
Segnalazione citoscheletrica
Gli inibitori della segnalazione del citoscheletro sono composti che interrompono le vie di segnalazione che regolano il citoscheletro, cruciale per la forma, la motilità, la divisione delle cellule e il trasporto intracellulare. Questi inibitori vengono utilizzati per studiare la dinamica delle proteine del citoscheletro, come actina e tubulina, e il loro ruolo in processi come la migrazione cellulare, l'adesione e la metastasi del cancro. Gli inibitori della segnalazione del citoscheletro sono preziosi nella ricerca sulla biologia cellulare, sul cancro e sulla neurobiologia. Presso CymitQuimica, offriamo una gamma completa di inibitori della segnalazione del citoscheletro di alta qualità per supportare le tue ricerche in questi ambiti.
Trovati 1591 prodotti per "Segnalazione citoscheletrica".
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CMPD101
CAS:CMPD101 is a membrane-permeable small-molecule inhibitor of GRK2/3 (IC50: 18 nM and 5.4 nM).Formula:C24H21F3N6OPurezza:99.01% - 99.04%Colore e forma:SolidPeso molecolare:466.46TINK-IN-1
CAS:TINK-IN-1 is a selective and potent TNIK inhibitor (IC50: 8 nM).TINK-IN-1 inhibits colorectal cancer cell viability and can be used to study mental retardation.Formula:C24H24N4O3Purezza:99.8%Colore e forma:SolidPeso molecolare:416.47Ref: TM-T77660
1mg39,00€2mg50,00€5mg82,00€10mg120,00€25mg236,00€50mg353,00€100mg517,00€500mg1.099,00€A-3 hydrochloride
CAS:A-3 hydrochloride: potent, reversible kinase antagonist; permeable; inhibits PKC, CKI, PKA, CKII, MLCK; Ki: 4.3-80 μM.Formula:C12H14Cl2N2O2SPurezza:99.32%Colore e forma:SolidPeso molecolare:321.22Danicamtiv
CAS:Danicamtiv (MYK-491) is an inotropic agent and it also is a selective allosteric activator of cardiac myosin.Formula:C16H20F3N5O4SPurezza:99.38%Colore e forma:SolidPeso molecolare:435.42Ref: TM-T15050
1mg129,00€5mg260,00€1mL*10mM (DMSO)286,00€10mg430,00€25mg710,00€50mg973,00€100mg1.333,00€ATN-161 acetate
CAS:ATN-161 acetate, a pentapeptide compound derived from the synergistic region of fibronectin, is an integrin-alpha5 antagonist with antitumor activity.Formula:C25H39N9O10SPurezza:98.27%Colore e forma:White SolidPeso molecolare:657.7Delcasertib
CAS:Delcasertib (KAI-9803) is a potent and selective inhibitor of δ-protein kinase C (δPKC).Formula:C120H199N45O34S2Purezza:99.96%Colore e forma:SolidPeso molecolare:2880.28Ref: TM-T11740
1mg192,00€5mg485,00€10mg700,00€25mg1.063,00€50mg1.459,00€1mL*10mM (DMSO)1.603,00€100mg1.963,00€ADH-1 trifluoroacetate
CAS:ADH-1 trifluoroacetate (Exherin trifluoroacetate) is a cyclic pentapeptide vascular-targeting agent with potential antineoplastic and antiangiogenic activities.Formula:C24H35F3N8O8S2Purezza:90.08% - 99.98%Colore e forma:White SolidPeso molecolare:684.71Ref: TM-T1608
2mg42,00€5mg62,00€10mg89,00€1mL*10mM (DMSO)89,00€25mg167,00€50mg227,00€100mg339,00€200mg482,00€BNC105
CAS:BNC105 is a tubulin polymerization inhibitor. It has potent antiproliferative and tumor vascular disrupting properties.Formula:C20H20O7Purezza:96.57%Colore e forma:SolidPeso molecolare:372.37Ref: TM-T14694
1mg79,00€5mg152,00€1mL*10mM (DMSO)167,00€10mg215,00€25mg351,00€50mg494,00€100mg665,00€200mg893,00€Abciximab
CAS:Abciximab: chimeric antibody, anti-platelet, blocks glycoprotein IIb/IIIa, vitronectin, Mac-1.Purezza:SDS-PAGE:95.2%;SEC-HPLC:95.9%Colore e forma:Transparent LiquidPeso molecolare:95.18 kDaCC-99677
CAS:CC-99677 (Gamcemetinib) is a MK2 inhibitor targeting autoimmune diseases; potent in rat assays with IC50=156.3 nM & EC50=89 nM.Formula:C22H20ClN5O3SPurezza:99.59%Colore e forma:SolidPeso molecolare:469.94Bosutinib
CAS:Bosutinib (SKI-606) is a synthetic quinolone derivative and dual kinase inhibitor that targets both Abl (IC50: 1 nM) and Src (IC50: 1.2 nM) kinases.Formula:C26H29Cl2N5O3Purezza:98.98% - 99.9%Colore e forma:Yellow SolidPeso molecolare:530.45Mps1-IN-3
CAS:Mps1-IN-3 is an effective and selective inhibitor of MPS1 kinase (IC50: 50 nM).Formula:C26H31N7O4SPurezza:99.25%Colore e forma:SolidPeso molecolare:537.63Ref: TM-T16130
2mg34,00€5mg54,00€1mL*10mM (DMSO)64,00€10mg87,00€25mg149,00€50mg255,00€100mg384,00€200mg538,00€RWJ 50271
CAS:RWJ 50271 inhibits LFA-1/ICAM-1 interaction with IC50 5.0 μM in HL60 cells.Formula:C18H17F3N4O2SPurezza:99.09%Colore e forma:White SolidPeso molecolare:410.41Ref: TM-T12783
1mg120,00€5mg295,00€1mL*10mM (DMSO)326,00€10mg447,00€25mg707,00€50mg964,00€100mg1.243,00€200mg1.693,00€AS1949490
CAS:AS1949490, a selective SHIP-2 inhibitor with IC50 of 620 nM, boosts glucose metabolism by upregulating GLUT1 in L6 myotubes.Formula:C20H18ClNO2SPurezza:99.94%Colore e forma:SolidPeso molecolare:371.88Ref: TM-T14327
1mg38,00€2mg50,00€5mg84,00€1mL*10mM (DMSO)93,00€10mg119,00€25mg236,00€50mg380,00€100mg555,00€PKC β pseudosubstrate acetate
PKC β pseudosubstrate acetate (PKC β pseudosubstrate acetate (172308-76-8 Free base)) is a selective cell-permeable inhibitor of PKC.Purezza:95.42%Colore e forma:SoildEntasobulin
CAS:Entasobulin is an inhibitor of β-tubulin polymerization. It has a potential anticancer activity.Formula:C26H18ClN3O2Purezza:98.40%Colore e forma:SolidPeso molecolare:439.89Dasatinib
CAS:Dasatinib (BMS-354825) is a tyrosine kinase inhibitor that inhibits Src and Bcr-Abl (Ki=16/30 pM) and is orally active and ATP-competitive.Formula:C22H26ClN7O2SPurezza:99.59% - 99.86%Colore e forma:Pale-Yellow SolidPeso molecolare:488.01Imatinib Mesylate
CAS:Imatinib Mesylate (STI-571) is a tyrosine kinase receptor inhibitor with antineoplastic activity (IC50s: 0.6 μM, 0.1 μM and 0.1 μM for v-Abl, c-Kit and PDGFR,Formula:C29H31N7O·CH4SO3Purezza:98% - >99.99%Colore e forma:White SolidPeso molecolare:589.71CCT251545
CAS:CCT251545 is an potent and oral-bioavailable WNT signaling inhibitor(IC50 of 5 nM in 7dF3 cells).Formula:C23H24ClN5OPurezza:98.29% - 98.69%Colore e forma:White SolidPeso molecolare:421.92Teplizumab
CAS:Teplizumab (MGA-031) is a humanized monoclonal antibody against CD3 that slows the loss of beta cell function.Teplizumab is used to treat type 1 diabetes.Purezza:SDS-PAGE:95.8%;SEC-HPLC:99.7%Colore e forma:LiquidPeso molecolare:145.79 kDa

