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Recettore dell'istamina

Recettore dell'istamina

I recettori dell'istamina sono GPCR che mediano gli effetti dell'istamina, un'ammina biogena coinvolta nelle risposte immunitarie, nella secrezione acida gastrica e nella neurotrasmissione. Esistono quattro sottotipi di recettori dell'istamina (H1, H2, H3 e H4), ognuno dei quali svolge ruoli distinti nelle reazioni allergiche, nella funzione gastrica e nell'attività del sistema nervoso centrale. Gli antagonisti dei recettori dell'istamina sono ampiamente utilizzati nel trattamento delle allergie, delle ulcere peptiche e della cinetosi. Presso CymitQuimica, offriamo una selezione completa di modulatori dei recettori dell'istamina di alta qualità per supportare la tua ricerca in immunologia, gastroenterologia e neurofarmacologia.

Trovati 385 prodotti di "Recettore dell'istamina"

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  • Bamirastine
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    Bamirastine

    CAS:
    Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect on
    Formula:C31H37N5O3
    Purezza:96.68%
    Colore e forma:Solid
    Peso molecolare:527.66

    Ref: TM-T13566

  • CP-66948
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    CP-66948

    CAS:
    CP-66948 is a potent histamine H2 receptor antagonist with inhibitory effect on gastric acid secretion and can be used to protect gastric and intestinal mucosa.
    Formula:C13H20N6S
    Purezza:99.14%
    Colore e forma:Solid
    Peso molecolare:292.4

    Ref: TM-T15005

  • PF-03654764
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    PF-03654764

    CAS:
    PF-03654764, an oral H3 receptor blocker, Ki: human 1.2 nM, rat 7.9 nM, used with Fexofenadine for allergic rhinitis.
    Formula:C20H28F2N2O
    Purezza:>99.99%
    Colore e forma:Solid
    Peso molecolare:350.45

    Ref: TM-T61213

  • Lavoltidine
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    Lavoltidine

    CAS:
    Lavoltidine (Loxtidine) is potent and selective H2 receptor antagonist, oral and irreversible,inhibits gastric acid secretion, gastroesophageal reflux disease.
    Formula:C19H29N5O2
    Purezza:98.30% - 98.36%
    Colore e forma:Solid
    Peso molecolare:359.47

    Ref: TM-T15722

  • H3R-IN-1 Hydrochloride
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    H3R-IN-1 Hydrochloride

    CAS:
    H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .
    Formula:C19H24ClN3O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:377.86

    Ref: TM-T11531

  • Propiomazine HCl
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    Propiomazine HCl

    CAS:
    Propiomazine HCl is an analgesia adjunct.
    Formula:C20H25ClN2OS
    Colore e forma:Solid
    Peso molecolare:376.94

    Ref: TM-T34152L

  • Vapitadine dihydrochloride
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    Vapitadine dihydrochloride

    CAS:
    Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on histamine H1.
    Formula:C17H22Cl2N4O
    Purezza:98.28% - 99.30%
    Colore e forma:Solid
    Peso molecolare:369.29

    Ref: TM-T29096

  • JNJ 10191584 maleate
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    JNJ 10191584 maleate

    CAS:
    JNJ 10191584 maleate (VUF6002 maleate) is an orally active and selective antagonist of H4 receptor (Ki = 26 nM).
    Formula:C17H19ClN4O5
    Purezza:99.37%
    Colore e forma:Solid
    Peso molecolare:394.81

    Ref: TM-T22879

  • Azatadine
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    Azatadine

    CAS:
    Azatadine is histamine and cholinergic inhibitor (IC50: 6.5 nM and 10 nM, respectively).
    Formula:C20H22N2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:290.4

    Ref: TM-T22593

  • Impromidine
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    Impromidine

    CAS:
    Impromidine is a highly potent and specific agonist of the histamine H2 receptor.
    Formula:C14H23N7S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:321.44

    Ref: TM-T24162

  • VUF14862
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    VUF14862

    CAS:
    VUF14862 is a robust and fatigue-resistant photoswitchable GPCR antagonist.
    Formula:C26H32N4O2
    Colore e forma:Solid
    Peso molecolare:432.56

    Ref: TM-T69775

  • Sch 44643
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    Sch 44643

    CAS:
    Sch 44643 is an antagonist of platelet activating factor with oral activity.
    Formula:C25H22ClN3O2
    Colore e forma:Solid
    Peso molecolare:431.91

    Ref: TM-T28720

  • UR-PI376
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    UR-PI376

    CAS:
    UR-PI376 is a selective histamine H4 receptor agonist with low H1/H2 activity and moderate H3 affinity.
    Formula:C17H22N6S
    Colore e forma:Solid
    Peso molecolare:342.46

    Ref: TM-T35003

  • Brl 22321
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    Brl 22321

    CAS:
    Brl 22321 is a mast cell stabilizer.
    Formula:C12H9N3O2
    Colore e forma:Solid
    Peso molecolare:227.22

    Ref: TM-T30587

  • BL 6341A
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    BL 6341A

    CAS:
    BL 6341A is related to Tumor data and H2-antagonists or anti-histamins
    Formula:C9H14N8OS3
    Colore e forma:Solid
    Peso molecolare:346.46

    Ref: TM-T68703

  • (R)-Azelastine
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    (R)-Azelastine

    CAS:
    (R)-Azelastine, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.
    Formula:C22H24ClN3O
    Colore e forma:Solid
    Peso molecolare:381.9

    Ref: TM-T70675

  • Aceprometazine
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    Aceprometazine

    CAS:
    Aceprometazine (1664CB) is an antipsychotic which is orally active. Aceprometazine can be used in psychiatric disorders research, for example, depression [1].
    Formula:C19H22N2OS
    Colore e forma:Solid
    Peso molecolare:326.46

    Ref: TM-T60913

  • Noberastine maleate
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    Noberastine maleate

    CAS:
    Noberastine maleate, a fast-acting furan-derived H1 antagonist, peaks at 4 hours with minimal CNS effects and maximal efficacy at 30 mg/day.
    Formula:C25H29N5O9
    Colore e forma:Solid
    Peso molecolare:543.53

    Ref: TM-T71425

  • ROS 234 dioxalate
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    ROS 234 dioxalate

    CAS:
    ROS 234 dioxalate is a potent antagonist of H3(pKB of 9.46 for Guinea-pig ileum H3-receptor)
    Formula:C17H19N5O8
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:421.37

    Ref: TM-T12756

  • Fenspiride-d5
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    Fenspiride-d5

    CAS:
    Fenspiride-d5: internal standard for GC/LC-MS quantification, H1 antagonist, NSAID, anti-inflammatory, selective PDE4,5,3 inhibitor.
    Formula:C15H15D5N2O2
    Colore e forma:Solid
    Peso molecolare:265.36

    Ref: TM-T71141