
Recettore della dopamina
I recettori della dopamina sono un gruppo di recettori accoppiati alle proteine G (GPCR) che rispondono al neurotrasmettitore dopamina, svolgendo un ruolo chiave nella regolazione del movimento, della motivazione, della ricompensa e di diverse funzioni cognitive. Questi recettori sono divisi in famiglie simili a D1 e D2, ognuna con funzioni e profili farmacologici distinti. I modulatori dei recettori della dopamina sono ampiamente studiati per le loro applicazioni nel trattamento del morbo di Parkinson, della schizofrenia, della dipendenza e di altri disturbi neuropsichiatrici. Presso CymitQuimica, offriamo una vasta gamma di modulatori dei recettori della dopamina di alta qualità per supportare la tua ricerca in neuroscienze, salute mentale e segnalazione GPCR.
Trovati 435 prodotti di "Recettore della dopamina"
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Mefexamide hydrochloride
CAS:Mefexamide hydrochloride is a central stimulant.Formula:C15H25ClN2O3Purezza:99.95%Colore e forma:SolidPeso molecolare:316.83Benserazide hydrochloride
CAS:<p>Benserazide hydrochloride (Ro 4-4602) is a peripherally-acting L-amino acid decarboxylase (AAAD) or DOPA decarboxylase inhibitor.</p>Formula:C10H15N3O5·HClPurezza:98.63% - 99.74%Colore e forma:White Crystalline SolidPeso molecolare:293.7Benztropine mesylate
CAS:<p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>Formula:C21H25NO·CH4SO3Purezza:98.41% - 99.96%Colore e forma:White Crystalline Powder; Odourless Or Almost OdourlessPeso molecolare:403.53Ro 10-5824 dihydrochloride
CAS:Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).Formula:C17H22Cl2N4Purezza:99.79%Colore e forma:SolidPeso molecolare:353.29Thioridazine hydrochloride
CAS:Thioridazine hydrochloride (Mellaril) , an antipsychotic drug, is used in the therapy of psychosis and schizophrenia and shows serotonin antagonism or D4Formula:C21H27ClN2S2Purezza:99.55% - 99.957%Colore e forma:White To Off-White SolidPeso molecolare:407.04Iloperidone
CAS:Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.Formula:C24H27FN2O4Purezza:99.42%Colore e forma:SolidPeso molecolare:426.48L-741626
CAS:<p>L-741626 (3-(4-(4-Chlorophenyl-4-hydroxypiperidino)methyl)indole) is a selective antagonist of D2 dopamine receptor (Ki: 2.4, 100, and 220 nM for human D2, D3</p>Formula:C20H21ClN2OPurezza:98.57%Colore e forma:SolidPeso molecolare:340.85Perphenazine
CAS:<p>Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.</p>Formula:C21H26ClN3OSPurezza:99.3% - 99.99%Colore e forma:SolidPeso molecolare:403.97Bendazol
CAS:<p>Bendazol (Dibazol) is always used as the drug for hypertension and cerebral Angiospasm.</p>Formula:C14H12N2Purezza:98.7% - 99.87%Colore e forma:White Or Almost White Crystalline PowderPeso molecolare:208.26Blonanserin
CAS:Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.Formula:C23H30FN3Purezza:99.85%Colore e forma:SolidPeso molecolare:367.5Domperidone
CAS:<p>Domperidone (R33812)(Motilium) is a dopamine blocker and an antidopaminergic reagent.</p>Formula:C22H24ClN5O2Purezza:98% - 99.82%Colore e forma:SolidPeso molecolare:425.91Loxapine succinate
CAS:Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.Formula:C22H24ClN3O5Purezza:99.69%Colore e forma:White To Of-White SolidPeso molecolare:445.9Levosulpiride
CAS:Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.Formula:C15H23N3O4SPurezza:98.20% - 99.88%Colore e forma:White Crystalline PowderPeso molecolare:341.43Talipexole dihydrochloride
CAS:Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical andFormula:C10H17Cl2N3SPurezza:99.89%Colore e forma:Light Yellow SolidPeso molecolare:282.23NEO 376
CAS:<p>NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.</p>Formula:C20H24ClN3OPurezza:99.56%Colore e forma:SolidPeso molecolare:357.88Amisulpride
CAS:Amisulpride (Solian/Deniban), a dopamine antagonist antipsychotic, treats psychosis and schizophrenia in Europe/Australia, not in the US.Formula:C17H27N3O4SPurezza:99.97% - 99.99%Colore e forma:White Or Almost White Crystalline PowderPeso molecolare:369.48Tipepidine hydrochloride
CAS:Tipepidine hydrochloride: reversible DA D2 receptor inhibitor, IC50 7.0 μM, with antidepressant effects.Formula:C15H18ClNS2Purezza:99.97%Colore e forma:SolidPeso molecolare:311.89Tetrabenazine
CAS:Tetrabenazine (Ro 1-9569) is a drug formerly used as an antipsychotic and treatment of various movement disorders.Formula:C19H27NO3Purezza:98% - 99.91%Colore e forma:White To Off-White White To Off-White SolidPeso molecolare:317.42Clozapine
CAS:<p>Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.</p>Formula:C18H19ClN4Purezza:99.91% - 99.93%Colore e forma:Yellow Crystals From Acetone-Petroleum Ether SolidPeso molecolare:326.82Ziprasidone
CAS:<p>Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.</p>Formula:C21H21ClN4OSPurezza:99.55%Colore e forma:Tan SolidPeso molecolare:412.94Quetiapine
CAS:<p>Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.</p>Formula:C21H25N3O2SPurezza:99.14% - 99.63%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:383.51Prochlorperazine Maleate
CAS:Prochlorperazine Maleate (Capazine) is a phenothiazine antipsychotic used principally in the treatment of NAUSEA; VOMITING; and VERTIGO.Formula:C28H32ClN3O8SPurezza:99.78%Colore e forma:Off-White PowderPeso molecolare:606.09Metoclopramide hydrochloride
CAS:Metoclopramide hydrochloride (Metoclopramide HCl) is a selective dopamine D2 receptor antagonist, used as an antiemetic.Formula:C14H22ClN3O2·HClPurezza:99.99%Colore e forma:White To Off-White PowderPeso molecolare:336.26Chlorprothixene hydrochloride
CAS:Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.Formula:C18H18ClNS·HClPurezza:99.76%Colore e forma:White PowderPeso molecolare:352.32Acetophenazine dimaleate
CAS:Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor.Formula:C31H37N3O10SPurezza:99.39% - 99.48%Colore e forma:SolidPeso molecolare:643.71Promazine hydrochloride
CAS:Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.Formula:C17H21ClN2SPurezza:99.90%Colore e forma:SolidPeso molecolare:320.88GR 103691
CAS:<p>GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).</p>Formula:C30H35N3O3Purezza:98.94% - 99.29%Colore e forma:SolidPeso molecolare:485.62Itopride hydrochloride
CAS:Itopride hydrochloride (Ganaton) is an AChE and D2DR inhibitor.Formula:C20H27ClN2O4Purezza:99.59%Colore e forma:White Or Pale Brownish CrystalPeso molecolare:394.9Pramipexole
CAS:<p>Pramipexole (SND 919), a dopamine agonist for Parkinson's, may cause mild, temporary enzyme spikes, not acute liver injury.</p>Formula:C10H17N3SPurezza:98% - 99.96%Colore e forma:SolidPeso molecolare:211.33Risperidone
CAS:Risperidone (R 64 766) is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.Formula:C23H27FN4O2Purezza:99.73%Colore e forma:Crystalline SolidPeso molecolare:410.48L-DOPA
CAS:L-DOPA (Levodopa) is an amino acid precursor of dopamine with antiparkinsonian properties. Levodopa that is converted to dopamine by DOPA decarboxylase.Formula:C9H11NO4Purezza:98.99% - 99.93%Colore e forma:Colorless To White Crystals Or Crystalline Powder; Needles From Water SolidPeso molecolare:197.19Ziprasidone hydrochloride monohydrate
CAS:Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychoticFormula:C21H21ClN4OS·HCl·H2OPurezza:98% - 99.83%Colore e forma:Off-White PowderPeso molecolare:467.12Sulpiride
CAS:Sulpiride (Aiglonyl) is a dopamine D2-receptor antagonist, used therapeutically as an antidepressant, antipsychotic, and as a digestive aid.Formula:C15H23N3O4SPurezza:99.94%Colore e forma:White Crystalline PowderPeso molecolare:341.43(-)-GSK598809 hydrochloride
CAS:<p>(-)-GSK598809 hydrochloride, a DRD3 selective antagonist, may correct reward deficits in substance dependence.</p>Formula:C22H24ClF4N5OSPurezza:98.36%Colore e forma:SoildPeso molecolare:517.97Oxidopamine hydrochloride
CAS:Oxidopamine hydrochloride (6-Hydroxydopamine hydrochloride) is an neurotransmitter dopamine antagonist.Formula:C8H12ClNO3Purezza:98.34% - 99.85%Colore e forma:Physical Description Beige Solid (Ntp 1992)Peso molecolare:205.64Bromopride
CAS:Bromopride (Valopride), a metoclopramide-like dopamine antagonist and prokinetic, is an antiemetic not sold in the US or UK.Formula:C14H22BrN3O2Purezza:99.95%Colore e forma:SolidPeso molecolare:344.25Flunarizine dihydrochloride
CAS:<p>Flunarizine dihydrochloride: a calcium blocker also targeting calmodulin and histamine H1, used for migraine, vertigo, vascular disease, and epilepsy aid.</p>Formula:C26H28Cl2F2N2Purezza:99.53% - 99.89%Colore e forma:White Crystalline Powder Odorless And TastelessPeso molecolare:477.42Fosopamine(HCl)
CAS:<p>Fosopamine(HCl) is a DRDs agonist that can be used to study hypertension.</p>Formula:C9H15ClNO5PPurezza:99.84%Colore e forma:SolidPeso molecolare:283.65Pipamperone
CAS:<p>Pipamperone (McN-JR 3345) binds 5-HT2A closely as receptor.</p>Formula:C21H30FN3O2Purezza:99.85%Colore e forma:White PowderPeso molecolare:375.48Pericyazine
CAS:<p>Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist.</p>Formula:C21H23N3OSPurezza:99.61%Colore e forma:SolidPeso molecolare:365.49Dopamine hydrochloride
CAS:<p>Dopamine hydrochloride (ASL279) is a natural catecholamine neurotransmitter, dopamine receptors (D1-5 receptors) (EC50=2.7 nM). High-Quality, Low-Cost!</p>Formula:C8H12ClNO2Purezza:99.47% - 99.72%Colore e forma:SolidPeso molecolare:189.64Olanzapine
CAS:Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.Formula:C17H20N4SPurezza:99.86% - ≥95%Colore e forma:Yellowish Crystalline PowderPeso molecolare:312.43Droperidol
CAS:<p>Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as a Dopamine D2 Antagonist.</p>Formula:C22H22FN3O2Purezza:97.16% - 98%Colore e forma:SolidPeso molecolare:379.43Fluphenazine dihydrochloride
CAS:Fluphenazine dihydrochloride (Prolixin) is an inhibitor of phenothiazine-class D1DR and D2DR. Fluphenazine can be used to probe effects and metabolic process.Formula:C22H28Cl2F3N3OSPurezza:99.23%Colore e forma:Off-White SolidPeso molecolare:510.44Dexpramipexole dihydrochloride
CAS:Dexpramipexole dihydrochloride (KNS-760704 dihydrochloride) ((R)-Pramipexole dihydrochloride) is a neuroprotective agent and is a weak non-ergoline dopamineFormula:C10H19Cl2N3SPurezza:99.75% - 99.88%Colore e forma:SolidPeso molecolare:284.25Tiapride hydrochloride
CAS:<p>Tiapride is a selective blocker of D2/3 dopamine receptors in the brain.</p>Formula:C15H24N2O4S·HClPurezza:99.4% - 99.77%Colore e forma:SolidPeso molecolare:364.89Romergoline 2HCl
Romergoline 2HCl is a D1 agonist and D2 antagonist used in the study of Parkinson's disease.Formula:C20H24Cl2N4O2Purezza:99.01% - 99.40%Colore e forma:SoildPeso molecolare:423.34Trifluoperazine dihydrochloride
CAS:Trifluoperazine dihydrochloride (SKF5019) is a potent dopamine D2 receptor inhibitor used as an antipsychotic and an antiemetic.Formula:C21H26Cl2F3N3SPurezza:99.57% - 99.96%Colore e forma:Cream Fine PowderPeso molecolare:480.43Molindone hydrochloride
CAS:<p>Molindone hydrochloride (EN-1733A) is an indole derivative effective in schizophrenia and other psychoses by blocking the effects of dopamine in the brain.</p>Formula:C16H24N2O2·HClPurezza:99% - 99.99%Colore e forma:SolidPeso molecolare:312.84Bromperidol
CAS:Bromperidol (R-11333) is a butyrophenone derivative and it is a potent and long-acting neuroleptic.Formula:C21H23BrFNO2Purezza:99.89%Colore e forma:Tan SolidPeso molecolare:420.32Ziprasidone hydrochloride
CAS:<p>Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic</p>Formula:C21H22CL2N4OSPurezza:97.97% - 99.82%Colore e forma:SolidPeso molecolare:449.4Tetrahydropalmatine
CAS:Tetrahydropalmatine (DL-Tetrahydropalmatine) is an active component isolated from corydalis, suppressing amygdaloid release of dopamine to inhibit an epilepticFormula:C21H25NO4Purezza:99.59% - 99.95%Colore e forma:SolidPeso molecolare:355.43Talquetamab
CAS:Talquetamab (JNJ-64407564) is a T-cell retargeting GPRC5D bispecific antibody with antitumor activity for the treatment of multiple myeloma.Colore e forma:LiquidPeso molecolare:144.59 kDaSpiperone
CAS:Spiperone (Spiropitan) is a spiro butyrophenone analog similar to HALOPERIDOL and other related compounds.Formula:C23H26FN3O2Purezza:99.34% - 99.91%Colore e forma:SolidPeso molecolare:395.47Quetiapine hemifumarate
CAS:Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.Formula:C46H54N6O8S2Purezza:99.32% - >99.99%Colore e forma:White Crystalline SolidPeso molecolare:883.09ONC206
CAS:<p>ONC206, an analogue of the TRAIL inducer ONC201, acts as a selective antagonist of the D2-like dopamine receptors (DRD2/3/4) at nanomolar concentrations and</p>Formula:C23H22F2N4OPurezza:99.38% - 99.81%Colore e forma:SolidPeso molecolare:408.44Oxidopamine hydrobromide
CAS:<p>Oxidopamine hydrobromide (6-OHDA hydrobromide) is a neurotransmitter dopamine antagonist.</p>Formula:C8H12BrNO3Purezza:98.22% - 99.88%Colore e forma:Beige To Brown Fine Crystalline PowderPeso molecolare:250.09Paliperidone
CAS:<p>Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic.</p>Formula:C23H27FN4O3Purezza:95% - 99.08%Colore e forma:Off White To Light Orange Coloured SolidPeso molecolare:426.48Haloperidol
CAS:Haloperidol (Serenace) is a highly potent neuroleptic by relieving nervous through the depression of nerve function.Formula:C21H23ClFNO2Purezza:98.69% - 98.97%Colore e forma:Crystals SolidPeso molecolare:375.86UCM-1306
CAS:<p>UCM-1306: an oral dopamine D1 receptor PAM; boosts DA efficacy, may enhance motor and cognitive function in PD.</p>Formula:C14H14FNO2SPurezza:99.98%Colore e forma:SoildPeso molecolare:279.33BP 897 hydrochloride
CAS:BP 897: potent D3 agonist (Ki: 0.92 nM), weak D2 antagonist (Ki: 61 nM), low affinity for D1/D4.Formula:C26H32ClN3O2Purezza:99.42%Colore e forma:SolidPeso molecolare:454D5R agonist 1
D5R Agonist 1 (Compound 5j) is a selective, orally active partial agonist of the D5 receptor that can penetrate the blood-brain barrier (EC50: 269.7 nM). It has been demonstrated to enhance cognitive abilities in a scopolamine-induced amnesia model.Colore e forma:Odour SolidDETQ
CAS:<p>DETQ enhances human D1 dopamine receptor signaling, EC50=5.8 nM, less effective in rats/mice, inactive on D5.</p>Formula:C22H25Cl2NO3Colore e forma:SolidPeso molecolare:422.34Octodrine
CAS:<p>Octodrine (2-Amino-6-methylheptane) is primarily used as a pharmaceutical intermediate for Octamylamine; it also functions as a local anesthetic and vasoconstrictor.</p>Formula:C8H19NPurezza:99.98%Colore e forma:Clear Colorless To Light Yellow LiquidPeso molecolare:129.24Losulazine
CAS:<p>Losulazine: a new antihypertensive, requires functional sympathetic nervous system; mechanism undefined.</p>Formula:C27H22F4N4O3SPurezza:98.83%Colore e forma:SolidPeso molecolare:558.55Vanicoside E
CAS:Vanicoside E is an antioxidant and antitumor agent. Vanicoside E inhibits L-Tyrosine and L-DOPA with IC 50 s of 45.23 μM and 189.96 μM, respectively [1] [2] .Formula:C53H52O22Colore e forma:SolidPeso molecolare:1040.97D3R/MOR antagonist 2
<p>Compound 121, a D3R/MOR antagonist with K i values of 361 nM and 85.2 nM for D3R and MOR respectively, has the potential for analgesic effects through MOR</p>Formula:C25H31ClN2OPurezza:98%Colore e forma:SolidPeso molecolare:410.98Neurotransmitter Receptor Compound Library
<p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening;</p>Colore e forma:Odour SolidABT 724 trihydrochloride
CAS:<p>ABT-724 trihydrochloride: selective D4 agonist; EC50=12.4nM(human),14.3nM(rat),23.2nM(ferret); for erectile dysfunction research.</p>Formula:C17H22Cl3N5Purezza:99.91%Colore e forma:SolidPeso molecolare:402.75D3R/MOR antagonist 1
<p>Compound 114 (D3R/MOR antagonist 1) exhibits dual antagonistic activity at dopamine D3 receptors (D3R) and mu-opioid receptors (MOR), with K i values of 46.5 nM</p>Formula:C22H27Cl2N3OPurezza:98%Colore e forma:SolidPeso molecolare:420.38Fenoldopam
CAS:Fenoldopam is a selective D1-like dopamine receptor partial agonist (EC50 = 57 nM).Formula:C16H16ClNO3Purezza:98%Colore e forma:SolidPeso molecolare:305.767-Hydroxy-PIPAT maleate
CAS:7-Hydroxy-PIPAT maleate is a D3R agonist.Formula:C16H22INOColore e forma:SolidPeso molecolare:371.262[18F]-Labeled L-dopa precursor
CAS:[18F]-Labeled L-dopa precursor is a precursor for synthesis of 18F-labeled L-dopa[1].Formula:C35H36N2O7Colore e forma:SolidPeso molecolare:596.67Neuromedin N
CAS:<p>Neuromedin N is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct expression and effects.</p>Formula:C38H63N7O8Purezza:98%Colore e forma:SolidPeso molecolare:745.95MLS1082
CAS:MLS1082 is a D1-like dopamine receptor (D1R) orthosteric modulatothat stimulates G-protein signaling upon dopamine activation for neurodegenerative disorders.Formula:C24H23N3O2Purezza:99.53%Colore e forma:SolidPeso molecolare:385.46D3R ligand 1
D3R Ligand 1 (compound 23b) is a potent, selective antagonist of the dopamine D3 receptor (Ki=66 nM), incorporating a THPB template.Formula:C27H37NO5Purezza:98%Colore e forma:SolidPeso molecolare:455.59Clomipramine D3
CAS:Clomipramine D3 is deuterium-labeled Clomipramine, blocking serotonin, norepinephrine, dopamine transporters (Ki: 0.14, 54, 3 nM).Formula:C19H23ClN2Purezza:98%Colore e forma:SolidPeso molecolare:317.87N-Methyl-2-phenylpropan-1-amine hydrochloride
CAS:N-Methyl-2-phenylpropan-1-amine hydrochloride is an analogue of β-methylphenethylamine (BMPEA) and demonstrates neurotransmitter-releasing properties in experiments involving NET and DAT.Formula:C10H16ClNPeso molecolare:185.69A 31472
CAS:A 31472 is a tetracyclic spiro amine that has affinity for dopamine D-2 receptors.Formula:C22H22ClNColore e forma:SolidPeso molecolare:335.87MOR agonist-3
MOR agonist-3 (Compound 84) is a dual D3R/MOR antagonist with K i values of 382 nM and 55.2 nM, respectively.Colore e forma:Odour SolidDopamine D2 receptor agonist-2
CAS:<p>Dopamine D2 receptor agonist-2 (Dopamine D2 Receptor) is a ligand targeting the dopamine D2 receptor.</p>Formula:C25H31Cl2N5OSPurezza:98.93%Colore e forma:SoildPeso molecolare:520.52A 77636 hydrochloride
CAS:<p>A 77636 hydrochloride is a potent, orally active, selective and long acting dopamine D1 receptor agonist (pKi=7.40; Ki=39.8 nM).</p>Formula:C20H28ClNO3Purezza:99.57%Colore e forma:SolidPeso molecolare:365.89ADTN hydrobromide
CAS:<p>ADTN hydrobromide (6,7-ADTN) is a dopamine receptor agonist (EC50s = 3.5 and 0.65 μM in rat striatal and nucleus accumbens homogenates, respectively).</p>Formula:C10H14BrNO2Colore e forma:SolidPeso molecolare:260.13Amisulpride hydrochloride
CAS:<p>Amisulpride is an antagonist of 5-HT7 receptor and dopamine D2 and D3 receptors. It modulates beta 2- arresting signaling and increases neurite outgrowth.</p>Formula:C17H28ClN3O4SColore e forma:SolidPeso molecolare:405.94MOR agonist-2
Compound 46, designated as MOR agonist-2, serves as a D3R antagonist and a MOR agonist with respective K i values of 7.26 nM and 564 nM.Formula:C37H47Cl2N5O3Purezza:98%Colore e forma:SolidPeso molecolare:680.71LE 300
CAS:<p>LE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.</p>Formula:C20H22N2Purezza:97.91% - 98.79%Colore e forma:SolidPeso molecolare:290.4S33084
CAS:S33084 is a potent, selective and competitive antagonist of dopamine D(3)-receptors.Formula:C29H29N3O2Purezza:98%Colore e forma:SolidPeso molecolare:451.56PF-4363467
CAS:PF-4363467 is a dopamine D3/D2 receptor antagonist that reduces opioid-seeking behavior without the side effects associated with D2 receptors. It has a Ki value of 3.1 nM for D3R and 692 nM for D2R.Formula:C22H30N2O3SColore e forma:SolidPeso molecolare:402.55O-2172
CAS:<p>O-2172 is a carbocyclic analogue serving as an inhibitor of dopamine transporter (DAT), exhibiting IC50 values of 47 nM for DAT and 7000 nM for the serotonin transporter (SERT).</p>Formula:C14H16Cl2O2Colore e forma:SolidPeso molecolare:287.18Cabergoline
CAS:<p>Cabergoline (FCE-21336), an ergot-derived dopamine D2-like agonist, targets D2/D3/5-HT2B, normalizes prolactin, controls pituitary tumors.</p>Formula:C26H37N5O2Purezza:97.69% - 99.86%Colore e forma:White Crystalline SolidPeso molecolare:451.6(R)-Preclamol hydrochloride
CAS:<p>(R)-Preclamol HCl is a dopamine agonist stimulating both auto and postsynaptic receptors.</p>Formula:C14H22ClNOColore e forma:SolidPeso molecolare:255.78Secretoneurin, rat
CAS:Secretoneurin, rat, a 33-amino acid polypeptide, is generated by proteolytic processing of secretogranin II (SgII).Formula:C159H252N40O58Purezza:98%Colore e forma:SolidPeso molecolare:3651.95ADTN
CAS:ADTN is an agonist of the dopamine receptor.Formula:C10H13NO2Purezza:98%Colore e forma:SolidPeso molecolare:179.22Haloperidol D4
CAS:<p>Haloperidol D4 is deuterium-labeled haloperidol.</p>Formula:C21H23ClFNO2Purezza:98%Colore e forma:SolidPeso molecolare:379.89Preclamol hydrochloride
CAS:Preclamol hydrochloride: selective dopamine agonist with research potential in schizophrenia.Formula:C14H22ClNOColore e forma:SolidPeso molecolare:255.78Quinelorane
CAS:Quinelorane is dextrorotary isomer.Formula:C14H22N4Colore e forma:SolidPeso molecolare:246.35Fluphenazine free base
CAS:Flufenazine: antipsychotic for schizophrenia, blocks dopamine D2 receptors, reduces hallucinations and delusions.Formula:C22H26F3N3OSColore e forma:SolidPeso molecolare:437.52Adrogolide HCl
CAS:Adrogolide Hydrochloride is a selective dopamine receptor D1 agonist.Formula:C22H26ClNO4SColore e forma:SolidPeso molecolare:435.96N-0500 HCl
CAS:<p>N-0500 HCl, a potent DA receptor agonist, displaces [3H]DP_x005f_x0002_5,6-ADTN with an IC50 of 3nM.</p>Formula:C15H22ClNO2Purezza:98.85% - 99.54%Colore e forma:SolidPeso molecolare:283.79Moperone
CAS:Moperone (R 1658) is an antagonist of both the D2 dopamine receptor (D2 dopamine receptor) and the D3 dopamine receptor (D3 dopamine receptor), with IC50 values for each of 1.0 nM.Formula:C22H26FNO2Colore e forma:SolidPeso molecolare:355.45

