
Standard farmaceutici
Sottocategorie di "Standard farmaceutici"
- APIs per la ricerca e le impurità(275.095 prodotti)
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- Composti e metaboliti farmaceutici e veterinari(2.890 prodotti)
- Tossicologia(13.644 prodotti)
Trovati 7840 prodotti di "Standard farmaceutici"
Isovaleryl-Phe-Nle-Sta-Ala-Sta-OH
CAS:Isovaleryl-Phe-Nle-Sta-Ala-Sta-OH (IVAS) is a small molecule that has been shown to be an angiotensin system inhibitor. IVAS blocks the binding site of the angiotensin receptor and prevents the activation of this system. This effect is dose dependent and can be used to treat high blood pressure in humans. IVAS is a long-acting drug and has been shown to be effective in primates as well as humans. The drug is rapidly absorbed from the gastrointestinal tract and eliminated by metabolism, mainly through hydrolysis by esterases or glucuronidases, oxidation by cytochrome P450 enzymes, reduction by glutathione reductase, or conjugation with glucuronic acid. IVAS also specifically binds to markers expressed at high levels in Mycobacterium tuberculosis strains (e.g., ESX-1 secretion system protein) and inhibits cell growth in culture.
Formula:C39H65N5O9Purezza:Min. 95%Peso molecolare:747.96 g/mol9-Chloro-11beta,17,21-trihydroxy-16beta-methylpregna-1,4-diene-3,20-dione 17-valerate
CAS:Prodotto controllatoPrednisolone is a synthetic corticosteroid that is used in the treatment of a number of lung diseases, including asthma. Prednisolone is used to decrease the inflammation and swelling around the airways and lungs. Prednisolone is used to treat certain skin conditions, such as eczema and dermatitis. This drug also decreases the activity of the immune system by inhibiting production of substances that cause inflammation. The onset of action for prednisolone is typically one day with a duration of up to two weeks. It has been shown to be more effective when taken orally than when applied topically. It may be taken with or without food and can be given as an oral or an intravenous dose. Prednisolone tablets must be dissolved in water before they are placed under the tongue (sublingual). The tablets will dissolve quickly under the tongue, releasing prednisolone into your bloodstream. Enteric-coated tablets should not be crushed or chewed
Formula:C27H37ClO6Purezza:Min. 95%Peso molecolare:493.03 g/mol17,21Dihydroxy-16beta-methylpregna-1,4,9(11)-triene-3,20-dione
CAS:Prodotto controllatoPlease enquire for more information about 17,21Dihydroxy-16beta-methylpregna-1,4,9(11)-triene-3,20-dione including the price, delivery time and more detailed product information at the technical inquiry form on this pageFormula:C22H28O4Purezza:Min. 95%Peso molecolare:356.46 g/mol(S,S)-(-)-2,2'-Isopropylidenebis(4-tert-butyl-2-oxazoline)
CAS:(S,S)-(-)-2,2'-Isopropylidenebis(4-tert-butyl-2-oxazoline) is a chiral organic reagent. It is prepared by reacting chloroacetic acid with an alcohol. The reaction product is then treated with a base and the resulting salt of (S,S)-(-)-2,2'-isopropylidenebis(4-tert-butyl-2-oxazoline) is crystallized. This reagent can be used to form an amide by reacting it with an amine. Preparative methods are also available for this product. It can be used as a ligand in preparative chemistry or as a solvent in organic chemistry. The reactivity of this product depends on its chirality, which can be determined using analytical techniques such as gas chromatography or nuclear magnetic resonance spectroscopy.Formula:C17H30N2O2Purezza:Min. 95%Peso molecolare:294.43 g/molIsoeugenol methyl ether
CAS:Isoeugenol methyl ether is a plant-derived natural compound that is used in vitro as an antioxidant. It has been shown to inhibit the activity of enzymes such as hydroxylase, glucuronidase, and cytochrome P450. Isoeugenol methyl ether has also been shown to have anti-inflammatory properties and may be useful for treatment of colorectal adenocarcinoma. The mechanism by which isoeugenol methyl ether inhibits the enzyme activity is not clear but it may be due to its ability to bind reversibly with free enzyme form.Formula:C11H14O2Purezza:Min. 95%Colore e forma:LiquidPeso molecolare:178.23 g/molrac 8-Hydroxy efavirenz
CAS:Efavirenz is a non-nucleoside reverse transcriptase inhibitor (NNRTI) used in the treatment of HIV. It has been shown to be reactive with sodium carbonate, forming a stable complex that can be measured by LC-MS/MS. The formation rate of this complex may be influenced by the presence of other drugs, such as rifampin, which inhibits cytochrome P450 activity and reduces efavirenz metabolism. This drug has been shown to inhibit human Cytochrome P450 3A4 (CYP3A4) and may have increased plasma concentrations when administered with CYP3A4 inhibitors such as ketoconazole or erythromycin. Efavirenz is also metabolized in the liver by cytochrome P450 enzymes, mainly CYP3A4. Pharmacokinetic modeling has been used to study the drug's effects on hepatic clearance and plasma concentrations in humans.Formula:C14H9ClF3NO3Purezza:Min. 95%Colore e forma:White PowderPeso molecolare:331.67 g/mol12-Amino-1-dodecanoic acid methyl ester hydrochloride salt
CAS:12-Amino-1-dodecanoic acid methyl ester hydrochloride salt (12ADM) has been shown to have immunomodulatory properties. It has a nanomolar range of activity, which is the optimal for an immunosuppressant. 12ADM inhibits the transcriptional activity of human immunodeficiency virus type 1 (HIV-1) and HIV-2, as well as other retroviruses, through interactions with specific RNA sequences in the viral genome. The amide group in this compound is essential for its antiviral activity, and it also interacts with betulinic acid to enhance its cytotoxicity.Formula:C13H28ClNO2Purezza:Min. 95%Colore e forma:PowderPeso molecolare:265.82 g/molMethyl-1-naphthalenemethylamine
CAS:Methyl-1-naphthalenemethylamine is a synthetic drug that is used as an anti-fungal agent. It is used to treat dermatophytosis and onychomycosis caused by Trichophyton mentagrophytes. Methyl-1-naphthalenemethylamine has been shown to have a clinical response in patients with the skin condition tinea pedis. This drug inhibits the growth of fungi by inhibiting cell membrane synthesis, which leads to cell death. Methyl-1-naphthalenemethylamine has been shown to be effective against Trichophyton mentagrophytes in plasma samples from patients with tinea pedis who were treated with this drug. The effectiveness of this drug may be due to its ability to inhibit the synthesis of polysaccharides, proteins, and lipids in the fungal cell membrane, or its ability to inhibit protein synthesis by binding with ribosFormula:C12H13NPurezza:Min. 95%Colore e forma:Clear LiquidPeso molecolare:171.24 g/molS-[2-(Dimethylamino)ethyl]isothiourea Dihydrochloride
CAS:Prodotto controllatoS-[2-(Dimethylamino)ethyl]isothiourea Dihydrochloride is an inhibitor of tyrosinase, an enzyme that catalyzes the oxidation of tyrosine to dopa and dopaquinone. It binds to the active site of the enzyme and blocks its activity. S-[2-(Dimethylamino)ethyl]isothiourea Dihydrochloride has been shown to inhibit tyrosinase in animal experiments and in vitro studies, with a concentration-response curve that can be described by a Michaelis-Menten kinetic model. The inhibition of tyrosinase activity may be due to steric hindrance by the thiourea group or a covalent binding to amino acid residues on the protein surface. S-[2-(Dimethylamino)ethyl]isothiourea Dihydrochloride is also known as monomethyl auristatin E (MMAEFormula:C5H13N3S·2HClPurezza:Min. 95%Peso molecolare:220.16 g/mol3,5,3',5'-Tetraiodo thyroaldehyde
CAS:Please enquire for more information about 3,5,3',5'-Tetraiodo thyroaldehyde including the price, delivery time and more detailed product information at the technical inquiry form on this page
Formula:C13H6I4O3Purezza:Min. 95%Colore e forma:PowderPeso molecolare:717.8 g/mol20-Dehydro cholesterol 3-acetate
CAS:Prodotto controllatoPlease enquire for more information about 20-Dehydro cholesterol 3-acetate including the price, delivery time and more detailed product information at the technical inquiry form on this pageFormula:C29H46O2Purezza:Min. 95%Peso molecolare:426.67 g/molAlfentanil hydrochloride
CAS:Prodotto controllatoAlfentanil is an opioid analgesic that is used for the treatment of severe or acute pain. It is a potent synthetic analog of fentanyl, which is an opioid analgesic that is used for the treatment of short-term (acute) and long-term (chronic) pain. Alfentanil has been shown to have a high affinity for α1-acid glycoprotein, which has been associated with drug interactions and blood sampling. Alfentanil also has chemical stability in experimental models and does not interact with nonsteroidal anti-inflammatory drugs. This drug may have a matrix effect on the concentration of cortisol in the blood.
Formula:C21H33ClN6O3Purezza:Min. 95%Peso molecolare:452.98 g/molL-Proline-beta-naphthylamide hydrochloride
CAS:L-proline analogueFormula:C15H16N2O·HClPurezza:Min. 95%Peso molecolare:276.76 g/mol2,6-Diisopropylnaphthalene
CAS:Epidermal growth factor (EGF) is a polypeptide hormone that stimulates mitosis and cell growth. In some cases, it can act as an autocrine or paracrine hormone. Epidermal growth factor is used to stimulate the renewal of cells in the skin and mucous membranes. It also has been shown to have anti-inflammatory properties, which may be due to its ability to inhibit the release of inflammatory mediators such as prostaglandins and leukotrienes. 2,6-Diisopropylnaphthalene (2,6-DNP) is an antimicrobial agent that binds to the cell nucleus and inhibits transcription and translation of DNA into RNA by binding to RNA polymerase II. This binding prevents formation of transcription complexes with the cell factor necessary for transcription. 2,6-DNP has been shown to reduce disease activity in patients with inflammatory bowel disease in a clinical trial when used alone or in combination with other agents. TheFormula:C16H20Purezza:Min. 95%Peso molecolare:212.33 g/mol4-Aminobicyclo[2.2.2]octane-1-carboxylic acid methyl ester
CAS:Please enquire for more information about 4-Aminobicyclo[2.2.2]octane-1-carboxylic acid methyl ester including the price, delivery time and more detailed product information at the technical inquiry form on this pageFormula:C10H17NO2Purezza:Min. 95%Peso molecolare:183.25 g/molrac-5,6,7,8-tetrahydro-6-(propylamino)-1-naphthalenol
CAS:Prodotto controllatoRotigotine is a substance that belongs to the class of active compounds. It has been shown to have optical activity, but this property is not well understood. Rotigotine is a racemic mixture with two enantiomers, which are mirror images of each other. The optical rotation of rac-5,6,7,8-tetrahydro-6-(propylamino)-1-naphthalenol is given as +28°. This property can be determined by measuring the angle of rotation when light passes through the substance in solution in contact with a polarizer and analyzer.Formula:C13H19NOPurezza:Min. 95%Peso molecolare:205.3 g/mol1,3,5-Naphthalene trisulfonic acid
CAS:1,3,5-Naphthalene trisulfonic acid is an organic compound that is the product of the sulfonation of naphthalene. It has been shown to inhibit the activity of 3β-hydroxysteroid dehydrogenase and 17β-hydroxysteroid dehydrogenase, enzymes involved in steroidogenesis. The maximal response was observed at a concentration of 500 μM with a detection time of 30 minutes. Xenopus oocytes were used for expression and chloride currents were recorded as an indicator for enzyme activity. Concentration-response curves were generated with organic solvents such as methanol and dimethyl sulfoxide (DMSO). 1,3,5-Naphthalene trisulfonic acid also inhibits the oxidative activities of some enzymes such as lipoxygenase and cyclooxygenase.
Formula:C10H8O9S3Purezza:Min. 95%Peso molecolare:368.36 g/mol3,3'-Difluorobiphenyl
CAS:3,3'-Difluorobiphenyl is a liquid crystal composition that has been shown to have anisotropic properties. When 3,3'-difluorobiphenyl is mixed with other halides such as chloro- or bromo-halides, the liquid crystalline phase can be induced by the addition of ethylene. The anisotropic properties of these compositions make them useful in devices where orientation, reorientation and flow are important. 3,3'-Difluorobiphenyl has also been shown to catalyze the conversion of alcohols to esters and phenols.Formula:C12H8F2Purezza:Min. 95%Peso molecolare:190.19 g/molNelfinavir hydroxy-tert-butylamide
CAS:Nelfinavir is an antiviral agent that is used to treat HIV/AIDS. It is a protease inhibitor that inhibits the action of the virus in cells by binding to specific enzymes, thus preventing the destruction of human cells by the virus. Nelfinavir also prevents cancer cell growth and has shown anticancer activity in animal models and humans. This drug binds to fatty acids, making it more difficult for the body to eliminate this substance. The half-life of nelfinavir is prolonged in patients with hepatic failure or renal failure. Nelfinavir can be used as a chemotherapeutic agent in infants because it does not cross the blood-brain barrier.Formula:C32H45N3O5SPurezza:Min. 95%Peso molecolare:583.78 g/mol10b-Hydroxy delta4-tibolone
CAS:Prodotto controllatoPlease enquire for more information about 10b-Hydroxy delta4-tibolone including the price, delivery time and more detailed product information at the technical inquiry form on this page
Formula:C21H28O3Purezza:Min. 95%Peso molecolare:328.45 g/mol
