
Recettore degli oppioidi
I recettori degli oppioidi sono un gruppo di recettori accoppiati alle proteine G che mediano gli effetti degli oppioidi endogeni ed esogeni. Questi recettori svolgono un ruolo centrale nella modulazione del dolore, nella regolazione dell'umore e nei comportamenti di dipendenza. Gli agonisti e antagonisti dei recettori degli oppioidi sono ampiamente utilizzati nella gestione del dolore e nel trattamento delle dipendenze, nonché nella ricerca sui disturbi neurologici e psichiatrici. Presso CymitQuimica, offriamo una selezione completa di modulatori dei recettori degli oppioidi di alta qualità per supportare la tua ricerca in neurobiologia, gestione del dolore e terapia delle dipendenze.
Trovati 328 prodotti per "Recettore degli oppioidi".
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
BTRX-335140
CAS:BTRX-335140 (CYM-53093) is a potent and selective orally active κ-opioid receptor (KOR) antagonist with antagonistic activity.Cost-effective and quality-assured.Formula:C25H32FN5O2Purezza:98% - 99.89%Colore e forma:SolidPeso molecolare:453.55Ref: TM-T14835
1mg100,00€2mg146,00€5mg236,00€1mL*10mM (DMSO)268,00€10mg385,00€25mg797,00€50mg1.305,00€100mg1.783,00€200mg2.493,00€Naltrexone hydrochloride
CAS:Naltrexone hydrochloride (Naltrexone HCl) is a synthetic opioid antagonist used in the prevention of relapse of opiate addiction and alcoholism.Formula:C20H24ClNO4Purezza:98.72% - 99.65%Colore e forma:White Crystalline PowderPeso molecolare:377.862Matrine
CAS:Matrine (Vegard), an alkaloid isolated from the Sophora genus, acts as a kappa opioid receptor agonist.Formula:C15H24N2OPurezza:99.77% - >99.99%Colore e forma:SolidPeso molecolare:248.36Samidorphan HCl
CAS:Samidorphan HCl is an orally active and highly potent modulator of the opioid system that binds to μ‐opioid, κ‐opioid, and delta-opioid receptors.Formula:C21H27ClN2O4Purezza:96.79% - 97.85%Colore e forma:SolidPeso molecolare:406.9Moguisteine
CAS:Moguisteine (BBR-2173) is a new-type peripheral non-narcotic antitussive drug.Formula:C16H21NO5SPurezza:99.98%Colore e forma:SolidPeso molecolare:339.41LY2940094
CAS:LY2940094 (LY-2940094) decreases ethanol self-administration in animal models.Formula:C22H23ClF2N4O2SPurezza:99.4%Colore e forma:SolidPeso molecolare:480.96Ref: TM-T15799
1mg77,00€2mg101,00€5mg155,00€1mL*10mM (DMSO)170,00€10mg259,00€25mg513,00€50mg737,00€100mg1.018,00€Loperamide hydrochloride
CAS:Loperamide hydrochloride (ADL 2-1294) is a synthetic, piperidine derivative and opioid agonist with antidiarrheal activity.Formula:C29H34Cl2N2O2Purezza:99.91% - >99.99%Colore e forma:Crystals Practically Insoluble In WaterPeso molecolare:513.50Apitegromab
CAS:Apitegromab (SRK-015) is a new myostatin inhibitor, an antibody targeting myostatin precursor, which can be used to study neuromuscular diseases includingPurezza:97.59% (SDS-PAGE); 99.78% (SEC-HPLC) - >95.0% (SDS-PAGE); 99.62% (SEC-HPLC)Colore e forma:LiquidPeso molecolare:145.06 kDaMeptazinol hydrochloride
CAS:Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic antagonist with analgesic properties.Formula:C15H23NO·HClPurezza:99.75%Colore e forma:White SolidPeso molecolare:269.81CP 866087
CAS:CP 866087 is an opioid receptor antagonist for the study of female sexual dysfunction.Formula:C24H30N2O3SPurezza:99.22% - 99.74%Colore e forma:SolidPeso molecolare:426.57Alvimopan
CAS:Alvimopan is a potent opioid antagonist targeting gut receptors to reverse opioid effects on motility.Formula:C25H32N2O4Purezza:99.47% - 99.78%Colore e forma:SolidPeso molecolare:424.53Ref: TM-T1242
1mg44,00€2mg57,00€5mg93,00€1mL*10mM (DMSO)94,00€10mg120,00€25mg220,00€50mg356,00€100mg530,00€200mg755,00€Trimebutine maleate
CAS:Trimebutine maleate (Polibutin) is a weak mu-opioid agonist and has antimuscarinic effects.Formula:C26H33NO9Purezza:99.89% - 99.98%Colore e forma:White SolidPeso molecolare:503.55Sinomenine hydrochloride
CAS:Sinomenine hydrochloride (Kukoline hydrochloride) is extracted from Sinomenium Acutum Rehderett Wilson.Formula:C19H24ClNO4Purezza:99.43%Colore e forma:SolidPeso molecolare:365.85ZT 52656A hydrochloride
CAS:ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or alleviation of pain in the eye.Formula:C19H26ClF3N2OPurezza:98.78%Colore e forma:SolidPeso molecolare:390.87Ref: TM-T13414
1mg94,00€5mg222,00€1mL*10mM (DMSO)245,00€10mg356,00€25mg715,00€50mg1.144,00€100mg1.783,00€δ opioid receptor antagonist 1
Compound 6-Cy3, a δ-opioid receptor antagonist, serves as a highly selective fluorescent probe for δ-opioid receptors (DOR), showcasing an affinity (Ki=1.7 nM). This compound is used in the study of pain perception mechanisms.Colore e forma:Odour SolidDermorphin
CAS:Dermorphin is agonist of μ-opioid receptor (MOR) agonist.Formula:C40H50N8O10Purezza:98.82%Colore e forma:SolidPeso molecolare:802.87μ/κ/δ opioid receptor agonist 1
μ/κ/δopioid receptor agonist1 is an agonist for the μ opioid receptor (MOR), κ opioid receptor (KOR), and δ opioid receptor (DOR). It produces potent and long-lasting analgesic effects in the tail flick test through peripheral MOR and KOR activation.Formula:C35H45FN8O8Colore e forma:SolidPeso molecolare:724.33444UFP-101
CAS:Strong, selective NOP receptor antagonist with pKi=10.24; >3000x selectivity over δ, μ, κ receptors; blocks nociceptin effects.
Formula:C82H138N32O21Purezza:98%Colore e forma:SolidPeso molecolare:1908.19DPDPE
CAS:DPDPE is selective δ-opioid receptor agonist peptide.Formula:C30H39N5O7S2Purezza:98%Colore e forma:SolidPeso molecolare:645.79NP-5497-KA
NP-5497-KA is a κ-opioid receptor agonist with oral bioavailability.Formula:C26H39Cl3N4O2Peso molecolare:544.21386

