CAS 1443983-36-5

2-[4-[2-[3-(Fluoromethyl)-1-azetidinyl]ethoxy]phenyl]-3-(3-hydroxyphenyl)-4-methyl-2H-1-benzopyran-6-ol

CAS: 1443983-36-5

2-[4-[2-[3-(Fluoromethyl)-1-azetidinyl]ethoxy]phenyl]-3-(3-hydroxyphenyl)-4-methyl-2H-1-benzopyran-6-ol is a potent antagonist for the ion channels TRPC1 and TRPC5. It is also an inhibitor of the human receptor, Ligand, Research tool, Pharmacology, Protein interactions, Peptides, Antibody, Cell Biology, Activator. The ligand has been shown to activate TRPC5 channels in sensory neurons and inhibit TRPC1 channels in bladder cells.

Fórmula: C₂₈H₂₈FNO₄

Pureza: Min. 95%

Peso molecular: 461.5 g/mol

Ref: 3D-THC98336

GDC-0927 Racemate

CAS: 1443983-36-5

GDC-0927 Racemate is a degrader of estrogen receptor, is used in the research of ER-related diseases, potently inhibits ER-α activity, with an IC50 of 0.2 nM.

Fórmula: C₂₈H₂₈FNO₄

Pureza: 98%

Cor e Forma: Solid

Peso molecular: 461.52

Ref: TM-T13700