Recettore degli oppioidi
I recettori degli oppioidi sono un gruppo di recettori accoppiati alle proteine G che mediano gli effetti degli oppioidi endogeni ed esogeni. Questi recettori svolgono un ruolo centrale nella modulazione del dolore, nella regolazione dell'umore e nei comportamenti di dipendenza. Gli agonisti e antagonisti dei recettori degli oppioidi sono ampiamente utilizzati nella gestione del dolore e nel trattamento delle dipendenze, nonché nella ricerca sui disturbi neurologici e psichiatrici. Presso CymitQuimica, offriamo una selezione completa di modulatori dei recettori degli oppioidi di alta qualità per supportare la tua ricerca in neurobiologia, gestione del dolore e terapia delle dipendenze.
Trovati 325 prodotti di "Recettore degli oppioidi"
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Ro 48-6791
CAS:Ro 48-6791, a GABA receptor agonist, is used potentially for anesthesia.Formula:C21H25FN6O2Colore e forma:SolidPeso molecolare:412.46Trap-101 hydrochloride
CAS:nociceptin/orphanin FQ (NOP) receptor antagonistFormula:C24H36ClN3O2Purezza:98%Colore e forma:SolidPeso molecolare:434.02μ opioid receptor agonist 1
CAS:μ opioid receptor agonist 1 (Compound H-1a) is an optically pure oxyheterocyclic substituted pyrroloxypyrazole derivative and an MOR receptor agonist that canFormula:C26H38N4OColore e forma:SolidPeso molecolare:422.61FK 33-824
CAS:FK 33-824, a stable synthetic analog of methionine enkephalin, reversible with naloxone.Formula:C29H41N5O7SPurezza:98%Colore e forma:SolidPeso molecolare:603.73DPI-3290
CAS:DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively) with potentFormula:C30H34FN3O2Purezza:98%Colore e forma:SolidPeso molecolare:487.61N-Benzylnaltrindole hydrochloride
CAS:δ2 opioid receptor antagonistFormula:C33H33ClN2O3Purezza:98%Colore e forma:SolidPeso molecolare:541.08Salvinorin A Carbamate
CAS:Salvinorin A carbamate, a potent κ-opioid receptor (KOR) full agonist, exhibits nearly the same potency as salvinorin A, with EC50 values of 6.2 and 4.5 nM, respectively, for activating the human KOR to augment the binding of [35S]GTPγS. Enhancing biological stability, the addition of a carbamate group to salvinorin A reduces deacetylation.Formula:C22H27NO8Colore e forma:SolidPeso molecolare:433.457Naloxonazine dihydrochloride
CAS:μ1 receptor antagonistFormula:C38H43ClN4O6Purezza:98%Colore e forma:SolidPeso molecolare:687.22SNC 162
CAS:SNC 162 is a potent and selective delta-opioid receptor (δ-opioid) agonist with analgesic, antidepressant and antiarrhythmic effects.Formula:C27H37N3OPurezza:98%Colore e forma:SolidPeso molecolare:419.6MR2034
CAS:MR2034 is an agonist of kappa-Opioid receptor. MR2034 stimulates hypothalamic-pituitary-adrenal axis.Formula:C19H27NO2Colore e forma:SolidPeso molecolare:301.42Naloxonazine
CAS:Naloxonazine, a potent, selective opiate mu-1 (μ1) antagonist, also influences leishmania through the modulation of host coding function.Formula:C38H42N4O6Colore e forma:SolidPeso molecolare:650.76Mu opioid receptor antagonist 7
CAS:Compound 24, also known as Mu opioid receptor antagonist 7, is a potent, centrally-acting µ-opioid receptor (µOR) antagonist with an inhibitory concentration (Formula:C22H27ClN2O2Purezza:98%Colore e forma:SolidPeso molecolare:386.91ICI 204448
CAS:ICI 204448 is a potent and peripherally selective κ-opioid agonist.Formula:C23H26Cl2N2O4Colore e forma:SolidPeso molecolare:465.37μ opioid receptor agonist 3
CAS:Compound 20, identified as μ opioid receptor agonist 3, is a potent µOR agonist that exhibits an EC50 value of 0.87 nM.Formula:C22H28N2O2Purezza:98%Colore e forma:SolidPeso molecolare:352.47ADL-08-0011
CAS:ADL-08-0011 is an metabolite of alvimopan.Formula:C23H29NO3Colore e forma:SolidPeso molecolare:367.49R-84760 hydrochloride
CAS:R-84760, a potent κ-opioid receptor agonist, relieves tonic pain via supraspinal/spinal pathways, activating noradrenergic descent.Formula:C19H25Cl3N2OSColore e forma:SolidPeso molecolare:435.84Prodilidine hydrochloride
CAS:Prodilidine hydrochloride is an opioid analgesic.Formula:C15H22ClNO2Colore e forma:SolidPeso molecolare:283.79CYT-1010
CAS:CYT-1010, a mu-opioid receptor agonist; EC50: β-arrestin, 13.1 nM; cAMP, 0.0053 nM. Extracted from patent WO2013173730A2.Formula:C35H40N6O5Purezza:98%Colore e forma:SolidPeso molecolare:624.73BU72
CAS:BU72 is a potent, long-lasting agonist for μ and κ opioid receptors, with partial agonistic activity at the δ opioid receptor (EC50 values of 0.054, 0.033, and 0.58 nM, respectively). It provides strong, enduring analgesic effects primarily mediated through μ opioid receptors. BU72 also exhibits a prolonged duration of activity and can partially reverse morphine-induced analgesia. It is applicable in studies of opioid dependence.Formula:C28H32N2O2Colore e forma:SolidPeso molecolare:428.57SB-612111
CAS:SB-612111: potent ORL-1 antagonist, Ki=0.33 nM; μ-, κ-, δ-receptor Ki=57.6, 160.5, 2109 nM; blocks nociceptin's pain effect.Formula:C24H29Cl2NOColore e forma:SolidPeso molecolare:418.40
