
Receptor de Androgénio
O receptor de andrógenos (AR) é um receptor hormonal nuclear que é ativado pela ligação a andrógenos, como a testosterona e a diidrotestosterona. Este receptor desempenha um papel crucial no desenvolvimento e na manutenção das características masculinas, bem como na regulação de vários processos fisiológicos, incluindo o crescimento muscular, a libido e a densidade óssea. Inibidores do receptor de andrógenos são amplamente estudados no contexto do câncer de próstata, onde a sinalização do AR é frequentemente aumentada. Na CymitQuimica, oferecemos uma gama de moduladores do receptor de andrógenos de alta qualidade para apoiar sua pesquisa em endocrinologia, biologia do câncer e regulação hormonal.
Foram encontrados 207 produtos de "Receptor de Androgénio"
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MI-136
CAS:<p>MI-136 inhibits expression of androgen receptor (AR) target genes that DHT induced.</p>Fórmula:C23H21F3N6SPureza:98.63% - 99.12%Cor e Forma:SolidPeso molecular:470.51Apalutamide
CAS:<p>Apalutamide (ARN-509) is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.</p>Fórmula:C21H15F4N5O2SPureza:99.03% - 99.91%Cor e Forma:SolidPeso molecular:477.43S-23
CAS:<p>S-23 ((S)-3-(4-chloro-3-fluorophenoxy)-N-(4-cyano-3-(trifluoromethyl)phenyl)-2-hydroxy-2-methylpropanamide) is an oral selective androgen receptor modulator (</p>Fórmula:C18H13ClF4N2O3Pureza:99.55%Cor e Forma:SolidPeso molecular:416.75Iprodione
CAS:<p>Iprodione is a fungicide. Iprodione is also used in cannabis testing kits as a component of pesticide mixes.</p>Fórmula:C13H13Cl2N3O3Pureza:98.82%Cor e Forma:Colorless Crystals Cream To Colorless Odorless PowderPeso molecular:330.17Testosterone undecanoate
CAS:<p>Testosterone undecanoate is a metabolite of Testosterone, which is a promising androgen for male hormonal contraception.</p>Fórmula:C30H48O3Pureza:99.45% - 99.788%Cor e Forma:White Crystalline PowderPeso molecular:456.7CLP-3094
CAS:<p>CLP-3094 (2-([2-(4-CHLOROPHENOXY)ETHYL]THIO)-1H-BE) is a potent androgen receptor BF3 (binding function 3) inhibitor.</p>Fórmula:C15H13ClN2OSPureza:99.84%Cor e Forma:SolidPeso molecular:304.79AC-262536
CAS:<p>AC-262536 is a selective androgen receptor (SAR) modulator and exhibits potent agonist activity at the androgen receptor.</p>Fórmula:C18H18N2OPureza:99.88%Cor e Forma:SolidPeso molecular:278.35Triptophenolide
CAS:<p>Triptophenolide (Hypolide) is a compound isolated from Tripterygium wilfordii Hook with anti-inflammatory activity.</p>Fórmula:C20H24O3Pureza:98.07% - ≥95%Cor e Forma:White PowderPeso molecular:312.4Boldenone Undecylenate
CAS:<p>Boldenone Undecylenate (Parenabol) is a synthetic steroid.</p>Fórmula:C30H44O3Pureza:99.39%Cor e Forma:Light Yellow Oily MatterPeso molecular:452.67JNJ-63576253 free base
CAS:<p>JNJ-63576253 free base (TRC253) is a potent and orally active full antagonist of androgen receptor (AR). JNJ-63576253 can be used for the research of CRPC.</p>Fórmula:C23H21F3N6O2SPureza:98.32%Cor e Forma:SolidPeso molecular:502.51Dimethylcurcumin
CAS:<p>Dimethylcurcumin (ASC-J9) (ASC-J9) is an androgen receptor degradation enhancer.</p>Fórmula:C23H24O6Pureza:97.36% - 98.96%Cor e Forma:SolidPeso molecular:396.43Nandrolone phenylpropionate
CAS:<p>Nandrolone phenylpropionate (Nandrolone phenpropionate) is an androgen receptor agonist. It mainly used to treat women with breast cancer and osteoporosis</p>Fórmula:C27H34O3Pureza:99.2% - 99.46%Cor e Forma:White Or Milky Crystalline PowderPeso molecular:406.56JNJ-63576253
CAS:<p>JNJ-63576253 is a Clinical Stage Androgen Receptor Antagonist for F877L Mutant and Wild-Type Castration-Resistant Prostate Cancer (mCRPC).</p>Fórmula:C23H22ClF3N6O2SPureza:98.71%Cor e Forma:SolidPeso molecular:538.97Ailanthone
CAS:<p>Ailanthone (Δ13-Dehydrochaparrinone) is an effective inhibitor of both full-length androgen receptor (AR) (IC50: 69 nM) and constitutively active truncated AR</p>Fórmula:C20H24O7Pureza:99.71% - 99.96%Cor e Forma:SolidPeso molecular:376.43-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile
CAS:<p>3-[7 ,7- dimethyl-5-oxo -6H-pyrrolo[3,4-b]pyridin-2-yI]-1H-indole-7 -carbonitrile is an androgen receptor modulator.</p>Fórmula:C18H14N4OPureza:98.41%Cor e Forma:SolidPeso molecular:302.33ARD-2128
CAS:<p>ARD-2128: potent oral PROTAC that degrades AR, curbing prostate cancer growth with no toxicity.</p>Fórmula:C45H50ClN7O6Pureza:98.8%Cor e Forma:SolidPeso molecular:820.372-hydroxy Flutamide
CAS:<p>2-hydroxy Flutamide is competitive inhibition of androgen receptor (AR) for the treatment of prostate cancer</p>Fórmula:C11H11F3N2O4Pureza:99.45% - 99.82%Cor e Forma:SolidPeso molecular:292.21AH-3960
CAS:<p>AH-3960 是一种甲状腺激素受体 1 (PTHR1) 激动剂。</p>Fórmula:C13H22N4O3Pureza:98.44%Cor e Forma:SolidPeso molecular:282.34DSRM-3716
CAS:<p>Isoquinoline, 5-iodo- (9CI) is a potent and selective inhibitor of SARM1(IC50 = 75 nM) by preventing axonal degeneration and by allowing functional recovery of</p>Fórmula:C9H6INPureza:97.28% - 99.785%Cor e Forma:SolidPeso molecular:255.06Bavdegalutamide
CAS:<p>Bavdegalutamide (ARV-110) is a PROTAC degrader of androgen receptor (AR).</p>Fórmula:C41H43ClFN9O6Pureza:97.17% - 99.04%Cor e Forma:SolidPeso molecular:812.29
