
Recettore della bradichinina
I recettori della bradichinina sono GPCR che mediano gli effetti della bradichinina, un peptide coinvolto nelle risposte infiammatorie, nella percezione del dolore e nella regolazione della pressione sanguigna. Esistono due principali tipi di recettori della bradichinina, B1 e B2, ognuno dei quali svolge ruoli distinti nei processi fisiopatologici. Gli antagonisti dei recettori della bradichinina sono utilizzati nel trattamento di condizioni come l'angioedema ereditario, il dolore cronico e l'ipertensione. Presso CymitQuimica, offriamo una varietà di modulatori dei recettori della bradichinina di alta qualità per supportare la tua ricerca in infiammazione, gestione del dolore e biologia cardiovascolare.
Trovati 63 prodotti per "Recettore della bradichinina".
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5-Hydroxy-1-methylhydantoin
CAS:5-Hydroxy-1-methylhydantoin (HD-003) is an antioxidant potentially for the treatment of renal failure.Formula:C4H6N2O3Purezza:99.99%Colore e forma:SolidPeso molecolare:130.1Bradykinin
CAS:Bradykinin is an inflammatory mediator.Formula:C50H73N15O11Purezza:99.68%Colore e forma:White SolidPeso molecolare:1060.21Lys-[Des-Arg9]Bradykinin,TFA
Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2Formula:C54H75F6N13O15Purezza:97.35%Colore e forma:White OilPeso molecolare:1260.24[Des-Arg9]-Bradykinin TFA
CAS:[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.Formula:C46H62F3N11O12Purezza:>99.99%Colore e forma:SolidPeso molecolare:1018.05Lys-[Des-Arg9]Bradykinin acetate
Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 andFormula:C52H77N13O13Purezza:99.93%Colore e forma:SolidPeso molecolare:1092.27Sar-[D-Phe8]-des-Arg9-Bradykinin acetate
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate is a potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant toFormula:C49H70N12O13Purezza:99.93%Colore e forma:SolidPeso molecolare:1035.15R715 TFA(185052-09-9 free base)
R715 TFA(185052-09-9 free base) is a potent and selective bradykinin B1 receptor antagonist (pA2 = 8.49).Formula:C59H82F3N13O14Purezza:>99.99%Colore e forma:White SolidPeso molecolare:1254.36Emorfazone
CAS:Emorfazone (PH011085) has an anti-nociceptive effect.Formula:C11H17N3O3Purezza:99.89%Colore e forma:SolidPeso molecolare:239.27Ref: TM-T9132
1mg84,00€1mL*10mM (DMSO)152,00€5mg168,00€10mg245,00€25mg404,00€50mg567,00€100mg767,00€200mg1.018,00€ELN-441958
CAS:ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM.Formula:C29H29ClN4O2Purezza:99.88%Colore e forma:SolidPeso molecolare:501.02Ref: TM-T2086
1mg58,00€5mg128,00€1mL*10mM (DMSO)141,00€10mg200,00€25mg339,00€50mg485,00€100mg658,00€200mg889,00€SSR240612
CAS:SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors,Formula:C42H53ClN4O7SPurezza:98.59% - 99.16%Colore e forma:SolidPeso molecolare:793.41Ref: TM-T5048
1mg222,00€5mg512,00€1mL*10mM (DMSO)612,00€10mg700,00€25mg982,00€50mg1.333,00€100mg1.783,00€Icatibant Acetate
CAS:Icatibant Acetate, an antagonist of the bradykinin B2 receptor, is used in the treatment of hereditary angioedema.Formula:C61H93N19O15SPurezza:99.68% - 99.90%Colore e forma:White SolidPeso molecolare:1364.57Ref: TM-T22344
1mg66,00€2mg92,00€5mg177,00€10mg281,00€1mL*10mM (DMSO)355,00€25mg475,00€50mg677,00€100mg888,00€Bradykinin (2-9)
CAS:Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin.Formula:C44H61N11O10Purezza:>99.99%Colore e forma:White SolidPeso molecolare:904.02BKM-570
CAS:BKM-570, a bradykinin antagonist, causes impressive growth inhibition of lung and prostate tumors.Formula:C34H34Cl2F5N3O3Purezza:98%Colore e forma:SolidPeso molecolare:698.55Anatibant
CAS:Anatibant: a strong non-peptide, inhibits bradykinin B2; lowers brain swelling and damage post-trauma.Formula:C34H36Cl2N6O5SPurezza:98%Colore e forma:SolidPeso molecolare:711.66B 4148
CAS:B 4148 is a bradykinin inhibitor.Formula:C62H95N19O14S2Colore e forma:SolidPeso molecolare:1394.67NPC 17731
CAS:NPC 17731 is a bradykinin receptor antagonist.Formula:C59H95N19O14Colore e forma:SolidPeso molecolare:1294.5FK-3657
CAS:FK-3657 is a non-peptide antagonist of bradykinin (BK)-B2 receptor.Formula:C30H27Cl2N5O4Colore e forma:SolidPeso molecolare:592.47Fulimetibant
CAS:Fulimetibant is a bradykinin receptor antagonist.Formula:C25H21F4N3O3Colore e forma:SolidPeso molecolare:487.45MK-0686
CAS:MK-0686 is an orally available bradykinin B1 receptor antagonist with potential anti-inflammatory activity.Formula:C22H19ClF4N2O4Purezza:99.88%Colore e forma:White SolidPeso molecolare:486.84Safotibant
CAS:Safotibant (LF-22-0542) is a bradykinin B1 receptor antagonist with anti-inflammatory and analgesic activity for the topical treatment of diabetic macular edemaFormula:C25H34N4O5SPurezza:99.62% - 99.67%Colore e forma:SolidPeso molecolare:502.63
