
Recettore della dopamina
I recettori della dopamina sono un gruppo di recettori accoppiati alle proteine G (GPCR) che rispondono al neurotrasmettitore dopamina, svolgendo un ruolo chiave nella regolazione del movimento, della motivazione, della ricompensa e di diverse funzioni cognitive. Questi recettori sono divisi in famiglie simili a D1 e D2, ognuna con funzioni e profili farmacologici distinti. I modulatori dei recettori della dopamina sono ampiamente studiati per le loro applicazioni nel trattamento del morbo di Parkinson, della schizofrenia, della dipendenza e di altri disturbi neuropsichiatrici. Presso CymitQuimica, offriamo una vasta gamma di modulatori dei recettori della dopamina di alta qualità per supportare la tua ricerca in neuroscienze, salute mentale e segnalazione GPCR.
Trovati 443 prodotti di "Recettore della dopamina"
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Oxidopamine hydrobromide
CAS:Oxidopamine hydrobromide (6-OHDA hydrobromide) is a neurotransmitter dopamine antagonist.Formula:C8H12BrNO3Purezza:98.22% - 99.88%Colore e forma:Beige To Brown Fine Crystalline PowderPeso molecolare:250.09Levosulpiride
CAS:Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.Formula:C15H23N3O4SPurezza:98.20% - 99.88%Colore e forma:White Crystalline PowderPeso molecolare:341.43Tetrabenazine
CAS:Tetrabenazine (Ro 1-9569) is a drug formerly used as an antipsychotic and treatment of various movement disorders.Formula:C19H27NO3Purezza:98% - 99.91%Colore e forma:White To Off-White White To Off-White SolidPeso molecolare:317.42NEO 376
CAS:NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.Formula:C20H24ClN3OPurezza:99.56%Colore e forma:SolidPeso molecolare:357.88Ref: TM-T12207
1mg74,00€5mg140,00€10mg215,00€25mg373,00€50mg522,00€100mg702,00€200mg944,00€1mL*10mM (DMSO)156,00€Promazine hydrochloride
CAS:Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.Formula:C17H21ClN2SPurezza:99.90%Colore e forma:SolidPeso molecolare:320.88Itopride hydrochloride
CAS:Itopride hydrochloride (Ganaton) is an AChE and D2DR inhibitor.Formula:C20H27ClN2O4Purezza:99.59%Colore e forma:White Or Pale Brownish CrystalPeso molecolare:394.9Sulpiride
CAS:Sulpiride (Aiglonyl) is a dopamine D2-receptor antagonist, used therapeutically as an antidepressant, antipsychotic, and as a digestive aid.Formula:C15H23N3O4SPurezza:99.94%Colore e forma:White Crystalline PowderPeso molecolare:341.43Perphenazine
CAS:<p>Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.</p>Formula:C21H26ClN3OSPurezza:99.3% - 99.99%Colore e forma:SolidPeso molecolare:403.97Paliperidone
CAS:<p>Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic.</p>Formula:C23H27FN4O3Purezza:95% - 99.08%Colore e forma:Off White To Light Orange Coloured SolidPeso molecolare:426.48Flunarizine dihydrochloride
CAS:<p>Flunarizine dihydrochloride: a calcium blocker also targeting calmodulin and histamine H1, used for migraine, vertigo, vascular disease, and epilepsy aid.</p>Formula:C26H28Cl2F2N2Purezza:99.53% - 99.89%Colore e forma:White Crystalline Powder Odorless And TastelessPeso molecolare:477.42Quetiapine
CAS:<p>Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.</p>Formula:C21H25N3O2SPurezza:99.14% - 99.63%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:383.51Domperidone
CAS:<p>Domperidone (R33812)(Motilium) is a dopamine blocker and an antidopaminergic reagent.</p>Formula:C22H24ClN5O2Purezza:98% - 99.82%Colore e forma:SolidPeso molecolare:425.91Mefexamide hydrochloride
CAS:Mefexamide hydrochloride is a central stimulant.Formula:C15H25ClN2O3Purezza:99.95%Colore e forma:SolidPeso molecolare:316.83Molindone hydrochloride
CAS:<p>Molindone hydrochloride (EN-1733A) is an indole derivative effective in schizophrenia and other psychoses by blocking the effects of dopamine in the brain.</p>Formula:C16H24N2O2·HClPurezza:99% - 99.99%Colore e forma:SolidPeso molecolare:312.84Romergoline 2HCl
Romergoline 2HCl is a D1 agonist and D2 antagonist used in the study of Parkinson's disease.Formula:C20H24Cl2N4O2Purezza:99.01% - 99.40%Colore e forma:SoildPeso molecolare:423.34Metoclopramide hydrochloride
CAS:Metoclopramide hydrochloride (Metoclopramide HCl) is a selective dopamine D2 receptor antagonist, used as an antiemetic.Formula:C14H22ClN3O2·HClPurezza:99.99%Colore e forma:White To Off-White PowderPeso molecolare:336.26Pericyazine
CAS:<p>Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist.</p>Formula:C21H23N3OSPurezza:99.61%Colore e forma:SolidPeso molecolare:365.49Ref: TM-T16472
1mg46,00€2mg59,00€5mg93,00€10mg124,00€25mg235,00€50mg389,00€100mg567,00€500mg1.225,00€GR 103691
CAS:GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).Formula:C30H35N3O3Purezza:98.94% - 99.29%Colore e forma:SolidPeso molecolare:485.62Ref: TM-T11463
2mg42,00€5mg62,00€10mg97,00€25mg187,00€50mg305,00€100mg487,00€200mg692,00€1mL*10mM (DMSO)66,00€Ro 10-5824 dihydrochloride
CAS:Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).Formula:C17H22Cl2N4Purezza:99.79%Colore e forma:SolidPeso molecolare:353.29Prochlorperazine Maleate
CAS:Prochlorperazine Maleate (Capazine) is a phenothiazine antipsychotic used principally in the treatment of NAUSEA; VOMITING; and VERTIGO.Formula:C28H32ClN3O8SPurezza:99.78%Colore e forma:Off-White PowderPeso molecolare:606.09Fosopamine(HCl)
CAS:Fosopamine(HCl) is a DRDs agonist that can be used to study hypertension.Formula:C9H15ClNO5PPurezza:99.84%Colore e forma:SolidPeso molecolare:283.65Bromopride
CAS:Bromopride (Valopride), a metoclopramide-like dopamine antagonist and prokinetic, is an antiemetic not sold in the US or UK.Formula:C14H22BrN3O2Purezza:99.95%Colore e forma:SolidPeso molecolare:344.25Ref: TM-T1175
2mg39,00€5mg58,00€10mg93,00€25mg167,00€50mg260,00€100mg409,00€200mg595,00€1mL*10mM (DMSO)64,00€ONC206
CAS:ONC206, an analogue of the TRAIL inducer ONC201, acts as a selective antagonist of the D2-like dopamine receptors (DRD2/3/4) at nanomolar concentrations andFormula:C23H22F2N4OPurezza:99.38% - 99.81%Colore e forma:SolidPeso molecolare:408.44L-741626
CAS:L-741626 (3-(4-(4-Chlorophenyl-4-hydroxypiperidino)methyl)indole) is a selective antagonist of D2 dopamine receptor (Ki: 2.4, 100, and 220 nM for human D2, D3Formula:C20H21ClN2OPurezza:98.57%Colore e forma:SolidPeso molecolare:340.85Iloperidone
CAS:Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.Formula:C24H27FN2O4Purezza:99.42%Colore e forma:SolidPeso molecolare:426.48Pramipexole
CAS:Pramipexole (SND 919), a dopamine agonist for Parkinson's, may cause mild, temporary enzyme spikes, not acute liver injury.Formula:C10H17N3SPurezza:98% - 99.96%Colore e forma:SolidPeso molecolare:211.33L-DOPA
CAS:L-DOPA (Levodopa) is an amino acid precursor of dopamine with antiparkinsonian properties. Levodopa that is converted to dopamine by DOPA decarboxylase.Formula:C9H11NO4Purezza:98.99% - 99.93%Colore e forma:Colorless To White Crystals Or Crystalline Powder; Needles From Water SolidPeso molecolare:197.19Talquetamab
CAS:Talquetamab (JNJ-64407564) is a T-cell retargeting GPRC5D bispecific antibody with antitumor activity for the treatment of multiple myeloma.Colore e forma:LiquidPeso molecolare:144.59 kDaHaloperidol
CAS:Haloperidol (Serenace) is a highly potent neuroleptic by relieving nervous through the depression of nerve function.Formula:C21H23ClFNO2Purezza:98.69% - 98.97%Colore e forma:Crystals SolidPeso molecolare:375.86UCM-1306
CAS:UCM-1306: an oral dopamine D1 receptor PAM; boosts DA efficacy, may enhance motor and cognitive function in PD.Formula:C14H14FNO2SPurezza:99.98%Colore e forma:SoildPeso molecolare:279.33Talipexole dihydrochloride
CAS:Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical andFormula:C10H17Cl2N3SPurezza:99.89%Colore e forma:Light Yellow SolidPeso molecolare:282.23Ref: TM-T14490
2mg35,00€5mg52,00€10mg80,00€25mg144,00€50mg225,00€100mg359,00€200mg532,00€1mL*10mM (DMSO)52,00€Chlorprothixene hydrochloride
CAS:Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.Formula:C18H18ClNS·HClPurezza:99.76%Colore e forma:White PowderPeso molecolare:352.32Olanzapine
CAS:Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.Formula:C17H20N4SPurezza:99.86% - ≥95%Colore e forma:Yellowish Crystalline PowderPeso molecolare:312.43Risperidone
CAS:Risperidone (R 64 766) is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.Formula:C23H27FN4O2Purezza:99.73%Colore e forma:Crystalline SolidPeso molecolare:410.48Ref: TM-T0351
10mg50,00€25mg59,00€50mg93,00€100mg128,00€200mg202,00€500mg340,00€1mL*10mM (DMSO)Prezzo su richiestaDopamine hydrochloride
CAS:Dopamine hydrochloride (ASL279) is a natural catecholamine neurotransmitter, dopamine receptors (D1-5 receptors) (EC50=2.7 nM). High-Quality, Low-Cost!Formula:C8H12ClNO2Purezza:99.47% - 99.72%Colore e forma:SolidPeso molecolare:189.64(-)-GSK598809 hydrochloride
CAS:<p>(-)-GSK598809 hydrochloride, a DRD3 selective antagonist, may correct reward deficits in substance dependence.</p>Formula:C22H24ClF4N5OSPurezza:98.36%Colore e forma:SoildPeso molecolare:517.97Quetiapine hemifumarate
CAS:Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.Formula:C46H54N6O8S2Purezza:99.32% - >99.99%Colore e forma:White Crystalline SolidPeso molecolare:883.09Clozapine
CAS:Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.Formula:C18H19ClN4Purezza:99.91% - 99.93%Colore e forma:Yellow Crystals From Acetone-Petroleum Ether SolidPeso molecolare:326.82Ref: TM-T0455
1g425,00€10mg34,00€25mg49,00€50mg66,00€100mg90,00€200mg161,00€500mg286,00€1mL*10mM (DMSO)44,00€Thioridazine hydrochloride
CAS:Thioridazine hydrochloride (Mellaril) , an antipsychotic drug, is used in the therapy of psychosis and schizophrenia and shows serotonin antagonism or D4Formula:C21H27ClN2S2Purezza:99.55% - 99.957%Colore e forma:White To Off-White SolidPeso molecolare:407.04Amisulpride
CAS:Amisulpride (Solian/Deniban), a dopamine antagonist antipsychotic, treats psychosis and schizophrenia in Europe/Australia, not in the US.Formula:C17H27N3O4SPurezza:99.97% - 99.99%Colore e forma:White Or Almost White Crystalline PowderPeso molecolare:369.48Tipepidine hydrochloride
CAS:Tipepidine hydrochloride: reversible DA D2 receptor inhibitor, IC50 7.0 μM, with antidepressant effects.Formula:C15H18ClNS2Purezza:99.97%Colore e forma:SolidPeso molecolare:311.89Ziprasidone
CAS:Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.Formula:C21H21ClN4OSPurezza:99.55%Colore e forma:Tan SolidPeso molecolare:412.94Oxidopamine hydrochloride
CAS:Oxidopamine hydrochloride (6-Hydroxydopamine hydrochloride) is an neurotransmitter dopamine antagonist.Formula:C8H12ClNO3Purezza:98.34% - 99.85%Colore e forma:Physical Description Beige Solid (Ntp 1992)Peso molecolare:205.64Tiapride hydrochloride
CAS:<p>Tiapride is a selective blocker of D2/3 dopamine receptors in the brain.</p>Formula:C15H24N2O4S·HClPurezza:99.4% - 99.77%Colore e forma:SolidPeso molecolare:364.89Loxapine succinate
CAS:Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.Formula:C22H24ClN3O5Purezza:99.69%Colore e forma:White To Of-White SolidPeso molecolare:445.9Spiperone
CAS:Spiperone (Spiropitan) is a spiro butyrophenone analog similar to HALOPERIDOL and other related compounds.Formula:C23H26FN3O2Purezza:99.34% - 99.91%Colore e forma:SolidPeso molecolare:395.47Blonanserin
CAS:Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.Formula:C23H30FN3Purezza:99.85%Colore e forma:SolidPeso molecolare:367.5Fluphenazine dihydrochloride
CAS:Fluphenazine dihydrochloride (Prolixin) is an inhibitor of phenothiazine-class D1DR and D2DR. Fluphenazine can be used to probe effects and metabolic process.Formula:C22H28Cl2F3N3OSPurezza:99.23%Colore e forma:Off-White SolidPeso molecolare:510.44Benztropine mesylate
CAS:<p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>Formula:C21H25NO·CH4SO3Purezza:98.41% - 99.96%Colore e forma:White Crystalline Powder; Odourless Or Almost OdourlessPeso molecolare:403.53Dexpramipexole dihydrochloride
CAS:Dexpramipexole dihydrochloride (KNS-760704 dihydrochloride) ((R)-Pramipexole dihydrochloride) is a neuroprotective agent and is a weak non-ergoline dopamineFormula:C10H19Cl2N3SPurezza:99.75% - 99.88%Colore e forma:SolidPeso molecolare:284.25Ref: TM-T11011
2mg35,00€5mg52,00€10mg79,00€25mg144,00€50mg216,00€100mg309,00€200mg462,00€1mL*10mM (DMSO)52,00€Acetophenazine dimaleate
CAS:Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor.Formula:C31H37N3O10SPurezza:99.39% - 99.48%Colore e forma:SolidPeso molecolare:643.71BP 897 hydrochloride
CAS:BP 897: potent D3 agonist (Ki: 0.92 nM), weak D2 antagonist (Ki: 61 nM), low affinity for D1/D4.Formula:C26H32ClN3O2Purezza:99.42%Colore e forma:SolidPeso molecolare:454Pipamperone
CAS:Pipamperone (McN-JR 3345) binds 5-HT2A closely as receptor.Formula:C21H30FN3O2Purezza:99.85%Colore e forma:White PowderPeso molecolare:375.48Ref: TM-T12480
1mg62,00€2mg85,00€5mg119,00€10mg170,00€25mg283,00€50mg430,00€100mg622,00€1mL*10mM (DMSO)131,00€Droperidol
CAS:Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as a Dopamine D2 Antagonist.Formula:C22H22FN3O2Purezza:97.16% - 98%Colore e forma:SolidPeso molecolare:379.43Benserazide hydrochloride
CAS:<p>Benserazide hydrochloride (Ro 4-4602) is a peripherally-acting L-amino acid decarboxylase (AAAD) or DOPA decarboxylase inhibitor.</p>Formula:C10H15N3O5·HClPurezza:98.63% - 99.74%Colore e forma:White Crystalline SolidPeso molecolare:293.7Bromperidol
CAS:Bromperidol (R-11333) is a butyrophenone derivative and it is a potent and long-acting neuroleptic.Formula:C21H23BrFNO2Purezza:99.89%Colore e forma:Tan SolidPeso molecolare:420.32Ziprasidone hydrochloride
CAS:Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychoticFormula:C21H22CL2N4OSPurezza:97.97% - 99.82%Colore e forma:SolidPeso molecolare:449.4Bendazol
CAS:<p>Bendazol (Dibazol) is always used as the drug for hypertension and cerebral Angiospasm.</p>Formula:C14H12N2Purezza:98.7% - 99.87%Colore e forma:White Or Almost White Crystalline PowderPeso molecolare:208.26Trifluoperazine dihydrochloride
CAS:Trifluoperazine dihydrochloride (SKF5019) is a potent dopamine D2 receptor inhibitor used as an antipsychotic and an antiemetic.Formula:C21H26Cl2F3N3SPurezza:99.57% - 99.96%Colore e forma:Cream Fine PowderPeso molecolare:480.43Tetrahydropalmatine
CAS:Tetrahydropalmatine (DL-Tetrahydropalmatine) is an active component isolated from corydalis, suppressing amygdaloid release of dopamine to inhibit an epilepticFormula:C21H25NO4Purezza:99.59% - 99.95%Colore e forma:SolidPeso molecolare:355.43Ziprasidone hydrochloride monohydrate
CAS:Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychoticFormula:C21H21ClN4OS·HCl·H2OPurezza:98% - 99.83%Colore e forma:Off-White PowderPeso molecolare:467.12Preclamol hydrochloride
CAS:Preclamol hydrochloride: selective dopamine agonist with research potential in schizophrenia.Formula:C14H22ClNOColore e forma:SolidPeso molecolare:255.78(R)-Preclamol hydrochloride
CAS:(R)-Preclamol HCl is a dopamine agonist stimulating both auto and postsynaptic receptors.Formula:C14H22ClNOColore e forma:SolidPeso molecolare:255.78D5R agonist 1
D5R Agonist 1 (Compound 5j) is a selective, orally active partial agonist of the D5 receptor that can penetrate the blood-brain barrier (EC50: 269.7 nM). It has been demonstrated to enhance cognitive abilities in a scopolamine-induced amnesia model.Colore e forma:Odour SolidHaloperidol D4
CAS:<p>Haloperidol D4 is deuterium-labeled haloperidol.</p>Formula:C21H23ClFNO2Purezza:98%Colore e forma:SolidPeso molecolare:379.89ABT 724 trihydrochloride
CAS:ABT-724 trihydrochloride: selective D4 agonist; EC50=12.4nM(human),14.3nM(rat),23.2nM(ferret); for erectile dysfunction research.Formula:C17H22Cl3N5Purezza:99.91%Colore e forma:SolidPeso molecolare:402.75Ref: TM-T22019
5mg40,00€10mg65,00€25mg126,00€50mg188,00€100mg283,00€200mg419,00€1mL*10mM (DMSO)44,00€Fenoldopam
CAS:Fenoldopam is a selective D1-like dopamine receptor partial agonist (EC50 = 57 nM).Formula:C16H16ClNO3Purezza:98%Colore e forma:SolidPeso molecolare:305.76Losulazine
CAS:<p>Losulazine: a new antihypertensive, requires functional sympathetic nervous system; mechanism undefined.</p>Formula:C27H22F4N4O3SPurezza:98.83%Colore e forma:SolidPeso molecolare:558.55Neurotransmitter Receptor Compound Library
<p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening;</p>Colore e forma:Odour Solid7-Hydroxy-PIPAT maleate
CAS:7-Hydroxy-PIPAT maleate is a D3R agonist.Formula:C16H22INOColore e forma:SolidPeso molecolare:371.262D3R/MOR antagonist 1
Compound 114 (D3R/MOR antagonist 1) exhibits dual antagonistic activity at dopamine D3 receptors (D3R) and mu-opioid receptors (MOR), with K i values of 46.5 nMFormula:C22H27Cl2N3OPurezza:98%Colore e forma:SolidPeso molecolare:420.38MOR agonist-2
Compound 46, designated as MOR agonist-2, serves as a D3R antagonist and a MOR agonist with respective K i values of 7.26 nM and 564 nM.Formula:C37H47Cl2N5O3Purezza:98%Colore e forma:SolidPeso molecolare:680.71Dopamine D2 receptor agonist-2
CAS:<p>Dopamine D2 receptor agonist-2 (Dopamine D2 Receptor) is a ligand targeting the dopamine D2 receptor.</p>Formula:C25H31Cl2N5OSPurezza:98.93%Colore e forma:SoildPeso molecolare:520.52A 77636 hydrochloride
CAS:<p>A 77636 hydrochloride is a potent, orally active, selective and long acting dopamine D1 receptor agonist (pKi=7.40; Ki=39.8 nM).</p>Formula:C20H28ClNO3Purezza:99.57%Colore e forma:SolidPeso molecolare:365.89Neuromedin N
CAS:Neuromedin N is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct expression and effects.Formula:C38H63N7O8Purezza:98%Colore e forma:SolidPeso molecolare:745.95[18F]-Labeled L-dopa precursor
CAS:[18F]-Labeled L-dopa precursor is a precursor for synthesis of 18F-labeled L-dopa[1].Formula:C35H36N2O7Colore e forma:SolidPeso molecolare:596.67Vanicoside E
CAS:Vanicoside E is an antioxidant and antitumor agent. Vanicoside E inhibits L-Tyrosine and L-DOPA with IC 50 s of 45.23 μM and 189.96 μM, respectively [1] [2] .Formula:C53H52O22Colore e forma:SolidPeso molecolare:1040.97Clomipramine D3
CAS:Clomipramine D3 is deuterium-labeled Clomipramine, blocking serotonin, norepinephrine, dopamine transporters (Ki: 0.14, 54, 3 nM).Formula:C19H23ClN2Purezza:98%Colore e forma:SolidPeso molecolare:317.87DETQ
CAS:DETQ enhances human D1 dopamine receptor signaling, EC50=5.8 nM, less effective in rats/mice, inactive on D5.Formula:C22H25Cl2NO3Colore e forma:SolidPeso molecolare:422.34S33084
CAS:S33084 is a potent, selective and competitive antagonist of dopamine D(3)-receptors.Formula:C29H29N3O2Purezza:98%Colore e forma:SolidPeso molecolare:451.56Cabergoline
CAS:<p>Cabergoline (FCE-21336), an ergot-derived dopamine D2-like agonist, targets D2/D3/5-HT2B, normalizes prolactin, controls pituitary tumors.</p>Formula:C26H37N5O2Purezza:97.69% - 99.86%Colore e forma:White Crystalline SolidPeso molecolare:451.6ADTN hydrobromide
CAS:<p>ADTN hydrobromide (6,7-ADTN) is a dopamine receptor agonist (EC50s = 3.5 and 0.65 μM in rat striatal and nucleus accumbens homogenates, respectively).</p>Formula:C10H14BrNO2Colore e forma:SolidPeso molecolare:260.13MOR agonist-3
MOR agonist-3 (Compound 84) is a dual D3R/MOR antagonist with K i values of 382 nM and 55.2 nM, respectively.Colore e forma:Odour SolidA 31472
CAS:A 31472 is a tetracyclic spiro amine that has affinity for dopamine D-2 receptors.Formula:C22H22ClNColore e forma:SolidPeso molecolare:335.87N-Methyl-2-phenylpropan-1-amine hydrochloride
CAS:N-Methyl-2-phenylpropan-1-amine hydrochloride is an analogue of β-methylphenethylamine (BMPEA) and demonstrates neurotransmitter-releasing properties in experiments involving NET and DAT.Formula:C10H16ClNPeso molecolare:185.69Adrogolide HCl
CAS:Adrogolide Hydrochloride is a selective dopamine receptor D1 agonist.Formula:C22H26ClNO4SColore e forma:SolidPeso molecolare:435.96D3R ligand 1
D3R Ligand 1 (compound 23b) is a potent, selective antagonist of the dopamine D3 receptor (Ki=66 nM), incorporating a THPB template.Formula:C27H37NO5Purezza:98%Colore e forma:SolidPeso molecolare:455.59MLS1082
CAS:MLS1082 is a D1-like dopamine receptor (D1R) orthosteric modulatothat stimulates G-protein signaling upon dopamine activation for neurodegenerative disorders.Formula:C24H23N3O2Purezza:99.53%Colore e forma:SolidPeso molecolare:385.46D3R/MOR antagonist 2
<p>Compound 121, a D3R/MOR antagonist with K i values of 361 nM and 85.2 nM for D3R and MOR respectively, has the potential for analgesic effects through MOR</p>Formula:C25H31ClN2OPurezza:98%Colore e forma:SolidPeso molecolare:410.98PF-4363467
CAS:PF-4363467 is a dopamine D3/D2 receptor antagonist that reduces opioid-seeking behavior without the side effects associated with D2 receptors. It has a Ki value of 3.1 nM for D3R and 692 nM for D2R.Formula:C22H30N2O3SColore e forma:SolidPeso molecolare:402.55Moperone
CAS:Moperone (R 1658) is an antagonist of both the D2 dopamine receptor (D2 dopamine receptor) and the D3 dopamine receptor (D3 dopamine receptor), with IC50 values for each of 1.0 nM.Formula:C22H26FNO2Colore e forma:SolidPeso molecolare:355.45Quinelorane
CAS:Quinelorane is dextrorotary isomer.Formula:C14H22N4Colore e forma:SolidPeso molecolare:246.35Secretoneurin, rat
CAS:Secretoneurin, rat, a 33-amino acid polypeptide, is generated by proteolytic processing of secretogranin II (SgII).Formula:C159H252N40O58Purezza:98%Colore e forma:SolidPeso molecolare:3651.95Fluphenazine free base
CAS:Flufenazine: antipsychotic for schizophrenia, blocks dopamine D2 receptors, reduces hallucinations and delusions.Formula:C22H26F3N3OSColore e forma:SolidPeso molecolare:437.52O-2172
CAS:O-2172 is a carbocyclic analogue serving as an inhibitor of dopamine transporter (DAT), exhibiting IC50 values of 47 nM for DAT and 7000 nM for the serotonin transporter (SERT).Formula:C14H16Cl2O2Colore e forma:SolidPeso molecolare:287.18Amisulpride hydrochloride
CAS:Amisulpride is an antagonist of 5-HT7 receptor and dopamine D2 and D3 receptors. It modulates beta 2- arresting signaling and increases neurite outgrowth.Formula:C17H28ClN3O4SColore e forma:SolidPeso molecolare:405.94Octodrine
CAS:Octodrine (2-Amino-6-methylheptane) is primarily used as a pharmaceutical intermediate for Octamylamine; it also functions as a local anesthetic and vasoconstrictor.Formula:C8H19NPurezza:99.98%Colore e forma:Clear Colorless To Light Yellow LiquidPeso molecolare:129.24ADTN
CAS:ADTN is an agonist of the dopamine receptor.Formula:C10H13NO2Purezza:98%Colore e forma:SolidPeso molecolare:179.22N-0500 HCl
CAS:N-0500 HCl, a potent DA receptor agonist, displaces [3H]DP_x005f_x0002_5,6-ADTN with an IC50 of 3nM.Formula:C15H22ClNO2Purezza:98.85% - 99.54%Colore e forma:SolidPeso molecolare:283.79LE 300
CAS:LE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.Formula:C20H22N2Purezza:97.91% - 98.79%Colore e forma:SolidPeso molecolare:290.4Trimethobenzamide
CAS:Trimethobenzamide (Ro 2-9578) is a D2 antagonist used to prevent nausea and vomiting.Formula:C21H28N2O5Colore e forma:SolidPeso molecolare:388.46ST-836 hydrochloride
CAS:ST-836 hydrochloride is a dopamine receptor ligand; Antiparkinsonian agent .Formula:C23H35ClN4OSPurezza:98%Colore e forma:SolidPeso molecolare:451.07Haloperidol (D4')
CAS:Haloperidol D4' is deuterium-labeled haloperidol. Haloperidol is a dopamine D2 receptor antagonist.Formula:C21H23ClFNO2Purezza:98%Colore e forma:SolidPeso molecolare:379.89Tiapride-d3
Tiapride-d3 is a deuterated form of Tiapride, a selective dopamine D2 receptor antagonist and an antipsychotic compound.Formula:C15H21D3N2O4SColore e forma:SolidPeso molecolare:331.45Eticlopride hydrochloride
CAS:Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM).Formula:C17H25ClN2O3·HClPurezza:98%Colore e forma:SolidPeso molecolare:377.31(-)-Apomorphine hydrochloride hydrate
CAS:(-)-Apomorphine hydrochloride hydrate is a broad-spectrum dopamine agonist and ferroptosis inhibitor.Formula:C17H17NO2HClXH2OColore e forma:SolidPeso molecolare:303.8SKF-82958 hydrobromide
CAS:SKF-82958 hydrobromide is a D1/D5 receptor full agonist.Formula:C19H21BrClNO2Purezza:98%Colore e forma:SolidPeso molecolare:410.73Docosahexaenoic acid ethyl ester
CAS:Docosahexaenoic acid ethyl ester (Ethyl docosahexaenoate) enhances 6-hydroxydopamine-induced neuronal damage by inducing lipid peroxidation in the mouse striatum, and can be used to study oxidative diseases of the retina or neurons.Formula:C24H36O2Purezza:98.35%Colore e forma:SolidPeso molecolare:356.54Clomipramine D3 hydrochloride
CAS:Clomipramine D3 hydrochloride is the deuterium-labeled Clomipramine. Clomipramine is a serotonin transporter, norepinephrine transporter dopamine transporter blocker (Ki: 0.14, 54 and 3 nM).Formula:C19H24Cl2N2Colore e forma:SolidPeso molecolare:354.333-O-Methyldopa-d3
CAS:3-O-Methyldopa-d3 is a deuterated compound of 3-O-Methyldopa. 3-O-Methyldopa has a CAS number of 300-48-1.Formula:C10H10D3NO4Peso molecolare:214.23Sumanirole maleate
CAS:Sumanirole maleate (PNU-95666E) is a D2 receptor full agonist with high selectivity that plays a vital role in Parkinson's disease and restless leg syndrome.Formula:C15H17N3O5Purezza:98%Colore e forma:SolidPeso molecolare:319.31GRK2 Inhibitor
CAS:GRK2 Inhibitor is an inhibitor of β-Adrenergic Receptor Kinase 1 (β ARK1).Formula:C12H9NO6Colore e forma:SolidPeso molecolare:263.2cis-(Z)-Flupentixol dihydrochloride
CAS:cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist.Formula:C23H27Cl2F3N2OSPurezza:98.07%Colore e forma:SolidPeso molecolare:507.44Pramipexole dihydrochloride
CAS:Pramipexole dihydrochloride could be used to treat Parkinson disease.Formula:C10H18ClN3SPurezza:98%Colore e forma:White Crystalline PowderPeso molecolare:247.79PD128907 HCl
CAS:PD128907 HCl is a potent and selective dopamine D3 receptor agonist, with EC50 of 0.64 nM, exhibits 53-fold selectivity over dopamine D2 receptor.Formula:C14H20ClNO3Purezza:98%Colore e forma:SolidPeso molecolare:285.77UCSF924
CAS:UCSF924 is a potent and specific agonist of dopamine D4 receptor (DRD4) partial (EC50: 4.2 nM, Ki: 3 nM).Formula:C20H22N2O2Purezza:98%Colore e forma:SolidPeso molecolare:322.4ABT-724
CAS:ABT-724 is an agonist of dopamine D4 receptor(EC50: 12.4 nM)Formula:C17H19N5Purezza:99.73%Colore e forma:SolidPeso molecolare:293.37Lurasidone hydrochloride
CAS:Lurasidone HCl: Atypical antipsychotic, treats schizophrenia & bipolar, affects dopamine, serotonin & adrenergic receptors.Formula:C28H36N4O2S·HClPurezza:99.51%Colore e forma:SolidPeso molecolare:529.14Ref: TM-T1735
5mg42,00€10mg63,00€25mg80,00€50mg96,00€100mg144,00€200mg225,00€500mg472,00€1mL*10mM (DMSO)Prezzo su richiestaPergolide
CAS:Pergolide is a long-acting and orally active dopamine receptor D1/D2 agonist and ergoline derivative, used in the study of Parkinson's diseaseFormula:C19H26N2SPurezza:99.95%Colore e forma:SolidPeso molecolare:314.49Ref: TM-T21340
2mg38,00€5mg57,00€10mg80,00€25mg116,00€50mg167,00€100mg250,00€200mg370,00€1mL*10mM (DMSO)64,00€Tavapadon
CAS:Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist.Formula:C19H16F3N3O3Purezza:99.33% - 99.8%Colore e forma:SolidPeso molecolare:391.34Ref: TM-T16999
1mg81,00€5mg170,00€10mg274,00€25mg502,00€50mg705,00€100mg938,00€1mL*10mM (DMSO)188,00€Neuromedin N acetate(92169-45-4 free base)
Neuromedin N acetate(92169-45-4 free base) is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinctFormula:C40H67N7O10Purezza:99.95%Colore e forma:SolidPeso molecolare:805.9Nomifensine maleate
CAS:<p>Nomifensine maleate (Nomifensine (maleate)) is a selective inhibitor of dopamine uptake. Nomifensine maleate is used in adult attention deficit disorder.</p>Formula:C20H22N2O4Purezza:98.46%Colore e forma:SolidPeso molecolare:354.4GBR 12935
CAS:GBR-12935: selective dopamine inhibitor, used in Parkinson's research.Formula:C28H34N2OColore e forma:SolidPeso molecolare:414.58Alizapride hydrochloride
CAS:Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting.Formula:C16H21N5O2·HClPurezza:99.35% - 99.48%Colore e forma:CoaPeso molecolare:351.83D-tetrahydropalmatine
CAS:D-Tetrahydropalmatine inhibits OCT1, reducing MCT uptake and hepatocyte damage in MDCK-hOCT1 cells and rat livers.Formula:C21H25NO4Purezza:99.34%Colore e forma:SolidPeso molecolare:355.43Ref: TM-T4S0779
2mg44,00€5mg64,00€10mg97,00€25mg182,00€50mg273,00€100mg393,00€200mg558,00€1mL*10mM (DMSO)65,00€Raclopride tartrate
CAS:Raclopride is a selective antagonist on D2 dopamine receptor ( D2 Ki: 1.8 nm, D3 Ki: 3.5 nm, D4 Ki: 2400, D1 Ki: 18000 nM).Formula:C19H26Cl2N2O9Colore e forma:SolidPeso molecolare:497.32Bisacodyl
CAS:Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for bowel evacuation.Formula:C22H19NO4Purezza:99.45% - 99.78%Colore e forma:Smaller Than 50 Microns Predominate White To Off-White Crystalline PowderPeso molecolare:361.39Dimethocaine
CAS:Dimethocaine (Larocaine) is a local anesthetic which also effects on the central nervous system acting as dopamine-reuptake-inhibitor.Formula:C16H26N2O2Purezza:99.52%Colore e forma:SolidPeso molecolare:278.39Ritanserin
CAS:Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.Formula:C27H25F2N3OSPurezza:99.77% - 99.89%Colore e forma:SolidPeso molecolare:477.57Bromocriptine mesylate
CAS:Bromocriptine mesylate (CB-154) is a potent dopamine receptor agonist that binds the D2 receptor with highest affinity (Ki = 2.5 nM)Formula:C33H44BrN5O8SPurezza:99.85% - 99.96%Colore e forma:White SolidPeso molecolare:750.7BisfluoroModafinil
CAS:CRL-40940 is a selective dopaminergic reuptake inhibitorFormula:C15H13F2NO2SPurezza:99.19%Colore e forma:SolidPeso molecolare:309.339-FLUORENOL
CAS:9-FLUORENOL is a dopamine reuptake inhibitor with IC50 of 9 μM, and a major metabolite of a compound developed as a wakefulness-promoting agent.Formula:C13H10OPurezza:99.98%Colore e forma:Off-White Crystalline PowderPeso molecolare:182.22Butyrophenone
CAS:Butyrophenone (NSC-8463) is a chemical compound. Some of its derivatives are used to treat various psychiatric disorders.Formula:C10H12OPurezza:99.84%Colore e forma:Colourless To Yellow LiquidPeso molecolare:148.2J-147
CAS:J-147, a curcumin derivative, is an experimental drug with reported effects against both Alzheimer's disease and ageing in mouse models of accelerated aging.Formula:C18H17F3N2O2Purezza:99.61% - >99.99%Colore e forma:SolidPeso molecolare:350.333-CPMT
CAS:3-CPMT (FC-1) is a dopamine uptake inhibitor and a potent long-acting antihistaminic agent.Formula:C21H25Cl2NOPurezza:99.03%Colore e forma:SolidPeso molecolare:378.33NGB 2904
CAS:NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).Formula:C28H29Cl2N3OPurezza:98.79%Colore e forma:SolidPeso molecolare:494.46Ref: TM-T28167
2mg40,00€5mg58,00€10mg90,00€25mg163,00€50mg279,00€100mg394,00€500mgPrezzo su richiesta1mL*10mM (DMSO)75,00€ML417
CAS:ML417 is a selective and brain penetrant agonist of D3 Dopamine (EC50 : 38 nM).Formula:C22H25N3O3Purezza:98.4% - 99.42%Colore e forma:SolidPeso molecolare:379.45SKF-83566
CAS:SKF-83566: Blood-brain permeable, orally active D1 dopamine antagonist; weaker 5-HT2 antagonist, Ki=11 nM.Formula:C17H18BrNOPurezza:95.00% - 99.82%Colore e forma:SolidPeso molecolare:332.23GSK163090
CAS:GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).Formula:C25H29N5OPurezza:99.2%Colore e forma:SolidPeso molecolare:415.53Ref: TM-TQ0311
1mg37,00€2mg52,00€5mg80,00€10mg125,00€25mgPrezzo su richiesta50mgPrezzo su richiesta1mL*10mM (DMSO)87,00€Metoclopramide
CAS:Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.Formula:C14H22ClN3O2Purezza:99.75%Colore e forma:SolidPeso molecolare:299.80Nomifensine
CAS:Nomifensine ((±)-Nomifensin) is a norepinephrine-dopamine reuptake inhibitor that prevents dopamine reuptake into synaptosomes.Formula:C16H18N2Purezza:99.83% - ≥95%Colore e forma:SolidPeso molecolare:238.33Propionylpromazine hydrochloride
CAS:Propionylpromazine hydrochloride (Propiopromazine hydrochloride) is a dopamine receptor D2 (DRD2) antagonist.Formula:C20H25ClN2OSPurezza:99.17%Colore e forma:SolidPeso molecolare:376.94Sultopride hydrochloride
CAS:Sultopride hydrochloride (LIN-1418 hydrochloride) is a selective dopamine D2 and D3 receptor antagonist.Formula:C17H27ClN2O4SPurezza:≥95%Colore e forma:White Or Yellowish PowderPeso molecolare:390.93Zotepine
CAS:Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,Formula:C18H18ClNOSPurezza:99.78%Colore e forma:SolidPeso molecolare:331.86Decynium 22
CAS:Decynium 22 is a plasma membrane monoamine transporter (PMAT) inhibitorFormula:C23H23IN2Purezza:99.92%Colore e forma:Dark Red CrystalsPeso molecolare:454.35Fenoldopam mesylate
CAS:Fenoldopam mesylate (Corlopam mesylate) is a selective dopamine-1 receptor (DA1) agonist with natriuretic/diuretic properties.Formula:C16H16ClNO3·CH4O3SPurezza:99.19% - 99.94%Colore e forma:SolidPeso molecolare:401.86GBR 12935 dihydrochloride
CAS:GBR 12935 dihydrochloride (GBR 12935) can induce the increase of the extracellular levels of dopamine to basal levels.Formula:C28H36Cl2N2OPurezza:99.09% - ≥95%Colore e forma:SolidPeso molecolare:487.5Cariprazine
CAS:<p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>Formula:C21H32Cl2N4OPurezza:99.68% - 99.87%Colore e forma:SolidPeso molecolare:427.41GSK 789472 hydrochloride
CAS:GSK 789472 hydrochloride is both a dopamine D3 receptor antagonist and a D2 partial agonist.Formula:C15H22ClN3OPurezza:99.89%Colore e forma:SolidPeso molecolare:295.81Chlorprothixene
CAS:Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.Formula:C18H18ClNSPurezza:98.77% - 99.756%Colore e forma:Pale Yellow Crystals SolidPeso molecolare:315.86Pramipexole dihydrochloride hydrate
CAS:Pramipexole dihydrochloride hydrate (Mirapex) is a selective, blood-brain barrier-crossing D2 dopamine receptor agonist, and is used in the study of PD.Formula:C10H17N3S·2HCl·H2OPurezza:99.68%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:302.26Ref: TM-T6951
10mg47,00€25mg74,00€50mg119,00€100mg170,00€200mg255,00€500mg430,00€1mL*10mM (DMSO)47,00€PD-168077 maleate
CAS:PD-168077 maleate is a selective agonist of dopamine D4 receptor(Ki : 9 nM)Formula:C24H26N4O5Purezza:99.13%Colore e forma:SolidPeso molecolare:450.49Ref: TM-T5047
2mg35,00€5mg52,00€10mg80,00€25mg150,00€50mg245,00€100mg364,00€200mg517,00€1mL*10mM (DMSO)58,00€Sonepiprazole mesylate
CAS:Sonepiprazole mesylate is a selective D4 antagonistFormula:C22H31N3O6S2Colore e forma:SolidPeso molecolare:497.63Azaperone
CAS:Azaperone, a sedative and antiemetic veterinary tranquilizer, belongs to pyridinylpiperazine and butyrophenone classes.Formula:C19H22FN3OPurezza:98.73%Colore e forma:White Or Off-White CrystallinePeso molecolare:327.4Ocaperidone
CAS:Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.Formula:C24H25FN4O2Purezza:99.33%Colore e forma:SolidPeso molecolare:420.48Brexpiprazole
CAS:Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.Formula:C25H27N3O2SPurezza:99.06% - 99.96%Colore e forma:SolidPeso molecolare:433.57Ref: TM-T2306
5mg50,00€10mg63,00€25mg75,00€50mg88,00€100mg94,00€200mg140,00€500mg259,00€1mL*10mM (DMSO)Prezzo su richiestaMetoclopramide dihydrochloride
CAS:Metoclopramide dihydrochloride is a dopamine D2 antagonist that is used as an antiemetic.Formula:C14H24Cl3N3O2Colore e forma:SolidPeso molecolare:372.72FAUC 346
CAS:FAUC 346 is a highly selective D3 partial agonist with EC50 of 1.5 nM.Formula:C24H29N3O2SPurezza:99.46%Colore e forma:SolidPeso molecolare:423.57Ref: TM-T9081
2mg35,00€5mg49,00€10mg81,00€25mg145,00€50mg235,00€100mg379,00€200mg517,00€1mL*10mM (DMSO)55,00€Diclofensine hydrochloride
CAS:Diclofensine hydrochloride (Ro 8-4650 hydrochloride) 是一种高效单胺再摄取抑制剂,在大鼠脑突触体中能够阻断多巴胺 (IC50=0.74 nM)、去甲肾上腺素 (IC50=2.3 nM) 和 5-羟色胺 (IC50=3.7 nM)。Formula:C17H18Cl3NOPurezza:98.86% - 99.93%Colore e forma:SolidPeso molecolare:358.69Fluphenazine decanoate
CAS:<p>Fluphenazine decanoate is dopamine D2 receptor blocke,and is a long-acting phenothiazine neuroleptic that used to treat schizophrenia.</p>Formula:C32H44F3N3O2SPurezza:98.14%Colore e forma:SolidPeso molecolare:591.77Aplindore
CAS:Aplindore is a dopamine receptor agonist used in the therapeutic treatment of Parkinson's Disease.Formula:C18H18N2O3Colore e forma:SolidPeso molecolare:310.35Fluoroclebopride
CAS:Fluoroclebopride is a dopamine (DA) D2 receptor ligand.Formula:C20H23ClFN3O2Purezza:99.68% - 99.91%Colore e forma:SolidPeso molecolare:391.87Ref: TM-T3187
1mg35,00€5mg74,00€10mg96,00€25mg159,00€50mg235,00€100mg376,00€500mg867,00€1mL*10mM (DMSO)96,00€L-745870 trihydrochloride
CAS:<p>L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.</p>Formula:C18H22Cl4N4Purezza:97.52%Colore e forma:SolidPeso molecolare:436.21Rotundine
CAS:Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.Formula:C21H25NO4Purezza:99.8% - 99.91%Colore e forma:Off-White SolidPeso molecolare:355.43Valbenazine dihydrochloride
CAS:Valbenazine dihydrochloride inhibits vesicular monoamine transporter 2 (VMAT2); used to treat tardive dyskinesia.Formula:C24H40Cl2N2O4Colore e forma:SolidPeso molecolare:491.49FAUC 213
CAS:<p>FAUC 213 is a selective full antagonist of the dopamine D4 receptor.</p>Formula:C18H19ClN4Purezza:99.84%Colore e forma:SolidPeso molecolare:326.82Piribedil
CAS:Piribedil (Trivastan) is a dopamine D2 agonist, used in the treatment of Parkinson's disease.Formula:C16H18N4O2Purezza:99.79% - 99.82%Colore e forma:SolidPeso molecolare:298.34Lurasidone
CAS:Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6Formula:C28H36N4O2SPurezza:99.78% - 99.91%Colore e forma:SolidPeso molecolare:492.68SKF38393 hydrobromide
CAS:SKF38393 hydrobromide is the salt form of SKF38393.a dopamine D1 receptor agonist that increases the expression of Shati/Nat8L mRNA in the NAc of mice;Formula:C16H18BrNO2Purezza:98.99%Colore e forma:SolidPeso molecolare:336.22Rimcazole
CAS:Rimcazole is a sigma receptor antagonist. It also binds to the dopamine transporter and inhibiting dopamine uptake.Formula:C21H27N3Purezza:98%Colore e forma:SolidPeso molecolare:321.46Dasotraline
CAS:Dasotraline: a triple reuptake inhibitor targeting DA, NE, and 5-HT with IC50 values of 4, 6, 11 nM. Possible new antidepressant class.Formula:C16H15Cl2NColore e forma:SolidPeso molecolare:292.2Haloperidol hydrochloride
CAS:Haloperidol hydrochloride is a potent dopamine D2 receptor antagonist which is a potent antipsychotic agent.Formula:C21H24Cl2FNO2Colore e forma:SolidPeso molecolare:412.33PD 168568
CAS:PD 168568: Oral DRD4 antagonist, selective over D2/D3, K_i - 8.8 nM. Used in GBM research.Formula:C22H27N3OColore e forma:SolidPeso molecolare:349.47Alizapride
CAS:Alizapride is an antagonist of dopamine receptor. Alizapride can be used in human digestive disorders which is a potent antiemetic [1] [3].Formula:C16H21N5O2Colore e forma:SolidPeso molecolare:315.37OS-3-106
CAS:OS-3-106 is a novel arylamide phenylpiperazines, as partial agonists at the D3R in the adenylyl cyclase inhibition assay.Formula:C25H30N4O2SPurezza:99.4% - 99.57%Colore e forma:SolidPeso molecolare:450.6JNJ-37822681
CAS:JNJ-37822681 is a novel, highly selective dopamine D₂ receptor antagonist characterized by a rapid dissociation rate from the dopamine D₂ receptor.Formula:C17H17F5N4Purezza:99.84%Colore e forma:SolidPeso molecolare:372.34Ansofaxine hydrochloride
CAS:Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).Formula:C24H32ClNO3Purezza:99.57% - 99.77%Colore e forma:SolidPeso molecolare:417.97Tiapride
CAS:Tiapride, an atypical neuroleptic, is a selective dopamine D2-receptor antagonist with varying IC50 values for D1-D4.Formula:C15H24N2O4SColore e forma:SolidPeso molecolare:328.43Rotigotine Hydrochloride
CAS:<p>Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.</p>Formula:C19H26ClNOSPurezza:99.53% - 99.56%Colore e forma:Almost White To White Crystalline PowderPeso molecolare:351.93Pergolide mesylate
CAS:Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.Formula:C20H30N2O3S2Purezza:99.70%Colore e forma:White To Off-White SolidPeso molecolare:410.59BP 897
CAS:BP 897: potent selective dopamine D3 agonist, weak D2 antagonist. Ki: 0.92 nM (D3), 61 nM (D2), low affinity at D1/D4.Formula:C26H31N3O2Purezza:99.44%Colore e forma:SolidPeso molecolare:417.54Ref: TM-T9100
1mg80,00€5mg162,00€10mg227,00€25mg379,00€50mg540,00€100mg730,00€200mg938,00€1mL*10mM (DMSO)177,00€Rotigotine-
CAS:Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.Formula:C19H25NOSPurezza:98.08% - 99.59%Colore e forma:SolidPeso molecolare:315.47Ref: TM-T6647
5mg52,00€10mg78,00€25mg145,00€50mg255,00€100mg378,00€200mg552,00€500mg868,00€1mL*10mM (DMSO)55,00€Perospirone
CAS:Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.Formula:C23H30N4O2SPurezza:99.23%Colore e forma:White PowderPeso molecolare:426.57carfenazine
CAS:<p>carfenazine targets the Dopamine receptor and is used for schizophrenia research.</p>Formula:C24H31N3O2SPurezza:98.06%Colore e forma:SolidPeso molecolare:425.59Sonepiprazole hydrochloride
CAS:Sonepiprazole HCl is a a selective dopamine D4 antagonist.Formula:C21H28ClN3O3SColore e forma:SolidPeso molecolare:437.98SK609
CAS:SK609: selective dopamine D3 agonist; enhances impaired paw function, corrects asymmetry in hemiparkinson rats.Formula:C10H14ClNColore e forma:SolidPeso molecolare:183.68Nuciferine
CAS:Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.Formula:C19H21NO2Purezza:98.76% - 99.79%Colore e forma:SolidPeso molecolare:295.38Raclopride
CAS:Raclopride is a selective antagonist of dopamine D2/D3 receptor.Formula:C15H20Cl2N2O3Purezza:99.17%Colore e forma:SolidPeso molecolare:347.24Haloperidol lactate
CAS:Haloperidol lactate: a potent antipsychotic for acute/chronic schizophrenia and polyarousal syndrome research.Formula:C24H29ClFNO5Colore e forma:SolidPeso molecolare:465.95L-DOPA methyl ester (hydrochloride)
CAS:<p>L-DOPA methyl ester (LDME) is an agonist of dopamine D1 receptor.</p>Formula:C10H14ClNO4Purezza:98.69% - 99.81%Colore e forma:White SolidPeso molecolare:247.675Tetrahydropalmatine hydrochloride
CAS:Tetrahydropalmatine HCl (Gindarine) is a muscle relaxant alkaloid from Corydalis plants.Formula:C21H26ClNO4Purezza:98% - 99.59%Colore e forma:SolidPeso molecolare:391.888Zuclopenthixol dihydrochloride
CAS:Zuclopenthixol dihydrochloride is an D1 and D2 dopamine receptors antagonist.Formula:C22H27Cl3N2OSPurezza:98%Colore e forma:SolidPeso molecolare:473.89AHN 1-055 hydrochloride
CAS:AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).Formula:C21H24ClF2NOPurezza:99.89%Colore e forma:SolidPeso molecolare:379.87Ref: TM-T39429
2mg35,00€5mg52,00€10mg80,00€25mg137,00€50mg202,00€100mg311,00€200mg467,00€1mL*10mM (DMSO)52,00€Clebopride
CAS:Clebopride is antidopaminergic. Clebopride also has an effect of antiemetic.Formula:C20H24ClN3O2Colore e forma:SolidPeso molecolare:373.88L-745870 hydrochloride
CAS:L-745870 hydrochloride has excellent brain penetration. L-745870 hydrochloride is a high-affinity, selective and orally active human dopamine D4 receptorFormula:C18H20Cl2N4Purezza:97.36%Colore e forma:SolidPeso molecolare:363.28Ref: TM-T11799
5mg40,00€10mg65,00€25mg111,00€50mg178,00€100mg259,00€200mg374,00€1mL*10mM (DMSO)34,00€Vanoxerine dihydrochloride
CAS:Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) is a potent inhibitor that blocks dopamine uptake (IC50 : 1-51 nM)Formula:C28H34Cl2F2N2OPurezza:98.16% - 98.35%Colore e forma:White SolidPeso molecolare:523.49Domperidone monomaleate
CAS:Domperidone monomaleate, a selective oral dopamine-2 antagonist, aids gastric motility and has antiemetic properties.Formula:C26H28ClN5O6Colore e forma:SolidPeso molecolare:541.98Mesdopetam
CAS:Mesdopetam (IRL790), a D3 antagonist, has Ki=90 nM, IC50=9.8 μM, stabilizes psychomotors, used in Parkinson's research.Formula:C12H18FNO3SColore e forma:SolidPeso molecolare:275.34Metergoline
CAS:Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.Formula:C25H29N3O2Purezza:99.83% - 99.97%Colore e forma:SolidPeso molecolare:403.52Bromopride hydrochloride
CAS:Bromopride HCl: Salt of a D2 blocker used for upper GI disorders, like dyspepsia and emesis.Formula:C14H23BrClN3O2Colore e forma:SolidPeso molecolare:380.71

