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Recettore degli oppioidi

Recettore degli oppioidi

I recettori degli oppioidi sono un gruppo di recettori accoppiati alle proteine G che mediano gli effetti degli oppioidi endogeni ed esogeni. Questi recettori svolgono un ruolo centrale nella modulazione del dolore, nella regolazione dell'umore e nei comportamenti di dipendenza. Gli agonisti e antagonisti dei recettori degli oppioidi sono ampiamente utilizzati nella gestione del dolore e nel trattamento delle dipendenze, nonché nella ricerca sui disturbi neurologici e psichiatrici. Presso CymitQuimica, offriamo una selezione completa di modulatori dei recettori degli oppioidi di alta qualità per supportare la tua ricerca in neurobiologia, gestione del dolore e terapia delle dipendenze.

Trovati 328 prodotti per "Recettore degli oppioidi".

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  • BTRX-335140

    CAS:
    BTRX-335140 (CYM-53093) is a potent and selective orally active κ-opioid receptor (KOR) antagonist with antagonistic activity.Cost-effective and quality-assured.
    Formula:C25H32FN5O2
    Purezza:98% - 99.89%
    Colore e forma:Solid
    Peso molecolare:453.55

    Ref: TM-T14835

    1mg
    100,00€
    2mg
    146,00€
    5mg
    236,00€
    1mL*10mM (DMSO)
    268,00€
    10mg
    385,00€
    25mg
    797,00€
    50mg
    1.305,00€
    100mg
    1.783,00€
    200mg
    2.493,00€
  • Naltrexone hydrochloride

    CAS:
    Naltrexone hydrochloride (Naltrexone HCl) is a synthetic opioid antagonist used in the prevention of relapse of opiate addiction and alcoholism.
    Formula:C20H24ClNO4
    Purezza:98.72% - 99.65%
    Colore e forma:White Crystalline Powder
    Peso molecolare:377.862

    Ref: TM-T0963

    25mg
    34,00€
    50mg
    42,00€
    1mL*10mM (DMSO)
    44,00€
    100mg
    52,00€
    500mg
    105,00€
    1g
    155,00€
  • Matrine

    CAS:
    Matrine (Vegard), an alkaloid isolated from the Sophora genus, acts as a kappa opioid receptor agonist.
    Formula:C15H24N2O
    Purezza:99.77% - >99.99%
    Colore e forma:Solid
    Peso molecolare:248.36

    Ref: TM-T2870

    25mg
    40,00€
    1mL*10mM (DMSO)
    50,00€
    50mg
    55,00€
    100mg
    77,00€
    200mg
    111,00€
    500mg
    236,00€
  • Samidorphan HCl

    CAS:
    Samidorphan HCl is an orally active and highly potent modulator of the opioid system that binds to μ‐opioid, κ‐opioid, and delta-opioid receptors.
    Formula:C21H27ClN2O4
    Purezza:96.79% - 97.85%
    Colore e forma:Solid
    Peso molecolare:406.9

    Ref: TM-T67888L

    1mg
    156,00€
    5mg
    371,00€
    10mg
    552,00€
    25mg
    882,00€
    50mg
    1.189,00€
    100mg
    1.603,00€
  • Moguisteine

    CAS:
    Moguisteine (BBR-2173) is a new-type peripheral non-narcotic antitussive drug.
    Formula:C16H21NO5S
    Purezza:99.98%
    Colore e forma:Solid
    Peso molecolare:339.41

    Ref: TM-T1169

    50mg
    33,00€
    1mL*10mM (DMSO)
    33,00€
  • LY2940094

    CAS:
    LY2940094 (LY-2940094) decreases ethanol self-administration in animal models.
    Formula:C22H23ClF2N4O2S
    Purezza:99.4%
    Colore e forma:Solid
    Peso molecolare:480.96

    Ref: TM-T15799

    1mg
    77,00€
    2mg
    101,00€
    5mg
    155,00€
    1mL*10mM (DMSO)
    170,00€
    10mg
    259,00€
    25mg
    513,00€
    50mg
    737,00€
    100mg
    1.018,00€
  • Loperamide hydrochloride

    CAS:
    Loperamide hydrochloride (ADL 2-1294) is a synthetic, piperidine derivative and opioid agonist with antidiarrheal activity.
    Formula:C29H34Cl2N2O2
    Purezza:99.91% - >99.99%
    Colore e forma:Crystals Practically Insoluble In Water
    Peso molecolare:513.50

    Ref: TM-T0209

    50mg
    42,00€
    100mg
    52,00€
    1mL*10mM (DMSO)
    52,00€
    500mg
    80,00€
    1g
    102,00€
  • Apitegromab

    CAS:
    Apitegromab (SRK-015) is a new myostatin inhibitor, an antibody targeting myostatin precursor, which can be used to study neuromuscular diseases including
    Purezza:97.59% (SDS-PAGE); 99.78% (SEC-HPLC) - >95.0% (SDS-PAGE); 99.62% (SEC-HPLC)
    Colore e forma:Liquid
    Peso molecolare:145.06 kDa

    Ref: TM-T77445

    1mg
    152,00€
    5mg
    447,00€
    10mg
    715,00€
    25mg
    1.063,00€
    50mg
    1.423,00€
  • Meptazinol hydrochloride

    CAS:
    Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic antagonist with analgesic properties.
    Formula:C15H23NO·HCl
    Purezza:99.75%
    Colore e forma:White Solid
    Peso molecolare:269.81

    Ref: TM-T0201

    5mg
    46,00€
    10mg
    52,00€
    1mL*10mM (DMSO)
    52,00€
    25mg
    82,00€
    50mg
    110,00€
    100mg
    159,00€
    200mg
    215,00€
  • CP 866087

    CAS:
    CP 866087 is an opioid receptor antagonist for the study of female sexual dysfunction.
    Formula:C24H30N2O3S
    Purezza:99.22% - 99.74%
    Colore e forma:Solid
    Peso molecolare:426.57

    Ref: TM-T31081L

    1mg
    175,00€
    5mg
    434,00€
    10mg
    622,00€
    25mg
    973,00€
    50mg
    1.341,00€
  • Alvimopan

    CAS:
    Alvimopan is a potent opioid antagonist targeting gut receptors to reverse opioid effects on motility.
    Formula:C25H32N2O4
    Purezza:99.47% - 99.78%
    Colore e forma:Solid
    Peso molecolare:424.53

    Ref: TM-T1242

    1mg
    44,00€
    2mg
    57,00€
    5mg
    93,00€
    1mL*10mM (DMSO)
    94,00€
    10mg
    120,00€
    25mg
    220,00€
    50mg
    356,00€
    100mg
    530,00€
    200mg
    755,00€
  • Trimebutine maleate

    CAS:
    Trimebutine maleate (Polibutin) is a weak mu-opioid agonist and has antimuscarinic effects.
    Formula:C26H33NO9
    Purezza:99.89% - 99.98%
    Colore e forma:White Solid
    Peso molecolare:503.55

    Ref: TM-T1197

    1g
    33,00€
    1mL*10mM (DMSO)
    33,00€
  • Sinomenine hydrochloride

    CAS:
    Sinomenine hydrochloride (Kukoline hydrochloride) is extracted from Sinomenium Acutum Rehderett Wilson.
    Formula:C19H24ClNO4
    Purezza:99.43%
    Colore e forma:Solid
    Peso molecolare:365.85

    Ref: TM-T2921

    200mg
    33,00€
    500mg
    49,00€
    1g
    66,00€
  • ZT 52656A hydrochloride

    CAS:
    ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or alleviation of pain in the eye.
    Formula:C19H26ClF3N2O
    Purezza:98.78%
    Colore e forma:Solid
    Peso molecolare:390.87

    Ref: TM-T13414

    1mg
    94,00€
    5mg
    222,00€
    1mL*10mM (DMSO)
    245,00€
    10mg
    356,00€
    25mg
    715,00€
    50mg
    1.144,00€
    100mg
    1.783,00€
  • δ opioid receptor antagonist 1


    Compound 6-Cy3, a δ-opioid receptor antagonist, serves as a highly selective fluorescent probe for δ-opioid receptors (DOR), showcasing an affinity (Ki=1.7 nM). This compound is used in the study of pain perception mechanisms.
    Colore e forma:Odour Solid

    Ref: TM-T89132

    10mg
    Prezzo su richiesta
    50mg
    Prezzo su richiesta
  • Dermorphin

    CAS:
    Dermorphin is agonist of μ-opioid receptor (MOR) agonist.
    Formula:C40H50N8O10
    Purezza:98.82%
    Colore e forma:Solid
    Peso molecolare:802.87

    Ref: TM-T7404

    1mg
    42,00€
  • μ/κ/δ opioid receptor agonist 1


    μ/κ/δopioid receptor agonist1 is an agonist for the μ opioid receptor (MOR), κ opioid receptor (KOR), and δ opioid receptor (DOR). It produces potent and long-lasting analgesic effects in the tail flick test through peripheral MOR and KOR activation.
    Formula:C35H45FN8O8
    Colore e forma:Solid
    Peso molecolare:724.33444

    Ref: TM-TP3501

    10mg
    Prezzo su richiesta
    50mg
    Prezzo su richiesta
  • UFP-101

    CAS:

    Strong, selective NOP receptor antagonist with pKi=10.24; >3000x selectivity over δ, μ, κ receptors; blocks nociceptin effects.

    Formula:C82H138N32O21
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1908.19

    Ref: TM-TP2105

    1mg
    1.549,00€
  • DPDPE

    CAS:
    DPDPE is selective δ-opioid receptor agonist peptide.
    Formula:C30H39N5O7S2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:645.79

    Ref: TM-TP2036

    1mg
    515,00€
  • NP-5497-KA


    NP-5497-KA is a κ-opioid receptor agonist with oral bioavailability.
    Formula:C26H39Cl3N4O2
    Peso molecolare:544.21386

    Ref: TM-T208331

    10mg
    Prezzo su richiesta
    50mg
    Prezzo su richiesta