Proteasi HIV
Gli inibitori della proteasi dell'HIV sono una classe di farmaci antiretrovirali che bersagliano specificamente l'enzima proteasi del virus dell'immunodeficienza umana (HIV). Inibendo questo enzima, questi composti impediscono al virus di elaborare le sue poliproteine in proteine mature e funzionali, bloccando così la produzione di nuovi virioni infettivi. Gli inibitori della proteasi dell'HIV sono una pietra miliare della terapia antiretrovirale altamente attiva (HAART) utilizzata per gestire l'HIV/AIDS. Presso CymitQuimica, offriamo una varietà di inibitori della proteasi dell'HIV per supportare la vostra ricerca nel trattamento dell'HIV, nella resistenza ai farmaci e nella virologia.
Trovati 489 prodotti di "Proteasi HIV"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
(S)-(+)-N-3-Benzylnirvanol
CAS:<p>(S)-(+)-N-3-Benzylnirvanol is a cytochrome P450 CYP2C19 inhibitor with a ki value of 82.5μM for CYP2C9 and 0.25μM for CYP2C19.Cost-effective and quality-assured.</p>Formula:C18H18N2O2Purezza:98.90%Colore e forma:SoildPeso molecolare:294.35Atazanavir
CAS:<p>Atazanavir (BMS-232632)(BMS-232632) is an highly effective HIV-1 protease inhibitor.</p>Formula:C38H52N6O7Purezza:98% - 99.95%Colore e forma:Crystalline SolidPeso molecolare:704.86(Rac)-Telinavir
CAS:<p>N1 compound with anti-HIV activity; contains dimethyl, phenyl, quinoline groups.</p>Formula:C33H44N6O5Purezza:99.30%Colore e forma:SolidPeso molecolare:604.74NBD-556
CAS:NBD-556 is a small molecule mimetic of CD4. NBD-556 recognizes the HIV-1 envelope protein gp120 and induces restructuring of gp120 analogous to CD4 binding.Formula:C17H24ClN3O2Purezza:99.79%Colore e forma:SolidPeso molecolare:337.84Fostemsavir Tris
CAS:Fostemsavir Tris (BMS-663068 Tris) is the prodrug of BMS-626529,is a oral, safe and effective inhibitor of HIV-1 attachment.Formula:C29H37N8O11PPurezza:99.45%Colore e forma:SolidPeso molecolare:704.623-Deazaadenosine hydrochloride
CAS:3-Deazaadenosine HCl blocks SAH hydrolase (Ki: 3.9 μM), with anti-inflammatory, anti-proliferative, and anti-HIV effects.Formula:C11H15ClN4O4Purezza:98.48%Colore e forma:SolidPeso molecolare:302.71Ibalizumab
CAS:<p>Ibalizumab(TMB-355) is a humanized IgG4 monoclonal antibody that acts as a CD4 receptor inhibitor, blocking the entry of HIV-1 into cells by binding to the CD4</p>Purezza:SDS-PAGE:96.4%;SEC-HPLC:97.7%Colore e forma:LiquidPeso molecolare:147.3 kDaGSK2838232
CAS:<p>GSK2838232 inhibit HIV reverse transcriptase activity across a broad panel of HIV-1 isolates,GSK2838232 is novel human immune virus (HIV) maturation inhibitor.</p>Formula:C48H73ClN2O6Purezza:97.97%Colore e forma:SolidPeso molecolare:809.56Elsulfavirine
CAS:Elsulfavirine (VM-1500) is an HIV-1 infection reverse transcriptase inhibitor. It is a new anti-HIV drug.Formula:C24H17BrCl2FN3O5SPurezza:99.66%Colore e forma:SolidPeso molecolare:629.28Probenecid
CAS:<p>Probenecid (Benemid) is a benzoic acid derivative with antihyperuricemic property.</p>Formula:C13H19NO4SPurezza:98.95% - 99.84%Colore e forma:Crystals From Dil Alcohol Pleasant Aftertaste (Ntp 1992)Peso molecolare:285.36Nevirapine
CAS:<p>Nevirapine (NVP) is a benzodiazepine non-nucleoside reverse transcriptase inhibitor.</p>Formula:C15H14N4OPurezza:99.58% - 99.59%Colore e forma:White Or Off-White Crystalline PowderPeso molecolare:266.3BRD-6929
CAS:BRD-6929, a brain-targeted HDAC1/2 inhibitor (IC50 1/8 nM), enhances gnidimacrin's anti-HIV effect, useful in mood behavior studies.Formula:C19H17N3O2SPurezza:98.01% - 99.05%Colore e forma:SolidPeso molecolare:351.42Dolutegravir intermediate-1
CAS:Dolutegravir intermediate-1 is a synthetic precursor for HIV-1 treatment from patent WO 2016125192 A2.Formula:C13H17NO8Purezza:99.52%Colore e forma:SolidPeso molecolare:315.28Salicylanilide
CAS:<p>Salicylanilide (2-Hydroxybenzanilide)s are a group of compounds with antiviral potency, antibacterial and antifungal activities.</p>Formula:C13H11NO2Purezza:99.55%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:213.23Pepstatin
CAS:Pepstatin (Pepsin Inhibitor S 735A) is a specific and orally aspartate protease inhibitor that also inhibits HIV protease activity. Cost effective and quality assured.Formula:C34H63N5O9Purezza:96.74% - 99.94%Colore e forma:SolidPeso molecolare:685.89Benfotiamine
CAS:Benfotiamine (S-Benzoylthiamine O-monophosphate) is a synthetic S-acyl derivative of thiamine (vitamin B1), used as an antioxidant dietary supplement.Formula:C19H23N4O6PSPurezza:99.2% - 99.91%Colore e forma:Shinning Black PowderPeso molecolare:466.45PF-3450074
CAS:<p>PF-3450074 (PF-74) is a specific HIV-1 inhibitor, blocking viral replication and uncoating at submicromolar EC50=8-640 nM.</p>Formula:C27H27N3O2Purezza:99.92%Colore e forma:SolidPeso molecolare:425.52Ritonavir
CAS:<p>Ritonavir (ABT 538) inhibits HIV-1/2 proteases; serum proteins limit it but it enhances other HIV drugs by hindering P450 degradation.</p>Formula:C37H48N6O5S2Purezza:99.38% - 99.96%Colore e forma:White PowderPeso molecolare:720.94TERT-IN-1
CAS:TERT-IN-1 has anti-HIV activity and can be used to study HIV infection.Formula:C16H20ClN3SPurezza:99.31%Colore e forma:SoildPeso molecolare:321.87Atazanavir sulfate
CAS:Atazanavir sulfate, an azapeptide HIV-protease inhibitor, treats HIV/AIDS alongside other anti-HIV drugs.Formula:C38H52N6O7·H2SO4Purezza:99.31% - 99.40%Colore e forma:SolidPeso molecolare:802.93Zalcitabine
CAS:<p>Zalcitabine (ddC) is a nucleoside analog inhibiting HIV by blocking reverse transcriptase and halting viral DNA synthesis.</p>Formula:C9H13N3O3Purezza:99.08% - ≥95%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:211.22Islatravir
CAS:<p>Islatravir (MK-8591) is an effective anti-HIV-1 agent.</p>Formula:C12H12FN5O3Purezza:98.77%Colore e forma:SolidPeso molecolare:293.25L 754394
CAS:L 754394 is an effective and specific inhibitor of the HIV-1 protease.Formula:C38H47N5O5Colore e forma:SolidPeso molecolare:653.81Globotriaosylceramides (porcine)
CAS:Globotriaosylceramides, cell membrane glycosphingolipids, act as Shiga toxin receptors and accumulate in Fabry disease, resisting HIV by blocking gp120.Formula:C60H113NO18Colore e forma:SolidPeso molecolare:1136.553HIV-1 protease-IN-10
<p>HIV-1 protease-IN-10 (Compound 2), exhibiting HIV-1 latency reversing activity (IC50: 0.22 μM), selectively binds to the PKCδ C1b domain (IC50: 0.69 μM) and</p>Formula:C23H40O5Purezza:98%Colore e forma:SolidPeso molecolare:396.56Protease Inhibitor Library
A unique collection of 343 protease and proteasome inhibitors for research in chemical genomics, and drug screening;Colore e forma:Odour SolidBictegravir Sodium
CAS:Bictegravir Sodium is an HIV-1 integrase inhibitor with 7.5 nM IC50, offering strong, selective anti-HIV effects and minimal toxicity.Formula:C21H17F3N3NaO5Purezza:99.97%Colore e forma:SolidPeso molecolare:471.36HIV p17 Gag (77-85)
CAS:<p>Targeting HIV Gag p17 (77-85) with intracellular Ab cDNA disrupts viral replication pre/post-integration.</p>Formula:C44H72N10O15Purezza:98%Colore e forma:SolidPeso molecolare:981.1HIV-1 protease-IN-14
<p>HIV-1protease-IN-14 (compound 5ae) is an effective inhibitor of HIV-1protease, exhibiting Ki values of 0.28 nM and 56.9 nM against WTHIV-1PR and R41THIV-1PR, respectively. This compound also demonstrates low cytotoxicity.</p>Colore e forma:Odour SolidHIV-1 inhibitor-81
HIV-1inhibitor-81 (Compound 14g) is an HIV-1 protease inhibitor with a Ki of 1.6 nM. This compound exhibits antiviral activity against HIV-1, with an EC50 value of 250 nM.Formula:C32H44N2O8SColore e forma:SolidPeso molecolare:616.77Scirpusin A
CAS:Scirpusin A is a hydroxystilbene dimer from the rhizome of Scirpus fluviatilis and Xinjiang wine grape.Formula:C28H22O7Colore e forma:SolidPeso molecolare:470.4712-Oxocalanolide A
12-Oxocalanolide A is a useful organic compound for research related to life sciences and the catalog number is T125675.Formula:C22H24O5Colore e forma:SolidPeso molecolare:368.429HIV gag peptide (197-205)
CAS:HIV gag peptide (197-205) is a H-2Kd-restricted epitope derived from the p24 portion of the HIV-1 gag protein and composed of the amino acid 197-205 (AMQMLKETIFormula:C45H81N11O14S2Purezza:98%Colore e forma:SolidPeso molecolare:1064.32Kuguacin N
Kuguacin N is a useful organic compound for research related to life sciences and the catalog number is T126345.Formula:C30H46O4Colore e forma:SolidPeso molecolare:470.694MPG, HIV related
CAS:MPG: 27-amino acid peptide from HIV-1 gp41 & SV40 T antigen, delivers nucleic acids into cells efficiently.Formula:C126H201N35O33SPurezza:98%Colore e forma:SolidPeso molecolare:2766.22ICeD-2
<p>ICeD-2 triggers death in HIV-1 infected cells, requires HIV protease, inhibits DPP8/9, and stabilizes DPP9 in PBMCs.</p>Formula:C20H29N3OColore e forma:SolidPeso molecolare:327.46VIR-165
VIR-165, a derivative of VIRIP (353-372 of alpha1-antitrypsin), blocks several HIV-1 strains.Formula:C109H158N22O25S2Purezza:98%Colore e forma:SolidPeso molecolare:2240.7MB-66
MB-66 (MAPP-66) is a fully human IgG1 antibody targeting HSV and HIV. It is a monoclonal antibody membrane intended for vaginal application. The isotype control for MB-66 can be referred to as HumanIgG1kappa, Isotype Control.Colore e forma:Odour LiquidHinnuliquinone
CAS:Hinnuliquinone is an anti-HIV agent.Formula:C32H30N2O4Purezza:98%Colore e forma:SolidPeso molecolare:506.59SPD-756
CAS:<p>SPD-756, a nucleoside reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection.</p>Formula:C12H16N6O3Purezza:98%Colore e forma:SolidPeso molecolare:292.29Peptide T
CAS:Peptide T, an HIV-1 derived octapeptide, may inhibit gp120 binding to CD4 and cytokines, and affect VIP receptors.Formula:C35H55N9O16Purezza:98%Colore e forma:SolidPeso molecolare:857.86HIV-1 inhibitor-59
<p>HIV-1 Inhibitor-59 (Compound I-5b) effectively inhibits both wild-type and mutant strains of HIV-1, with EC50 values ranging from 5.62 to 171 nM.</p>Formula:C28H28FN5O3SColore e forma:SolidPeso molecolare:533.62Delavirdine
CAS:<p>Delavirdine, an NNRTI for HIV-1, is used in HAART.</p>Formula:C22H28N6O3SColore e forma:SolidPeso molecolare:456.56Cys-TAT(47-57)
CAS:Cys-TAT(47-57): arginine-rich peptide from HIV-1 TAT protein's transduction domain.Formula:C67H124N34O14SPurezza:98%Colore e forma:SolidPeso molecolare:1661.99NNRT-IN-6
<p>NNRT-IN-6 (Compound 13a) is a non-nucleoside reverse transcriptase inhibitor (NNRT) used to inhibit HIV-1 reverse transcriptase (HIV-1RT), with an IC50 of 0.41 μM. It effectively suppresses both wild-type HIV-1 and mutants L100I, K103N, Y181C, Y188L, E138K, F227L/V106A, and RES056, with an EC50 range of 6.2-250 nM.</p>Formula:C32H31N9O3SColore e forma:SolidPeso molecolare:621.71HIV-1 inhibitor-11
HIV-1 inhibitor-11, a fused pyridine ring derivative, is a HIV-1 inhibitor.Formula:C42H36ClF10N7O5S2Colore e forma:SolidPeso molecolare:1008.35HIV-IN-9
HIV-IN-9 (Compound 2b) is an HIV inhibitor with an IC50 value of 6.65 μg/mL, demonstrating high binding affinity for HIV-RT.Colore e forma:Odour SolidPeptide T TFA
CAS:Peptide T (TFA), an octapeptide from HIV-1 gp120, inhibits HIV binding to CD4.Formula:C37H56F3N9O18Purezza:98%Colore e forma:SolidPeso molecolare:971.89HIV-1 inhibitor-6
CAS:<p>HIV-1 inhibitor-6 (3-Pyridinecarboxamide, 1,4-dihydro-1-methyl-N-(5-nitro-1,2-benzisothiazol-3-yl)-4-oxo-) is a potent HIV-1 pre-mRNA selective splicing</p>Formula:C14H10N4O4SPurezza:99.33%Colore e forma:SolidPeso molecolare:330.32AL-470
CAS:AL-470 demonstrates significant antiviral efficacy, exhibiting EC50 values of 0.27 µM against HIV-1, 0.63 µM against HIV-2, and 0.35 µM against EV-A71, asFormula:C67H57N7O23Colore e forma:SolidPeso molecolare:1328.2
