Receptor GABA
Os receptores de GABA são os principais receptores de neurotransmissores inibitórios no sistema nervoso central, desempenhando um papel crítico na regulação da excitabilidade neuronal e na manutenção do equilíbrio entre excitação e inibição. A disfunção dos receptores de GABA está implicada em vários distúrbios neurológicos e psiquiátricos, incluindo epilepsia, ansiedade e depressão. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores de GABA para apoiar sua pesquisa em neurobiologia, saúde mental e desenvolvimento terapêutico.
Foram encontrados 372 produtos de "Receptor GABA"
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Primidone (Standard)
CAS:Primidone (Standard) is the standard substance of Primidone, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Primidone (NCI-C56360) is a potent anticonvulsant agent. It is a neuronal voltage-gated sodium channel blocker and has value in the study of epilepsy, essential tremor, and psychiatric disorders.Fórmula:C12H14N2O2Cor e Forma:Crystals (Ntp 1992)Peso molecular:218.25Vigabatrin Hydrochloride
CAS:Vigabatrin Hydrochloride (γ-Vinyl-GABA hydrochloride) is a structural analog of the GABA, irreversibly inhibiting the catabolism of GABA by GABA transaminase.Fórmula:C6H11NO2·HClPureza:98%Cor e Forma:SolidPeso molecular:165.62CGP 36742
CAS:CGP 36742 blocks GABAB receptor, crosses blood-brain barrier, aids depression treatment (IC50: 32 μM).Fórmula:C7H18NO2PCor e Forma:SolidPeso molecular:179.2MRK-016
CAS:MRK-016 is a selective GABAA α5 receptor inverse agonist/ negative allosteric modulator, orally available and penetrating the BBB. MRK-016 is antidepressant.Fórmula:C17H20N8O2Pureza:99.76%Cor e Forma:SolidPeso molecular:368.39L-655708
CAS:L-655708 is a selective and highly potent GABAA receptor reverse agonist with a Ki value of 0.45 nM.Fórmula:C18H19N3O4Pureza:99.36%Cor e Forma:PowderPeso molecular:341.36Furosemide-d5
CAS:Furosemide-d5 is a deuterium marker for Furosemide and used in isotope tracer experiments. orally active inhibitor of Na+/K+/2Cl- (NKCC) diuretic reagent.Fórmula:C12H11ClN2O5SCor e Forma:SolidPeso molecular:335.78(2S)-6-Prenylnaringenin
CAS:(2S)-6-Prenylnaringenin (6-Prenylnaringenin) is an isomer of the potent phytoestrogen, 8-prenylnaringenin.Fórmula:C20H20O5Pureza:99.47%Cor e Forma:SolidPeso molecular:340.37Acamprosate calcium
CAS:Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.Fórmula:C10H20CaN2O8S2Pureza:98% - 99.93%Cor e Forma:White Odorless Or Nearly Odorless PowderPeso molecular:400.48Acetoxyvalerensre
CAS:Acetoxyvalerensre (acetylvalerenolic acid) (acetylvalerenolic acid) is a derivative of valerenic acid, which is a a GABAA receptor modulator.Fórmula:C17H24O4Pureza:98.22%Cor e Forma:SolidPeso molecular:292.37Piperazine citrate
CAS:Piperazine citrate, an organic compound, consists of a six-membered ring, containing two nitrogen atoms at opposite positions in the ring.Fórmula:C24H46N6O14Pureza:99.8%Cor e Forma:Crystals IndicationPeso molecular:642.65AZD7325
CAS:AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.
Fórmula:C19H19FN4O2Pureza:99.83%Cor e Forma:SolidPeso molecular:354.38Ginkgolide A
CAS:Ginkgolide A (BN-52020), from Ginkgo biloba leaves, is an active PAF antagonist with potential in treating inflammation and immune disorders.Fórmula:C20H24O9Pureza:98.76% - 99.81%Cor e Forma:White PowderPeso molecular:408.40Guvacine hydrochloride
CAS:Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)Fórmula:C6H10ClNO2Pureza:98.42%Cor e Forma:SolidPeso molecular:163.602CL 218872
CAS:CL 218872: selective α1 GABAA receptor agonist, anxiolytic, and anticonvulsant; Ki=130 nM for α1, less potent for α2-α6.Fórmula:C13H9F3N4Pureza:99.92%Cor e Forma:SolidPeso molecular:278.23Pipequaline hydrochloride
CAS:Pipequaline hydrochloride (PK-8165 hydrochloride) is an anticonflict & anticonvulsant quinoline derivative.Fórmula:C22H25ClN2Pureza:99.46%Cor e Forma:SolidPeso molecular:352.9Arecaidine hydrochloride
CAS:Arecaidine hydrochloride may have carcinogenesis.Fórmula:C7H12ClNO2Pureza:99.69% - ≥95%Cor e Forma:SolidPeso molecular:177.63Ref: TM-T5799
2mg34,00€5mg48,00€10mg67,00€25mg100,00€50mg149,00€100mg213,00€200mg316,00€1mL*10mM (DMSO)49,00€(R)-baclofen
CAS:(R)-baclofen (STX209), a derivative of gamma-aminobutyric acid, is commonly utilized for the treatment of spasticity.Fórmula:C10H12ClNO2Pureza:97.20% - 98.94%Cor e Forma:SolidPeso molecular:213.66Ocinaplon
CAS:Ocinaplon (DOV 273547) is a GABAA receptors modulator.Fórmula:C17H11N5OPureza:99.81%Cor e Forma:SolidPeso molecular:301.3L-DABA
CAS:L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 > 500 μM).Fórmula:C4H10N2O2Pureza:99.32%Cor e Forma:SolidPeso molecular:118.13Kavain
CAS:Kavain, a compound extracted from the Kava plant, Piper methysticum, is found to be involved in TNF-α expression in human and mouse cells via regulation ofFórmula:C14H14O3Pureza:99.93% - ≥95%Cor e Forma:SolidPeso molecular:230.26Songorine
CAS:Songorine (Napellonine) shows anti-tumor activity in preliminary pharmacological verification trials including cell proliferation and molecular docking assays.Fórmula:C22H31NO3Pureza:98% - 99.92%Cor e Forma:SolidPeso molecular:357.49AZD-6280
CAS:AZD6280 is a novel, subtype-selective GABAAα2/3 receptor positive modulators, used for treatment of generalized anxiety disorder.Fórmula:C20H22N4O3Pureza:98.99%Cor e Forma:SolidPeso molecular:366.41Ref: TM-T7136
1mg215,00€5mg439,00€10mg640,00€25mg1.018,00€50mg1.423,00€100mg1.935,00€1mL*10mM (DMSO)484,00€Cholesterol myristate
CAS:Cholesterol myristate, a natural steroid in Chinese medicine, affects GABAA, nicotinic receptors, and potassium channels.
Fórmula:C41H72O2Pureza:99.65%Cor e Forma:SolidPeso molecular:597.01α-Thujone
CAS:α-Thujone is an inhibitor of ACh with an IC50 value of 24.7μM.Fórmula:C10H16OPureza:97.02% - 98.41%Cor e Forma:Less Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996) Colorless Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996)Peso molecular:152.23Temgicoluril
CAS:Temgicoluril (mebikar) acts on GABA Receptor.Fórmula:C8H14N4O2Pureza:99.8%Cor e Forma:SolidPeso molecular:198.226-Aminonicotinic acid
CAS:6-Aminonicotinic acid is a natural product.
Fórmula:C6H6N2O2Pureza:99.94%Cor e Forma:SoildPeso molecular:138.1238rac-BHFF
CAS:rac-BHFF, a GABA B receptor modulator, boosts GABA potency >15x, efficacy >149%, has anxiolytic effects, and is orally active.Fórmula:C17H21F3O3Pureza:99.69% - >99.99%Cor e Forma:SolidPeso molecular:330.34Ref: TM-T4176
2mg43,00€5mg60,00€10mg96,00€25mg187,00€50mg311,00€100mg472,00€200mg657,00€1mL*10mM (DMSO)71,00€α-Asarone
CAS:alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.Fórmula:C12H16O3Pureza:99.64% - 99.64%Cor e Forma:Monoclinic Needles From Water Monoclinic Needles From WaterPeso molecular:208.25Fipronil
CAS:Fipronil (Fluocyanobenpyrazole) is a broad-use insecticide that belongs to the phenylpyrazole chemical family.Fórmula:C12H4Cl2F6N4OSPureza:97.21%Cor e Forma:Solid PowderPeso molecular:437.15Thiocolchicoside
CAS:Thiocolchicoside, a muscle relaxant, has anti-inflammatory and analgesic properties; not for seizure-prone people.Fórmula:C27H33NO10SPureza:99.11% - 99.39%Cor e Forma:SolidPeso molecular:563.62γ-Acetylenic GABA
CAS:γ-Acetylenic GABA (4-Aminohex-5-ynoic acid) is a potent, irreversible inhibitor of GABA-transaminase.Fórmula:C6H9NO2Cor e Forma:SolidPeso molecular:127.143Tiagabine hydrochloride
CAS:Tiagabine hydrochloride, a nipecotic acid derivative, is an anticonvulsant and selective GABA reuptake inhibitor.Fórmula:C20H25NO2S2·HClPureza:99.09% - 99.77%Cor e Forma:White To Off-White SolidPeso molecular:412.01Gabazine free base
CAS:Gabazine free base is a specific antagonist of the GABA receptor. It does not affect GABA-transaminase or glutamate-decarboxylase activities.Fórmula:C15H17N3O3Cor e Forma:SolidPeso molecular:287.31Lorediplon
CAS:Lorediplon is a novel hypnotic drug acting as a GABAA receptor modulator, differentially active at the α1-subunit, associated with promoting sleep.Fórmula:C20H15FN4O2SPureza:99.12% - 99.19%Cor e Forma:SolidPeso molecular:394.42Loreclezole hydrochloride
CAS:Loreclezole hydrochloride is an antiepileptic, enhancing GABA A receptors with β2/β3 subunits.Fórmula:C10H7Cl4N3Cor e Forma:SolidPeso molecular:310.99Tiagabine hydrochloride hydrate
CAS:Tiagabine HCl hydrate, IC50: 67-446 nM, selectively inhibits GABA uptake, acts as an anticonvulsant.Fórmula:C20H28ClNO3S2Cor e Forma:SolidPeso molecular:430.022'MeO6MF
CAS:2'MeO6MF is a brain-penetrant positive allosteric modulator at α2β1γ2L and all α1-containing GABAA receptors.It offers neuroprotection and improved functionalFórmula:C17H14O3Pureza:99.28% - 99.63%Cor e Forma:SolidPeso molecular:266.29Ref: TM-T8887
1mg49,00€5mg102,00€10mg152,00€25mg243,00€50mg340,00€100mg460,00€200mg627,00€1mL*10mM (DMSO)96,00€Piperazine
CAS:Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.Fórmula:C4H10N2Cor e Forma:SolidPeso molecular:86.14Pikamilone
CAS:Pikamilone (Picamilon) is an intelligent medicine.Fórmula:C10H12N2O3Pureza:99.38%Cor e Forma:White Crystalline PowderPeso molecular:208.21(+)-Kavain
CAS:(+)-Kavain ((R)-KAWAIN) is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.Fórmula:C14H14O3Pureza:97% - ≥95%Cor e Forma:White Fine PowderPeso molecular:230.26(-)-Securinine
CAS:(-)-Securinine (Securinine) is plant-derived alkaloid and also a GABAA receptor antagonist.Fórmula:C13H15NO2Pureza:99.58% - 99.87%Cor e Forma:SolidPeso molecular:217.26Isonipecotic acid
CAS:Isonipecotic acid (4-Piperidinecarboxylic acid) is a heterocyclic compound. Isonipecotic acid mainly characterized as a GABAA receptor partial agonist.Fórmula:C6H11NO2Pureza:99.82%Cor e Forma:White To Faint Pink-Beige PowderPeso molecular:129.16SKF89976A hydrochloride
CAS:SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) andFórmula:C22H26ClNO2Pureza:98.02%Cor e Forma:SolidPeso molecular:371.9Ref: TM-T12930
1mg34,00€5mg65,00€10mg89,00€25mg167,00€50mg264,00€100mg409,00€200mg590,00€1mL*10mM (DMSO)71,00€Miltirone
CAS:Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.Fórmula:C19H22O2Pureza:99.22% - 99.66%Cor e Forma:SolidPeso molecular:282.38Phenibut (hydrochloride)
CAS:Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors.Fórmula:C10H14ClNO2Pureza:99.93%Cor e Forma:White Crystalline PowderPeso molecular:215.684-Acetamidobutanoic acid
CAS:4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.Fórmula:C6H11NO3Pureza:98.51%Cor e Forma:SolidPeso molecular:145.16CGP52432
CAS:CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).Fórmula:C15H24Cl2NO4PPureza:98.75%Cor e Forma:SolidPeso molecular:384.24(E)-3,4,5-Trimethoxycinnamic acid
CAS:(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium incisum.Fórmula:C12H14O5Pureza:99.83%Cor e Forma:SolidPeso molecular:238.24Imidazenil
CAS:Imidazenil is an modulator of GABA-A that blocks the sedative effects without lowering the convulsion threshold.Fórmula:C18H12BrFN4OPureza:98.4%Cor e Forma:SolidPeso molecular:399.22Isoflurane
CAS:Isoflurane (Forane) is a stable, non-explosive inhalation anesthetic that has been reported to induce caspase-3 activation.Fórmula:C3H2ClF5OPureza:98%Cor e Forma:Clear Colorless Liquid LiquidPeso molecular:184.49Cyclothiazide
CAS:Cyclothiazide enhances AMPA receptors, prevents desensitization, and boosts glutamic acid response (EC50 = 3.8µM).Fórmula:C14H16ClN3O4S2Pureza:98.23% - 99.49%Cor e Forma:Crystals From Dilute Alcohol SolidPeso molecular:389.88SSD114 HCl
CAS:SSD114 is a novel GABAB receptor positive allosteric modulator.Fórmula:C18H21ClF3N3OPureza:99.03% - 99.95%Cor e Forma:SolidPeso molecular:387.83Ref: TM-T4522
2mg34,00€5mg50,00€10mg75,00€25mg111,00€50mg172,00€100mg290,00€200mg419,00€1mL*10mM (DMSO)46,00€p-Hydroxybenzaldehyde
CAS:1.Fórmula:C7H6O2Pureza:99.05% - 99.86%Cor e Forma:SolidPeso molecular:122.12Aminooxyacetic acid hemihydrochloride
CAS:Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABAFórmula:C2H5NO3·5HClPureza:98.03%Cor e Forma:Light Beige Crystalline PowderPeso molecular:109.3Amentoflavone
CAS:Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.Fórmula:C30H18O10Pureza:98.21% - 99.22%Cor e Forma:Odourless Whitish SolidPeso molecular:538.46Ref: TM-T3417
2mg34,00€5mg50,00€10mg80,00€25mg126,00€50mg215,00€100mg349,00€200mg512,00€1mL*10mM (DMSO)59,00€Tiagabine
CAS:Tiagabine (NO050328) is an Anti-epileptic Agent.Fórmula:C20H25NO2S2Pureza:99.25% - 99.67%Cor e Forma:White To Off-White Crystalline SolidPeso molecular:375.55Gaboxadol hydrochloride
CAS:Gaboxadol (hydrochloride) is a GABAA receptor agonist.Fórmula:C6H9ClN2O2Pureza:99.39%Peso molecular:176.601SKF89976A HCl
CAS:SKF89976A: GABA uptake inhibitor, selective for GAT-1, passes blood-brain barrier, active in vivo (IC50: 0.13 μM hGAT-1).Fórmula:C22H25NO2Cor e Forma:SolidPeso molecular:335.44Gabazine
CAS:Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)Fórmula:C15H18BrN3O3Pureza:98.51% - 99.24%Cor e Forma:SolidPeso molecular:368.236-(4-Methoxyphenyl)-3-pyridazinamine
CAS:6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonistFórmula:C11H11N3OPureza:99.03%Cor e Forma:SolidPeso molecular:201.22L-838417 D9
CAS:L-838417 D9 (C-21191) is a novel deuterated subtype-selective GABAA positive allosteric modulator, acting as a partial agonist at α2, α3 and α5 subtypes[1].Fórmula:C19H10D9F2N7OPureza:99.65%Cor e Forma:SolidPeso molecular:408.45Ref: TM-T22301
2mg34,00€5mg52,00€10mg71,00€25mg128,00€50mg200,00€100mg323,00€200mg447,00€1mL*10mM (DMSO)58,00€2'-O-Methylisoliquiritigenin
CAS:2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-Fórmula:C16H14O4Pureza:98.75%Cor e Forma:SolidPeso molecular:270.28Baclofen hydrochloride
CAS:Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.Fórmula:C10H13Cl2NO2Pureza:99.55%Cor e Forma:SolidPeso molecular:250.1226-Methylflavone
CAS:6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.Fórmula:C16H12O2Pureza:99.69%Cor e Forma:SolidPeso molecular:236.27Neurotensin TFA
Neurotensin TFA (39379-15-2) is a 13-amino acid neuropeptide with opioid-independent pain relief, acting in the CNS and gut, linked to numerous disorders.Fórmula:C80H122F3N21O22Pureza:99.41%Cor e Forma:SolidPeso molecular:1786.98DL-Menthol
CAS:DL-Menthol ((±)-Menthol) is a racemic mixture of the monoterpene alcohols (–)-menthol and (+)-menthod, which have been found in Cannabis.Fórmula:C10H20OPureza:99.74%Cor e Forma:White Crystals /89-78-1/ Physical Description White Crystalline Solid With A Peppermint Odor And Taste (Ntp 1992)Peso molecular:156.27Saclofen
CAS:Saclofen is a GABA analog and GABAB receptor antagonist, useful for studying inhibitory brain signals. IC50: 7.8 μM.Fórmula:C9H12ClNO3SPureza:99.17%Cor e Forma:White Crystalline SolidPeso molecular:249.71Ref: TM-T4440
1mg52,00€5mg113,00€10mg177,00€25mg340,00€50mg550,00€100mg860,00€200mg1.161,00€1mL*10mM (DMSO)108,00€Imepitoin
CAS:Imepitoin (AWD 131-138), a new low-affinity partial benzodiazepine receptor agonist, shows potent anticonvulsant and anxiolytic properties in rodent models.Fórmula:C13H14ClN3O2Pureza:99.82%Cor e Forma:SolidPeso molecular:279.72U93631
CAS:GABAA antagonist; binds picrotoxin site, stabilizes inactive channel. Speeds GABA-induced Cl- decay, minor peak effect. Inhibits 5-HT3A receptors.Fórmula:C17H21N3O2Pureza:99.65% - 99.76%Cor e Forma:SolidPeso molecular:299.37Fluralaner
CAS:Fluralaner (A1443) is an isoxazoline ectoparasiticide.Fórmula:C22H17Cl2F6N3O3Pureza:99.72% - 99.99%Cor e Forma:Solid PowderPeso molecular:556.29Ginsenoside Rc
CAS:Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.
Fórmula:C53H90O22Pureza:98.83% - 99.56%Cor e Forma:White PowderPeso molecular:1079.27NS11394
CAS:NS11394 is a effective and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of α(5) > α(3) > α(2) > α(Fórmula:C23H19N3OPureza:99.44% - 99.86%Cor e Forma:SolidPeso molecular:353.42Ref: TM-T2067
2mg34,00€5mg50,00€10mg80,00€25mg131,00€50mg212,00€100mg321,00€200mg460,00€1mL*10mM (DMSO)58,00€ONO-8590580
CAS:ONO-8590580 (CS-2894) is a negative allosteric modulator of GABAA α5.Fórmula:C21H21FN6Pureza:99.43%Cor e Forma:SolidPeso molecular:376.43Ref: TM-TQ0040
1mg57,00€5mg119,00€10mg166,00€25mg356,00€50mg532,00€100mg760,00€1mL*10mM (DMSO)133,00€Jujuboside A
CAS:Jujuboside A: glycoside from Semen Ziziphi Spinosae, may treat Alzheimer's, has neuro-inhibitory effects.Fórmula:C58H94O26Pureza:98% - >99.99%Cor e Forma:SolidPeso molecular:1207.35Suritozole
CAS:Suritozole (MDL-26479) is a negative modulator at the gamma-aminobutyric acidA (GABAA) receptorFórmula:C10H10FN3SPureza:99.25%Cor e Forma:SolidPeso molecular:223.27Ref: TM-T8568
1mg58,00€5mg116,00€10mg172,00€25mg281,00€50mg396,00€100mg537,00€200mg712,00€1mL*10mM (DMSO)104,00€Basmisanil
CAS:Basmisanil (RG1662) is a negative allosteric modulator/inverse agonist of GABAAα5 receptors.Formulations containing basmisanil are in clinical trials for theFórmula:C21H20FN3O5SPureza:99.21% - 99.42%Cor e Forma:SolidPeso molecular:445.46Ref: TM-T7165
2mg35,00€5mg52,00€10mg74,00€25mg116,00€50mg187,00€100mg356,00€500mg802,00€1mL*10mM (DMSO)49,00€Dihydroergotoxine mesylate
CAS:Dihydroergotoxine mesylate (Ergoloid mesylates) is mainly used to improve symptoms and physical symptoms of mental degeneration related to aging.Fórmula:C20H29N3O5SPureza:99.39% - ≥95%Cor e Forma:SolidPeso molecular:423.53Bicuculline
CAS:Bicuculline, a plant-derived GABAA receptor antagonist, identified in 1932, reacts to light.Fórmula:C20H17NO6Pureza:98% - 99.99%Cor e Forma:Light Yellow PowderPeso molecular:367.35Loreclezole
CAS:Loreclezole is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit-containing receptors.Fórmula:C10H6Cl3N3Pureza:99.78%Cor e Forma:SolidPeso molecular:274.53Afloqualone
CAS:Afloqualone (HQ-495) is a GABA Receptor agonist with sedative and muscle-relaxant properties.Fórmula:C16H14FN3OPureza:99.72%Cor e Forma:SolidPeso molecular:283.3Riluzole
CAS:Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.Fórmula:C8H5F3N2OSPureza:99.71% - 99.88%Cor e Forma:PowderPeso molecular:234.2Darigabat
CAS:Darigabat (PF-06372865) is a GABAA receptor modulator with anxiolytic activity that inhibits α2, α1 PAM, and α2 PAM.Fórmula:C22H21FN4O3SPureza:98.42% - 99.29%Cor e Forma:SolidPeso molecular:440.49PNU-107484A
CAS:PNU-107484A is a unique GABA(A) receptor ligand.Fórmula:C18H23ClN6Pureza:98%Cor e Forma:SolidPeso molecular:358.87ABP-700
CAS:ABP-700 is a positive allosteric modulator of the GABAA receptor.Fórmula:C17H18N2O4Pureza:98%Cor e Forma:SolidPeso molecular:314.34DAA-1097
CAS:DAA-1097 is a novel ligand of peripheral benzodiazepine receptor.Fórmula:C24H24ClNO3Pureza:98%Cor e Forma:SolidPeso molecular:409.91(S)-3-Carboxy-4-hydroxyphenylglycine
CAS:group I metabotropic glutamate receptor antagonist and group II mGlu agonistFórmula:C9H9NO5Pureza:98%Cor e Forma:SolidPeso molecular:211.17BGT1-IN-9
CAS:BGT1-IN-9 is an M1 muscarinic agonist.Fórmula:C5H10ClN3O2Cor e Forma:SolidPeso molecular:179.605GABAA receptor agent 5
CAS:Compound 018 is a potent γ-GABAAR antagonist, Ki of 0.020 μM, with low membrane permeability.Fórmula:C21H25N3O2SPureza:99.39%Cor e Forma:SolidPeso molecular:383.51CGP 46381
CAS:CGP 46381 is a GABAB receptor antagonist.Fórmula:C10H22NO2PPureza:98%Cor e Forma:White SolidPeso molecular:219.26RO 4938581
CAS:RO 4938581: potent GABAA α5 inverse agonist (Ki 4.6 nM); lower affinity for α1β3γ2a, α2β3γ2a, α3β3γ2a (Ki: 174, 185, 80 nM).Fórmula:C13H8BrF2N5Pureza:98%Cor e Forma:SolidPeso molecular:352.14GS 39783
CAS:GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties of alcohol and the conditioned reinforcement andFórmula:C15H23N5O2SPureza:99.92%Cor e Forma:SolidPeso molecular:337.44PF-0713
CAS:PF 0713, a GABAA receptor agonist, is used as an intravenous sedative-hypnotic for general anaesthesia, ICU sedation, procedural sedation, chemotherapy.Fórmula:C14H22OPureza:98%Cor e Forma:SolidPeso molecular:206.32Ro 41-3290
CAS:Ro 41-3290 is the desethylated derivative of Ro 41-3696, which is an agonist of nonbenzodiazepine partial at the benzodiazepine receptor.Fórmula:C24H21ClN2O3Pureza:98%Cor e Forma:SolidPeso molecular:420.89SCH 50911
CAS:SCH 50911 is a selective GABA(B) receptor antagonist with IC50: 1.1 μM, boosting 3H overflow at IC50: 3 μM.Fórmula:C8H15NO3Pureza:98%Cor e Forma:SolidPeso molecular:173.21Anxiolytic/nonsedative agent-1
CAS:TCS 1205: Selective GABAA agonist, BzR affinity in bovine brain (Kis: 14-239 nM), α2 efficacy in vitro, anxioselective in vivo.Fórmula:C18H15N3O4Pureza:98.61%Cor e Forma:SolidPeso molecular:337.33Ref: TM-T23445
1mg64,00€2mg96,00€5mg115,00€10mg150,00€25mg330,00€50mg472,00€100mg655,00€500mg1.293,00€CP-409092 hydrochloride
CAS:CP-409092 hydrochloride is a partial agonist of the GABAA receptor with anti-anxiety activity.Fórmula:C17H20ClN3O2Cor e Forma:SolidPeso molecular:333.81Ciclotizolam
CAS:Ciclotizolam, a thienotriazolodiazepine derivative and partial GABAA receptor agonist, has low efficacy but similar affinity as brotizolam.Fórmula:C20H18BrClN4SCor e Forma:SolidPeso molecular:461.81Arbaclofen placarbil
CAS:Arbaclofen placarbil is a GABA(B) receptor agonist with better ADMET than R-baclofen, reducing postprandial reflux in GERD.Fórmula:C19H26ClNO6Cor e Forma:SolidPeso molecular:399.87SH-053-S-CH3-2'F
CAS:SH-053-S-CH3-2'F is a potent and selective agonist of GABAA receptors.Fórmula:C23H18FN3O2Cor e Forma:SolidPeso molecular:387.41
