Recettore dei cannabinoidi
I recettori dei cannabinoidi sono GPCR che mediano gli effetti dei cannabinoidi endogeni (endocannabinoidi) e fitocannabinoidi, come quelli presenti nella cannabis. I due principali tipi di recettori dei cannabinoidi, CB1 e CB2, sono coinvolti nella regolazione di una vasta gamma di processi fisiologici, tra cui la percezione del dolore, l'appetito, l'umore e la funzione immunitaria. I modulatori dei recettori dei cannabinoidi hanno un potenziale terapeutico nel trattamento di condizioni come il dolore cronico, l'epilessia e la sclerosi multipla. Presso CymitQuimica, offriamo una vasta gamma di modulatori di recettori dei cannabinoidi di alta qualità per supportare la tua ricerca in neurofarmacologia, gestione del dolore e immunologia.
Trovati 217 prodotti di "Recettore dei cannabinoidi"
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PGN36
CAS:PGN36 (Compound 18) is a potent CB2 receptor antagonist with a high affinity (Ki=0.09 μM).Formula:C21H23N3O3Colore e forma:SolidPeso molecolare:365.43CB1R Allosteric modulator 4
CAS:Modulates CB1R positively; inhibits cAMP production; strong β-arrestin-2 recruitment.Formula:C20H17N3O2SColore e forma:SolidPeso molecolare:363.43CB1R Allosteric modulator 2
CAS:Compound 18 is a potent CB1R allosteric modulator that acts as a negative modulator (NAM) for CB1R orthosteric ligands.Formula:C19H15ClFN3OColore e forma:SolidPeso molecolare:355.79GAT229
CAS:GAT229 is a CB1 positive modulator, enhancing CB agonist activity without direct activation; influences binding, signaling, and lowers ocular pressure in mice.Formula:C22H18N2O2Colore e forma:SolidPeso molecolare:342.39CB1-IN-2
CAS:CB1-IN-2 (4g) inhibits CB1 receptor with 0.644 μM IC50; crosses blood-brain barrier, may cause CNS side effects like Rimonabant.Formula:C17H19Cl2N5OColore e forma:SolidPeso molecolare:380.27COR167
CAS:COR167 is a CB2 agonist with immunomodulatory effects, protective brain properties, and antinociception.Formula:C28H38N2O2Colore e forma:SolidPeso molecolare:434.61UCM 707
CAS:endocannabinoid transport inhibitorFormula:C25H37NO2Purezza:98%Colore e forma:SolidPeso molecolare:383.57SMM-189
CAS:SMM-189 is a potent and selective CB2 inverse agonist.Formula:C19H12Cl2O3Colore e forma:SolidPeso molecolare:359.2CAY10412
CAS:Anandamide (AEA) is an endocannabinoid with neural reuptake. CAY10412, an AEA analog, inhibits this reuptake without binding to CB receptors.Formula:C25H36O2SColore e forma:SolidPeso molecolare:400.62(S)-SLV 319
CAS:Ibipinabant (SLV319), a potent CB1 antagonist, K i = 7.8 nM, >1000x selective over CB2, for obesity and diabetic research.Formula:C23H20Cl2N4O2SColore e forma:SolidPeso molecolare:487.4LEI-101
CAS:LEI-101: potent CB2 agonist, pEC50=8, bioavailable, >100x selective over CB1, potential for inflammatory diseases.Formula:C23H25FN4O4SPurezza:98%Colore e forma:SolidPeso molecolare:472.53Palmitoyl serinol
CAS:Anticancer agent 110 is an anticancer compound with cytotoxic, antitumor and antileukemic activities.Formula:C19H39NO3Colore e forma:SolidPeso molecolare:329.52ZCZ011
CAS:ZCZ011 enhances CB1 receptor effects, crosses blood-brain barrier, and potentiates cannabimimetic behaviors in mice.Formula:C21H18N2O2SPurezza:98%Colore e forma:SolidPeso molecolare:362.44KLS-13019
CAS:KLS-13019 is a highly effective and orally active GPR55 receptor antagonist, neuroprotective can reverse chemotherapy-induced peripheral neuropathy (CIPN).Formula:C22H29NO3Purezza:>99.99% - >99.99%Colore e forma:SolidPeso molecolare:355.47LEI 101 hydrochloride
CAS:LEI 101 hydrochloride is potent and selective CB2 partial agonist.Formula:C23H26ClFN4O4SColore e forma:SolidPeso molecolare:508.99OMDM-6
CAS:OMDM-6 is a dual agonist of TRPV1(EC50 = 75 nM) and CB1 (Ki = 3.2 μM). OMDM-6 inhibits anandamide cellular uptake with a Ki of 7.0 μM.Formula:C28H42N2O3Purezza:99.66%Colore e forma:SolidPeso molecolare:454.64Ref: TM-T12307
1mg89,00€5mg178,00€10mg264,00€25mg393,00€50mg552,00€100mg752,00€200mg1.008,00€1mL*10mM (DMSO)197,00€Virodhamine trifluoroacetate
CAS:Virodhamine trifluoroacetate: full GPR55 & CB2 agonist, partial CB1 antagonist, cannabinoid receptor mixed antagonist.Formula:C24H38F3NO4Purezza:98%Colore e forma:SolidPeso molecolare:461.56LBP-1
CAS:LBP-1 is a cannabinoid receptor type 1 (CB1) agonist.Formula:C23H29ClN6O3Colore e forma:SolidPeso molecolare:472.97N-Arachidonyldopamine
CAS:N-Arachidonyldopamine (NADA) is a selective and potent endogenous CB1 receptor agonist (Ki: 250 nM).N-Arachidonyldopamine is also a potent and selective TRPV1Formula:C28H41NO3Purezza:97.65%Colore e forma:SolidPeso molecolare:439.632-Arachidonoylglycerol
CAS:In the central nervous system, 2-Arachidonoylglycerol is a second endogenous cannabinoid ligandFormula:C23H38O4Purezza:95%Colore e forma:LiquidPeso molecolare:378.55GPR55 agonist 3
CAS:Compound 26, a GPR55 agonist, exhibits potent activity with EC50 values of 0.239 nM for hGPR55 and 1.76 nM for rGPR55.Formula:C19H16F4N4Colore e forma:SolidPeso molecolare:376.35AM404
CAS:AM404 is a cannabinoid reuptake inhibitor and a TRPV (1) activator with neuroprotective and anticancer activities that blocks anandamide transport.Formula:C26H37NO2Colore e forma:SolidPeso molecolare:395.58CB2 modulator 1
CAS:CB2 modulator 1 is a potent CB2 modulator. It can be used for the research for immune disorders, osteoporosis, inflammation, renal ischemia.Formula:C18H19F3N4O2Purezza:99.6%Colore e forma:SolidPeso molecolare:380.36MJ 15
CAS:MJ 15 is a CB1 receptor antagonist with specificity for the study of obesity-induced diseases.Formula:C23H17Cl3N4OPurezza:99.63%Colore e forma:SolidPeso molecolare:471.77CB1/2 agonist 4
CAS:CB1/2 agonist 4 is a potent CB1 full agonist (EC50: 15.09 nM) and CB2 partial agonist (EC50: 1.16 nM), with anti-pain and TRPV1 activation properties.Formula:C27H45NO3Colore e forma:SolidPeso molecolare:431.65CB1R Allosteric modulator 1
CAS:CB1R modulator 1 (compound 11), a potent CB1R inhibitor, decreases activity of orthosteric ligands.Formula:C24H24ClN3OColore e forma:SolidPeso molecolare:405.92UCM710
CAS:UCM710 is a dual inhibitor of α/β hydrolase domain 6 (ABHD6) and fatty acid amide hydrolase (FAAH).Formula:C19H34O3Purezza:98%Colore e forma:SolidPeso molecolare:310.47MM-22
CAS:biotinylated anandamide analog acts as a probe for visualizing the accumulation and intracellular trafficking of anandamideFormula:C36H60N4O5SPurezza:98%Colore e forma:SolidPeso molecolare:660.95CB2R agonist 1
CAS:CB2R agonist 1 selectively binds human CB2R, EC50 of 0.56 µM, modulates inflammatory cytokines.Formula:C22H32N2OColore e forma:SolidPeso molecolare:340.5S-777469
CAS:S-777469: Selective CB2 agonist, oral, inhibits itching in mice (Ki: 36 nM). Anti-pruritic.Formula:C23H27FN2O4Colore e forma:SolidPeso molecolare:414.47PM226
CAS:CB2 agonist with Ki of 12.8 nM; EC50 of 38.67 nM. Negligible CB1 affinity, no GPR55 activity. Anti-inflammatory, neuroprotective, crosses BBB.Formula:C22H31NO3Colore e forma:SolidPeso molecolare:357.49AZD-2207
CAS:AZD-2207 is a cannabinoid receptor CB1 antagonist and highly lipophilic compound for the treatment of type 2 diabetes mellitus and obesity.Formula:C25H25Cl2F3N4O4SColore e forma:SolidPeso molecolare:605.46Cannabicitran
CAS:Cannabicitran is a cannabinoid that can decrease rabbits intraocular pressure [1] [2].Formula:C21H30O2Colore e forma:SolidPeso molecolare:314.46CB1 inverse agonist 2
CAS:CB1 inverse agonist 2, an oral drug, counters CB1 effects, reducing CP55940-induced hypothermia and anorexia in mice.Formula:C24H20ClFN2OSColore e forma:SolidPeso molecolare:438.94GAT228
CAS:GAT228, an allosteric ligand for the cannabinoid receptor 1 (CB1), functions as the enantiomer of GAT211 [1].Formula:C22H18N2O2Colore e forma:SolidPeso molecolare:342.39AM-6538
CAS:AM6538: long-acting, high-affinity CB antagonist similar to rimonabant, useful for studying cannabinoid agonists.Formula:C26H25Cl2N5O4Colore e forma:SolidPeso molecolare:542.41COR 170
CAS:<p>inverse agonist of CB2 receptors</p>Formula:C31H36N2O2Purezza:98%Colore e forma:SolidPeso molecolare:468.63NIDA 41020
CAS:NIDA 41020 is a CB1 receptor antagonist.Formula:C23H24Cl2N4O2Purezza:98%Colore e forma:SolidPeso molecolare:459.37LH 21
CAS:LH-21, a strong CB1 receptor antagonist, curbs eating and lessens weight gain in obese rats.Formula:C20H20Cl3N3Colore e forma:SolidPeso molecolare:408.75CID1792197
CAS:CID1792197 is a selective agonist of GPR55.Formula:C24H23N3O4S2Purezza:98%Colore e forma:SolidPeso molecolare:481.59O-2093
CAS:anandamide uptake inhibitorFormula:C34H43Cl2NO3Purezza:98%Colore e forma:SolidPeso molecolare:584.62CID1172084
CAS:CID1172084, a novel high-potent GPR55 agonist, interacts with cannabinoid receptors.Formula:C23H18FN5O2S2Colore e forma:SolidPeso molecolare:479.55CB2 receptor agonist 3
CAS:GP 2A is a selective agonist of CB2 receptor.Formula:C24H23Cl2N3OColore e forma:SolidPeso molecolare:440.36TC-C 14G
CAS:CB1 receptor inverse agonistFormula:C24H17Cl2F2NO4Purezza:98%Colore e forma:SolidPeso molecolare:492.3(R)-SLV 319
CAS:(R)-SLV 319: potent CB1 antagonist, K i of 894 nM, dextrorotatory isomer.Formula:C23H20Cl2N4O2SColore e forma:SolidPeso molecolare:487.4Olorinab
CAS:Olorinab (APD 371) (APD 371) is a highly potent, selective and fully efficacious cannabinoid receptor type 2 (CB2) agonist. With an EC50 of 6.2 nM for hCB2.Formula:C18H23N5O3Purezza:97.67% - 98.47%Colore e forma:SolidPeso molecolare:357.41AM-1235
CAS:AM-1235 is a potent and selective cannabinoid receptor CB1 agonist.Formula:C24H21FN2O3Purezza:99.92%Colore e forma:SolidPeso molecolare:404.43CB1 agonist 1
CAS:CB1 agonist 1 is a potent CB1 agonist with a pIC50 value of 5.7 for CB1 receptors.CB1 agonist 1 can be used to study brain disorders, pain, and inflammation.Formula:C24H24N2O5SPurezza:98.56%Colore e forma:SolidPeso molecolare:452.52SR144528
CAS:SR144528 is an antagonist of the CB2 receptor (Ki = 0.6 nM) and inhibits microsomal ACAT activity (IC50 = 3.6 μM).Formula:C29H34ClN3OPurezza:99.63%Colore e forma:SolidPeso molecolare:476.05Nonabine
CAS:Nonabine is a compound with strong antiemetic properties that can be used to prevent nausea and vomiting associated with cancer chemotherapy.Formula:C25H33NO2Purezza:99.82% - 99.94%Colore e forma:SolidPeso molecolare:379.54CB1R antagonist 1
CAS:CB1R antagonist 1 is a potent CB1R antagonist that can be used to study diseases related to the nervous system.Formula:C18H23F3N2O3SPurezza:99.65%Colore e forma:SolidPeso molecolare:404.45CB2R PAM
CAS:CB2R PAM, an oral drug, boosts CB2 receptor response to specific agonists, showing potential in neuropathic pain relief.Formula:C21H24BrFN2O2Purezza:99.09%Colore e forma:SolidPeso molecolare:435.33SCH-336
CAS:<p>SCH-336: potent, selective CB2 agonist (Ki=1.8 nM, EC50=2 nM), orally active, 100x CB2 vs. CB1 preference, reduces leukocyte migration and eosinophilia.</p>Formula:C23H25NO8S3Purezza:95.01%Colore e forma:SolidPeso molecolare:539.64PSB-CB5
CAS:PSB-CB5 (GPR18-IN-32)2 is a GRP18 antagonist with anti-inflammatory activity and can be used to study obesity and metabolic disorders.Formula:C20H17ClN2O2SPurezza:99.26%Colore e forma:SolidPeso molecolare:384.88AZD1940
CAS:AZD1940 (UNII-0J0035E9FT) is a high affinity CB(1)/CB(2) receptor agonist of the cannabinoid with oral activity. Application in the study of orofacial pain.Formula:C20H29F2N3O2SPurezza:98.68%Colore e forma:SolidPeso molecolare:413.52Ref: TM-T30252
1mg130,00€5mg311,00€10mg535,00€25mg847,00€50mg1.169,00€100mg1.586,00€1mL*10mM (DMSO)344,00€JTE-907
CAS:JTE-907 是一种具有高度选择性和口服活性的 CB2 受体反向激动剂。JTE-907在体内展现出抗炎活性。Formula:C24H26N2O6Purezza:99.93%Colore e forma:SolidPeso molecolare:438.47Ref: TM-T19705
1mg56,00€5mg126,00€10mg187,00€25mg329,00€50mg490,00€100mg700,00€1mL*10mM (DMSO)150,00€O-2050
CAS:O-2050: strong CB1 antagonist (Ki 2.5 nM), CB2 inhibitor (Ki 0.2 nM); reduces mouse food intake, increases activity.Formula:C23H31NO4SPurezza:98%Colore e forma:SolidPeso molecolare:417.56Heptadecanoyl ethanolamide
CAS:Heptadecanoyl ethanolamide, an endogenous cannabinoid, serves as a synthetic analog of PEA, featuring an odd-numbered (17-carbon) fatty acid chain [1].Formula:C19H39NO2Colore e forma:SolidPeso molecolare:313.52COR659
CAS:COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.Formula:C16H16ClNO3SPurezza:99.75%Colore e forma:SolidPeso molecolare:337.82Ref: TM-T36520
1mg40,00€5mg90,00€10mg130,00€25mg227,00€50mg316,00€100mg434,00€200mg590,00€1mL*10mM (DMSO)89,00€PF-03550096
CAS:PF-03550096, an orally active synthetic cannabinoid (CB), selectively binds to peripheral CB2 receptors with a Ki value of 7.9 nM, demonstrating analgesic activity [1].Formula:C19H28N4O4Colore e forma:SolidPeso molecolare:376.45URB447
CAS:URB447, a peripherally restricted CB1 cannabinoid antagonist with IC50 values of 313 nM for rat CB1 receptor and 41 nM for human CB2 receptor, effectively reduces food intake and body weight gain in mice. It achieves these effects without penetrating the brain or antagonizing central CB1-dependent responses, making it a potential research tool for obesity studies [1].Formula:C25H21ClN2OColore e forma:SolidPeso molecolare:400.9Tedalinab
CAS:Tedalinab is an effective and selective cannabinoid receptor 2 agonist.Formula:C19H21F2N3OPurezza:98%Colore e forma:SolidPeso molecolare:345.39GW405833 hydrochloride
CAS:GW405833 hydrochloride, a potent and selective agonist of the cannabinoid-2 (CB2) receptor (EC 50 = 0.65 nM; maximum inhibition = 44.6%), exhibits significant antihyperalgesic effects in various rodent pain models [1] [2] [3].Formula:C23H25Cl3N2O3Colore e forma:SolidPeso molecolare:483.822-Linoleoyl Glycerol
CAS:2-Arachidonoyl glycerol (2-AG), a natural endocannabinoid ligand for the CB1 receptor, was isolated from porcine brain and characterized. Its congener, 2-linoleoyl glycerol (2-LG), which has a linoleoyl group instead of an arachidonoyl group, also exists alongside 2-AG in vivo. While 2-LG exhibits low intrinsic activity, it enhances the activity of 2-AG and other endocannabinoids through an "entourage" effect, attributed to the inhibition of breakdown and reuptake pathways that typically decrease endocannabinoid levels post-release.Formula:C21H38O4Colore e forma:SolidPeso molecolare:354.531GSK494581A
CAS:GSK494581A is a GPR55 agonist and glycine transporter subtype 1 inhibitor.Formula:C27H28F2N2O4SPurezza:98%Colore e forma:SolidPeso molecolare:514.58PF 514273
CAS:PF 514273 is a CB1 receptor antagonist.Formula:C21H17Cl2F2N3O2Purezza:98%Colore e forma:SolidPeso molecolare:452.28PSNCBAM-1
CAS:PSNCBAM-1 (PSNCBAM 1) is a CB1 receptor negative allosteric modulator (EC50 = 0.1 μM) with hypophagic effects in vivo.Formula:C22H21ClN4OPurezza:99.86%Colore e forma:SolidPeso molecolare:392.88Hemopressin(rat) TFA
CAS:Hemopressin(rat) TFA, a nonapeptide from hemoglobin α1-chain, selectively inhibits CB1 receptors and reduces inflammatory pain.Formula:C55H78F3N13O14Colore e forma:SolidPeso molecolare:1202.2811(Z),14(Z)-Eicosadienoic Acid Ethanolamide
CAS:11(Z),14(Z)-Eicosadienoic acid ethanolamide is an ethanolamide derivative of 11(Z),14(Z)-eicosadienoic acid.Formula:C22H41NO2Colore e forma:SolidPeso molecolare:351.57SAD-448
CAS:SAD-448 is a cannabinoid receptor type 1 (CB1) agonist. SAD-448 controls spasticity via action on the peripheral nerve CB1 receptor.Formula:C24H28N4O8SColore e forma:SolidPeso molecolare:532.57O-2545 hydrochloride
CAS:O-2545 is a potent water-soluble central cannabinoid (CB1) and peripheral cannabinoid (CB2) receptor agonist with Ki values of 1.5 and 0.32 nM, respectively. Typically, cannabinoid agonists are highly lipophilic and require solubilization through surfactant agents or binding to water miscible substances like albumin, Tween 80, or Emulphor for use. When dissolved in saline, O-2545 has shown high efficacy in mouse behavioral models, administered either intravenously or intracerebroventricularly.Formula:C26H36N2O2HClColore e forma:SolidPeso molecolare:445Tricosanoyl Ethanolamide
CAS:Tricosanoyl ethanolamide, a fatty N-acyl ethanolamine within the endocannabinoid family, has an ethanolamine metabolite whose significance remains to be established.Formula:C25H51NO2Colore e forma:SolidPeso molecolare:397.688Isopropyl dodec-11-enylfluorophosphonate
CAS:Isopropyl dodec-11-enylfluorophosphonate (IDEFP) is an organophosphorus ester functioning as a central cannabinoid receptor (CB1) antagonist and exhibitsFormula:C15H30FO2PPurezza:98%Colore e forma:SolidPeso molecolare:292.37MCHB-1
CAS:MCHB-1, a potent agonist of the human cannabinoid 2 (CB2) receptor (EC50= 0.52 nM), demonstrates high selectivity for CB2 over CB1 (Kis = 3.7 and 110 nM, respectively), distinguishing itself from similar benzimidazole compounds that significantly alleviate peripheral pain while minimizing central nervous system side effects in mice.Formula:C28H37N3O2Colore e forma:SolidPeso molecolare:447.623CB1 antagonist 1
CAS:CB1 antagonist 1 is a CB1 receptor antagonist, used in the research of obesity and metabolic syndrome, neuroinflammatory disorders, cognitive disorders, andFormula:C26H22Cl2N4Purezza:98%Colore e forma:SolidPeso molecolare:461.39Amauromine
CAS:Amauromine is a peripherally selective and potent cannabinoid receptor type 1 (CB1) receptor antagonist, a novel alkaloid with vasodilatory activity.Formula:C32H36N4O2Colore e forma:SolidPeso molecolare:508.65CB 65
CAS:CB 65 is a high affinity and selective CB2 receptor agonist with Ki values of 3.3 and > 1000 nM for CB2 and CB1 receptors respectively.Formula:C22H28ClN3O3Purezza:99.53%Colore e forma:SolidPeso molecolare:417.93(R)-Monlunabant
CAS:<p>(R)-Monlunabant ((R)-MRI-1891) serves as a CB1 receptor antagonist utilized in obesity and metabolic disease research [1].</p>Formula:C26H22ClF3N6O3SPurezza:98%Colore e forma:SolidPeso molecolare:591CB1 inverse agonist 1
CAS:MRL-650 is an oral, selective CB1 agonist; IC50: CB1=7.5 nM, CB2=4100 nM; anorexigenic effects noted.Formula:C25H18Cl3N3O3Purezza:99.92%Colore e forma:SolidPeso molecolare:514.79Ref: TM-T10694
1mg52,00€5mg111,00€10mg163,00€25mg235,00€50mg330,00€100mg452,00€200mg608,00€1mL*10mM (DMSO)136,00€AM841
CAS:AM841, a high-affinity electrophilic ligand, covalently interacts with a cysteine residue in helix six, thus activating the CB1 cannabinoid receptor.Formula:C26H39NO3SPurezza:98%Colore e forma:SolidPeso molecolare:445.66γ-Linolenoyl monoethanolamide
CAS:γ-Linolenoyl monoethanolamide, a fatty N-acyl ethanolamine, acts as an endocannabinoid [1] [2].Formula:C20H35NO2Colore e forma:SolidPeso molecolare:321.505Prostaglandin E2-1-glyceryl ester
CAS:Prostaglandin E2-1-glyceryl ester, a member of the Prostaglandin Glycerol Ester family, serves as an endocannabinoid ligand targeting the CB1 receptor. This compound triggers a swift and transient surge in intracellular free calcium levels [1] [2].Formula:C23H38O7Colore e forma:SolidPeso molecolare:426.55PSB-SB1202
CAS:PSB-SB1202 (Compound 21a), a phenyl coumarin compound, acts as a CB1/CB2 agonist. It demonstrates EC50 values of 56 and 14 nM and K i values of 32 and 49 nM for CB1 and CB2 receptors, respectively [1].Formula:C23H26O4Colore e forma:SolidPeso molecolare:366.45CB2R-IN-1
CAS:CB2R-IN-1 is a potent inverse agonist of the cannabinoid CB2 receptor (Ki: 0.9 nM).Formula:C23H27F3N4O6S3Purezza:98%Colore e forma:SolidPeso molecolare:608.67CB-25
CAS:CB-25 is a partial agonist ligand of CB1 cannabinoid receptors, augmenting Forskolin-induced cAMP formation in cancer cells, though not affecting hCB1-CHO cellsFormula:C25H41NO3Purezza:98%Colore e forma:SolidPeso molecolare:403.6CB-52
CAS:CB-52 acts as a neutral antagonist and ligand for the CB2 cannabinoid receptor [1].Formula:C26H43NO3Colore e forma:SolidPeso molecolare:417.62OMDM-5
CAS:OMDM-5 is a potent vanilloid receptor type 1 (TRPV1, EC50 = 75 nM) agonist, showing weak ligand activity at cannabinoid type 1 receptor (CB1, Ki=4.9 μM).Formula:C26H44N2O3Purezza:99.73%Colore e forma:SolidPeso molecolare:432.64Ref: TM-T12306
1mg87,00€5mg187,00€10mg284,00€25mg452,00€50mg645,00€100mg867,00€200mg1.130,00€1mL*10mM (DMSO)221,00€O-Arachidonoyl glycidol
CAS:O-Arachidonoyl glycidol (compound 1), a 2-arachidonoylglycerol (2-AG) analog, effectively inhibits the hydrolysis of cytosolic 2-oleoylglycerol (2-OG) with an IC50 value of 4.5 µM, and also blocks 2-OG and anandamide hydrolysis in membrane fractions with IC50 values of 19 µM and 12 µM, respectively [1].Formula:C23H36O3Colore e forma:SolidPeso molecolare:360.53GSK-554418A
CAS:GSK-554418A, a novel azaindole CB(2) agonists, is used for the treatment of chronic pain. It is efficacious in the acute model and the chronic joint pain model.Formula:C19H19ClN4O2Colore e forma:SolidPeso molecolare:370.83CAY10508
CAS:CAY10508 is a potent and selective inverse agonist for the central cannabinoid (CB1) receptor with therapeutic potential for treating obesity and drug dependence, lacking psychotropic effects. It exhibits a Ki value of 243 nM and an EC50 of 195 nM. At a concentration of 10 µM, CAY10508 displaces [3H]-CP-55,940 with 100% efficacy at the CB1 receptor and 35% at the peripheral cannabinoid (CB2) receptor. Its inverse agonist activity at the CB1 receptor was confirmed through a [35S]-GTPγS binding assay.Formula:C21H14Br2N2O2Colore e forma:SolidPeso molecolare:486.2GP 1a
CAS:<p>GP 1a: potent CB2 receptor agonist (EC50=7.1), 30x CB2 over CB1 preference, boosts P-ERK1/2, aids skin healing, anti-inflammatory.</p>Formula:C23H22Cl2N4OPurezza:99.79%Colore e forma:SolidPeso molecolare:441.35GW 833972A
CAS:<p>GW 833972A: selective CB2 agonist; reduces neural depolarization and citric acid cough in animals.</p>Formula:C18H14Cl2F3N5OPurezza:99.93%Colore e forma:SoildPeso molecolare:444.24Bzo-poxizid
CAS:Bzo-poxizid is a synthetic cannabinoid and a psychoactive substance.Formula:C20H21N3O2Colore e forma:SolidPeso molecolare:335.40BAY 38-7271
CAS:BAY 38-7271: potent neuroprotective, selective CB1/CB2 agonist, Ki of 1.85 nM (CB1) & 5.96 nM (CB2).Formula:C20H21F3O5SPurezza:98%Colore e forma:SolidPeso molecolare:430.44AM8936
AM8936: potent CB1 agonist, EC50 rCB1=8.6nM/hCB1=1.4nM, Ki rat CB1=0.55nM; potential for CNS, metabolic, pain, glaucoma research.Formula:C25H33NO3Colore e forma:SolidPeso molecolare:395.53CBR Agonist-2
CBR Agonist-2: CB1 receptor agonist, EC50 - 960 nM, Ki - 970 nM, useful for hCB1R-related disease research.Formula:C27H27FN4OColore e forma:SolidPeso molecolare:442.53PSB-KK1415
CAS:PSB-KK1415 is a selective agonist for the human orphan G protein-coupled receptor GPR18, with an EC50 of 19.1 nM.Formula:C24H23ClN6O2Peso molecolare:462.93Cannabigerovarin
CAS:Cannabigerovarin (CBGV) is a compound categorized as a phytocannabinoid.Formula:C19H28O2Peso molecolare:288.42Ac-Atovaquone
CAS:Ac-Atovaquone, an ester-acetylated derivative of atovaquone, acts as a potent inhibitor of cytochrome bc1 (cytochrome bc1). This compound shows potential for use in malaria research.Formula:C24H21ClO4Colore e forma:SolidPeso molecolare:408.87CBR Agonist-1
CBR Agonist-1 targets CB1R and CB2R with Ki of 0.18 μM and 1.22 μM, useful for studying cannabinoid-related diseases.Formula:C27H27FN4OColore e forma:SolidPeso molecolare:442.53
