
Recettore della bradichinina
I recettori della bradichinina sono GPCR che mediano gli effetti della bradichinina, un peptide coinvolto nelle risposte infiammatorie, nella percezione del dolore e nella regolazione della pressione sanguigna. Esistono due principali tipi di recettori della bradichinina, B1 e B2, ognuno dei quali svolge ruoli distinti nei processi fisiopatologici. Gli antagonisti dei recettori della bradichinina sono utilizzati nel trattamento di condizioni come l'angioedema ereditario, il dolore cronico e l'ipertensione. Presso CymitQuimica, offriamo una varietà di modulatori dei recettori della bradichinina di alta qualità per supportare la tua ricerca in infiammazione, gestione del dolore e biologia cardiovascolare.
Trovati 61 prodotti di "Recettore della bradichinina"
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Emorfazone
CAS:Emorfazone (PH011085) has an anti-nociceptive effect.Formula:C11H17N3O3Purezza:99.89%Colore e forma:SolidPeso molecolare:239.27Ref: TM-T9132
1mg88,00€5mg172,00€10mg259,00€25mg425,00€50mg598,00€100mg810,00€200mg1.074,00€1mL*10mM (DMSO)160,00€ELN-441958
CAS:ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM.Formula:C29H29ClN4O2Purezza:99.88%Colore e forma:SolidPeso molecolare:501.02Ref: TM-T2086
1mg62,00€5mg135,00€10mg212,00€25mg359,00€50mg512,00€100mg695,00€200mg939,00€1mL*10mM (DMSO)149,00€SSR240612
CAS:SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors,Formula:C42H53ClN4O7SPurezza:98.59% - 99.16%Colore e forma:SolidPeso molecolare:793.41Ref: TM-T5048
1mg235,00€5mg540,00€10mg740,00€25mg1.035,00€50mg1.406,00€100mg1.882,00€1mL*10mM (DMSO)645,00€Bradykinin (acetate)
CAS:Bradykinin (acetate) is an active peptide that is generated by the kallikrein-kinin system.Formula:C52H77N15O13Purezza:>99.99%Colore e forma:SolidPeso molecolare:1120.26Lys-[Des-Arg9]Bradykinin,TFA
Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2Formula:C54H75F6N13O15Purezza:97.35%Colore e forma:SolidPeso molecolare:1260.24[Des-Arg9]-Bradykinin TFA
CAS:[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.Formula:C46H62F3N11O12Purezza:>99.99%Colore e forma:SolidPeso molecolare:1018.05Bradykinin (2-9)
CAS:Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin.Formula:C44H61N11O10Purezza:>99.99%Colore e forma:SolidPeso molecolare:904.02Ref: TM-TP1181
1mg42,00€5mg93,00€10mg137,00€25mg221,00€50mg329,00€100mg490,00€200mg697,00€1mL*10mM (DMSO)153,00€R715 TFA(185052-09-9 free base)
R715 TFA(185052-09-9 free base) is a potent and selective bradykinin B1 receptor antagonist (pA2 = 8.49).Formula:C59H82F3N13O14Purezza:>99.99%Colore e forma:SolidPeso molecolare:1254.36Lys-Bradykinin acetate(342-10-9 free base)
CAS:Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.Formula:C58H89N17O14Purezza:99.86%Colore e forma:SolidPeso molecolare:1248.43Lys-[Des-Arg9]Bradykinin acetate
<p>Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and</p>Formula:C52H77N13O13Purezza:99.93%Colore e forma:SolidPeso molecolare:1092.27B 4148
CAS:B 4148 is a bradykinin inhibitor.Formula:C62H95N19O14S2Colore e forma:SolidPeso molecolare:1394.67NPC 17731
CAS:NPC 17731 is a bradykinin receptor antagonist.Formula:C59H95N19O14Colore e forma:SolidPeso molecolare:1294.5BKM-570
CAS:BKM-570, a bradykinin antagonist, causes impressive growth inhibition of lung and prostate tumors.Formula:C34H34Cl2F5N3O3Purezza:98%Colore e forma:SolidPeso molecolare:698.55Anatibant
CAS:Anatibant: a strong non-peptide, inhibits bradykinin B2; lowers brain swelling and damage post-trauma.Formula:C34H36Cl2N6O5SPurezza:98%Colore e forma:SolidPeso molecolare:711.66Fulimetibant
CAS:Fulimetibant is a bradykinin receptor antagonist.Formula:C25H21F4N3O3Colore e forma:SolidPeso molecolare:487.45MK-0686
CAS:MK-0686 is an orally available bradykinin B1 receptor antagonist with potential anti-inflammatory activity.Formula:C22H19ClF4N2O4Purezza:99.88%Colore e forma:SolidPeso molecolare:486.84Safotibant
CAS:Safotibant (LF-22-0542) is a bradykinin B1 receptor antagonist with anti-inflammatory and analgesic activity for the topical treatment of diabetic macular edemaFormula:C25H34N4O5SPurezza:99.62% - 99.67%Colore e forma:SolidPeso molecolare:502.63NVP-SAA164
CAS:NVP-SAA164 is a nonpeptide bradykinin B1 receptor antagonist agent.Formula:C36H45N5O5SPurezza:98%Colore e forma:SolidPeso molecolare:659.84FK-3657
CAS:FK-3657 is a non-peptide antagonist of bradykinin (BK)-B2 receptor.Formula:C30H27Cl2N5O4Colore e forma:SolidPeso molecolare:592.47BI-113823
CAS:BI-113823 is an orally active and selective bradykinin B1 receptor antagonist. It alleviates mechanical hyperalgesia induced by complete Freund's adjuvant in rats. BI-113823 is applicable for research on chronic inflammatory pain.Formula:C26H44N4O5SColore e forma:SolidPeso molecolare:524.716
