Recettore della bradichinina
I recettori della bradichinina sono GPCR che mediano gli effetti della bradichinina, un peptide coinvolto nelle risposte infiammatorie, nella percezione del dolore e nella regolazione della pressione sanguigna. Esistono due principali tipi di recettori della bradichinina, B1 e B2, ognuno dei quali svolge ruoli distinti nei processi fisiopatologici. Gli antagonisti dei recettori della bradichinina sono utilizzati nel trattamento di condizioni come l'angioedema ereditario, il dolore cronico e l'ipertensione. Presso CymitQuimica, offriamo una varietà di modulatori dei recettori della bradichinina di alta qualità per supportare la tua ricerca in infiammazione, gestione del dolore e biologia cardiovascolare.
Trovati 61 prodotti di "Recettore della bradichinina"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Anatibant 2HCl
CAS:<p>Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological disorders and may be used in the study of brain injury.</p>Formula:C34H36Cl2N6O5S·2ClHPurezza:99.17% - 99.58%Colore e forma:SoildPeso molecolare:784.58Bradykinin (1-7)
CAS:Bradykinin (1-7), an amino-truncated peptide derived from Bradykinin, is a metabolite formed through enzymatic cleavage by endopeptidase.Formula:C35H52N10O9Purezza:98%Colore e forma:White Lyophilized PowderPeso molecolare:756.85FR167344 free base
CAS:FR167344 free base: oral, nonpeptide B2 bradykinin receptor antagonist, high-affinity (IC50: 65 nM), no B1 affinity.Formula:C30H28BrCl2N5O4Purezza:98%Colore e forma:SolidPeso molecolare:673.38Bradykinin (1-6)
CAS:Bradykinin (1-6) is a stable, CPY-cleaved metabolite that triggers pain, induces muscle contractions, and activates NO synthetase.Formula:C30H45N9O8Purezza:98%Colore e forma:SolidPeso molecolare:659.73Labradimil
CAS:Labradimil, a bradykinin B2 agonist, boosts brain drug delivery and tumor survival rates.Formula:C49H75N15O12SPurezza:98%Colore e forma:SolidPeso molecolare:1098.29MEN 11270
CAS:B2 bradykinin receptor peptide antagonist, pKi 10.3; improves hypotension, bronchoconstriction; B2-selective over 29 receptors/ion channels.Formula:C60H90N20O11SPurezza:98%Colore e forma:SolidPeso molecolare:1299.56Bradykinin (1-3)
CAS:<p>Bradykinin (1-3) is a fragment of Bradykinin. Bradykinin is an activates pain receptors.</p>Formula:C16H28N6O4Purezza:98%Colore e forma:SolidPeso molecolare:368.43[Des-Arg9]-Bradykinin
CAS:<p>[Des-Arg9]-Bradykinin ([Des-Arg9]-Bradykinin(2TFA))(2TFA) is an agonist of Bradykinin (B1) receptor.</p>Formula:C44H61N11O10Purezza:98%Colore e forma:SolidPeso molecolare:904.02Sar-[D-Phe8]-des-Arg9-Bradykinin
CAS:Potent bradykinin B1 agonist, EC50 = 9.02 nM, enzyme resistant, induces hypotension and angiogenesis.Formula:C47H66N12O11Purezza:98%Colore e forma:SolidPeso molecolare:975.11Icatibant
CAS:Icatibant is a selective and specific antagonist of the bradykinin B2 receptor (IC50 and Ki: 1.07 nM and 0.798 nM respectively).Formula:C59H89N19O13SPurezza:98%Colore e forma:White SolidPeso molecolare:1304.52Lys-[Des-Arg9]Bradykinin
CAS:Selective bradykinin B1 agonist with Ki 0.12 nM; inactive at B2 (>30,000 nM). Lowers blood pressure, more potent than Des-Arg9-Bradykinin.Formula:C50H73N13O11Purezza:98%Colore e forma:SolidPeso molecolare:1032.21[Des-Arg10]-HOE I40 TFA
<p>[Des-Arg10]-HOE I40 TFA is a potent antagonist of the bradykinin B1 receptor.</p>Formula:C53H77N15O12S·xC2HF3O2Colore e forma:SolidBombinakinin M
CAS:Potent, selective bradykinin receptor agonist 50x stronger than bradykinin, contracts guinea pig ileum muscle at EC50 4.0 nM.Formula:C100H159N31O24Purezza:98%Colore e forma:SolidPeso molecolare:2179.55[Phe8Ψ(CH-NH)-Arg9]-Bradykinin
CAS:Selective bradykinin B2 receptor agonist that is resistant to carboxypeptidase cleavage.Formula:C50H75N15O10Purezza:98%Colore e forma:SolidPeso molecolare:1046.23Fasitibant chloride
CAS:<p>Fasitibant chloride, a potent B2R blocker, alleviates pain and swelling in arthritis.</p>Formula:C36H49Cl3N6O6SColore e forma:SolidPeso molecolare:800.23NPC 567
CAS:NPC 567 is an antagonist of the bradykinin receptor.Formula:C60H87N19O13Purezza:98%Colore e forma:SolidPeso molecolare:1282.48Fasitibant chloride hydrochloride
CAS:Fasitibant chloride( MEN16132) is an effective and selective non-peptide antagonist of kinin B2 receptor.Formula:C36H50Cl4N6O6SColore e forma:SolidPeso molecolare:836.7Lys-Bradykinin
CAS:Endogenous bradykinin receptor agonistFormula:C56H85N17O12Purezza:98%Colore e forma:SolidPeso molecolare:1188.38Zoliprofen
CAS:Zoliprofen: potent, oral NSAID with anti-inflammatory, antipyretic, analgesic effects. Exceeds ibuprofen's efficacy in rats and rabbits.Formula:C12H11NO3SPurezza:99.62%Colore e forma:SolidPeso molecolare:249.29Ref: TM-T68025
1mg85,00€5mg170,00€10mg256,00€25mg480,00€50mg655,00€100mg933,00€500mg1.872,00€1mL*10mM (DMSO)168,00€Retrobradykinin
CAS:Bradykinin analog nonapeptide. Reverse sequence of Bradykinin. Exhibits no significant kinin activity. Can be used as a negative control.Formula:C50H73N15O11Colore e forma:SolidPeso molecolare:1060.228
![[Des-Arg9]-Bradykinin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT7645.webp&w=3840&q=75)
![Sar-[D-Phe8]-des-Arg9-Bradykinin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1917.webp&w=3840&q=75)
![Lys-[Des-Arg9]Bradykinin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1918.webp&w=3840&q=75)
![[Phe8Ψ(CH-NH)-Arg9]-Bradykinin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP2076.webp&w=3840&q=75)
