CymitQuimica logo
Canais de Cálcio

Canais de Cálcio

Os canais de cálcio são proteínas de membrana que regulam o fluxo de íons de cálcio para dentro e fora das células, o que é essencial para várias funções celulares, incluindo a contração muscular, a liberação de neurotransmissores e a expressão gênica. A desregulação da atividade dos canais de cálcio está associada a condições como hipertensão, arritmias cardíacas e distúrbios neurológicos. Na CymitQuimica, oferecemos uma ampla seleção de moduladores de canais de cálcio para apoiar sua pesquisa em saúde cardiovascular, neurobiologia e transdução de sinais.

Foram encontrados 541 produtos de "Canais de Cálcio"

Ordenar por

Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
produtos por página.
  • Penfluridol

    CAS:
    Penfluridol (TLP-607) is a highly potent antipsychotic.
    Fórmula:C28H27ClF5NO
    Pureza:98.9% - 99.87%
    Cor e Forma:Off-White To White Crystalline Powder
    Peso molecular:523.97
  • Praziquantel

    CAS:
    Praziquantel (Droncit) is an anthelmintic that paralyzes worms by increasing calcium in muscle cells, causing tegument damage and immune response.
    Fórmula:C19H24N2O2
    Pureza:99.67% - 99.69%
    Cor e Forma:Solid
    Peso molecular:312.41
  • Brompheniramine maleate

    CAS:
    Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.
    Fórmula:C16H19BrN2·C4H4O4
    Pureza:99.80%
    Cor e Forma:Crystal Powder
    Peso molecular:435.31
  • Ethacrynic acid D5

    CAS:
    Ethacrynic acid: a diuretic, anti-inflammatory, inhibits calcium channels, GSTs, NF-kB pathway, and modulates leukotriene; has deuterium-labeled form.
    Fórmula:C13H12Cl2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:308.17
  • sFTX-3.3

    CAS:
    sFTX-3.3 is a calcium ion channel antagonist, exhibiting IC50 values of approximately 0.24 mM and 0.70 mM against P-type and N-type channels respectively.
    Fórmula:C12H29N7O
    Cor e Forma:Solid
    Peso molecular:287.412
  • NSC156529

    CAS:
    NSC156529 suppresses AKT1, reduces cancer cell growth in vitro, and inhibits prostate tumors in vivo.
    Fórmula:C28H21ClS2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:457.05
  • Sulcardine 2HCl

    CAS:
    Sulcardine 2HCl is a multi-ion channel blocker that blocks the properties of hERG and hNav1.5 channels and can be used to study atrial fibrillation.
    Fórmula:C24H35Cl2N3O4S
    Pureza:99.33% - 99.76%
    Cor e Forma:Soild
    Peso molecular:532.523
  • Cyclic ADP-ribose ammonium


    cADPR ammonium is a second messenger that boosts cytosolic calcium via Ryanodine receptors and TRPM2 channels.
    Cor e Forma:Liquid
  • UK-59811 hydrochloride

    CAS:
    UK-59811 hydrochloride, Br-dihydropyridine derivative, blocks Ca V Ab channels in bacteria, IC50: 194 nM.
    Fórmula:C22H30BrClN2O5
    Cor e Forma:Solid
    Peso molecular:517.85
  • Calcium Ionophore I

    CAS:
    <p>Calcium Ionophore I has a wide range of applications in life science related research.</p>
    Fórmula:C38H72N2O8
    Cor e Forma:Solid
    Peso molecular:685.0
  • PACAP-38 (31-38), human, mouse, rat

    CAS:
    <p>PACAP-38 (31-38), human, mouse, rat demonstrates potent, efficacious, and sustained stimulatory effects on sympathetic neuronal NPY and catecholamine production</p>
    Fórmula:C47H83N17O11
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1062.27
  • MMK 1

    CAS:
    Potent hFPR2 agonist; EC50: 1 nM (mFPR2), 2 nM (hFPR2), >10,000 nM (hFPR1). Induces monocyte/neutrophil migration, boosts IL-1β/IL-6, activates NADPH-oxidase.
    Fórmula:C75H123N19O18S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1610.97
  • BTT-266

    CAS:
    <p>BTT-266 is a blocker of voltage-gated calcium channel for pain management.</p>
    Fórmula:C34H28N4O4
    Pureza:98.34%
    Cor e Forma:Solid
    Peso molecular:556.61
  • ILS-920

    CAS:
    ILS-920, a Rapamycin analog, has reduced immunosuppression, enhanced neuroprotection, and preferentially binds FKBP52 and L-type VGCC β1.
    Fórmula:C57H86N2O14
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1023.3
  • PDDHV

    CAS:
    PDDHV: a capsaicin-like vanilloid selective for rat TRPV1; induces Ca2+ uptake in neurons, EC50 of 70 nM.
    Fórmula:C49H72O11
    Cor e Forma:Solid
    Peso molecular:837.09
  • GTx1-15


    GTx1-15, an inhibitor cystine knot (ICK) peptide, antagonizes the voltage-dependent calcium channel Cav3.1, as well as voltage-dependent sodium channels Nav1.3
    Fórmula:C176H271N53O45S7
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:4073.82
  • SNX-482

    CAS:
    Potent CaV2.3 calcium channel blocker, selective, voltage-dependent, with 30 nM IC50. Offers antinociceptive effects on C and Aδ fibres.
    Fórmula:C192H274N52O60S7
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:4495.01
  • Levamlodipine besylate Hemipentahydrate

    CAS:
    <p>Levamlodipine besylate hemipentahydrate is the besylate hemipentahydrate salt form of Levamlodipine. It is an orally effective calcium channel blocker with antioxidative and vasodilatory properties. This compound can reduce serum malondialdehyde (MDA) levels, enhance the activity of superoxide dismutase (SOD), and alleviate oxidative stress. Levamlodipine besylate hemipentahydrate is relevant for research in vascular dementia, hypertension, and cerebrovascular diseases.</p>
    Fórmula:C20H25ClN2O5·C6H6O3SH2O
    Cor e Forma:Solid
    Peso molecular:1224.18
  • ProTx-I

    CAS:
    <p>Selective blocker for CaV3.1 (IC50 = 0.2 μM), CaV3.2 (31.8 μM), also inhibits NaV1.8 and blocks KV2.1 channels.</p>
    Fórmula:C171H245N53O47S6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:3987.51
  • ω-Agatoxin IVA

    CAS:
    Selective blocker of P-type calcium channels (IC50 < 1 - 3 nM). Also inhibits N-type channels at micromolar concentrations.
    Fórmula:C217H360N68O60S10
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:5202.25