CAS 1404562-17-9

BRD6688

CAS: 1404562-17-9

BRD6688

Pureza: ≥95%

Peso molecular: 282.34g/mol

Ref: 54-BUP00613

BRD6688

CAS: 1404562-17-9

BRD6688 is a selective HDAC2 inhibitor that acts by enhancing the learning and memory processes

Fórmula: C₁₆H₁₈N₄O

Pureza: 98.36%

Cor e Forma: Solid

Peso molecular: 282.34

Ref: TM-T21715

BRD6688

CAS: 1404562-17-9

BRD6688 is a protein inhibitor that binds to and inhibits the activity of GABA transporters. It is a potent inhibitor of the gaba transporter (GAT) with an IC50 of 0.2 μM. BRD6688 has been shown to inhibit the acetylation of histone proteins, which are important for transcriptional regulation and gene expression. BRD6688 also has a thermodynamic inhibitory constant (Ki) of 1.4 μM and a kinetic inhibitory constant (Ki) of 0.3 μM, indicating that it binds tightly to GATs and does not dissociate easily from it. The Ki values were determined by measuring the inhibition of GAT-mediated chloride transport in cells cultured in vitro. This drug also inhibits antigen presentation in T cells by inhibiting protein synthesis and cell division, as well as histone methylation during mitosis, leading to downregulation of cell-surface antigens on B cells.

Fórmula: C₁₆H₁₈N₄O

Pureza: Min. 95%

Cor e Forma: Powder

Peso molecular: 282.34 g/mol

Ref: 3D-EGC56217