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Recettore dell'istamina

Recettore dell'istamina

I recettori dell'istamina sono GPCR che mediano gli effetti dell'istamina, un'ammina biogena coinvolta nelle risposte immunitarie, nella secrezione acida gastrica e nella neurotrasmissione. Esistono quattro sottotipi di recettori dell'istamina (H1, H2, H3 e H4), ognuno dei quali svolge ruoli distinti nelle reazioni allergiche, nella funzione gastrica e nell'attività del sistema nervoso centrale. Gli antagonisti dei recettori dell'istamina sono ampiamente utilizzati nel trattamento delle allergie, delle ulcere peptiche e della cinetosi. Presso CymitQuimica, offriamo una selezione completa di modulatori dei recettori dell'istamina di alta qualità per supportare la tua ricerca in immunologia, gastroenterologia e neurofarmacologia.

Trovati 385 prodotti di "Recettore dell'istamina"

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  • GSK-239512
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    GSK-239512

    CAS:
    GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.
    Formula:C23H27N3O2
    Purezza:99.62% - 99.74%
    Colore e forma:Solid
    Peso molecolare:377.48

    Ref: TM-T27462

  • S-1-Propenyl-L-cysteine
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    S-1-Propenyl-L-cysteine

    CAS:
    S-1-Propenyl-L-cysteine, a stereoisomer of S-allyl-l-cysteine, exhibits immunomodulatory effects and has been shown to decrease blood pressure in hypertensive
    Formula:C6H11NO2S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:161.22

    Ref: TM-T12789

  • Dacemazine
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    Dacemazine

    CAS:
    Dacemazine is used to treat depression.
    Formula:C16H16N2OS
    Colore e forma:Solid
    Peso molecolare:284.38

    Ref: TM-T31181

  • VUF14738
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    VUF14738

    CAS:
    VUF14738 is a robust and fatigue-resistant photoswitchable GPCR antagonist.
    Formula:C25H32N4O2
    Colore e forma:Solid
    Peso molecolare:420.55

    Ref: TM-T69774

  • Nedocromil
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    Nedocromil

    CAS:
    Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).
    Formula:C19H17NO7
    Purezza:95% - 97.34%
    Colore e forma:Solid
    Peso molecolare:371.34

    Ref: TM-T16280

  • Dothiepin HCl
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    Dothiepin HCl

    CAS:
    Dothiepin HCl: TCA, SNRI, with antihistamine, antiadrenergic, anticholinergic, and sodium block properties.
    Formula:C19H22ClNS
    Colore e forma:Solid
    Peso molecolare:331.9

    Ref: TM-T69579

  • FR-A 19
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    FR-A 19

    CAS:
    FR-A 19: Histamine H2 agonist, nanomolar inhibition of basophil histamine release; potent anti-allergic.
    Formula:C25H34Cl3F2N5
    Colore e forma:Solid
    Peso molecolare:548.93

    Ref: TM-T27388

  • KY 234
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    KY 234

    CAS:
    KY 234 is a thromboxane synthetase antagonist.
    Formula:C33H35N5O2
    Colore e forma:Solid
    Peso molecolare:533.676

    Ref: TM-T70241

  • (S)-Azelastine
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    (S)-Azelastine

    CAS:
    (S)-Azelastine is an antihistamine reducing receptors H1R, M1R, M3R, and inhibiting HNEpC cell growth.
    Formula:C22H24ClN3O
    Colore e forma:Solid
    Peso molecolare:381.9

    Ref: TM-T70674

  • VUF 8328
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    VUF 8328

    CAS:
    VUF 8328 is an agonist of histamine H(3) receptor.
    Formula:C7H12N4S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:184.26

    Ref: TM-T29145

  • ReN-1869
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    ReN-1869

    CAS:
    ReN-1869 is a novel selective histamine H(1) receptor antagonist with anti-neurogenic pain and anti-inflammatory activity for the study of neurological diseases
    Formula:C24H27NO2
    Purezza:99.83% - 99.98%
    Colore e forma:Solid
    Peso molecolare:361.48

    Ref: TM-T28516

  • Immethridine dihydrobromide
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    Immethridine dihydrobromide

    CAS:
    Immethridine dihydrobromide is a histamine H3 receptor agonist.
    Formula:C9H11Br2N3
    Purezza:97.61% - 98.14%
    Colore e forma:Solid
    Peso molecolare:321.01

    Ref: TM-T22864

  • Proxyfan
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    Proxyfan

    CAS:
    Proxyfan is a high-affinity protean antagonist/agonist of H3 receptors from full agonist to full inverse agonist, depending on given tissue or brain region.
    Formula:C13H16N2O
    Purezza:99.68%
    Colore e forma:Solid
    Peso molecolare:216.28

    Ref: TM-T23190

  • DF-1111301
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    DF-1111301

    CAS:
    DF-1111301 is a novel anti-allergic compound with anti-histamine H1 and anti-PAF activity.
    Formula:C15H25Cl2N3O
    Purezza:99.17%
    Colore e forma:Solid
    Peso molecolare:334.29

    Ref: TM-T27159

  • Noberastine
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    Noberastine

    CAS:
    Noberastine (R 64947) is a novel histamine H1 antagonist with potent and specific peripheral antihistamine activity.
    Formula:C17H21N5O
    Purezza:99.72% - >99.99%
    Colore e forma:Solid
    Peso molecolare:311.38

    Ref: TM-T25875

  • KP136
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    KP136

    CAS:
    KP136 is an orally effective antiallergic compound (IC50: 76.1 μg/mL for histamine release and 63 ug/mL for degranulation).
    Formula:C16H18N4O3
    Purezza:98.3% - 98.61%
    Colore e forma:Solid
    Peso molecolare:314.34

    Ref: TM-T15666

  • JZP-361
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    JZP-361

    CAS:
    JZP-361: selective MAGL inhibitor (IC50 = 46 nM); weaker on FAAH, hABHD6; anti-histamine; for asthma research.
    Formula:C22H20ClN5O
    Purezza:99.82%
    Colore e forma:Solid
    Peso molecolare:405.88

    Ref: TM-T27703

  • Pitolisant
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    Pitolisant

    CAS:
    Pitolisant is a potent and selective nonimidazole inverse agonist that acts on the recombinant human histamine H3 receptor with Ki of 0.16 nM.
    Formula:C17H26ClNO
    Purezza:99.84%
    Colore e forma:Solid
    Peso molecolare:295.85

    Ref: TM-T60636

  • KSK94
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    KSK94

    CAS:
    KSK94 is an H3 receptor antagonist that inhibits sigma-2 receptors , with a Ki value of 75.2 nM, and can be used to study injurious pain.
    Formula:C25H26N4O
    Purezza:99.60%
    Colore e forma:Solid
    Peso molecolare:398.5

    Ref: TM-T79500

  • Impromidine hydrochloride
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    Impromidine hydrochloride

    CAS:
    <p>Impromidine hydrochloride is a very potent and specific histamine H2 receptor agonist for conducting cardiovascular studies.</p>
    Formula:C14H26Cl3N7S
    Purezza:99.82%
    Colore e forma:Solid
    Peso molecolare:430.83

    Ref: TM-T68921