CAS 2929345-46-8

MKLP2-IN-1

CAS: 2929345-46-8

MKLP2-IN-1 (compound 12a) is an inhibitor of MKLP2 that demonstrates excellent oral bioactivity. In vitro, MKLP2-IN-1 inhibits the ATPase activity stimulated by recombinant MKLP2 microtubules and, in a mouse Calu-6 lung cancer model, it effectively suppresses tumor growth.

Fórmula: C₂₃H₁₉BrFN₃O₂

Cor e Forma: Solid

Peso molecular: 468.318

Ref: TM-T205538