Altri inibitori
Questa categoria comprende una vasta gamma di inibitori che non rientrano nelle classificazioni standard ma sono comunque fondamentali per varie ricerche biochimiche e farmacologiche. Questi inibitori possono bersagliare vie, enzimi e interazioni molecolari uniche o meno studiate, fornendo strumenti preziosi per aree di ricerca specializzate. Presso CymitQuimica, offriamo una selezione diversificata di inibitori di alta qualità che coprono molteplici bersagli biologici e discipline di ricerca, permettendoti di esplorare nuove strade terapeutiche e approfondire la tua comprensione dei processi biologici complessi.
Trovati 37928 prodotti di "Altri inibitori"
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Fos-Choline-9
CAS:<p>Fos-Choline-9 is a useful organic compound for research related to life sciences. The catalog number is TF0065 and the CAS number is 253678-64-7.</p>Formula:C14H32NO4PColore e forma:SolidPeso molecolare:309.44-(Trifluoromethoxy)cinnamic Acid
CAS:<p>4-(Trifluoromethoxy)cinnamic Acid is a useful organic compound for research related to life sciences. The catalog number is T66196 and the CAS number is 783-13-1.</p>Formula:C10H7F3O3Colore e forma:SolidPeso molecolare:232.158CLEC12A/MICL/CLL-1 Protein, Human, Recombinant (hFc)
<p>CLEC12A/MICL/CLL-1 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag.</p>Colore e forma:Lyophilized PowderPeso molecolare:50.38 kDa (predicted); 65.49 kDa (reducing conditions)Valiloxibic acid
CAS:<p>Valiloxibic acid is a prodrug for GHB, a natural psychoactive neurotransmitter and weak GABAB agonist.</p>Formula:C9H17NO4Colore e forma:SolidPeso molecolare:203.238BSPII Protein, Mouse, Recombinant (His)
<p>Osteopontin (OPN), bone sialoprotein (BSPII), and osteonectin (ON) belong to a family of glycoproteins, which have been linked to cancer metastasis and</p>Colore e forma:Lyophilized PowderPeso molecolare:34.9 kDa (predicted). Due to glycosylation, the protein migrates to 68-80 kDa based on Tris-Bis PAGE result.Ref: TM-TMPK-01028
Prodotto fuori produzioneCLEC12A/MICL/CLL-1 Protein, Mouse, Recombinant (His)
<p>CLEC12A/MICL/CLL-1 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag.</p>Colore e forma:Lyophilized PowderPeso molecolare:25.12 kDa (predicted); 33.68 kDa (reducing conditions)Omilancor
CAS:<p>Omilancor,BT-11 is a direct LANCL2 activator with oral activity for Crohn's Disease (CD), Inflammatory Bowel Disease (IBD) and Ulcerative Colitis (UC).</p>Formula:C30H24N8O2Purezza:99.73%Colore e forma:SolidPeso molecolare:528.56N-Octylmaleimide
CAS:<p>N-Octylmaleimide is an alkylmaleimide, which can inhibit rat liver glucose 6-phosphatase.</p>Formula:C12H19NO2Colore e forma:SolidPeso molecolare:209.28Ref: TM-T40509
Prodotto fuori produzione4',5'-Dibromofluorescein
CAS:<p>4',5'-Dibromofluorescein (Eosinic acid) is a fluorescent dye that can be used as a ligand for protein characterization by spectroscopic analysis.</p>Formula:C20H10Br2O5Colore e forma:Orange Solid PowderPeso molecolare:490.10Ref: TM-T20030
Prodotto fuori produzioneBCL-W Protein, Human, Recombinant (His)
<p>BCL-W Protein, Human, Recombinant (His) is expressed in E.</p>Colore e forma:Lyophilized PowderPeso molecolare:20 kDa (predicted); 18 kDa (reducing conditions)sodium 4-pentynoate
CAS:<p>sodium 4-pentynoate is a alkynylacetate analogue.</p>Formula:C5H5NaO2Purezza:98%Colore e forma:SolidPeso molecolare:120.08Ref: TM-T13893
Prodotto fuori produzioneAniline-2,4-diphosphonic acid tetraethyl ester;
CAS:<p>Intermediates and building blocks - phosphorous compounds; nucleophile</p>Formula:C14H25NO6P2Colore e forma:SolidPeso molecolare:365.33,5-Diphenyl pyridine
CAS:<p>Heterocyclic compounds-pyridine,</p>Formula:C17H13NColore e forma:SolidPeso molecolare:231.29STAT2 Protein, Human, Recombinant (His)
<p>Signal transducer and activator of transcription that mediates signaling by type I IFNs (IFN-alpha and IFN-beta).</p>Colore e forma:Odour Lyophilized PowderRef: TM-TMPU-00003
Prodotto fuori produzioneMuzolimine
CAS:<p>Muzolimine: a long-acting, high-capacity diuretic for kidney failure/hypertension; withdrawn due to serious neurological side effects.</p>Formula:C11H11Cl2N3OColore e forma:SolidPeso molecolare:272.13Metrizoic acid
CAS:<p>Metrizoic acid is an ionic contrast medium. Metrizoic acid displays high osmolality and has a risk of inducing allergic reactions.</p>Formula:C12H11I3N2O4Purezza:98%Colore e forma:SolidPeso molecolare:627.9402Ref: TM-T16067
Prodotto fuori produzione2-Nitrosopyridine
CAS:<p>2-Nitrosopyridine: used in antibiotic synthesis, Click/Diels-Alder reactions, excellent dienophile.</p>Formula:C5H4N2OColore e forma:SolidPeso molecolare:108.1Golgicide A-1
CAS:<p>Golgicide A-1 (GCA-1) is a moderately potent cis-diastereomer variant of Golgicide A (GCA) specifically designed to inhibit mosquito reproduction.</p>Formula:C17H14F2N2Colore e forma:SolidPeso molecolare:284.31Bikunin/AMBP Protein, Human, Recombinant (aa 1-203, His)
<p>Bikunin/AMBP Protein, Human, Recombinant (aa 1-203, His) is expressed in HEK293 mammalian cells with His tag.</p>Colore e forma:Lyophilized PowderPeso molecolare:22.3 kDa (predicted); 32.8 kDa (reducing conditions)5-OxoETE
CAS:<p>5-OxoETE, a dehydrogenase-oxidized 5-HETE, raises neutrophil Ca²⁺ (EC50=2nM) & drives eosinophil migration & MAPK pathway.</p>Formula:C20H30O3Purezza:98.59%Colore e forma:SolidPeso molecolare:318.45PIH
CAS:<p>PIH inhibits ciliogenesis by destabilizing microtubules and blocking Hh signaling, hindering cilia formation and alpha-tubulin disassembly.</p>Formula:C20H19N5SPurezza:98%Colore e forma:SolidPeso molecolare:361.46STING agonist-23
CAS:<p>CF502 (STING agonist-23) is a non-nucleotide that activates STING pathway, boosts immune responses, and shows activity against SARS-CoV.</p>Formula:C33H35N13O4Colore e forma:SolidPeso molecolare:677.72SIRT-IN-3
CAS:<p>SIRT-IN-3: potent SIRT1 inhibitor (IC50=17μM), 4x selective over SIRT2, 14x over SIRT3 (IC50s: 74μM & 235μM).</p>Formula:C13H12N2OColore e forma:SolidPeso molecolare:212.25Benzylacyclouridine
CAS:<p>Benzylacyclouridine (BAU) is a specific UrdPase inhibitor, uridine metabolism and potentiate toxicity of 5-Fu against human prostate cancer cells antitumor.</p>Formula:C14H16N2O4Colore e forma:SolidPeso molecolare:276.29Ref: TM-T40932
Prodotto fuori produzioneHT-2 Toxin
CAS:<p>HT-2 Toxin, a deacetylated metabolite of T-2 toxin, impairs protein synthesis and hinders cell proliferation in plants.</p>Formula:C22H32O8Purezza:98%Colore e forma:SolidPeso molecolare:424.49Ref: TM-T13726
Prodotto fuori produzioneL-690330
CAS:<p>L-690330 inhibits human/bovine inositol monophosphatase; Ki: 0.19-0.42 μM. 10x potency vs. mouse/rat IMPase.</p>Formula:C8H12O8P2Colore e forma:SolidPeso molecolare:298.12Ref: TM-T15685
Prodotto fuori produzione4-Hydroxy-6-methylcoumarin
CAS:<p>4-Hydroxy-6-methylcoumarin (4-HMC) is a naturally occurring phenolic compound, a derivative of coumarin, found in a variety of plants, fungi, and bacteria. It has anti-inflammatory and anti-tumor activity.4-HMC is used as a flavoring agent, preservative and antioxidant in the food industry.</p>Formula:C10H8O3Purezza:99.95%Colore e forma:White PowderPeso molecolare:176.17Ref: TM-FR12277
Prodotto fuori produzioneElamipretide 2TFA
CAS:<p>Elamipretide 2TFA (RX-31 2TFA) is a novel mitochondrion-targeted antioxidant.</p>Formula:C36H51F6N9O9Purezza:>99.99%Colore e forma:SolidPeso molecolare:867.84Ref: TM-T8831
Prodotto fuori produzioneMTP 131 acetate
CAS:<p>MTP 131 (acetate) is a small mitochondrially-targeted tetrapeptide.</p>Formula:C34H53N9O7Purezza:99.9%Colore e forma:SolidPeso molecolare:699.844-Methoxycoumarine
CAS:<p>4-Methoxycoumarine has antitumour effects.</p>Formula:C10H8O3Purezza:99.88%Colore e forma:SolidPeso molecolare:176.17Ref: TM-FR12290
Prodotto fuori produzioneElamipretide
CAS:<p>Elamipretide (SS-31, MTP-131, Bendavia) is a mitochondria-focused peptide that curbs toxic ROS and stabilizes cardiolipin.</p>Formula:C32H49N9O5Purezza:98.53% - 99.85%Colore e forma:SolidPeso molecolare:639.797-Methoxy-1-tetralone
CAS:<p>7-Methoxy-1-tetralone may have insecticidal activity.</p>Formula:C11H12O2Purezza:99.93%Colore e forma:White CrystalPeso molecolare:176.21Danoprevir sodium
CAS:<p>Danoprevir sodium is an NS3/4A protease inhibitor used in the treatment of Hepatitis C</p>Formula:C35H45FN5NaO9SColore e forma:SolidPeso molecolare:753.82Ref: TM-T68354
Prodotto fuori produzioneCompound T69202(SC)
CAS:<p>NBQX (FG9202), an AMPA/kainate receptor blocker, counters glutamate toxicity; water-soluble as disodium salt, has anticonvulsant properties.</p>Formula:C12H6N4Na2O6SColore e forma:SolidPeso molecolare:380.2415Ref: TM-T69202
Prodotto fuori produzione10Z-Nonadecenoic acid
CAS:<p>10Z-Nonadecenoic acid is a long-chain fatty acid with anti-tumor activity.</p>Formula:C19H36O2Purezza:99.43%Colore e forma:SolidPeso molecolare:296.49Tropinone
CAS:<p>Tropinone used as an intermediate in the synthesis of atropine sulfate, and is a decane alkaloid.</p>Formula:C8H13NOPurezza:99.90%Colore e forma:Beige To Brown Crystalline PowderPeso molecolare:139.19Dimethylamine hydrochloride
CAS:<p>Dimethylamine hydrochloride, found in urine, comes from food compound TMAO and NO synthesis inhibitor ADMA, processed by DDAH enzyme.</p>Formula:C2H8ClNPurezza:98% - 99.89%Colore e forma:White Solid CrystallinePeso molecolare:81.54Decyl-TPP bromide
CAS:<p>Decyl-TPP bromide ((1-Decyl)triphenylphosphonium bromide) may be used as an intermediate for chemical synthesis and an inactive control or as a reference to</p>Formula:C28H36BrPPurezza:98%Colore e forma:SolidPeso molecolare:483.46Oxindole
CAS:<p>Oxindole (Indolin-2-one) is an aromatic heterocyclic building block. 2-indolinone derivatives have become lead compounds in the research of kinase inhibitors.Oxindole structure has been used in receptor tyrosine kinases (RTKs) inhibitors such as SU4984 and intedanib, the RTK family represents an important therapeutic target for anti-cancer drug development.</p>Formula:C8H7NOPurezza:99.34%Colore e forma:Off-White Crystalline PowderPeso molecolare:133.15Ethyl 4-hydroxyphenylacetate
CAS:<p>Ethyl 4-hydroxyphenylacetate is a selective inhibitor of monoamine oxidase A.</p>Formula:C10H12O3Purezza:99.89%Colore e forma:Slightly Yellow LiquidPeso molecolare:180.2IGFBP-1 Protein, Rat, Recombinant
<p>IGF-binding proteins prolong the half-life of the IGFs and have been shown to either inhibit or stimulate the growth promoting effects of the IGFs on cell culture. They alter the interaction of IGFs with their cell surface receptors. Promotes cell migration. IGFBP-1 Protein, Rat, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 26.9 kDa and the accession number is P21743.</p>Peso molecolare:26.9 kDa (predicted)CTHRC1 Protein, Mouse, Recombinant (aa 33-245, His)
<p>May act as a negative regulator of collagen matrix deposition.</p>Colore e forma:Lyophilized PowderPeso molecolare:25.9 kDa (predicted)Ref: TM-TMPH-02592
Prodotto fuori produzioneSLC1A2 Protein, Mouse, Recombinant (GST)
<p>SLC1A2 Protein, Mouse, Recombinant (GST) is expressed in E. coli. The accession number is P43006.</p>Colore e forma:Lyophilized PowderPeso molecolare:37.6 kDa (Predicted)Pomalidomide 4'-PEG5-azide
CAS:<p>Pomalidomide 4'-PEG5-azide, a cereblon (CRBN) ligand based on Pomalidomide, facilitates the recruitment of CRBN protein. It can be conjugated through a linker to another ligand, forming a proteolysis-targeting chimera (PROTAC) [1].</p>Formula:C25H34N6O9Colore e forma:SolidPeso molecolare:562.5709Ref: TM-T84902
Prodotto fuori produzione(S)-Coriolic acid
CAS:<p>(S)-Coriolic acid, a 15-LOX metabolite and signaling molecule, modulates cell growth, tumor adhesion, receptor expression, and can cause mitochondrial damage.</p>Formula:C18H32O3Purezza:97.67% - 98.04%Colore e forma:SolidPeso molecolare:296.44Phenamil methanesulfonate
CAS:<p>TRPP3 channel inhibitor</p>Formula:C13H16ClN7O4SPurezza:98%Colore e forma:SolidPeso molecolare:401.83Questiomycin A derivatives 18 TFA
<p>Questiomycin A derivative 18 TFA exhibits antibacterial, anticancer properties and inhibits GRP78.</p>Formula:C16H12F3N3O5Purezza:98.45%Colore e forma:SoildPeso molecolare:383.07Ref: TM-T67717L
Prodotto fuori produzioneH 35-25
CAS:<p>H 35-25 is a beta 2-antagonist.</p>Formula:C13H21NOColore e forma:SolidPeso molecolare:207.31Ref: TM-T70895
Prodotto fuori produzioneDioxifedrine
CAS:<p>Dioxifedrine is a beta-2 -adrenergic agonist with bronchodilator activity.</p>Formula:C10H15NO3Colore e forma:SolidPeso molecolare:197.23Ref: TM-T71575
Prodotto fuori produzioneGuancydine
CAS:<p>Guancydine is an antihypertensive agent.</p>Formula:C7H14N4Purezza:98%Colore e forma:SolidPeso molecolare:154.21CH-100
CAS:<p>CH-100 is a Chinese herbal medicine previously used in the treatment of human hepatitis C.</p>Formula:C14H22ClNO3Colore e forma:SolidPeso molecolare:287.78Ref: TM-T30866
Prodotto fuori produzioneIDX-375
CAS:<p>IDX-375, a HCV NS5B polymerase inhibitor, is used potentially for the treatment of HCV infection.</p>Formula:C29H50N5O7PSPurezza:98%Colore e forma:SolidPeso molecolare:643.78PAD4-IN-2
CAS:<p>PAD4-IN-2 (compound 5i) is a PAD4 inhibitor with an IC50 value of 1.94 μM, shown to suppress tumor growth in mice through specific inhibition of the PAD4-H3cit-</p>Formula:C20H23BClN7O6Colore e forma:SolidPeso molecolare:503.7Ref: TM-T79276
Prodotto fuori produzioneFM-24 HCl
CAS:<p>FM-24 HCl is a long acting beta-adrenergic receptor antagonist.</p>Formula:C19H30ClNO2Colore e forma:SolidPeso molecolare:339.9Ref: TM-T68856
Prodotto fuori produzioneSaxitoxinol
CAS:<p>Saxitoxinol is an analog of saxitoxin, a known voltage-gated sodium channel blocker.</p>Formula:C10H17N7O3Purezza:98%Colore e forma:SolidPeso molecolare:283.29Ref: TM-T68748
Prodotto fuori produzioneRadafaxine hydrochloride
CAS:<p>Radafaxine hydrochloride is an inhibitor of DAT and NET transporters, and nAChR family modulator.</p>Formula:C13H19Cl2NO2Purezza:98%Peso molecolare:292.2Tifenazoxide
CAS:<p>Tifenazoxide is an effective and SUR1/Kir6.2 selective KATP channels opener. Tifenazoxide has an anti-diabetic effect, can inhibit glucose-stimulated insulin release in vitro and in vivo.</p>Formula:C9H10ClN3O2S2Purezza:98%Colore e forma:SolidPeso molecolare:291.78anti-TNBC agent-3
CAS:<p>Anti-TNBC agent-3 (compound 3g) is a compound that induces apoptosis and possesses anti-cancer cell proliferation properties.</p>Formula:C29H39F2N7OColore e forma:SolidPeso molecolare:539.66Ref: TM-T79410
Prodotto fuori produzioneD(-)-Octopamine CSA salt
CAS:<p>D(-)-Octopamine CSA salt is an agonist of octopamine receptors.</p>Formula:C18H27NO6SPurezza:98%Colore e forma:SolidPeso molecolare:385.48Ref: TM-T27116
Prodotto fuori produzioneCK176
CAS:<p>CK176 is an HIV-1 inhibitor, 11x more effective than I-XW-053 in human PBMCs.</p>Formula:C21H12IN3O2Purezza:98%Colore e forma:SolidPeso molecolare:465.24Ref: TM-T27030
Prodotto fuori produzionePS372424 HCl
CAS:<p>PS372424 activates CXCR3, triggers ERK phosphorylation, and inhibits CXCL11's effect on CD45+ cell migration in humanized mice.</p>Formula:C33H45ClN6O4Colore e forma:SolidPeso molecolare:625.21Ref: TM-T70411
Prodotto fuori produzioneCebranopadol ((1α,4α)stereoisomer)
CAS:<p>Cebranopadol ((1α,4α)stereoisomer) is a stereoisomer of cebranopadol which is a potent ORL-1 agonist.</p>Formula:C24H27FN2OPurezza:98%Colore e forma:SolidPeso molecolare:378.48Ref: TM-T10749
Prodotto fuori produzioneAlbuterol stearate
CAS:<p>Albuterol stearate, a salt form of Albuterol, is a selective beta2 agonist for treating asthma and COPD, with 29x preference for beta2 over beta1.</p>Formula:C31H57NO5Purezza:98%Colore e forma:SolidPeso molecolare:523.799Ref: TM-T25030
Prodotto fuori produzioneCulmerciclib
CAS:<p>Culmerciclib is a cell cycle protein-dependent kinase (CDK) inhibitor that exhibits antitumour effects.</p>Formula:C24H27FN8Colore e forma:SolidPeso molecolare:446.52Ref: TM-T62650
Prodotto fuori produzione(E)-Crotylbarbital
CAS:<p>(E)-Crotylbarbital, a Crotylbarbital isomer, is a sedative with hypnotic, anticonvulsant properties, aiding sleep and mental stability.</p>Formula:C10H14N2O3Purezza:99.94%Colore e forma:SolidPeso molecolare:210.23Butabindide oxalate
CAS:<p>CCK-inactivating serine protease (tripeptidyl peptidase II) inhibitor</p>Formula:C19H27N3O6Purezza:98%Colore e forma:SolidPeso molecolare:393.43Aminobutane bisphosphonate
CAS:<p>Aminobutane bisphosphonate curbs bone loss; may manage hypercalcemia in cancer.</p>Formula:C4H13NO6P2Colore e forma:SolidPeso molecolare:233.1Ref: TM-T69443
Prodotto fuori produzioneBChE-IN-17
CAS:<p>BChE-IN-17 (compound 6n) is a potent, selective inhibitor of butyrylcholinesterase (BChE), demonstrating inhibitory half-maximal inhibitory concentrations (</p>Formula:C23H23BrN2O4S2Colore e forma:SolidPeso molecolare:535.47Ref: TM-T79342
Prodotto fuori produzioneHPK1-IN-18
CAS:<p>HPK1-IN-18: Potent, specific inhibitor of HPK1, a MAP4K enzyme, for cancer research and treatment.</p>Formula:C24H24N4Colore e forma:LiquidPeso molecolare:368.47Ref: TM-T61449
Prodotto fuori produzioneKP372-1
CAS:<p>KP372-1, an Akt inhibitor, blocks PI3K signaling, arrests cell growth, and triggers apoptosis in head/neck squamous cell carcinoma.</p>Formula:C20H8N12O2Colore e forma:SolidPeso molecolare:448.36DPX-3778
CAS:<p>DPX-3778, a triethanolamine salt, boosts tobacco callus growth 4-5x at 0.124-2.48 μM and slows aging with IAA and kinetin.</p>Formula:C16H23ClN4O6Colore e forma:SolidPeso molecolare:402.83Ref: TM-T31573
Prodotto fuori produzioneYM 298198 Hydrochloride
CAS:<p>YM 298198 HCl: non-competitive mGlu1 antagonist, Ki=19 nM. Inactive on mGlu2-7, stronger than CPCCOEt.</p>Formula:C18H22N4OSColore e forma:SolidPeso molecolare:342.46Ref: TM-T71764
Prodotto fuori produzioneFosfonet sodium
CAS:<p>Fosfonet sodium is a sodium salt of phosphonoacetic acid, effective against herpesviruses by inhibiting viral DNA polymerase.</p>Formula:C2H4NaO5PColore e forma:SolidPeso molecolare:162.01Ref: TM-T69345
Prodotto fuori produzioneSB251023
CAS:<p>SB251023 is an agonist of β3-adrenoceptor.</p>Formula:C28H34NO6PColore e forma:SolidPeso molecolare:511.55(Rac)-LM11A-31 dihydrochloride
CAS:<p>(Rac)-LM11A-31 dihydrochloride is an isomer of LM11A-31 dihydrochloride, a potent antagonist of proNGF (nerve growth factor).</p>Formula:C12H27Cl2N3O2Purezza:98%Colore e forma:SolidPeso molecolare:316.268Phenazolam
CAS:<p>Phenazolam is an analytical reference standard categorized as a benzodiazepine. [1] This product is intended for research and forensic applications.</p>Formula:C17H12BrClN4Colore e forma:SolidPeso molecolare:387.66MDK-2959
CAS:<p>MDK-2959 is a potent inhibitor of protein tyrosine phosphatase sigma (PTPsigma).</p>Formula:C15H11N3O4Purezza:98%Colore e forma:SolidPeso molecolare:297.27Erythrityl Tetranitrate
CAS:<p>Erythrityl Tetranitrate, a vasodilator similar to nitroglycerin, was first in "sustained release" tablets; may cause "nitro headache."</p>Formula:C4H6N4O12Colore e forma:SolidPeso molecolare:302.11Ref: TM-T31671
Prodotto fuori produzionePSB-6426
CAS:<p>PSB-6426 is the first potent and selective human nucleoside triphosphate diphosphohydrolase-2 inhibitor.</p>Formula:C22H29N4O10PPurezza:98%Colore e forma:SolidPeso molecolare:540.46Ref: TM-T24681
Prodotto fuori produzioneBenzovindiflupyr
CAS:<p>Benzovindiflupyr: a fungicide that inhibits SDH (IC50=5.2nM), halts S. sclerotiorum growth (EC50=0.011μg/ml), and protects crops like eggplants.</p>Formula:C18H15Cl2F2N3OColore e forma:SolidPeso molecolare:398.23PL265
CAS:<p>PL265 is a long-acting dual ENKephalinase inhibitor (DENKi) with analgesic potential.</p>Formula:C27H35N2O9PPurezza:98%Colore e forma:SolidPeso molecolare:562.55AKOS-22
CAS:<p>AKOS-22: potent VDAC1 inhibitor, Kd=15.4 μM; prevents mitochondrial dysfunction and apoptosis.</p>Formula:C22H21ClF3N3O3Purezza:98%Colore e forma:SolidPeso molecolare:467.87Trimetoquinol HCl hydrate
CAS:<p>Trimetoquinol hydrochloride possesses differential and selective beta-adrenergic properties.</p>Formula:C19H26ClNO6Colore e forma:SolidPeso molecolare:399.87Ref: TM-T34950
Prodotto fuori produzioneLM2I
CAS:<p>LM2I, a derivative of Spinosyn A (SPA), serves both as an argininosuccinate synthase (ASS1) enzyme activator and a tumor inhibitor through direct interaction</p>Formula:C47H77N3O11Colore e forma:SolidPeso molecolare:860.13Antitumor photosensitizer-1
CAS:<p>Antitumor Photosensitizer-1 (Compound 8) is a potent photosensitizer with remarkable photodynamic anti-tumor properties and minimal skin photo-toxicity,</p>Formula:C42H51N5O6Colore e forma:SolidPeso molecolare:721.88MDVN1003
CAS:<p>MDVN1003 inhibits BTK & PI3Kδ in B cells, blocking NHL growth; it kills lymphoma cells, not erythroblasts.</p>Formula:C22H20FN7OPurezza:98%Colore e forma:SolidPeso molecolare:417.44Ref: TM-T28008
Prodotto fuori produzioneAzilsartan mepixetil potassium
CAS:<p>Azilsartan medoxomil potassium (QR-01019K), an angiotensin II receptor antagonist, exhibits a potent and sustained antihypertensive effect, along with a more</p>Formula:C36H33KN6O8Colore e forma:SolidPeso molecolare:716.78Immune cell migration-IN-1
CAS:<p>Immune cell migration-IN-1 (compound 2) serves as a potent inhibitor of immune cell migration, with potential research applications for mitigating conditions</p>Formula:C30H25ClN4O6SColore e forma:SolidPeso molecolare:605.06Antitumor agent-136
CAS:<p>Antitumor Agent-136 (Compound 17), a broad-spectrum antitumor agent and NAMPT inhibitor, exhibits potent activity with an IC50 of 9.5 nM. It efficiently lowers intracellular and extracellular NAMPT protein levels via the ubiquitin proteasome pathway, achieving effective tumor inhibition [1].</p>Formula:C58H76N10O11S3Colore e forma:SolidPeso molecolare:1185.48URAT1 inhibitor 5
CAS:<p>URAT1 Inhibitor 5 (compound 16) serves as a powerful inhibitor of URAT1 and is utilized in hyperuricemia research [1].</p>Formula:C18H14BrN3O2SColore e forma:SolidPeso molecolare:416.29Anti-MI/R injury agent 1
CAS:<p>Anti-MI/R injury agent 1 (compound 18), derived from Panaxatriol, represents an orally administered, potent agent against myocardial ischemia/reperfusion (MI/R</p>Formula:C32H49NO6Colore e forma:SolidPeso molecolare:543.73Civorebrutinib
CAS:<p>Civorebrutinib (WS-413) is an inhibitor of Bruton's tyrosine kinase that exhibits antineoplastic activity [1].</p>Formula:C23H22ClN7O2Colore e forma:SolidPeso molecolare:463.92SHP2-IN-14
CAS:<p>SHP2-IN-14 (compound 27) is a potent, orally active allosteric inhibitor of SHP2, displaying strong anti-tumor activity with an IC50 of 7 nM.</p>Formula:C22H20Cl2N8OColore e forma:SolidPeso molecolare:483.35Ref: TM-T79108
Prodotto fuori produzionePF-05236216 hydrochloride
CAS:<p>PF-05236216 hydrochloride: Brain-penetrant, potent CK1δ/ε inhibitor affecting mouse circadian rhythms.</p>Formula:C18H15FN4OColore e forma:SolidPeso molecolare:322.34Ref: TM-T70812
Prodotto fuori produzionePD1-PDL1-IN 2
CAS:<p>PD1-PDL1-IN 2 (ZE132) is a potent, selective inhibitor of PD-1/PD-L1, exhibiting significant anti-tumor activity in vivo. It enhances cytotoxic T-cell tumor infiltration and stimulates IL-2 expression, while also strongly inhibiting TGF-β [1] mRNA expression, showcasing its comprehensive immunotherapeutic potential.</p>Formula:C37H41ClN4O7SColore e forma:SolidPeso molecolare:721.26HMR 1556
CAS:<p>HMR 1556 is a chromanol derivative and is an IKs blocker (IC50s of 10.5 nM and 34 nM in canine and guinea pig left ventricular myocytes, respectively).</p>Formula:C17H24F3NO5SColore e forma:SolidPeso molecolare:411.44Sakura 6
CAS:<p>Sakura 6, a synthetic serotonin transporter (SERT)-binding peptide, enhances the interaction between SERT and neuronal nitric oxide synthase.</p>Formula:C31H45N5O7Colore e forma:SolidPeso molecolare:599.73S-72
CAS:<p>S-72 acts as a microtubule polymerization inhibitor, effective in cell-free assays at concentrations of 1, 3, and 10 µM.</p>Formula:C20H22N4O3SColore e forma:SolidPeso molecolare:398.50Ref: TM-T83874
Prodotto fuori produzioneTauro-Obeticholic Acid sodium
CAS:<p>Tauro-obeticholic acid, a farnesoid X receptor (FXR) agonist and semisynthetic derivative of chenodeoxycholic acid, is an active metabolite of obeticholic acid.</p>Formula:C28H48NO6S·NaColore e forma:SolidPeso molecolare:549.74FOXM1-IN-2
CAS:<p>FOXM1-IN-2, a FOXM1 inhibitor, exhibits antineoplastic activity [1].</p>Formula:C48H47F4N7O12SColore e forma:SolidPeso molecolare:1021.99HPK1-IN-38
CAS:<p>HPK1-IN-38 (compound 15) is an inhibitor of MAP4K1/HPK1, suitable for research into disorders related to HPK1 [1].</p>Formula:C29H29N5O3Colore e forma:SolidPeso molecolare:495.57Antibacterial agent 160
CAS:<p>Antibacterial Agent 160 is a potent antibacterial agent that rapidly eradicates bacteria and inhibits the formation of bacterial biofilms.</p>Formula:C29H27ClFN3O6Colore e forma:SolidPeso molecolare:567.99ARN 077
CAS:<p>ARN 077 is a selective N-acylethanolamine acid amidase (NAAA) inhibitor (IC50: 7 nM for human NAAA). ARN 077 significantly increases palmitoyl ethanolamine (PEA) levels within the CNS.</p>Formula:C16H21NO4Colore e forma:SolidPeso molecolare:291.34L 689037
CAS:<p>L 689037 is an inhibitor of leukotriene biosynthesis.</p>Formula:C36H37ClN2O4Purezza:98%Colore e forma:SolidPeso molecolare:597.14Ref: TM-T24337
Prodotto fuori produzioneFAP-IN-2
CAS:<p>FAP-IN-2 is a 99mTc-labeled, isonitrile-containing derivative of a fibroblast activation protein (FAPI) inhibitor suitable for tumor imaging [1].</p>Formula:C24H28F2N6O3Colore e forma:SolidPeso molecolare:486.51Antibacterial agent 157
CAS:<p>Compound B12 (Antibacterial agent 157) is a fungicidal agent that can impact protein synthesis in Botrytis cinerea.</p>Formula:C26H23BrF4N2O3Colore e forma:SolidPeso molecolare:567.37RIOK2-IN-2
CAS:<p>RIOK2-IN-2 (8) functions as an inhibitor of RIOK2, exhibiting IC50 values of 3.02 μM in MKN-1 cells and 5.34 μM in MOLT4 cells [1].</p>Formula:C27H23F3N6O2Colore e forma:SolidPeso molecolare:520.51FLT3-IN-19
CAS:<p>FLT3-IN-19 (Comp 50) is a potent, selective inhibitor of FLT3, demonstrating an IC50 value of 0.213 nM, and is applicable in research pertaining to acute</p>Formula:C22H26N8OColore e forma:SolidPeso molecolare:418.49Antitumor photosensitizer-2
CAS:<p>Compound 11, also known as Antitumor Photosensitizer-2, is a potent photosensitizer with remarkable photodynamic anti-tumor properties and minimal skin photo-</p>Formula:C40H47N5O7Colore e forma:SolidPeso molecolare:709.83DiaFluo
CAS:<p>DiaFluo is a probe for protein S-sulfinylation from cells.</p>Formula:C32H32N4O9SColore e forma:SolidPeso molecolare:648.69LT-540-717
CAS:<p>LT-540-717 (compound 32), a potent FLT3 inhibitor (IC50=0.62 nM), exhibits antiproliferative activity and effectively inhibits various acquired FLT3 mutations,</p>Formula:C24H24N8O2Colore e forma:SolidPeso molecolare:456.5Ref: TM-T79490
Prodotto fuori produzioneOmeprazole acid
CAS:<p>Omeprazole treats GERD, ulcers, Zollinger-Ellison syndrome, prevents GI bleeding; it's a proton pump inhibitor.</p>Formula:C34H32N6Na2O10S2Colore e forma:SolidPeso molecolare:794.76Ref: TM-T71980
Prodotto fuori produzioneI-BET282
CAS:<p>BET-IN-1 is a bromodomain inhibitor extracted from patent WO/2013024104A1 (example 2, plC50: 6.0 - 7.0).</p>Formula:C25H30N4O4Purezza:98%Colore e forma:SolidPeso molecolare:450.53IDO/Tubulin-IN-2
CAS:<p>IDO/Tubulin-IN-2 inhibits TDO/tubulin, effective on U87, HepG2, A549, HCT-116, LO2 cancer cells; IC50 values 0.036-1.04 μM, boosts antitumor action.</p>Formula:C48H40N6O10Colore e forma:SolidPeso molecolare:860.87Ref: TM-T74536
Prodotto fuori produzioneCIAC001
CAS:<p>CIAC001, a pyruvate kinase PKM2 inhibitor, exhibits anti-neuroinflammatory properties.</p>Formula:C20H25N3O2Colore e forma:SolidPeso molecolare:339.43Ref: TM-T79637
Prodotto fuori produzioneAc4GalNAlk
CAS:<p>Ac4GalNAlk, a weakly alkyne-labeled reagent for metabolic oligosaccharide engineering (MOE), facilitates the detection of protein glycosylation by promoting nucleotide-sugar biosynthesis and enhancing bioorthogonal cell surface markers. It is activated by cellular biosynthetic machinery into nucleotide sugars, subsequently enabling the tracing of glycoproteins in bioorthogonal chemistry [1].</p>Formula:C19H25NO10Colore e forma:SolidPeso molecolare:427.4CYY292
CAS:<p>CYY292 is a chemical compound acting as an inhibitor of PDGFRα, PDGFRβ, FGFR1, -2, and -3, with respective IC50 values of 5.35, 4.6, 28, 28, and 78 nM.</p>Formula:C24H28N8OColore e forma:SolidPeso molecolare:444.53And1-IN-1
CAS:<p>And1-IN-1, also known as compound III, is a potent inhibitor of And1 [1].</p>Formula:C15H11BCl2O2Colore e forma:SolidPeso molecolare:304.9680-O16B
CAS:<p>80-O16B, an ionizable cationic lipid featuring disulfide bonds, is utilized in the preparation of lipid nanoparticles (LNP) [1].</p>Formula:C39H78N2O4S4Colore e forma:SolidPeso molecolare:767.31DDO-2213
CAS:<p>DDO-2213 is a potent, orally active inhibitor of the WDR5-MLL1 interaction, demonstrating an IC50 of 29 nM and a Kd of 72.9 nM against WDR5.</p>Formula:C24H27ClFN7OColore e forma:SolidPeso molecolare:483.97Ifetroban
CAS:<p>Ifetroban is a potent and selective TxA2/PGH2 receptor antagonist.</p>Formula:C25H32N2O5Colore e forma:SolidPeso molecolare:440.53Ref: TM-T27588
Prodotto fuori produzioneBB-Cl-Amidine hydrochloride
CAS:<p>BB-Cl-Amidine hydrochloride is an inhibitor of peptidylarginine deminase (PAD) [1].</p>Formula:C26H27Cl2N5OPurezza:98%Colore e forma:SolidPeso molecolare:496.43Cortivazol
CAS:<p>Cortivazol is an Anti-Inflammatory Drug.</p>Formula:C32H38N2O5Purezza:98%Colore e forma:SolidPeso molecolare:530.65Ref: TM-T25271
Prodotto fuori produzioneIfetroban sodium
CAS:<p>Ifetroban sodium (BMS-180291), oral TXA2/PGH2 antagonist for researching heart, stroke, BP, thrombosis.</p>Formula:C25H31N2NaO5Colore e forma:SolidPeso molecolare:462.522Ref: TM-T62924
Prodotto fuori produzione9,10-Phenanthrenequinone
CAS:<p>9,10-Phenanthrenequinone is an inhibitor of claudin-5/CLDN5, which induces apoptosis via an NO synthase/ROS-dependent mechanism. It also promotes caspase activation and DNA fragmentation while reducing CLDN5 expression and proteasome proteolysis, contributing to endothelial barrier dysfunction.</p>Formula:C14H8O2Colore e forma:SolidPeso molecolare:208.21DG026
CAS:<p>DG026 selectively inhibits IRAP, reducing its cross-presentation in dendritic cells without affecting ERAP1.</p>Formula:C35H40N3O4PPurezza:98%Colore e forma:SolidPeso molecolare:597.68Ref: TM-T27160
Prodotto fuori produzioneALS-I-41
CAS:<p>ALS-I-41 is a novel, potent and selective antagonist of oxytocin receptor.</p>Formula:C30H38FN3O6SPurezza:98%Colore e forma:SolidPeso molecolare:587.7Ref: TM-T26602
Prodotto fuori produzioneBPH-628
CAS:<p>BPH-628 is a bioactive chemical.</p>Formula:C20H20O7P2Colore e forma:SolidPeso molecolare:434.32
