
Canais de Cálcio
Os canais de cálcio são proteínas de membrana que regulam o fluxo de íons de cálcio para dentro e fora das células, o que é essencial para várias funções celulares, incluindo a contração muscular, a liberação de neurotransmissores e a expressão gênica. A desregulação da atividade dos canais de cálcio está associada a condições como hipertensão, arritmias cardíacas e distúrbios neurológicos. Na CymitQuimica, oferecemos uma ampla seleção de moduladores de canais de cálcio para apoiar sua pesquisa em saúde cardiovascular, neurobiologia e transdução de sinais.
Foram encontrados 541 produtos de "Canais de Cálcio"
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AMG-1
CAS:AMG-1 inhibits CRAC channels, blocks effector T cells, not regulatory ones, and reduces EAE progression.Fórmula:C18H9ClF5N3OCor e Forma:SolidPeso molecular:413.73NPS-2143
CAS:NPS-2143 (SB 262470A) is a novel potent and selective antagonist of Ca(2+) receptor.Fórmula:C24H25ClN2O2Pureza:99.56%Cor e Forma:SolidPeso molecular:408.92RQ-00311651
CAS:RQ-00311651 is a novel T-type Ca2+ channel blocker. RQ-00311651 also inhibited high K-induced Ca signaling in those cells.Fórmula:C19H18F3N5O2Cor e Forma:SolidPeso molecular:405.37(R)-Lercanidipine hydrochloride
CAS:(R)-Lercanidipine hydrochloride is the R-enantiomer of Lercanidipine. (R)-lercanidipine hydrochloride is a blocker of calcium channel.Fórmula:C36H42ClN3O6Pureza:98%Cor e Forma:SolidPeso molecular:648.2β-Amino Acid Imagabalin Hydrochloride
CAS:β-Amino Acid Imagabalin Hydrochloride is the voltage-dependent calcium channel ligand for the α2δ subunit.Fórmula:C9H20ClNO2Pureza:98%Cor e Forma:SolidPeso molecular:209.71TMB 8 (hydrochloride)
CAS:TMB 8 blocks nAChRs (IC50: 390-480 nM), reduces Ca2+ in muscles, hinders rabbit aorta contraction at 50 μM, and inhibits PKC dose-dependently.Fórmula:C22H38ClNO5Cor e Forma:White SolidPeso molecular:431.99Sadopine
CAS:Sadopine is a high-affinity radioligand for DHP receptor in L-type Ca2+ channels, suitable for tissue and membrane labeling.Fórmula:C30H40F3N3O7SCor e Forma:SolidPeso molecular:643.71Lercanidipine. (R)-
CAS:(R)-Lercanidipine enantiomer: antihypertensive, blocks L-type Ca2+ channels, dilates blood vessels.Fórmula:C36H41N3O6Cor e Forma:SolidPeso molecular:611.73PD0176078
CAS:PD0176078 () is a newly blocker of N-type Calcium channel.Fórmula:C23H30F2N2OPureza:99.72%Cor e Forma:SolidPeso molecular:388.49Lidoflazine
CAS:Lidoflazine: antianginal, blocks HERG K+ & Ca channels, risks QT prolongation & arrhythmia.Fórmula:C30H35F2N3OPureza:98%Cor e Forma:SolidPeso molecular:491.62Semotiadil recemate fumarate
CAS:Semotiadil recemate fumarate is the recemate of Semotiadil fumarate. Semotiadil fumarate is a novel antagonist of vasoselective Ca2+ channel.Fórmula:C33H36N2O10SPureza:98%Cor e Forma:SolidPeso molecular:652.71TTA-P2
CAS:TTA-P2: potent CNS-penetrating T-type Ca2+ channel blocker; eliminates Cav3.1 window currents.Fórmula:C21H29Cl2FN2O2Cor e Forma:SolidPeso molecular:431.37Leconotide
CAS:Leconotide is a calcium channel blocker and antihyperalgesia agent; isolated from the venom of the cone snail, Conus catus.Fórmula:C107H179N35O36S7Cor e Forma:SolidPeso molecular:2756.23ML218
CAS:ML218 is an inhibitor of T-type Ca2+ channels (Cav3.1, Cav3.2, Cav3.3).ML218 inhibits the synaptic activity of subthalamic nucleus (STN) neurons.Fórmula:C19H26Cl2N2OPureza:99.2% - 99.45%Cor e Forma:SolidPeso molecular:369.33Carboxyamidotriazole
CAS:Carboxyamidotriazole is a cytostatic inhibitor of non-voltage-operated calcium channels and calcium channel-mediated signaling pathways.Fórmula:C17H12Cl3N5O2Pureza:98%Cor e Forma:SolidPeso molecular:424.67IDO1-IN-19
CAS:IDO1-IN-19 (Compound 17) is a potent inhibitor of IDO1 and has potential for cancer disease research.Fórmula:C25H22F4N2O3Cor e Forma:SolidPeso molecular:474.45CXL-1020
CAS:CXL-1020, a HNO prodrug, enhances heart muscle function & relaxation, aiding in heart failure research.Fórmula:C7H9NO5S2Cor e Forma:SolidPeso molecular:251.28Halofuginone hydrobromide
CAS:Halofuginone specifically inhibits collagen type I and MMP-2 gene expression, which may result in the suppression of angiogenesis and tumor cell growth.Fórmula:C16H17BrClN3O3·HBrPureza:97.01% - 99.73%Cor e Forma:SolidPeso molecular:495.5918:0 LYSO-PE
CAS:18:0 LYSO-PE is a compound that induces an increase in [Ca2+]i and can be used as a phospholipid (PL) standard for lipid analysis by electrospray mass spectrometry (ESI-MS)/MS.Fórmula:C23H48NO7PPureza:98%Cor e Forma:SolidPeso molecular:481.6
