
Canais de Cálcio
Os canais de cálcio são proteínas de membrana que regulam o fluxo de íons de cálcio para dentro e fora das células, o que é essencial para várias funções celulares, incluindo a contração muscular, a liberação de neurotransmissores e a expressão gênica. A desregulação da atividade dos canais de cálcio está associada a condições como hipertensão, arritmias cardíacas e distúrbios neurológicos. Na CymitQuimica, oferecemos uma ampla seleção de moduladores de canais de cálcio para apoiar sua pesquisa em saúde cardiovascular, neurobiologia e transdução de sinais.
Foram encontrados 541 produtos de "Canais de Cálcio"
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Opc 8490
CAS:Opc 8490 is a cardiotonic agent and a positive inotropic vasodilator, which prolongs the atrial action potential in a concentration-dependent manner.Fórmula:C30H35N3O10Pureza:98.88%Cor e Forma:SolidPeso molecular:597.618-Bromo-cGMP sodium
CAS:<p>8-Bromo-cGMP sodium: PKG activator, eases pain, dilates vessels, reduces Ca2+ currents & insulin release.</p>Fórmula:C10H10BrN5NaO7PPureza:99.45%Cor e Forma:SolidPeso molecular:446.09AZD-1305
CAS:<p>AZD-1305: novel anti-arrhythmic blocking IKr, Ca, Na currents; useful in arrhythmia research.</p>Fórmula:C22H31FN4O4Pureza:99.31% - 99.86%Cor e Forma:SolidPeso molecular:434.5Diproteverine HCl
CAS:<p>Diproteverine HCl is a novel calcium antagonist with antianginal properties, antispasmodic and vasoactive.</p>Fórmula:C26H36ClNO4Pureza:98.55% - 99.84%Cor e Forma:SolidPeso molecular:462.02Sulcardine sulfate
CAS:<p>Sulcardine sulfate (B-87823) is a multi-ion channel blocker with antiarrhythmic activity that inhibits Na+, K+, and Ca2+ channels.</p>Fórmula:C24H35N3O8S2Pureza:98.74%Cor e Forma:SolidPeso molecular:557.68O-1602
CAS:O-1602 is a novel GPR55 agonist, an atypical cannabinoid associated with the central nervous system and obesity, and is a candidate compound for the treatmentFórmula:C17H22O2Pureza:99.85%Cor e Forma:SolidPeso molecular:258.36Cronidipine
CAS:<p>Cronidipine (LF 20254), a calcium channel antagonist, is used potentially for the treatment of hypertension and myocardia ischemia.</p>Fórmula:C30H32ClN3O8Pureza:99.47%Cor e Forma:SolidPeso molecular:598.04Upacicalcet
CAS:Upacicalcet (AJT-240) is a calcium mimetic for SHPT in dialysis, reducing PTH by targeting parathyroid receptors.Fórmula:C11H14ClN3O6SPureza:99.88%Cor e Forma:SolidPeso molecular:351.76Tamolarizine
CAS:<p>Tamolarizine (Tamolarizine free base) free base is a novel calcium antagonist.</p>Fórmula:C27H32N2O3Pureza:98.17%Cor e Forma:SoildPeso molecular:432.55Clopimozide
CAS:Clopimozide (R-29764), a long-acting oral antischizophrenic, blocks calcium channels and [3H] nilandipine binding.Fórmula:C28H28ClF2N3OPureza:98.99% - 99.66%Cor e Forma:SolidPeso molecular:495.99SERCA2a activator 1
CAS:SERCA2a activator 1 boosts heart function by reducing phospholamban restraint and enhancing cardiac contraction-relaxation cycles.Fórmula:C32H29N3O4SPureza:99.75%Cor e Forma:SolidPeso molecular:551.66Vatanidipine
CAS:Vatanidipine (AE0047) is a novel dihydropyridine (DHP)-type calcium channel blocker with slow-onset pharmacological actions.A slow-onset and long-lastingFórmula:C41H42N4O6Pureza:99.95%Cor e Forma:SolidPeso molecular:686.8Gallopamil
CAS:Gallopamil blocks acid secretion (IC50: 10.9 μM), acts as antiarrhythmic, vasodilator, and is a methoxy Verapamil derivative.Fórmula:C28H40N2O5Pureza:99.85%Cor e Forma:SolidPeso molecular:484.63R 56865
CAS:R 56865 is a weak potential-operated channel inhibitor that inhibits the late sodium current in human isolated cardiomyocytes.Fórmula:C23H28FN3OSPureza:99.52%Cor e Forma:SolidPeso molecular:413.55NecroX-5
CAS:<p>NecroX-5, a derivative of NecroX, exhibits anti-inflammatory and anti-cancer activities. NecroX-5 reduces intracellular calcium concentration.</p>Fórmula:C27H39N3O9S3Pureza:99.944%Cor e Forma:SolidPeso molecular:645.81Iganidipine
CAS:Iganidipine(NKY 722) is a new water-soluble Ca2+ antagonist with antihypertensive activity for research and neurological related diseases.Fórmula:C28H38N4O6Pureza:96.3%Cor e Forma:SolidPeso molecular:526.62A 425619
CAS:A 425619 (1-(4-(TRIFLUOROMETHYL)BENZYL)-3-(ISOQUINOLIN-5-YL)UREA) is a potent TRPV1 antagonistFórmula:C18H14F3N3OPureza:99.75%Cor e Forma:SolidPeso molecular:345.32N-type calcium channel blocker-1
CAS:N-type calcium channel blocker-1 is an orally active analgesic agent,shows high affinity to functionally block N-type calcium channels.Fórmula:C31H47N3Pureza:98%Cor e Forma:SolidPeso molecular:461.73Piprofurol
CAS:Piprofurol is used as a Calcium channel blocker.Fórmula:C26H33NO6Pureza:98%Cor e Forma:SolidPeso molecular:455.54LOE 908 hydrochloride
CAS:Broad spectrum cation channel blockerFórmula:C41H49ClN2O9Pureza:98%Cor e Forma:SolidPeso molecular:749.29
