A
CAS:GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).Formula:C21H25N3O2Purezza:98.71% - 99.858%Colore e forma:SolidPeso molecolare:351.44Ref: TM-TQ0066
1mg52,00€5mg88,00€10mg120,00€25mg216,00€50mg350,00€100mg505,00€200mg727,00€1mL*10mM (DMSO)67,00€Osthole
CAS:Osthole (Osthol), a potential inhibitor of histamine H1 receptor, has been shown to stimulate osteoblast proliferation and differentiation.Formula:C15H16O3Purezza:99.93% - 99.96%Colore e forma:Fine White PowderPeso molecolare:244.29Betazole
CAS:Betazole, an oral H2 receptor agonist, stimulates gastric acid and raises bile duct pressure, used for gastric secretory testing.Formula:C5H9N3Colore e forma:SolidPeso molecolare:111.15Betazole dihydrochloride
CAS:<p>Betazole dihydrochloride (Betazole hydrochloride) is an agonist of H2 receptor.</p>Formula:C5H11Cl2N3Purezza:99.12%Colore e forma:SolidPeso molecolare:184.067Mequitazine
CAS:Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.Formula:C20H22N2SPurezza:99.98%Colore e forma:SolidPeso molecolare:322.47Ciproxifan maleate
CAS:<p>Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity</p>Formula:C20H22N2O6Purezza:99.39%Colore e forma:SolidPeso molecolare:386.4Epinastine hydrochloride
CAS:Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.Formula:C16H15N3·HClPurezza:99.26% - 99.62%Colore e forma:White SolidPeso molecolare:285.77Mecamylamine hydrochloride
CAS:Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.Formula:C11H22ClNPurezza:99.76% - >99.99%Colore e forma:White SolidPeso molecolare:203.75JNJ-7777120
CAS:JNJ-7777120 is the first potent and selective non-imidazole histamine H4 receptor antagonist, exhibits >1000-fold selectivity over the other histamin receptors.Formula:C14H16ClN3OPurezza:99.83% - 99.96%Colore e forma:SolidPeso molecolare:277.75Chlorcyclizine
CAS:CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.Formula:C18H21ClN2Purezza:98.75%Colore e forma:SolidPeso molecolare:300.83Chlorprothixene
CAS:Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.Formula:C18H18ClNSPurezza:98.77% - 99.756%Colore e forma:Pale Yellow Crystals SolidPeso molecolare:315.86VUF10460
CAS:VUF10460 is a non-imidazole histamine H4 receptor agonist.Formula:C15H19N5Purezza:99.44% - 99.57%Colore e forma:SolidPeso molecolare:269.34Dimaprit dihydrochloride
CAS:Dimaprit dihydrochloride: selective H2 agonist, inhibits nNOS (IC50: 49 μM), boosts gastric acid.Formula:C6H15N3S·2HClPurezza:99.79%Colore e forma:SolidPeso molecolare:234.19Talastine HCl
CAS:Talastine is an antihistamine drug.Formula:C19H22ClN3OPurezza:98%Colore e forma:SolidPeso molecolare:343.86C-Type Natriuretic Peptide (CNP) (1-22), human
CAS:C-Type Natriuretic Peptide (CNP) (1-22), human is the 1-22 fragment of C-Type Natriuretic Peptide.Formula:C93H157N27O28S3Purezza:>99.99%Colore e forma:SolidPeso molecolare:2197.6Ref: TM-TP1187
1mg119,00€5mg414,00€10mg658,00€25mg945,00€50mg1.264,00€100mg1.700,00€200mg2.270,00€500µg88,00€Tiaramide hydrochloride
CAS:Tiaramide hydrochloride (FK-1160) is an anti-inflammatory that blocks mast cell mediators and relaxes smooth muscles.Formula:C15H19Cl2N3O3SPurezza:98.48%Colore e forma:SolidPeso molecolare:392.3Ref: TM-T28972
1mg70,00€5mg137,00€10mg187,00€25mg315,00€50mg472,00€100mg658,00€200mg930,00€1mL*10mM (DMSO)144,00€Tribenoside
CAS:Tribenoside (BG-356) is a vasoprotectant with mild anti-inflammatory, analgesic, and wound healing properties.Formula:C29H34O6Purezza:≥98%Colore e forma:LiquidPeso molecolare:478.58cicloprofen
CAS:cicloprofen is Cell division cycle 7-related protein kinase (human) inhibitor.Formula:C16H14O2Purezza:98.15%Colore e forma:SolidPeso molecolare:238.2812Ref: TM-T8586
1mg62,00€5mg123,00€10mg180,00€25mg298,00€50mg419,00€100mg567,00€200mg752,00€1mL*10mM (DMSO)111,00€Acitazanolast
CAS:<p>Acitazanolast (WP-871) is an anti-allergic drug candidate.</p>Formula:C9H7N5O3Purezza:98.25%Colore e forma:SolidPeso molecolare:233.182-Pyridylethylamine dihydrochloride
CAS:2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.Formula:C7H12Cl2N2Purezza:99.42%Colore e forma:SolidPeso molecolare:195.09Decloxizine
CAS:Decloxizine is a H1 receptor antagonistFormula:C21H28N2O2Purezza:99.53%Colore e forma:White Or Similar To White PowderPeso molecolare:340.46Zotepine
CAS:Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,Formula:C18H18ClNOSPurezza:99.78%Colore e forma:SolidPeso molecolare:331.86Pemirolast
CAS:Pemirolast: oral antiallergic, reduces paclitaxel reactions, inhibits neuropeptides, for asthma and conjunctivitis study.Formula:C10H8N6OColore e forma:SolidPeso molecolare:228.21Clemizole hydrochloride
CAS:Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.Formula:C19H21Cl2N3Purezza:>99.99%Colore e forma:SolidPeso molecolare:362.3Antazoline
CAS:Antazoline has antihistamine and anticholinergic effects.It used to treat a variety of arrhythmias.Formula:C17H19N3Purezza:≥95%Colore e forma:White Crystalline Powder SolidPeso molecolare:265.35Psoralenoside
CAS:Psoralenoside: a compound from Psoralea fruit; has estrogenic, osteoblastic, antitumor, and antibacterial properties.Formula:C17H18O9Purezza:99.03% - 99.49%Colore e forma:SolidPeso molecolare:366.32Ref: TM-TN1008
1mg96,00€2mg139,00€5mg227,00€10mg364,00€25mg600,00€50mg845,00€100mg1.121,00€1mL*10mM (DMSO)235,00€Betahistine EP Impurity C
CAS:Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.Formula:C15H19N3Purezza:≥95%Colore e forma:SolidPeso molecolare:241.33Dioxopromethazine hydrochloride
CAS:Dioxopromethazine is a target-based classification of drug and available in a number of countries worldwide.Formula:C17H20N2O2S·HClPurezza:99.58%Colore e forma:SolidPeso molecolare:352.88Betahistine
CAS:<p>Betahistine treats vertigo and balance issues in Ménière's disease; it's a histamine analog and H1 receptor agonist.</p>Formula:C8H12N2Purezza:99.87% - 99.87%Colore e forma:Yellowish Liquid Liquid LiquidPeso molecolare:136.19Buclizine dihydrochloride
CAS:Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic andFormula:C28H33ClN2·2HClPurezza:98.05%Colore e forma:Off-White PowderPeso molecolare:505.95S 38093
CAS:S 38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).Formula:C17H24N2O2Purezza:99.95%Colore e forma:SolidPeso molecolare:288.38Ref: TM-T4099
2mg38,00€5mg52,00€10mg80,00€25mg131,00€50mg210,00€100mg334,00€200mg467,00€1mL*10mM (DMSO)52,00€Dioxopromethazine
CAS:Dioxopromethazine (Dioxoprothazine) is a drug for the treatment of a cough and expectoration. It also can be used in local anesthesia.Formula:C17H20N2O2SPurezza:98%Colore e forma:SolidPeso molecolare:316.42Carcinine ditrifluoroacetate Acetate
Carcinine ditrifluoroacetate Acetate (β-Alanylhistamine dihydrochloride) is an H3 receptor antagonist.Formula:C14H20F6N4O7Purezza:98.18%Colore e forma:SolidPeso molecolare:470.32Decloxizine dihydrochloride
CAS:<p>Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.</p>Formula:C21H28N2O2·2ClHPurezza:99.73%Colore e forma:SolidPeso molecolare:413.39Histamine Phosphate
CAS:Histamine Phosphate (Histamine acid phosphate) acts directly on the blood vessels to dilate arteries and capillaries mediated by both H 1- and H 2-receptors.Formula:C5H9N·2H3O4PPurezza:>99.99%Colore e forma:White Crystal PowderPeso molecolare:307.14Alginic acid
CAS:Alginic acid, a polysaccharide from brown seaweed, has anti-anaphylactic and anti-inflammatory properties and is used in food industry.Formula:C14H22O13Purezza:≥98%Colore e forma:SolidPeso molecolare:398.317Betahistine dihydrochloride
CAS:Betahistine dihydrochloride (Betahistine 2HCl) is a histamine analog and H1 receptor agonist that serves as a vasodilator.Formula:C8H14Cl2N2Purezza:99.22% - 99.88%Colore e forma:White To Light Yellow Crystalline PowderPeso molecolare:209.12Thonzylamine
CAS:Thonzylamine is an antihistamine/anticholinergic, combined with Clofedanol or Phenylephrine for cold, hay fever, or allergy relief.Formula:C16H22N4OPurezza:99.45%Colore e forma:SolidPeso molecolare:286.37Alimemazine hemitartrate
CAS:Alimemazine hemitartrate (Trimeprazine hemitartrate) is aphenothiazine derivative that is used as an antipruritic.Formula:C18H22N2SC4H6O6Purezza:98.16% - 99.69%Colore e forma:SolidPeso molecolare:448.53JNJ-5207852
CAS:JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.Formula:C20H32N2OPurezza:97.19%Colore e forma:SolidPeso molecolare:316.48LML134
CAS:LML134 (LML-134) is an inverse agonist of Histamine 3 receptor (H3R)(hH3R cAMP and hH3R bdg with Kis of 0.3 nM and 12 nM).Formula:C19H29N5O3Purezza:99.36%Colore e forma:SolidPeso molecolare:375.47Ref: TM-T8514
1mg37,00€5mg82,00€10mg118,00€25mg215,00€50mg316,00€100mg472,00€200mg633,00€1mL*10mM (DMSO)90,00€S 38093 HCl
CAS:S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors.Formula:C17H25ClN2O2Purezza:97.91%Colore e forma:SolidPeso molecolare:324.85Ref: TM-T4087
1mg39,00€5mg74,00€10mg97,00€25mg167,00€50mg239,00€100mg340,00€200mg460,00€1mL*10mM (DMSO)74,00€Hydroxyzine dihydrochloride
CAS:<p>Hydroxyzine dihydrochloride treats allergies, pruritus, anxiety; causes drowsiness; also an antiemetic and sedative.</p>Formula:C21H27ClN2O2·2HClPurezza:99.46% - 99.79%Colore e forma:Oil PowderPeso molecolare:447.83OXOMEMAZINE
CAS:Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in cough research.Formula:C18H22N2O2SPurezza:99.58%Colore e forma:SolidPeso molecolare:330.44Ranitidine
CAS:Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors).Formula:C13H22N4O3SPurezza:99.52%Colore e forma:Solid SolidPeso molecolare:314.40Bepotastine
CAS:Bepotastine (Bepotastine free base) free base is a histamine 1 (H1) receptor antagonis.Formula:C21H25ClN2O3Purezza:99.75%Colore e forma:SolidPeso molecolare:388.89Ref: TM-T7893
2mg37,00€5mg52,00€10mg82,00€25mg149,00€50mg216,00€100mg329,00€200mg490,00€1mL*10mM (DMSO)59,00€Latrepirdine dihydrochloride
CAS:Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.Formula:C21H25N3·2HClPurezza:98.45%Colore e forma:SolidPeso molecolare:392.37Levocetirizine Dihydrochloride
CAS:<p>Levocetirizine Dihydrochloride is a third-gen antihistamine targeting H1-receptors, treating allergies and urticaria.</p>Formula:C21H27Cl3N2O3Purezza:99.89%Colore e forma:White Or Off-White Crystalline PowderPeso molecolare:461.81
