Recettore degli oppioidi
I recettori degli oppioidi sono un gruppo di recettori accoppiati alle proteine G che mediano gli effetti degli oppioidi endogeni ed esogeni. Questi recettori svolgono un ruolo centrale nella modulazione del dolore, nella regolazione dell'umore e nei comportamenti di dipendenza. Gli agonisti e antagonisti dei recettori degli oppioidi sono ampiamente utilizzati nella gestione del dolore e nel trattamento delle dipendenze, nonché nella ricerca sui disturbi neurologici e psichiatrici. Presso CymitQuimica, offriamo una selezione completa di modulatori dei recettori degli oppioidi di alta qualità per supportare la tua ricerca in neurobiologia, gestione del dolore e terapia delle dipendenze.
Trovati 326 prodotti di "Recettore degli oppioidi"
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Loperamide hydrochloride
CAS:Loperamide hydrochloride (ADL 2-1294) is a synthetic, piperidine derivative and opioid agonist with antidiarrheal activity.Formula:C29H34Cl2N2O2Purezza:99.91% - >99.99%Colore e forma:Crystals Practically Insoluble In WaterPeso molecolare:513.50BTRX-335140
CAS:<p>BTRX-335140 (CYM-53093) is a potent and selective orally active κ-opioid receptor (KOR) antagonist with antagonistic activity.Cost-effective and quality-assured.</p>Formula:C25H32FN5O2Purezza:98% - 99.89%Colore e forma:SolidPeso molecolare:453.55Ref: TM-T14835
1mg105,00€2mg155,00€5mg250,00€10mg406,00€25mg840,00€50mg1.378,00€100mg1.882,00€200mg2.632,00€Moguisteine
CAS:Moguisteine (BBR-2173) is a new-type peripheral non-narcotic antitussive drug.Formula:C16H21NO5SPurezza:99.98%Colore e forma:SolidPeso molecolare:339.41Meptazinol hydrochloride
CAS:Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic antagonist with analgesic properties.Formula:C15H23NO·HClPurezza:99.75%Colore e forma:White SolidPeso molecolare:269.81Matrine
CAS:Matrine (Vegard), an alkaloid isolated from the Sophora genus, acts as a kappa opioid receptor agonist.Formula:C15H24N2OPurezza:99.77% - >99.99%Colore e forma:SolidPeso molecolare:248.36Apitegromab
CAS:Apitegromab (SRK-015) is a new myostatin inhibitor, an antibody targeting myostatin precursor, which can be used to study neuromuscular diseases includingPurezza:97.59% (SDS-PAGE); 99.78% (SEC-HPLC) - >95.0% (SDS-PAGE); 99.62% (SEC-HPLC)Colore e forma:LiquidPeso molecolare:145.06 kDaTrimebutine maleate
CAS:<p>Trimebutine maleate (Polibutin) is a weak mu-opioid agonist and has antimuscarinic effects.</p>Formula:C26H33NO9Purezza:99.76% - 99.98%Colore e forma:White SolidPeso molecolare:503.55Alvimopan
CAS:<p>Alvimopan is a potent opioid antagonist targeting gut receptors to reverse opioid effects on motility.</p>Formula:C25H32N2O4Purezza:99.47% - 99.78%Colore e forma:SolidPeso molecolare:424.53Samidorphan HCl
CAS:<p>Samidorphan HCl is an orally active and highly potent modulator of the opioid system that binds to μ‐opioid, κ‐opioid, and delta-opioid receptors.</p>Formula:C21H27ClN2O4Purezza:96.79% - 97.85%Colore e forma:SoildPeso molecolare:406.9Sinomenine hydrochloride
CAS:Sinomenine hydrochloride (Kukoline hydrochloride) is extracted from Sinomenium Acutum Rehderett Wilson.Formula:C19H24ClNO4Purezza:99.43%Colore e forma:SolidPeso molecolare:365.85Naltrexone hydrochloride
CAS:<p>Naltrexone hydrochloride (Naltrexone HCl) is a synthetic opioid antagonist used in the prevention of relapse of opiate addiction and alcoholism.</p>Formula:C20H24ClNO4Purezza:98.72% - 99.65%Colore e forma:White Crystalline PowderPeso molecolare:377.862ZT 52656A hydrochloride
CAS:ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or alleviation of pain in the eye.Formula:C19H26ClF3N2OPurezza:98.78%Colore e forma:SolidPeso molecolare:390.87LY2940094
CAS:LY2940094 (LY-2940094) decreases ethanol self-administration in animal models.Formula:C22H23ClF2N4O2SPurezza:99.4%Colore e forma:SolidPeso molecolare:480.96Ref: TM-T15799
1mg81,00€2mg106,00€5mg163,00€10mg274,00€25mg542,00€50mg778,00€100mg1.074,00€1mL*10mM (DMSO)180,00€CP 866087
CAS:CP 866087 is an opioid receptor antagonist for the study of female sexual dysfunction.Formula:C24H30N2O3SPurezza:99.22% - 99.74%Colore e forma:SolidPeso molecolare:426.57Axelopran sulfate
CAS:Axelopran sulfate is used in Oral Therapies for Opioid-induced Bowel Dysfunction in Patients with Chronic Noncancer Pain.Formula:C26H41N3O8SColore e forma:SolidPeso molecolare:555.68SB 205607 dihydrobromide
CAS:non-peptide δ1 opioid receptor agonistFormula:C23H24N2OPurezza:98%Colore e forma:SolidPeso molecolare:344.45β-Lipotropin (61-69)
CAS:β-Lipotropin (61-69) is a potent opioid agonist [1] [2] .Formula:C45H66N10O15SPeso molecolare:1019.13PL-017 TFA
PL-017 TFA: μ opioid agonist, IC50 5.5 nM, long-lasting analgesia in rats.Formula:C31H38F3N5O7Peso molecolare:649.66Acetalin-3
CAS:Acetalin-3 (Ac-RFMWMT-NH2) is a hexapeptide that acts as a μ opioid receptor antagonist, displaying high affinity for μ and κ3 opioid receptors, weak affinity for κ1 receptors, and no affinity for κ2 receptors [1].Formula:C42H61N11O8S2Peso molecolare:912.13Neuropeptide AF (human) acetate
<p>Neuropeptide AF (human) acetate (Neuropeptide AF (human) acetate (192387-38-5 Free base)) is an anti-opioid neuropeptide, a Neuropeptide AF (human) derivative,</p>Purezza:99.89%Colore e forma:Soild[(pF)Phe4]Nociceptin(1-13)NH2 acetate
<p>[(pF)Phe4]Nociceptin(1-13)NH2 acetate is a selective agonist of NOP receptor with a pKi of 10.68 and a pEC50 of 9.31.</p>Formula:C63H103FN22O17Purezza:98.03%Colore e forma:SolidPeso molecolare:1459.63MOR agonist-4
MOR agonist-4 (2d), having an EC50 of 11 nM, is a G protein-biased agonist of the Kappa opioid receptor (KOR). This compound features a triazole-based, electron-withdrawing CF3 group and a bias factor of 38. MOR agonist-4 is utilized for antipruritic and analgesic applications.Bilaid C
CAS:Bilaid C: Tetrapeptide μ-opioid agonist from Penicillium (Ki=210 nM), inhibits cAMP (77% at 10 μM), induces Kir currents (EC50=4.2 μM).Formula:C28H38N4O6Peso molecolare:526.62K-Opioid receptor agonist-1
CAS:K-Opioid receptor agonist-1 (Compound 5a) acts as an agonist for the κ-Opioid receptor, exhibiting a K_i of 0.25 nM and an EC_50 of 2 nM. This compound is capable of crossing the blood-brain barrier (BBB), evidenced by brain/plasma ratios ranging from 0.50 to 0.65. Additionally, K-Opioid receptor agonist-1 demonstrates anti-inflammatory effects in dermatitis models induced by either Arachidonic acid or oxazolidinone.Formula:C22H29Cl2N3O3Peso molecolare:454.39[D-Ala2]-Met-Enkephalinamide
CAS:[D-Ala2]-Met-Enkephalinamide: potent opioid, reduces bile flow centrally, analgesic.Formula:C28H38N6O6SPeso molecolare:586.7BPRMU191
CAS:BPRMU191 is a distinct mu-opioid receptor (MOR) modulator with an EC50 of 2.17 μM in FLIPR Ca2+ assays conducted on CHO-K1/MOR/Gα15 cells. Additionally, BPRMU191 interacts with MOR in the presence of naloxone.Formula:C17H14FNO3SPeso molecolare:331.36Frakefamide TFA
Frakefamide TFA: potent, peripherally active μ-opioid agonist; doesn't cross blood-brain barrier.Formula:C32H35F4N5O7Colore e forma:SolidPeso molecolare:677.64DPDPE
CAS:DPDPE is selective δ-opioid receptor agonist peptide.Formula:C30H39N5O7S2Purezza:98%Colore e forma:SolidPeso molecolare:645.79[Met5]-Enkephalin, amide
CAS:[Met5]-Enkephalin, amide activates δ and ζ opioid receptors; has multiple forms and varying plasma levels.Formula:C27H36N6O6SPurezza:98%Colore e forma:SolidPeso molecolare:572.68Helianorphin-19
Helianorphin-19: Potent KOR agonist (Ki=25 nM; EC50=45 nM), 200x selective over μ/δ receptors, effective in mouse pain model, non-sedative.Colore e forma:LiquidEnkephalin-met, ala(2)-
CAS:Enkephalin-met, ala(2)- is a synthetic analog of methionine enkephalin.Formula:C28H37N5O7SPeso molecolare:587.69Acetalin-2
CAS:Acetalin-2, an opioid peptide with the sequence Ac-Arg-Phe-Met-Trp-Met-Arg-NH2, selectively binds to [3 H]DAMGO with a Ki value of 93.3 nM [1].Formula:C44H66N14O7S2Peso molecolare:967.21Dafphedyn
CAS:Dafphedyn (DAFPHEDYN), a potent endorphin 1-13 analog, induces diuresis and analgesia in rats via IV.Formula:C76H124F5N25O14Colore e forma:SolidPeso molecolare:1706.95BPR1M97
CAS:BPR1M97 is a mu opioid receptor (MOP) and neuropeptide-orphin FQ (NOP) receptor agonist with blood-brain barrier permeability and potency, with Kis values of 1.Formula:C18H18Cl2N2OPurezza:98.78% - 99.95%Colore e forma:SolidPeso molecolare:349.25D-Ala-Gly-Phe-Met-NH2 monoacetate
CAS:D-Ala-Gly-Phe-Met-NH2 monoacetate, an opioid peptide, serves as a potent agonist for the opiate δ-receptor [1].Formula:C21H33N5O6SPeso molecolare:483.58UFP-101 acetate
<p>UFP-101 acetate is a selective and competitive antagonist of the NOP receptor (pKi = 10.24) with >3000-fold selectivity over δ, μ, and κ opioid receptors.</p>Formula:C84H142N32O23Purezza:95.92%Colore e forma:SolidPeso molecolare:1968.23Ac-RYYRWK-NH2 TFA
CAS:Ac-RYYRWK-NH2: potent, specific NOP receptor partial agonist with 0.071 nM affinity; no affinity for μ/κ/δ-opioid receptors.Formula:C51H70F3N15O11Colore e forma:SolidPeso molecolare:1126.21Dynorphin B (1-13)
CAS:Dynorphin B (1-13) acts as an agonist on opioid κ-receptor.Formula:C74H115N21O17Purezza:98%Colore e forma:SolidPeso molecolare:1570.84Biphalin TFA
CAS:Biphalin TFA is an opioid peptide analog that penetrates the blood-brain barrier (BBB) and encompasses two active enkephalin pharmacophores.Formula:C46H56N10O10·xC2HF3O2Purezza:98%Colore e forma:SolidPeso molecolare:909.00 (free base)(N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8)
CAS:E-2078, known chemically as (N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8), is a stable analog of Dynorphin A (1–8) and functions as a kappa opioidFormula:C50H81N15O9Colore e forma:SolidPeso molecolare:1036.27DPI-287
CAS:DPI-287, a selective delta-opioid receptor (DOP) agonist, has a K\(_i\) value of 0.39 nM and is applicable for pain research [1].Formula:C31H39N3O2Peso molecolare:485.66Dynorphin A (1-13) amide
CAS:Dynorphin A (1-13) amide, an endogenous opioid peptide, counteracts the analgesic effects of morphine [1].Formula:C75H127N25O14Peso molecolare:1602.97[Phe1Ψ(CH2-NH)Gly2]Nociceptin(1-13)NH2
CAS:Potent agonist of the nociceptin (ORL1) receptor, demonstrated both in vitro and in vivo.Formula:C61H102N22O14Purezza:98%Colore e forma:SolidPeso molecolare:1367.6MT-7716 free base
CAS:MT-7716: selective NOP agonist, potential in preventing alcohol abuse/relapse.Formula:C27H28N4O2Purezza:98%Colore e forma:SolidPeso molecolare:440.54BAM-22P
CAS:Bovine adrenal medulla docosapeptide (BAM-22P) is a potent opioid agonist, derived from the proenkephalin A gene, which is present in the adrenal medulla.Formula:C130H184N38O31S2Purezza:98%Colore e forma:SolidPeso molecolare:2839.22N-Desmethyl Loperamide
CAS:N-Desmethyl Loperamide is the major metabolite of loperamide. It is also used as the precusor for radiolabelled loperamide.Formula:C28H31ClN2O2Colore e forma:SolidPeso molecolare:463.01Morphiceptin
CAS:Morphiceptin is a synthetic tetrapeptide with morphinelike activities, highly specific for morphine receptors, but not for enkephalin receptors.Formula:C28H35N5O5Peso molecolare:521.61β-Lipotropin (60-65)
CAS:<p>β-Lipotropin (60-65) (β-LPH (60-65)), an opioid agonist, is a significant [1] opioid peptide.</p>Formula:C33H47N9O8SColore e forma:SolidPeso molecolare:729.85KOR agonist 5
KOR agonist 5 (Compound 10a) is both a KOR/MOR modulator, exhibiting agonistic effects on KOR and antagonistic effects on MOR. It effectively blocks morphine-induced antinociception and gastrointestinal motility inhibition. KOR agonist 5 is applicable in research related to substance use disorder (SUD).Formula:C38H38N2O5Colore e forma:SolidPeso molecolare:602.72Clocinnamox mesylate
CAS:Clocinnamox mesylate: irreversible μ-opioid blocker; Ki: 0.7 nM (mouse μ), 1.9 nM (δ), 5.7 nM (κ).Formula:C30H33ClN2O7SColore e forma:SolidPeso molecolare:601.11N-Acetyl-α-Endorphin
CAS:N-Acetyl-α-Endorphin is a chemical compound consisting of α-Endorphin that has been acetylated at the N-terminal.Formula:C79H122N18O27SPurezza:98%Colore e forma:SolidPeso molecolare:1787.98HINT1-IN-1
HINT1-IN-1 (compound 8) is an inhibitor of histidine triad nucleotide-binding protein 1 (HINT1) with a Ki of 1.14 μM. It influences the cross-regulation between μ-opioid receptors (MOR) and NMDA receptors (NMDAR).Formula:C23H24N8O5Colore e forma:SolidPeso molecolare:492.49KOR agonist 4
<p>KOR agonist 4 (compound 39) is an agonist targeting the κ opioid receptor (Kappa Opioid Receptor) and activates G protein signaling. It has an EC50 of 14 nM and an Emax of 83% for binding to GTPγS. This compound demonstrates moderate to high intrinsic clearance in human liver cells and shows selectivity for the κ opioid receptor over the μ (MOR) and δ (DOR) opioid receptors by factors of 60 and 810, respectively. KOR agonist 4 is useful for research into central nervous system (CNS) disorders.</p>Formula:C21H25N3Colore e forma:SolidPeso molecolare:319.44β-Endorphin, equine TFA
β-Endorphin, equine TFA, an endogenous opioid peptide, demonstrates high affinity binding to μ/δ opioid receptors and possesses analgesic properties [1] [2] [3Formula:C156H249F3N42O46SColore e forma:SolidPeso molecolare:3537.96Akuammicine
CAS:Akuammicine, as an indole alkaloid from Catharanthus roseus, can be used in cancer cell eradication.Formula:C20H22N2O2Colore e forma:SolidPeso molecolare:322.408Nociceptin(1-7)
CAS:Bioactive metabolite of nociceptin, antagonist of nociceptin-induced hyperalgesiaFormula:C31H41N7O9Purezza:98%Colore e forma:SolidPeso molecolare:655.709[(pF)Phe4]Nociceptin(1-13)NH2
CAS:<p>Potent, selective OP4 agonist; pKi=10.68, pEC50=9.80. >8000x selectivity vs other opioid receptors; long-lasting in vivo effects.</p>Formula:C61H99FN22O15Purezza:98%Colore e forma:SolidPeso molecolare:1399.6Dermorphin Analog
Dermorphin Analog, a heptapeptide from amphibian skin, binds μ-opioid receptors selectively and strongly.Formula:C44H59N11O10Purezza:98%Colore e forma:SolidPeso molecolare:901.43Dynorphin B (1-13) (TFA)
Dynorphin B (1-13) TFA acts as an agonist on opioid κ-receptor .Formula:C76H116N21F3O19Colore e forma:SolidPeso molecolare:1684.86PL-017
CAS:μ opioid receptor agonist; IC50: 5.5 nM (μ), >10,000 nM (δ). Induces reversible analgesia, catalepsy, hyperthermia in rats.Formula:C29H37N5O5Purezza:98%Colore e forma:SolidPeso molecolare:535.64Nocistatin
CAS:Nocistatin, a neuropeptide, blocks Nociceptin effects and inhibits 5-HT release, acting on an opioid-related receptor.Formula:C32H56N10O12Colore e forma:SolidPeso molecolare:772.85Ro 64-6198
CAS:Ro 64-6198: Nonpeptide, selective NOP agonist, high brain uptake, EC50=25.6 nM, 100x NOP>opioid affinity.Formula:C26H31N3OPurezza:98%Colore e forma:SolidPeso molecolare:401.54Herkinorin
CAS:Herkinorin: μ-opioid agonist with 100x μ-affinity, 50x less κ-affinity than Salvinorin A, from Salvia divinorum. Semi-synthetic from Salvinorin B.Formula:C28H30O8Colore e forma:SolidPeso molecolare:494.53Gluten Exorphin B5
CAS:Gluten exorphin B5 (GE-B5) is a food-derived opioid peptide identified in digests of wheat gluten.Formula:C30H38N6O7Purezza:98%Colore e forma:SolidPeso molecolare:594.66β-Chlornaltrexamine dihydrochloride
CAS:β-Chlornaltrexamine dihydrochloride (β-CNA dihydrochloride) is an effective long-term antagonist of opioid receptors. It efficiently blocks the inhibition of dopamine release mediated by κ opioid receptor agonists. This compound is useful in the research of pain perception mechanisms.Formula:C24H34Cl4N2O3Peso molecolare:540.35ICI 174,864
CAS:Selective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.Formula:C38H53N5O7Purezza:98%Colore e forma:White SolidPeso molecolare:691.87U-54494A hydrochloride
CAS:U-54494A hydrochloride is a benzamide derivative related to kappa opioid receptor agonists. U-54494A hydrochloride has anticonvulsant activity.Formula:C18H25Cl3N2OColore e forma:SolidPeso molecolare:391.76CJ-15208
CAS:<p>CJ-15208: κ-opioid antagonist, IC50: 47 nM kappa, 260 nM mu, 2600 nM delta, reverses asimadoline effects in rabbits (ED50 1.3 µM).</p>Formula:C34H35N5O4Colore e forma:SolidPeso molecolare:577.67UFP-101
CAS:<p>Strong, selective NOP receptor antagonist with pKi=10.24; >3000x selectivity over δ, μ, κ receptors; blocks nociceptin effects.</p>Formula:C82H138N32O21Purezza:98%Colore e forma:SolidPeso molecolare:1908.19[Nphe1]Nociceptin(1-13)NH2
CAS:<p>Competitive nociceptin receptor antagonist with pKi=8.4; no agonist activity; blocks nociceptin effects in vitro/in vivo.</p>Formula:C61H100N22O15Purezza:98%Colore e forma:SolidPeso molecolare:1381.6PIPE-3297
PIPE-3297 (compound 25) is a selective kappa opioid receptor (KOR) agonist that activates the G protein signaling pathway with an EC50 of 1.1 nM and exhibits low β-arrestin-2 recruitment activity (10%). Additionally, PIPE-3297 promotes myelination and has anti-inflammatory properties.Formula:C23H30N2OPeso molecolare:350.23581N-terminally acetylated Endomorphin-1
N-terminally acetylated Endomorphin-1 is a modified Endomorphin-1.Formula:C36H40N6O6Purezza:98%Colore e forma:SolidPeso molecolare:652.74β-Endorphin (rat)
CAS:β-Endorphin (β-EP) is an endogenous opioid neuropeptide with diverse biological activities.Formula:C157H254N42O44SColore e forma:SolidPeso molecolare:3466.07Naldemedine
CAS:Naldemedine (S 297995), developed by Shionogi, is a drug for opioid side effects like constipation. It's well tolerated with minor GI issues.Formula:C32H34N4O6Colore e forma:SolidPeso molecolare:570.64MT-7716 hydrochloride
CAS:MT-7716 hydrochloride is a selective agonist of non-peptide nociceptin receptor (NOP)Formula:C27H29ClN4O2Purezza:98%Colore e forma:SolidPeso molecolare:477Neuropeptide AF (human)
CAS:Neuropeptide AF (93-110), Human is an endogenous antiopioid peptide.Formula:C90H132N26O25Purezza:98%Colore e forma:SolidPeso molecolare:1978.17CTAP
CAS:Potent μ opioid antagonist, IC50 3.5 nM, 1200x selectivity over δ and somatostatin, brain-penetrant, active in vivo.Formula:C51H69N13O11S2Purezza:98%Colore e forma:White Solid/PowderPeso molecolare:1104.32Dermorphin
CAS:<p>Dermorphin is agonist of μ-opioid receptor (MOR) agonist.</p>Formula:C40H50N8O10Purezza:98.82%Colore e forma:SolidPeso molecolare:802.87[DAla2, DArg6] Dynorphin A, (1-13) (porcine)
CAS:'[DAla2, DArg6] Dynorphin A (1-13) porcine is a potent opioid peptide resistant to enzymatic degradation.'Formula:C76H128N24O15Colore e forma:SolidPeso molecolare:1617.98β-Naltrexamine dihydrochloride
CAS:β-Naltrexamine dihydrochloride is an orally administered, irreversible opioid receptor antagonist. Its derivatives exhibit optimised subtype selectivity and can be used for pain research.Formula:C20H28Cl2N2O3Purezza:95.98%Colore e forma:SoildPeso molecolare:415.35Ac-RYYRIK-NH2
CAS:NOP site high affinity ligand (Ki=1.5 nM); blocks nociceptin effects in rat brain/heart; agonist in vivo, reduces mouse movement.Formula:C44H70N14O9Purezza:98%Colore e forma:SolidPeso molecolare:939.12CTOP
CAS:Potent μ-receptor antagonist, Ki=0.96nM, ineffective at δ (>10,000nM). Alters behavior in vivo, boosts K+ currents in rat neurons in vitro, μ-independent.Formula:C50H67N11O11S2Purezza:98%Colore e forma:SolidPeso molecolare:1062.28Nociceptin (1-13), amide
CAS:Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrainFormula:C61H100N22O15Purezza:98%Colore e forma:SolidPeso molecolare:1381.59Cebranopadol hemicitrate
CAS:Cebranopadol hemicitrate is a NOP and opioid receptor agonist that targets human NOP, MOP, KOP, and δ-opioid peptide (DOP) receptors, with Ki/EC50 values of 0.9 nM/13 nM, 0.7 nM/1.2 nM, 2.6 nM/17 nM, and 18 nM/110 nM, respectively. It is used in studies of acute and chronic pain.Colore e forma:Solid[DPro10] Dynorphin A (1-11)acetate,porcine
[DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value of 0.13 nM.Formula:C65H107N21O15Purezza:99.59%Colore e forma:SoildPeso molecolare:1422.7α-Neoendorphin (1-8)
CAS:α-Neoendorphin (1-8) is a 8-amino acid peptide derived from the N-terminal of α-Neoendorphin.Formula:C49H70N12O11Purezza:98%Colore e forma:SolidPeso molecolare:1003.15Neurotransmitter Receptor Compound Library
<p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；</p>Colore e forma:Odour Solid[Arg14,Lys15]Nociceptin
CAS:Potent NOP agonist (EC50 = 1 nM), >875x selective vs opioid receptors; outperforms nociceptin in vivo, increases pain perception, reduces movement.Formula:C82H137N31O22Purezza:98%Colore e forma:SolidPeso molecolare:1909.18SNC 80
CAS:SNC 80, a non-peptide δ-opioid agonist (Ki=1.78 nM, IC50=2.73 nM), also targets μ-δ heteromers (EC50=52.8 nM), with analgesic and antidepressant potential.Formula:C28H39N3O2Purezza:99.65%Colore e forma:SolidPeso molecolare:449.63β-Endorphin, equine
CAS:Endorphin Beta is A substance produced in the brain, especially in the pituitary gland, Endorphin Beta blocks the sensation of pain.Formula:C154H248N42O44SPurezza:98%Colore e forma:SolidPeso molecolare:3423.94Orphanin FQ(1-11)
CAS:<p>Nociceptin peptide fragment (1-11) with potent ORL1/KOR-3 receptor agonism (Ki = 55 nM), no opioid receptor affinity, and analgesic in mice.</p>Formula:C49H75N15O14Purezza:98%Colore e forma:SolidPeso molecolare:1098.2TAN67
CAS:<p>TAN67 is the first effective selective non-peptide delta1 opioid receptor.</p>Formula:C23H26Br2N2OColore e forma:SolidPeso molecolare:506.282Boc-ypgflt(O-tbu)
CAS:Boc-ypgflt(O-tbu) is a delta-receptor-selective opioid antagonist.Formula:C44H64N6O11Colore e forma:SolidPeso molecolare:853.01Axelopran
CAS:Axelopran (TD-1211) treats opioid constipation; it's a potent, selective peripheral opioid blocker.Formula:C26H39N3O4Colore e forma:SolidPeso molecolare:457.61[Nphe1]Nociceptin(1-13)NH2 TFA
[Nphe1]Nociceptin(1-13)NH2 is a selective nociceptin receptor antagonist with potential analgesic properties, pKi=8.4, pA2=6.0.Formula:C63H101F3N22O17Colore e forma:SolidPeso molecolare:1495.61(Rac)-SNC80
CAS:(Rac)-SNC80, a racemic δ-opioid agonist (K i 1.78 nM), shows potential for treating various headache disorders.Formula:C28H39N3O2Colore e forma:SolidPeso molecolare:449.63DAMGO (TFA)
CAS:DAMGO is a selective peptide agonist of the µ-opioid receptor .Formula:C28H36F3N5O8Purezza:98%Colore e forma:SolidPeso molecolare:627.61(S,S)-J-113397
CAS:(S,S)-J-113397 is an isomer of J-113397 . J-113397 is an Opioid Receptor antagonist [1] .Formula:C24H37N3O2Colore e forma:SolidPeso molecolare:399.57Ac-RYYRWK-NH2
CAS:Selective NOP receptor partial agonist peptide; Ki=0.71 nM; >4000 nM for μ, δ, κ receptors; boosts food intake in vivo.Formula:C49H69N15O9Purezza:98%Colore e forma:SolidPeso molecolare:1012.17Opioid receptor agonist 1
<p>Opioid receptor agonist1 (Compound 2638-28) is an orally active opioid receptor agonist that shows strong affinity for MOR, DOR, and KOR, with Ki values of 5, 24, and 212 nM, respectively. It exhibits analgesic activity in both the mouse warm water tail-flick model and the acetic acid writhing model.</p>Formula:C32H45N5OColore e forma:SolidPeso molecolare:515.73
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