CAS 106266-06-2

Risperidona

Descrição:

Risperidona é um medicamento antipsicótico atípico usado principalmente para tratar esquizofrenia, transtorno bipolar e irritabilidade associada ao autismo. Funciona como um antagonista de serotonina e dopamina, influenciando a atividade dos neurotransmissores no cérebro, particularmente os receptores de serotonina e dopamina. Risperidona é caracterizado pela sua fórmula química C23H27N3O2 e um peso molecular de aproximadamente 410,48 g/mol. A substância aparece como um pó cristalino branco a off-white e é tipicamente administrada por via oral, embora formulações injetáveis também estejam disponíveis. Sua farmacocinética indica uma meia-vida relativamente longa, permitindo a dosagem uma vez ao dia em muitos casos. Efeitos colaterais comuns podem incluir sedação, ganho de peso e alterações metabólicas, necessitando monitoramento durante o tratamento. O perfil de eficácia e segurança de Risperidona torna-o uma opção amplamente prescrita na assistência psiquiátrica, embora seja essencial adaptar o tratamento às necessidades individuais do paciente e monitorar possíveis efeitos adversos.

Fórmula: C₂₃H₂₇FN₄O₂

InChI: InChI=1/C23H27FN4O2/c1-15-18(23(29)28-10-3-2-4-21(28)25-15)9-13-27-11-7-16(8-12-27)22-19-6-5-17(24)14-20(19)30-26-22/h5-6,14,16H,2-4,7-13H2,1H3

Chave InChI: InChIKey=RAPZEAPATHNIPO-UHFFFAOYSA-N

SMILES: FC=1C=C2C(C(=NO2)C3CCN(CCC=4C(=O)N5C(=NC4C)CCCC5)CC3)=CC1

Sinónimos:

• 1,2-Benzisoxazole, 4H-pyrido[1,2-a]pyrimidin-4-one deriv.
• 3-(2-(4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-α]pyrimidin-4-one
• 3-[2-[4-(6-Fluor-1,2-benzisoxazol-3-yl)piperidino]ethyl]-2-methyl-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-4-on
• 3-{2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl}-2-methyl-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-4-one
• 4H-Pyrido[1,2-a]pyrimidin-4-one, 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-
• Apexidone
• Psychodal
• R 64766
• Rbp 7000
• Resperidone
• Ripedon
• Risbiodal
• Rispa
• Rispadal
• Risperdal
• Risperdal Consta
• Risperdine
• Risperid
• Risperid fort
• Risperidal
• Risperidone ACIS
• Risperidone intermediates
• Spiron
• Zophrenal
• Risperidone
• 4H-Pyrido[1,2-a]pyrimidin-4-one, 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-(9CI)
• 3-[2-4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-α]pyrimidin-4-one, R-64766, Belivon, Risperdal
• Risoeridone
• 3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-
• Kesperidone
• 3-[2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl]-2-methyl-6,7,8,9-tetrahydropyrido[2,1-b]pyrimidin-4-one
• 3-[2-4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one, R-64766, Belivon, Risperdal
• 4h-pyrido(1,2-a)pyrimidin-4-one,6,7,8,9-tetrahydro-3-(2-(4-(6-fluoro-1,2-benzi
• 3-[2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-
• soxazol-3-yl)-1-piperidinyl)ethyl)-2-methyl-
• 3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-ethyl}-2-methyl-6,7,8,9-tetrahydro-pyrido[1,2,a]pyrimidin-4-one

Risperidone - Bio-X ™

Produto Controlado

CAS: 106266-06-2

Risperidone can be used as an antipsychotic drug in the treatment of schizophrenia and mania. This is due to it binding to the 5-HT2 receptor and antagonizing serotonin, leading to a reduction in symptoms such as delusions and hallucinations. This product can also act on the D1 and D2 Dopamine receptors. It is thought, that as a result of Risperidone’s antagonistic activity against D2 receptors within the tuberoinfundibular pathway, an increase in the level of prolactin occurs.
Risperidone is part of our Bio-X ™ Range. These products are aimed at life science researchers who need high quality ready-to-use products for assay development, screening or other R&D work. With a solubility datasheet and convenient vials, all of our Bio-X ™ products are in stock across our global warehouses for rapid delivery and ease of use.

Fórmula: C₂₃H₂₇FN₄O₂

Pureza: Min. 99.0 Area-%

Cor e Forma: White Powder

Peso molecular: 410.48 g/mol

Ref: 3D-BR164349

Risperidone

Produto Controlado

CAS: 106266-06-2

Risperidone can be used as an antipsychotic drug in the treatment of schizophrenia and mania. This is due to it binding to the 5-HT2 receptor and antagonizing serotonin, leading to a reduction in symptoms such as delusions and hallucinations. This product can also act on the D1 and D2 Dopamine receptors. It is thought, that as a result of Risperidone’s antagonistic activity against D2 receptors within the tuberoinfundibular pathway, an increase in the level of prolactin occurs. Consequently leading to hyperprolactinemia, a negative adverse effect when Risperidone is used as a drug. Risperidone has been shown to have cardiac effects, including increasing heart rate and QT interval. It is also metabolized by cytochrome P450 enzymes and can be detected in wastewater after oral administration of a single dose (0.5 mg/kg).

Fórmula: C₂₃H₂₇FN₄O₂

Pureza: Min. 98.5 Area-%

Cor e Forma: White Off-White Powder

Peso molecular: 410.48 g/mol

Ref: 3D-FR27737

Risperidone

CAS: 106266-06-2

Fórmula: C₂₃H₂₇FN₄O₂

Pureza: 98%

Cor e Forma: Solid, White to off-white powder

Peso molecular: 410.212

Ref: 10-F036563