
Recettore dell'adenosina
I recettori dell'adenosina sono una classe di GPCR che rispondono al nucleoside endogeno adenosina. Questi recettori sono coinvolti nella regolazione di vari processi fisiologici, tra cui la funzione cardiovascolare, i cicli sonno-veglia e le risposte immunitarie. I modulatori dei recettori dell'adenosina hanno un potenziale terapeutico nel trattamento di condizioni come le aritmie cardiache, l'infiammazione e le malattie neurodegenerative. Presso CymitQuimica, offriamo una selezione di modulatori dei recettori dell'adenosina di alta qualità per supportare la tua ricerca in biologia cardiovascolare, neuroscienze e immunologia.
Trovati 249 prodotti di "Recettore dell'adenosina"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Xanthine amine congener trihydrochloride
CAS:Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.Formula:C21H29ClN6O4Purezza:98.81%Colore e forma:SolidPeso molecolare:464.95N6-Benzyl-5'-ethylcarboxamido adenosine
CAS:N6-Benzyl-5'-ethylcarboxamido adenosine is a selective A3 adenosine receptor agonist.Formula:C19H22N6O4Colore e forma:SolidPeso molecolare:398.428-Chloro caffeine
CAS:8-Chloro caffeine binds to adenosine receptors with a Ki of 30 µM. It enhances UV-induced chromosomal aberrations in the Cl-I type Chinese hamster embryo lung cells. 8-Chloro caffeine is a derivative of the methylxanthine alkaloid caffeine.Formula:C8H9ClN4O2Colore e forma:SolidPeso molecolare:228.64hA3AR agonist 2
hA3AR agonist 2 is a potent activator of A3AR, with a Ki value of 3.5 nM.Formula:C11H14ClN5O2SColore e forma:SolidPeso molecolare:315.78Apadenoson TFA
<p>Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.</p>Formula:C25H31F3N6O8Purezza:98.08%Colore e forma:SoildPeso molecolare:600.55A2A/A3 AR antagonist-1
A2A/A3 AR antagonist-1 is a dual fluorescent AR ligand with K i of 90 nM (hA2A) & 31.8 nM (hA3).Formula:C56H71N15O12S2Colore e forma:SolidPeso molecolare:1210.39MRS-3777 hemioxalate
CAS:<p>MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its corresponding agonist and serves as a valuable tool for studying inflammatory pain.</p>Formula:C17H19N5OC2H2O4Purezza:97.10%Colore e forma:SolidPeso molecolare:354.39(Rac)-Mirabegron-d5
CAS:(Rac)-Mirabegron D5 is a deuterium labeled (Rac)-Mirabegron. Mirabegron is a selective agonist of β3-adrenoceptor.Formula:C21H24N4O2SPurezza:98%Colore e forma:SolidPeso molecolare:401.54LAS101057
CAS:LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.Formula:C18H14FN5OPurezza:99.03% - >99.99%Colore e forma:SolidPeso molecolare:335.34GR79236
CAS:GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.Formula:C15H21N5O5Colore e forma:SolidPeso molecolare:351.36Theophylline-d6
CAS:Theophylline-d6, an internal standard for theophylline quantification in GC/LC-MS, relaxes bronchial muscles and treats asthma/COPD.Formula:C7H2D6N4O2Peso molecolare:186.2Norisoboldine
CAS:<p>Norisoboldine, potential rheumatoid arthritis therapy, protects joints and modulates immunity by inhibiting MAPKs, not NF-κB.</p>Formula:C18H19NO4Purezza:98.12% - 99.7%Colore e forma:SolidPeso molecolare:313.35Taminadenant
CAS:Taminadenant is an adenosine receptor antagonist.Formula:C10H8BrN7Purezza:99.11%Colore e forma:SolidPeso molecolare:306.125'-N-Ethylcarboxamidoadenosine
CAS:NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.Formula:C12H16N6O4Purezza:98.95% - ≥95%Colore e forma:PowderPeso molecolare:308.29Namodenoson
CAS:Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.Formula:C18H18ClIN6O4Purezza:98.97%Colore e forma:SolidPeso molecolare:544.73N6,N6-Dimethyladenosine
CAS:<p>N6,N6-Dimethyladenosine is find in mycobacterium bovis Bacille Calmette-Guérin tRNA.</p>Formula:C12H17N5O4Purezza:98.79%Colore e forma:White PowderPeso molecolare:295.29VPC171
CAS:VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).Formula:C18H12F3NOSPurezza:99.78%Colore e forma:SolidPeso molecolare:347.35BAY-545
CAS:BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).Formula:C18H22F3N3O4SPurezza:98.05%Colore e forma:SolidPeso molecolare:433.45Preladenant
CAS:<p>Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosine</p>Formula:C25H29N9O3Purezza:98.02% - 99.68%Colore e forma:SolidPeso molecolare:503.56Swertisin
CAS:Swertisin: an herbal molecule with antihyperglycemic, antidiabetic, anti-inflammatory, and antioxidant properties; blocks adenosine A1 receptor.Formula:C22H22O10Purezza:99.74% - 99.89%Colore e forma:SolidPeso molecolare:446.40

