Canais de Cálcio
Os canais de cálcio são proteínas de membrana que regulam o fluxo de íons de cálcio para dentro e fora das células, o que é essencial para várias funções celulares, incluindo a contração muscular, a liberação de neurotransmissores e a expressão gênica. A desregulação da atividade dos canais de cálcio está associada a condições como hipertensão, arritmias cardíacas e distúrbios neurológicos. Na CymitQuimica, oferecemos uma ampla seleção de moduladores de canais de cálcio para apoiar sua pesquisa em saúde cardiovascular, neurobiologia e transdução de sinais.
Foram encontrados 544 produtos de "Canais de Cálcio"
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Watanidipine dihydrochloride
CAS:Watanidipine dihydrochloride is a novel dihydropyridine (DHP)-type calcium channel blocker with slow-onset pharmacological actions.Fórmula:C41H44Cl2N4O6Pureza:98%Cor e Forma:SolidPeso molecular:759.73Levosemotiadil
CAS:Levosemotiadil（SA 3212） is a novel calcium antagonist and a very potent inhibitor of low-density lipoprotein oxidation.Levosemotiadil may be used to preventFórmula:C29H32N2O6SPureza:98.53% - 98.88%Cor e Forma:SolidPeso molecular:536.64BK 129
CAS:BK 129 is a local anesthetic with relaxant properties. BK 129 inhibits Ca2+ entry into the smooth muscle cell and Ca2+ release from sarcoplasmic reticulum.Fórmula:C22H36N2O4Pureza:98%Cor e Forma:SolidPeso molecular:392.53(R)-Amlodipine
CAS:(R)-Amlodipine is the R-enantiomer of Amlodipine and functions as an orally active dihydropyridine calcium channel blocker with antianginal properties.Fórmula:C20H25ClN2O5Pureza:99.977%Cor e Forma:SolidPeso molecular:408.88Diltiazem malate
CAS:Diltiazem malate is an ACE inhibitor and non-dihydropyridine calcium channel blocker used in the treatment of hypertension.Fórmula:C26H32N2O9SCor e Forma:SolidPeso molecular:548.60SCH00013
CAS:SCH00013 is a cardiotonic that enhances myofibrillar Ca++ sensitivity, with notable effects at pH 7.2-7.4.Fórmula:C18H20N4O2Pureza:98%Cor e Forma:SolidPeso molecular:324.38GZ4
CAS:GZ4 is a Ca2+ currents inhibitor, acting on cell surface channels.Fórmula:C11H17NO2Pureza:98%Cor e Forma:SolidPeso molecular:195.26AJG-049 HCl
CAS:AJG-049 HCl is a calcium channel antagonist that inhibits L-type Ca2+ channels via diltiazem-binding site(s).Fórmula:C27H31ClN2O2Cor e Forma:SolidPeso molecular:451.01ML218 hydrochloride
CAS:ML218 hydrochloride inhibits T-type Ca2+ channels Cav3.1-3.3; most effective on Cav3.2 and Cav3.3 (IC50s: 310 nM, 270 nM).Fórmula:C19H27Cl3N2OPureza:98%Cor e Forma:SolidPeso molecular:405.79ITH-12575
CAS:ITH-12575 is an inhibitor of Mitochondrial Na+/Ca2+ exchange (mNCX). ITH12575 reduces Ca(2+) influx through CALHM1 at low micromolar concentrations.Fórmula:C18H18ClNOSCor e Forma:SolidPeso molecular:331.86Dopropidil
CAS:Dopropidil: anti-angina calcium regulator with anti-ischemic properties in animal models.Fórmula:C20H35NO2Pureza:98%Cor e Forma:SolidPeso molecular:321.5CaV1.3 antagonist-1
CAS:CaV1.3 antagonist-1 is a selective CaV1.3L-type calcium channel antagonist useful for researching neurological disorders and cardiovascular diseases.Fórmula:C17H19ClN2O3Cor e Forma:SolidPeso molecular:334.8UK51656
CAS:UK51656 is an antagonist of calcium (IC50: 4 nM).Fórmula:C22H28ClN3O6Pureza:98%Cor e Forma:SolidPeso molecular:465.93RS 30026
CAS:RS 30026 is a potent calcium channel agonist.Fórmula:C23H21NO4SCor e Forma:SolidPeso molecular:407.48JTV-519 free base
CAS:JTV-519 free base (K201 free base), recognized for its antiarrhythmic and cardioprotective properties, functions as a Ca2+-dependent blocker of sarcoplasmicFórmula:C25H32N2O2SPureza:98%Cor e Forma:SolidPeso molecular:424.6Palonidipine
CAS:Palonidipine is an antagonist of calcium, is potential for the therapy of angina-pectoris and hypertension.Fórmula:C29H34FN3O6Pureza:98%Cor e Forma:SolidPeso molecular:539.6Ned-K
CAS:Ned-K blocks NAADP, reduces heart ischemia-reperfusion calcium waves.Fórmula:C31H31N5O3Cor e Forma:SolidPeso molecular:521.61NC 1100
CAS:NC 1100 is a calcium channel antagonist.Fórmula:C27H34Cl2N2O3Pureza:98%Cor e Forma:SolidPeso molecular:505.48BN 50341
CAS:BN 50341 is an inhibitor of antithrombotic platelet activating factor.Fórmula:C32H41ClN2O4Pureza:98%Cor e Forma:SolidPeso molecular:553.13Nemadipine-A
CAS:Nemadipine A blocks L-type Ca2+ channels, alters C. elegans morphology, boosts TRAIL's cancer kill rate, and lowers Survivin in A549 cells.Fórmula:C19H18F5NO4Cor e Forma:SolidPeso molecular:419.34Gallopamil, (-)-
CAS:Gallopamil, (-)- is an L-type calcium channel blocker. It is used in the treatment of abnormal heart rhythms.Fórmula:C28H40N2O5Pureza:98%Cor e Forma:SolidPeso molecular:484.63EO-122
CAS:EO-122, a calcium channel antagonist and sodium channel antagonist, is used potentially for the treatment of arrhythmia.Fórmula:C16H23ClN2OCor e Forma:SolidPeso molecular:294.82SQ-31765
CAS:SQ-31765 is a blocker of benzazepine calcium channel.Fórmula:C24H27F3N2O4Pureza:98%Cor e Forma:SolidPeso molecular:464.48TDN345
CAS:TDN345 is a antagonist of Ca2+, for the treatment of vascular and senile dementia including Alzheimer's disease.Fórmula:C28H34F2N2O2Pureza:98%Cor e Forma:SolidPeso molecular:468.58Cyclic ADP-ribose
CAS:cADPR, made from NAD+, boosts calcium in cells via Ryanodine receptors and TRPM2 channels.Fórmula:C15H21N5O13P2Pureza:98%Cor e Forma:Lyophilized PowderPeso molecular:541.3TTA-A8
CAS:TTA-A8 is an antagonist of T-type calcium channel.Fórmula:C22H21F3N4O2Pureza:99.22%Cor e Forma:SolidPeso molecular:430.42KB-130015
CAS:KB-130015, a activator of hERG1 potassium channels, blocks native and recombinant hERG1 channels at high voltages.Fórmula:C18H14I2O4Pureza:98%Cor e Forma:SolidPeso molecular:548.11McN5691
CAS:McN5691 is a voltage sensitive calcium channel blocker.Fórmula:C30H35NO3Pureza:98.93% - 99.38%Cor e Forma:SolidPeso molecular:457.6Gallopamil hydrochloride
CAS:Gallopamil hydrochloride (Methoxyverapamil hydrochloride) is an antagonist of phenylalkylamine calcium.Fórmula:C28H41ClN2O5Pureza:99.86%Cor e Forma:SolidPeso molecular:521.09Ref: TM-T11353L
1mg38,00€5mg73,00€10mg90,00€25mg140,00€50mg183,00€100mg283,00€500mg692,00€1mL*10mM (DMSO)90,00€(2R/S)-6-PNG
CAS:(2R/S)-6-PNG (6-Prenylnaringenin) from hops is a natural histone deacetylase inhibitor that blocks T-type calcium channels reducing neurogenicity in mice.Fórmula:C20H20O5Pureza:98%Cor e Forma:SolidPeso molecular:340.37Norverapamil
CAS:Norverapamil is a blocker of L-type calcium channel and an inhibitor of P-glycoprotein (P-gp) function .Fórmula:C26H36N2O4Pureza:98%Cor e Forma:SolidPeso molecular:440.58JTV-519 fumarate
CAS:Ryanodine receptor (RyR) inhibitor; stabilizes RyR2 in a closed conformation. Exhibits antiarrhythmic and cardioprotective properties in vivo.Fórmula:C29H36N2O6SCor e Forma:SolidPeso molecular:540.67Gallopamil HCl, (-)-
CAS:Gallopamil HCl, (-)- is an L-type calcium channel blocker. It is used in the treatment of abnormal heart rhythms.Fórmula:C28H41ClN2O5Pureza:98%Cor e Forma:SolidPeso molecular:521.09A 39355
CAS:A 39355 may specifically overcome multidrug resistance without the serious hypotensive effects associated with calcium antagonists.Fórmula:C28H39Cl2N3OPureza:98%Cor e Forma:SolidPeso molecular:504.54AH-1058 HCl
CAS:AH-1058 HCl is a lipophilic antiarrhythmic calcium channel blocker.Fórmula:C30H29ClN2O3Pureza:98%Cor e Forma:SolidPeso molecular:501.02Hns 32
CAS:Hns 32 possesses antiarrhythmic properties in dog and guinea pig hearts. It also has vasodilator action.Fórmula:C24H29N3Pureza:98%Cor e Forma:SolidPeso molecular:359.51A 80b
CAS:A-80b: synthetic pyridazinoindole; potent, lasting antihypertensive; lowers diastolic more; no change in heart rate; inhibits Ca2+-induced contraction.Fórmula:C16H17N7Pureza:98%Cor e Forma:SolidPeso molecular:307.35Methsuximide
CAS:Methsuximide is an anticonvulsant agent which appeared to be effective in petit mal, psychomotor and focal motor attacks [1].Fórmula:C12H13NO2Cor e Forma:Crystals From Dilute Alcohol SolidPeso molecular:203.243',4'-Dichlorobenzamil HCl
CAS:3',4'-Dichlorobenzamil HCl is an inhibitor of Na+ transport, Na+/Ca2+ exchanger, sarcoplasmic reticulum Ca2+ release channels.Fórmula:C13H12Cl3N7OPureza:98%Cor e Forma:Yellow SolidPeso molecular:388.64BAY-Y-5959
CAS:BAY-Y-5959, a calcium channel agonist, is used potentially for the treatment of arrhythmia, heart failure and myocardial.Fórmula:C26H24N4O2Cor e Forma:SolidPeso molecular:424.49AK-2-38
CAS:AK-2-38 is a nifedipine analogue with potent smooth muscle calcium antagonist action and partial agonist effects on isolated guinea pig left atrium.Fórmula:C26H30N2O4Pureza:98%Cor e Forma:SolidPeso molecular:434.53Aladorian
CAS:Aladorian (ARM036), a benzothiazepine, has anti-arrhythmic properties for heart failure and CPVT research.Fórmula:C12H13NO4SPureza:98%Cor e Forma:SolidPeso molecular:267.3Aprindine hydrochloride
CAS:Aprindine HCl, a Class 1b antiarrhythmic, treats heart arrhythmias, outperforming digoxin in delaying atrial fibrillation. It's effective orally.Fórmula:C22H31ClN2Cor e Forma:SolidPeso molecular:358.95Levamlodipine gentisate
CAS:Levamlodipine gentisate, an active amlodipine enantiomer, is a dihydropyridine calcium channel blocker for treating hypertension and angina.Fórmula:C27H31ClN2O9Pureza:98%Cor e Forma:SolidPeso molecular:563GSK205
CAS:GSK205 is a selective TRPV4 antagonist (IC50: 4.19 μM) for inhibiting TRPV4-mediated Ca2+ influx.Fórmula:C24H25BrN4SPureza:99.46%Cor e Forma:SolidPeso molecular:481.45Ref: TM-T11480
1mg70,00€5mg154,00€10mg235,00€25mg518,00€50mg847,00€100mg1.359,00€1mL*10mM (DMSO)162,00€R 56865
CAS:R 56865 is a weak potential-operated channel inhibitor that inhibits the late sodium current in human isolated cardiomyocytes.Fórmula:C23H28FN3OSPureza:99.52%Cor e Forma:SolidPeso molecular:413.55Cronidipine
CAS:Cronidipine (LF 20254), a calcium channel antagonist, is used potentially for the treatment of hypertension and myocardia ischemia.Fórmula:C30H32ClN3O8Pureza:99.47%Cor e Forma:SolidPeso molecular:598.04Enecadin
CAS:Enecadin is a neuroprotective agent.Fórmula:C21H28FN3OPureza:98.53%Cor e Forma:SolidPeso molecular:357.46Cerebrocrast
CAS:Cerebrocrast (IOS-11212) has anti-inflammatory and hypoglycemic activity, blocks human platelet activation, and is used in the study of diabetes.Fórmula:C26H35F2NO7Pureza:99.71%Cor e Forma:SolidPeso molecular:511.56Terflavoxate
CAS:<p>Terflavoxate is a novel, orally active, semisynthetic statin microtubule inhibitor commonly used in combination with capecitabine.</p>Fórmula:C26H29NO4Pureza:98%Cor e Forma:SolidPeso molecular:419.51Gallopamil
CAS:Gallopamil blocks acid secretion (IC50: 10.9 μM), acts as antiarrhythmic, vasodilator, and is a methoxy Verapamil derivative.Fórmula:C28H40N2O5Pureza:99.85%Cor e Forma:SolidPeso molecular:484.63Ref: TM-T11353
1mg38,00€5mg79,00€10mg119,00€25mg188,00€50mg283,00€100mg430,00€500mg938,00€1mL*10mM (DMSO)85,00€Vatanidipine
CAS:Vatanidipine (AE0047) is a novel dihydropyridine (DHP)-type calcium channel blocker with slow-onset pharmacological actions.A slow-onset and long-lastingFórmula:C41H42N4O6Pureza:99.95%Cor e Forma:SolidPeso molecular:686.8Ref: TM-T24932
1mg187,00€5mg454,00€10mg622,00€25mg940,00€50mg1.264,00€100mg1.663,00€1mL*10mM (DMSO)730,00€N106
CAS:N106 is an activator of the SUMO-activating enzyme, E1 ligase, and triggers intrinsic sumoylation of SERCA2a. N106 can be used in studies about heart failure.Fórmula:C17H14N4O3SPureza:99.69%Cor e Forma:SolidPeso molecular:354.38CERM-11956
CAS:Pelretin (BASF 43915) is a potential protein inhibitor for the study of dermatologic diseases.Fórmula:C29H38N2O7Pureza:99.38%Cor e Forma:SolidPeso molecular:526.62FPL-62129
CAS:FPL-62129 is a calcium channel antagonist and a novel angiotensin-converting enzyme inhibitor with vasodilator activity for the study of cardiovascular disease.Fórmula:C20H19ClF5NO4Pureza:98.27% - 99.34%Cor e Forma:SolidPeso molecular:467.81Opc 8490
CAS:Opc 8490 is a cardiotonic agent and a positive inotropic vasodilator, which prolongs the atrial action potential in a concentration-dependent manner.Fórmula:C30H35N3O10Pureza:98.88%Cor e Forma:SolidPeso molecular:597.61Sipatrigine
CAS:Sipatrigine (619C89) is an inhibitor of glutamate release, TREK ion channels, TRESK channels, sodium channels, and calcium channels.Fórmula:C15H16Cl3N5Pureza:98.64% - 99.77%Cor e Forma:SolidPeso molecular:372.68Ref: TM-T16887
1mg92,00€5mg192,00€10mg286,00€25mg480,00€50mg692,00€100mg973,00€200mg1.305,00€1mL*10mM (DMSO)212,00€AZD-1305
CAS:<p>AZD-1305: novel anti-arrhythmic blocking IKr, Ca, Na currents; useful in arrhythmia research.</p>Fórmula:C22H31FN4O4Pureza:99.31% - 99.86%Cor e Forma:SolidPeso molecular:434.5Tamolarizine
CAS:<p>Tamolarizine (Tamolarizine free base) free base is a novel calcium antagonist.</p>Fórmula:C27H32N2O3Pureza:98.17%Cor e Forma:SoildPeso molecular:432.55Sulcardine sulfate
CAS:<p>Sulcardine sulfate (B-87823) is a multi-ion channel blocker with antiarrhythmic activity that inhibits Na+, K+, and Ca2+ channels.</p>Fórmula:C24H35N3O8S2Pureza:98.74%Cor e Forma:SolidPeso molecular:557.68O-1602
CAS:O-1602 is a novel GPR55 agonist, an atypical cannabinoid associated with the central nervous system and obesity, and is a candidate compound for the treatmentFórmula:C17H22O2Pureza:99.85%Cor e Forma:SolidPeso molecular:258.36Ref: TM-T23097
1mg47,00€5mg90,00€10mg144,00€25mg268,00€50mg378,00€100mg567,00€200mg805,00€1mL*10mM (DMSO)100,00€Clopimozide
CAS:Clopimozide (R-29764), a long-acting oral antischizophrenic, blocks calcium channels and [3H] nilandipine binding.Fórmula:C28H28ClF2N3OPureza:98.99% - 99.66%Cor e Forma:SolidPeso molecular:495.99SERCA2a activator 1
CAS:SERCA2a activator 1 boosts heart function by reducing phospholamban restraint and enhancing cardiac contraction-relaxation cycles.Fórmula:C32H29N3O4SPureza:99.75%Cor e Forma:SolidPeso molecular:551.66Ref: TM-T16873
1mg187,00€5mg472,00€10mg660,00€25mg1.035,00€50mg1.483,00€100mg2.072,00€1mL*10mM (DMSO)563,00€VU 0240551
CAS:VU 0240551 is a selective antagonist of neuronal K-Cl cotransporter KCC2 inhibitor with an IC50 of 560 nM. VU 0240551 inhibits L-type calcium channels and hERG.Fórmula:C16H14N4OS2Pureza:99.9%Cor e Forma:SolidPeso molecular:342.44Ref: TM-TQ0139
1mg37,00€5mg78,00€10mg125,00€25mg255,00€50mg439,00€100mg705,00€200mg938,00€500mg1.415,00€1mL*10mM (DMSO)86,00€CP-060
CAS:CP-060 is a potent Ca2+ antagonist and inhibits Ca2+ overload with antioxidant and cardioprotective activities.Fórmula:C30H42N2O5SPureza:99.54%Cor e Forma:SolidPeso molecular:542.73Ref: TM-T10874
1mg239,00€5mg474,00€10mg638,00€25mg950,00€50mg1.283,00€100mg1.730,00€200mg2.337,00€1mL*10mM (DMSO)642,00€PD173212
CAS:PD 173212 is a blocker that blocks N-type voltage sensitive calcium channel (Cav2.2).Fórmula:C38H53N3O3Pureza:99.84%Cor e Forma:SolidPeso molecular:599.85Ref: TM-T16448
2mg46,00€5mg80,00€10mg116,00€25mg190,00€50mg284,00€100mg395,00€200mg560,00€1mL*10mM (DMSO)96,00€Ticolubant
CAS:Ticolubant: Oral LTB4 antagonist, Ki=0.78 nM; blocks Ca2+ migration, IC50=6.6 nM; anti-inflammatory in mice.Fórmula:C23H19Cl2NO3SPureza:99.5%Cor e Forma:SolidPeso molecular:460.37Lifarizine
CAS:Lifarizine (RS-87476), a calcium-sodium channel antagonist, shows neuroprotective activity in a simplified rat survival model of double vessel occlusion.Fórmula:C29H32N4Pureza:99.88%Cor e Forma:SolidPeso molecular:436.598-Bromo-cGMP sodium
CAS:<p>8-Bromo-cGMP sodium: PKG activator, eases pain, dilates vessels, reduces Ca2+ currents & insulin release.</p>Fórmula:C10H10BrN5NaO7PPureza:99.45%Cor e Forma:SolidPeso molecular:446.09Tiapamil hydrochloride
CAS:Tiapamil hydrochloride (Ro 11-1781 hydrochloride) is a calcium channel blocker with antihypertensive activity used in the study of angina pectoris.Fórmula:C26H38ClNO8S2Pureza:99.17%Cor e Forma:SolidPeso molecular:592.16Crobenetine
CAS:Crobenetine (BIII 890 CL) Free Base is a selective NaV channel blocker that eliminates VTD-induced [Ca2+] elevation.Fórmula:C25H33NO2Pureza:98.99%Cor e Forma:SolidPeso molecular:379.54Upacicalcet
CAS:Upacicalcet (AJT-240) is a calcium mimetic for SHPT in dialysis, reducing PTH by targeting parathyroid receptors.Fórmula:C11H14ClN3O6SPureza:99.88%Cor e Forma:SolidPeso molecular:351.76Fenoverine
CAS:Fenoverine (Spasmopriv) has antispasmodic activity and can be used to study gastrointestinal spasms.Fórmula:C26H25N3O3SPureza:98.34%Cor e Forma:SolidPeso molecular:459.56Ref: TM-T62889
1mg66,00€5mg142,00€10mg222,00€25mg447,00€50mg715,00€100mg1.063,00€200mg1.459,00€1mL*10mM (DMSO)145,00€NecroX-5
CAS:<p>NecroX-5, a derivative of NecroX, exhibits anti-inflammatory and anti-cancer activities. NecroX-5 reduces intracellular calcium concentration.</p>Fórmula:C27H39N3O9S3Pureza:99.944%Cor e Forma:SolidPeso molecular:645.81Diproteverine HCl
CAS:<p>Diproteverine HCl is a novel calcium antagonist with antianginal properties, antispasmodic and vasoactive.</p>Fórmula:C26H36ClNO4Pureza:98.55% - 99.84%Cor e Forma:SolidPeso molecular:462.02DS16570511
CAS:DS16570511 is a novel, cell-permeable inhibitor targeting the mitochondrial calcium uniporter.Fórmula:C30H25Cl2N3O4Pureza:98.34% - 98.45%Cor e Forma:SolidPeso molecular:562.44MONIRO-1
CAS:MONIRO-1 blocks T/N-type Ca²⁺ channels: hCav2.2 (IC50: 34μM), hCav3.1 (3.3μM), hCav3.2 (1.7μM), hCav3.3 (7.2μM).Fórmula:C23H24ClFN4O3Cor e Forma:SolidPeso molecular:458.92N-type calcium channel blocker-1
CAS:N-type calcium channel blocker-1 is an orally active analgesic agent,shows high affinity to functionally block N-type calcium channels.Fórmula:C31H47N3Pureza:98%Cor e Forma:SolidPeso molecular:461.73RS 5773
CAS:RS 5773 is a benzothiazepine derivative with antianginal effects.Fórmula:C29H33ClN2O4SPureza:98%Cor e Forma:SolidPeso molecular:541.1Piprofurol
CAS:Piprofurol is used as a Calcium channel blocker.Fórmula:C26H33NO6Pureza:98%Cor e Forma:SolidPeso molecular:455.54TMDJ-035
CAS:TMDJ-035 is a selective inhibitor of the RyR2 (ryanodine receptor 2).Fórmula:C16H12F3N5OPureza:98%Cor e Forma:SolidPeso molecular:347.29(S)-(-)-Bay-K-8644
CAS:(S)-(-)-Bay-K-8644 ((S)-(-)-Bay K 8644) is an agonist of L-type Ca2+ channel and activates Ba2+ currents with an EC50 of 32 nM.Fórmula:C16H15F3N2O4Pureza:98.28% - 99.37%Cor e Forma:SolidPeso molecular:356.3HA-1004 dihydrochloride
CAS:HA-1004 dihydrochloride is an inhibitor of PKA, PKC, cGKI, MYLK, and calcium channel proteinFórmula:C12H16ClN5O2SPureza:98%Cor e Forma:White Crystalline SolidPeso molecular:329.81Coelenterazine h
CAS:Coelenterazine H, a Ca2+ sensitive synthetic derivative, is a luminescent biomolecule used to measure Ca2+ changes.Fórmula:C26H21N3O2Pureza:99.58%Cor e Forma:Yellow To Brownish PowderPeso molecular:407.46Ref: TM-T14994
1mg87,00€5mg216,00€10mg354,00€25mg582,00€50mg825,00€100mg1.111,00€200mg1.491,00€500µg67,00€5J-4
CAS:<p>5J-4 is a potent a blocker of calcium release-activated calcium (CRAC) channel and store-operated calcium entry (SOCE).</p>Fórmula:C16H12N2O3SPureza:96.12%Cor e Forma:SolidPeso molecular:312.34Cav 3.2 inhibitor 4
CAS:<p>Cav 3.2 Inhibitor 4 (Compound 21) is a selective and potent inhibitor of the T-type calcium channel (Ca v 3.2), demonstrating peripheral restriction with an</p>Fórmula:C21H32Cl2N4O3Pureza:98%Cor e Forma:SolidPeso molecular:459.41Budiodarone
CAS:Budiodarone (ATI-2042) resembles amiodarone, potentially preventing atrial fibrillation.Fórmula:C27H31I2NO5Cor e Forma:SolidPeso molecular:703.35Halofuginone hydrochloride
CAS:Halofuginone hydrochloride (RU-19110), a derivative of Febrifugine, functions as a competitive inhibitor of prolyl-tRNA synthetase, displaying a Ki value of 18.3 nM. This compound effectively inhibits type-I collagen synthesis, providing therapeutic benefits in osteoarthritis (OA) by impeding TGF-β signaling. Additionally, it serves as a potent pulmonary vasodilator, mainly through the activation of Kv channels and the inhibition of various calcium channels including voltage-gated, receptor-operated, and store-operated ones. Beyond its vascular effects, Halofuginone hydrochloride exhibits a broad spectrum of biological activities, including anti-malarial, anti-inflammatory, anti-cancer, and anti-fibrotic properties, supported by multiple studies.Fórmula:C16H18BrCl2N3O3Cor e Forma:SolidPeso molecular:451.14Darodipine
CAS:Darodipine (PY-108068) is a dihydropyridine type Ca+2 antagonist.Fórmula:C19H21N3O5Pureza:99.67%Cor e Forma:SolidPeso molecular:371.39A 425619
CAS:A 425619 (1-(4-(TRIFLUOROMETHYL)BENZYL)-3-(ISOQUINOLIN-5-YL)UREA) is a potent TRPV1 antagonistFórmula:C18H14F3N3OPureza:99.75%Cor e Forma:SolidPeso molecular:345.32Ref: TM-T8562
1mg60,00€5mg130,00€10mg203,00€25mg404,00€50mg567,00€100mg767,00€200mg1.074,00€1mL*10mM (DMSO)137,00€BBT
CAS:BBT has anti-hyperglycemic activity, protecting beta cells from cytokine or streptozotocin-induced cell death, and restoring beta cell function.Fórmula:C18H12BrNO2SPureza:99.02%Cor e Forma:SolidPeso molecular:386.26Iganidipine HCl
CAS:NKY-722 (HCl), also known as Iganidipine, is a calcium channel blocker potentially for the treatment of glaucoma.Fórmula:C28H40Cl2N4O6Cor e Forma:SolidPeso molecular:599.55Iganidipine
CAS:Iganidipine（NKY 722） is a new water-soluble Ca2+ antagonist with antihypertensive activity for research and neurological related diseases.Fórmula:C28H38N4O6Pureza:96.3%Cor e Forma:SolidPeso molecular:526.62Naltiazem
CAS:Naltiazem, a calcium channel antagonist, is used potentially for the treatment of arrhythmias, hypertension and myocardial infarction.Fórmula:C26H28N2O4SPureza:98%Cor e Forma:SolidPeso molecular:464.588-bromo NAD+ sodium
CAS:8-Bromo NAD+ serves as a prodrug for the cyclic ADP-ribose (cADPR) inhibitor, 8-bromo cADPR, undergoing conversion to its active form by the enzyme CD38.Fórmula:C21H25BrN7O14P2·NaCor e Forma:SolidPeso molecular:764.30Mioflazine hydrochloride anhydrous
CAS:Mioflazine hydrochloride anhydrous is a nucleoside transport inhibitor that acts on adenosine to improve sleep.Fórmula:C29H32Cl4F2N4O2Cor e Forma:SolidPeso molecular:648.4ATI-22-107
CAS:ATI-22-107 is a positive cardiac inotropic agent which may affect myocyte calcium cycling and contractility.Fórmula:C31H32Cl2N4O8Cor e Forma:SolidPeso molecular:659.51TROX-1
CAS:TROX-1 is the activation state-dependent Cav2 channel antagonist.Fórmula:C22H16ClFN6OPureza:98%Cor e Forma:SolidPeso molecular:434.85
