Receptor de Androgénio
O receptor de andrógenos (AR) é um receptor hormonal nuclear que é ativado pela ligação a andrógenos, como a testosterona e a diidrotestosterona. Este receptor desempenha um papel crucial no desenvolvimento e na manutenção das características masculinas, bem como na regulação de vários processos fisiológicos, incluindo o crescimento muscular, a libido e a densidade óssea. Inibidores do receptor de andrógenos são amplamente estudados no contexto do câncer de próstata, onde a sinalização do AR é frequentemente aumentada. Na CymitQuimica, oferecemos uma gama de moduladores do receptor de andrógenos de alta qualidade para apoiar sua pesquisa em endocrinologia, biologia do câncer e regulação hormonal.
Foram encontrados 207 produtos de "Receptor de Androgénio"
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Fenarimol
CAS:<p>Fenarimol, a pyrimidine-type fungicide, exhibits potent inhibitory activity against BR biosynthesis.</p>Fórmula:C17H12Cl2N2OCor e Forma:SolidPeso molecular:331.2MK-0773
CAS:<p>MK-0773 (PF-05314882) is a selective androgen receptor modulator that binds to AR (IC50: 6.6 nM) for the study of diseases caused by endocrine abnormalities.</p>Fórmula:C27H34FN5O2Pureza:98.38% - 99.14%Cor e Forma:SolidPeso molecular:479.59Dehydroepiandrosterone-d2
CAS:<p>Dehydroepiandrosterone-d2 is a deuterated compound of Dehydroepiandrosterone.</p>Fórmula:C19H26D2O2Cor e Forma:SolidPeso molecular:290.44ARD-1676
CAS:<p>ARD-1676 is an orally administered androgen receptor (AR) PROTAC degrader that combines an AR ligand with a cereblon ligand.</p>Fórmula:C44H46ClN7O5Pureza:98%Cor e Forma:SolidPeso molecular:788.33Leelamine hydrochloride
CAS:<p>Leelamine hydrochloride, a pine bark extract, inhibits androgen receptor and CB1, reducing lipid synthesis in prostate cancer.</p>Fórmula:C20H32ClNPureza:98%Cor e Forma:SolidPeso molecular:321.93(Rac)-PF-998425
CAS:<p>(Rac)-PF-998425: nonsteroidal AR antagonist, potent & selective, IC50: 26 nM (binding), 90 nM (cellular), potential for androgenetic alopecia study.</p>Fórmula:C14H14F3NOCor e Forma:SolidPeso molecular:269.267Rezvilutamide
CAS:<p>Rezvilutamide (SHR3680) is an orally available androgen receptor inhibitor that crosses the blood-brain barrier and has antitumor activity.</p>Fórmula:C22H20F3N3O4SPureza:99.97%Cor e Forma:SolidPeso molecular:479.47D4-abiraterone
CAS:<p>D4-abiraterone is the active metabolite of abiraterone.Δ4-Abiraterone is a inhibitor of CYP17A1, 3β-HSD and SRD5A, and an antagonist of the androgen receptor.</p>Fórmula:C24H29NOPureza:99.75% - 99.8%Cor e Forma:SolidPeso molecular:347.49VPC-13566
CAS:<p>VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the</p>Fórmula:C18H14N2Pureza:99.55%Cor e Forma:SolidPeso molecular:258.323-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile
CAS:<p>3-[7 ,7- dimethyl-5-oxo -6H-pyrrolo[3,4-b]pyridin-2-yI]-1H-indole-7 -carbonitrile is an androgen receptor modulator.</p>Fórmula:C18H14N4OPureza:98.41%Cor e Forma:SolidPeso molecular:302.33AH-3960
CAS:<p>AH-3960 是一种甲状腺激素受体 1 (PTHR1) 激动剂。</p>Fórmula:C13H22N4O3Pureza:98.44%Cor e Forma:SolidPeso molecular:282.34Darolutamide
CAS:<p>Darolutamide (BAY-1841788) is an androgen receptor (AR) antagonist that blocks AR nuclear translocation (Ki: 11 nM).</p>Fórmula:C19H19ClN6O2Pureza:97.36% - >99.99%Cor e Forma:SolidPeso molecular:398.85Enzalutamide
CAS:<p>Enzalutamide (MDV3100) is an androgen receptor (AR) antagonist (IC50=36 nM in LNCaP).</p>Fórmula:C21H16F4N4O2SPureza:99% - 99.93%Cor e Forma:SolidPeso molecular:464.44Nandrolone phenylpropionate
CAS:<p>Nandrolone phenylpropionate (Nandrolone phenpropionate) is an androgen receptor agonist. It mainly used to treat women with breast cancer and osteoporosis</p>Fórmula:C27H34O3Pureza:99.2% - 99.46%Cor e Forma:White Or Milky Crystalline PowderPeso molecular:406.56CTK8A3536
CAS:<p>CTK8A3536 ((2-MORPHOLIN-4-YL-4-PHENYL-1,3-THIAZOL-5-YL)METHANOL) is an inhibitor of Androgen receptor.</p>Fórmula:C14H16N2O2SPureza:99.62%Cor e Forma:SolidPeso molecular:276.35MI-136
CAS:<p>MI-136 inhibits expression of androgen receptor (AR) target genes that DHT induced.</p>Fórmula:C23H21F3N6SPureza:98.63% - 99.12%Cor e Forma:SolidPeso molecular:470.51Lupeol
CAS:<p>Lupeol (Monogynol B) is a novel androgen receptor inhibitor with anti-inflammatory and antioxidant activity.</p>Fórmula:C30H50OPureza:98% - 99.96%Cor e Forma:Needles From Alcohol Acetone White PowderPeso molecular:426.72ARD-2128
CAS:<p>ARD-2128: potent oral PROTAC that degrades AR, curbing prostate cancer growth with no toxicity.</p>Fórmula:C45H50ClN7O6Pureza:98.8%Cor e Forma:SolidPeso molecular:820.37Dimethylcurcumin
CAS:<p>Dimethylcurcumin (ASC-J9) (ASC-J9) is an androgen receptor degradation enhancer.</p>Fórmula:C23H24O6Pureza:97.36% - 98.96%Cor e Forma:SolidPeso molecular:396.43Bavdegalutamide
CAS:<p>Bavdegalutamide (ARV-110) is a PROTAC degrader of androgen receptor (AR).</p>Fórmula:C41H43ClFN9O6Pureza:97.17% - 99.04%Cor e Forma:SolidPeso molecular:812.29
![3-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT9752.webp&w=3840&q=75)
