CAS 1786412-46-1

L-803087 TFA

CAS: 1786412-46-1

L-803087 TFA: potent sst4 agonist, Ki=0.7 nM, >280x selective vs other somatostatin receptors; boosts AMPA, heightens seizures.

Fórmula: C₂₇H₃₀F₅N₅O₅

Cor e Forma: Solid

Peso molecular: 599.55

Ref: TM-T39207

L-803,087 trifluoroacetate

CAS: 1786412-46-1

L-803,087 is a potent and selective activator of the TRPA1 ion channel. It acts as an agonist at TRPA1, which is a member of the transient receptor potential (TRP) family of ion channels. L-803,087 has been shown to activate TRPA1 in a dose-dependent manner. This compound also activates TRPA1 in the presence of elevated levels of extracellular calcium ions and was found to be a potent inhibitor of the phospholipase C enzyme phospholipase Cβ3. L-803,087 also inhibits cell proliferation in human breast cancer cells and has been shown to inhibit protein interactions with bovine serum albumin (BSA).

Fórmula: C₂₇H₃₀F₅N₅O₅

Pureza: Min. 95%

Peso molecular: 599.5 g/mol

Ref: 3D-LWC41246