Recettore dell'adenosina
I recettori dell'adenosina sono una classe di GPCR che rispondono al nucleoside endogeno adenosina. Questi recettori sono coinvolti nella regolazione di vari processi fisiologici, tra cui la funzione cardiovascolare, i cicli sonno-veglia e le risposte immunitarie. I modulatori dei recettori dell'adenosina hanno un potenziale terapeutico nel trattamento di condizioni come le aritmie cardiache, l'infiammazione e le malattie neurodegenerative. Presso CymitQuimica, offriamo una selezione di modulatori dei recettori dell'adenosina di alta qualità per supportare la tua ricerca in biologia cardiovascolare, neuroscienze e immunologia.
Trovati 218 prodotti per "Recettore dell'adenosina".
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A2A receptor antagonist 2
A2A receptor antagonist 2 is a highly selective and potent antagonist of the adenosine A2Areceptor (IC50: 8.3 nM).Formula:C25H28FN7O3Colore e forma:SolidPeso molecolare:493.53DMPX
CAS:DMPX (3,7-Dimethyl-1-propargylxanthine) is a caffeine-like compound capable of crossing the blood-brain barrier. It serves as an A2-selective adenosine receptor (AR) antagonist, effectively and selectively blocking the hypothermia and behavioral inhibition induced by A2 adenosine receptor agonists, such as NECA. DMPX is utilized in research on diseases like Parkinson's disease.Formula:C10H10N4O2Colore e forma:SolidPeso molecolare:218.212Neladenoson
CAS:Neladenoson is an effective and selective agonist of the Adenosine A1 Receptor (A1R). EGFR-IN-162 shows potential for research in heart failure.Formula:C29H24ClN5O2S2Colore e forma:SolidPeso molecolare:574.12M1069
M1069 is an oral A2A/A2B receptor antagonist, 100x more selective over A1/A3, with antitumor properties by blocking adenosine's immunosuppressive effects.Formula:C25H30N4O8SColore e forma:SolidPeso molecolare:546.59Zaladenant
CAS:Zaladenant is an adenosine receptor antagonist with antitumor properties.Formula:C19H15F3N6OColore e forma:SolidPeso molecolare:400.357N-(7H-Purin-6-yl)acetamide
CAS:N-(7H-Purin-6-yl)acetamide (Compound 25) is a selective adenosine receptor (AdeR) agonist with a Ki value of 0.515 μM for human adenosine receptors and 2.85 μM for rat adenosine receptors. It shows potential for research into adenosine receptor function, pain perception, inflammatory response, and kidney function.Formula:C7H7N5OPeso molecolare:177.1634ATL444
CAS:ATL444 is an adenosine receptor antagonist with affinity (Ki values) for rA1AR, rA2AAR, rA2BAR, and rA3AR of 7.0, 2.5, 61.8, and >1000 nM, respectively.Formula:C17H19N5OColore e forma:SolidPeso molecolare:309.37PSB 36
CAS:A1 adenosine receptor antagonistFormula:C21H30N4O3Purezza:98%Colore e forma:SolidPeso molecolare:386.49A3AR antagonist 5
CAS:A3AR antagonist 5 (Compound 16) acts as a selective antagonist for the human adenosine A3 receptor (human adenosine A3 receptor), with an affinity expressed as a pC value of 4.542 μM.Formula:C18H16N2O2SColore e forma:SolidPeso molecolare:324.40L-97-1
CAS:L-97-1 is an antagonist of the adenosine A1 receptor.Formula:C29H38N6O3Purezza:98%Colore e forma:SolidPeso molecolare:518.65MSX-3
CAS:MSX-3 is an antagonist of the A2A adenosine receptor and a prodrug of MSX-2.Formula:C21H23N4Na2O7PPurezza:98%Colore e forma:SolidPeso molecolare:520.389Tonapofylline
CAS:Tonapofylline, orally active, selectively blocks A1 adenosine receptor (Ki: 7.4 nM), used in heart failure research.Formula:C22H32N4O4Purezza:98.57%Colore e forma:SolidPeso molecolare:416.51MRS 5980
CAS:MRS 5980, an A3AR agonist with a K i value of 0.7 nM, exhibits oral activity [1].Formula:C20H19ClN6O3SColore e forma:SolidPeso molecolare:458.92KF26777
CAS:KF26777 is a potent and selective antagonist of adenosine A3 receptor.Formula:C16H16BrN5OPurezza:98%Colore e forma:SolidPeso molecolare:374.23LJ-4517
LJ-4517 is an effective A2AAR antagonist (Ki=18.3 nM). LJ-4517 can effectively replace the binding of [3H] ZM241385 at WT A2AAR.Formula:C19H21N5O3SColore e forma:SolidPeso molecolare:399.47A1/A3 AR antagonist 1
Compound 10 is a potent dual A1/A3 AR antagonist, with Ki values of 37.6 nM (hA1), 25.4 nM (hA3), and 1.47 nM (rA1), studied in renal, lung, and Alzheimer's.Formula:C24H18N2O3SColore e forma:SolidPeso molecolare:414.48A2A receptor antagonist 3
CAS:A2A receptor antagonist 3 (Example 92) is an adenosine A2a receptor antagonist (Ki: 0.4 nM). receptor (Ki: 1467 nM).Formula:C26H26N6O2Purezza:99.58%Colore e forma:SolidPeso molecolare:454.52hA3AR agonist 1
hA3AR agonist 1 is a potent human A 3 adenosine receptor (hA 3 AR) agonist (Ki = 2.40 nM) .Formula:C10H14N6OSColore e forma:SolidPeso molecolare:266.32
