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Receptor GABA

Receptor GABA

Os receptores de GABA são os principais receptores de neurotransmissores inibitórios no sistema nervoso central, desempenhando um papel crítico na regulação da excitabilidade neuronal e na manutenção do equilíbrio entre excitação e inibição. A disfunção dos receptores de GABA está implicada em vários distúrbios neurológicos e psiquiátricos, incluindo epilepsia, ansiedade e depressão. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores de GABA para apoiar sua pesquisa em neurobiologia, saúde mental e desenvolvimento terapêutico.

Foram encontrados 336 produtos de "Receptor GABA"

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  • CP-409092 hydrochloride

    CAS:
    <p>CP-409092 hydrochloride is a partial agonist of the GABAA receptor with anti-anxiety activity.</p>
    Fórmula:C17H20ClN3O2
    Cor e Forma:Solid
    Peso molecular:333.81
  • CGP 46381

    CAS:
    <p>CGP 46381 is a GABAB receptor antagonist.</p>
    Fórmula:C10H22NO2P
    Pureza:98%
    Cor e Forma:White Solid
    Peso molecular:219.26
  • GABAA receptor agent 5

    CAS:
    <p>Compound 018 is a potent γ-GABAAR antagonist, Ki of 0.020 μM, with low membrane permeability.</p>
    Fórmula:C21H25N3O2S
    Cor e Forma:Solid
    Peso molecular:383.51
  • BGT1-IN-9

    CAS:
    <p>BGT1-IN-9 is an M1 muscarinic agonist.</p>
    Fórmula:C5H10ClN3O2
    Cor e Forma:Solid
    Peso molecular:179.605
  • CCD-3693

    CAS:
    <p>CCD-3693 is a gamma-aminobutyric acid (GABA) receptor agonist.</p>
    Fórmula:C21H31F3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:372.46
  • GABA-AT-IN-1

    CAS:
    <p>GABA-AT-IN-1 (Compound 6) is an inhibitor of γ-aminobutyric acid transaminase (GABA-AT) that crosses the blood-brain barrier.</p>
    Fórmula:C23H18N2O6
    Cor e Forma:Solid
    Peso molecular:418.4
  • GABAA receptor agent 8

    CAS:
    <p>Compound 5e, a GABAA receptor modulator, shows potent anticonvulsant effects with low neurotoxicity for epilepsy research.</p>
    Fórmula:C19H16N4O
    Cor e Forma:Solid
    Peso molecular:316.36
  • ZAPA sulfate

    CAS:
    <p>GABAA receptors agonist</p>
    Fórmula:C4H8N2O6S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:244.25
  • TPMPA

    CAS:
    <p>GABAA-ρ antagonist</p>
    Fórmula:C6H12NO2P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:161.14
  • TG41

    CAS:
    <p>TG41 is a GABAA receptors positive modulator.</p>
    Fórmula:C18H13BrCl2N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:440.12
  • FG8119

    CAS:
    <p>FG8119 is a novel benzodiazepine agonist with potential anticonvulsant and antiepileptic activity for the study of neurological disorders.</p>
    Fórmula:C17H15N5O2
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:321.33
  • GABAA receptor agent 6

    CAS:
    <p>GABAA receptor agent 6 (compound 2027) is a potent γ-GABAAR antagonist with low cellular membrane permeability (Ki = 0.56 μM) [1].</p>
    Fórmula:C18H25N3O2
    Cor e Forma:Solid
    Peso molecular:315.41
  • TB 21007

    CAS:
    <p>GABAA receptor inverse agonist</p>
    Fórmula:C15H17NO2S3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:339.5
  • SL-651498

    CAS:
    <p>SL-651498, a GABAA receptor agonist, is used potentially for the treatment of anxiety.</p>
    Fórmula:C23H20FN3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:389.42
  • Bamaluzole

    CAS:
    <p>Bamaluzole is an agonist of GABA receptor.</p>
    Fórmula:C14H12ClN3O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:273.72
  • NAP-1

    CAS:
    <p>NAP-1 is an anesthetic that enhances CA1 brain inhibition in rats and causes tadpole sedation (EC50 = 0.53 μM).</p>
    Fórmula:C20H18ClNO2
    Cor e Forma:Solid
    Peso molecular:339.82
  • GABAA receptor agent 7

    CAS:
    <p>Compound 5c, a GABAA receptor modulator with anticonvulsant properties and low neurotoxicity, is promising for epilepsy research.</p>
    Fórmula:C18H13ClN4O
    Cor e Forma:Solid
    Peso molecular:336.77
  • MRK-623

    CAS:
    <p>MRK-623 (14k) is an oral GABA A agonist with high affinity for α1/α2/α3/α5 subunits and anxiolytic properties.</p>
    Fórmula:C20H17FN4O
    Cor e Forma:Solid
    Peso molecular:348.37
  • Etbicyphat

    CAS:
    <p>Etbicyphat: potent GABA(A) antagonist, induces epileptiform activity, binds to GABA/benzodiazepine receptors.</p>
    Fórmula:C6H11O4P
    Cor e Forma:Solid
    Peso molecular:178.12
  • TCS 1105

    CAS:
    <p>TCS 1105 is a GABAA BZR ligand, blocking Sema3A and altering mouse anxiety, aggression, and social dominance.</p>
    Fórmula:C17H13FN2O2
    Pureza:99.75%
    Cor e Forma:Solid
    Peso molecular:296.3
  • Pipazethate

    CAS:
    <p>Pipipyrazine is a nonnarcotic oral cough suppressant, cough suppressant.</p>
    Fórmula:C21H25N3O3S
    Cor e Forma:Solid
    Peso molecular:399.51
  • NNC052090

    CAS:
    <p>NNC052090 inhibits GABA uptake, favoring hBGT-1 (Ki=1.4μM), affects α1/D2 receptors (IC50=266/1632nM).</p>
    Fórmula:C27H30N2O2
    Cor e Forma:Solid
    Peso molecular:414.54
  • RU 33965

    CAS:
    <p>RU 33965, a 3-cyclopropyl carbonyl imidazobenzodiazepine, act as a low-efficacy benzodiazepine receptor inverse agonist.</p>
    Fórmula:C16H15N3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:281.31
  • ZK93423

    CAS:
    <p>ZK93423: potent benzodiazepine agonist, IC50=1nM, non-selective, Ki=4.1-6nM for α1-α5 GABAA subunits.</p>
    Fórmula:C23H22N2O4
    Cor e Forma:Solid
    Peso molecular:390.43
  • GABAA receptor modulator-2

    CAS:
    <p>Compound 20: Selective, oral α5-GABAAR inhibitor, Ki: 4.1 nM. High stability, CNS safe.</p>
    Fórmula:C22H22FN3O5S
    Cor e Forma:Solid
    Peso molecular:459.49
  • Carburazepam

    CAS:
    <p>Carburazepam is a derivate of benzodiazepines. Benzodiazepines are a class of psychoactive drugs.</p>
    Fórmula:C17H16ClN3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:329.78
  • UMB68 sodium

    CAS:
    <p>UMB-68 is a GHB receptor ligand with no affinity (IC(50) &gt;100 microM) at GABA(A) or GABA(B) receptors.</p>
    Fórmula:C6H12NaO3
    Cor e Forma:Solid
    Peso molecular:155.149
  • (+)-Nipecotic acid

    CAS:
    <p>(+)-Nipecotic acid ((+)-β-Homoproline) is a specific inhibitor of GABA transport and uptake, capable of activating GABAA receptors.</p>
    Fórmula:C6H11NO2
    Pureza:99.38%
    Cor e Forma:Solid
    Peso molecular:129.16
  • (S)-SNAP5114

    CAS:
    <p>(S)-SNAP5114 is a selective inhibitor of GABA transport with IC50s of 5 μM for hGAT-3 and 21 μM for rGAT-2. (S)-SNAP5114 has anticonvulsant properties.</p>
    Fórmula:C30H35NO6
    Pureza:97%
    Cor e Forma:Solid
    Peso molecular:505.6
  • Radequinil

    CAS:
    <p>Radequinil is a benzodiazepine receptor partial inverse agonist. Rade quinil binds to GABA(-) and GABA(+) ligand (Kis: 5.15 and 6.11 nM, respectively).</p>
    Fórmula:C18H14N4O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:334.33
  • 3α,21-Dihydroxy-5α-pregnan-20-one

    CAS:
    <p>3α,21-Dihydroxy-5α-pregnan-20-one (5alpha-THDOC) is a GABAA modulator that can be used in the study of Alzheimer's-like neurological diseases.</p>
    Fórmula:C21H34O3
    Pureza:98.00%
    Cor e Forma:Solid
    Peso molecular:334.49
  • Chlormethiazole edisylate

    CAS:
    <p>Chlormethiazole edisylate is a positive allosteric modulator of the GABAA receptor. Chlormethiazole edisylate is a sedative and hypnotic.</p>
    Fórmula:C8H14ClNO6S3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:351.85
  • COR628

    CAS:
    <p>COR628 is the GABA(B) receptor positive allosteric modulator.</p>
    Fórmula:C16H23NO3S
    Cor e Forma:Solid
    Peso molecular:309.42
  • trans-4-Hydroxycrotonic acid

    CAS:
    <p>ligand of γ-hydroxybutyric acid (GHB) receptor</p>
    Fórmula:C4H6O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:102.09
  • LY 81067

    CAS:
    <p>LY 81067, a new anticonvulsant, prevents PTZ- and picrotoxin-induced seizures in mice via picrotoxin site interaction.</p>
    Fórmula:C22H24N4O
    Cor e Forma:Solid
    Peso molecular:360.45
  • U 90042

    CAS:
    <p>GABAA receptor ligand</p>
    Fórmula:C17H13ClN6O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:352.78
  • COR627

    CAS:
    <p>COR627 is the GABA receptor positive allosteric modulator.</p>
    Fórmula:C20H27NO3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:361.5
  • CPP-115

    CAS:
    <p>CPP-115 is a GABA-aminotransferase inhibitor and a high-affinity vigabatrin analogue.</p>
    Fórmula:C7H9F2NO2
    Cor e Forma:Solid
    Peso molecular:177.15
  • JY-XHe-053

    CAS:
    <p>JY-XHe-053 is a selective modulator of GABAA receptors.</p>
    Fórmula:C22H16FN3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:373.38
  • HIE-124

    CAS:
    <p>HIE-124 is a central cervous system active anticonvulsant and ultra-short acting hypnotic.</p>
    Fórmula:C10H12N2O3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:240.28
  • Suclofenide

    CAS:
    <p>Suclofenide: a benzenesulfonamide anticonvulsant, effective in mouse seizure models, with side effects like lethargy and diarrhea.</p>
    Fórmula:C16H13ClN2O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:364.8
  • (S)-Baclofen

    CAS:
    <p>(S)-Baclofen may treat hyperacusis and tinnitus by reducing auditory pathway excitation.</p>
    Fórmula:C10H12ClNO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:213.66
  • ABP-700

    CAS:
    <p>ABP-700 is a positive allosteric modulator of the GABAA receptor.</p>
    Fórmula:C17H18N2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:314.34
  • DAA-1097

    CAS:
    <p>DAA-1097 is a novel ligand of peripheral benzodiazepine receptor.</p>
    Fórmula:C24H24ClNO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:409.91
  • (S)-3-Carboxy-4-hydroxyphenylglycine

    CAS:
    <p>group I metabotropic glutamate receptor antagonist and group II mGlu agonist</p>
    Fórmula:C9H9NO5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:211.17
  • PNU-107484A

    CAS:
    <p>PNU-107484A is a unique GABA(A) receptor ligand.</p>
    Fórmula:C18H23ClN6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:358.87
  • GS 39783

    CAS:
    <p>GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties of alcohol and the conditioned reinforcement and</p>
    Fórmula:C15H23N5O2S
    Pureza:99.92%
    Cor e Forma:Solid
    Peso molecular:337.44
  • SCH 50911

    CAS:
    <p>SCH 50911 is a selective GABA(B) receptor antagonist with IC50: 1.1 μM, boosting 3H overflow at IC50: 3 μM.</p>
    Fórmula:C8H15NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:173.21
  • Anxiolytic/nonsedative agent-1

    CAS:
    <p>TCS 1205: Selective GABAA agonist, BzR affinity in bovine brain (Kis: 14-239 nM), α2 efficacy in vitro, anxioselective in vivo.</p>
    Fórmula:C18H15N3O4
    Pureza:98.61%
    Cor e Forma:Solid
    Peso molecular:337.33
  • SCH 50911 hydrochloride

    CAS:
    <p>SCH 50911 hydrochloride is a selective, orally-active and competitive antagonist of γ-Aminobutyric acid B GABA(B) receptor(IC50 : 1.1 μM).</p>
    Fórmula:C8H16ClNO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:209.67
  • Bifenazate

    CAS:
    <p>Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.</p>
    Fórmula:C17H20N2O3
    Pureza:99.62%
    Cor e Forma:Solid Crystalline
    Peso molecular:300.35
  • E2730

    CAS:
    <p>E2730 is a non-competitive GABA transporter 1 (GAT1) inhibitor with anti-epileptic activity, useful in studying neurological disorders.</p>
    Fórmula:C9H8F4N2O2S
    Pureza:98.22% - 98.54%
    Cor e Forma:Solid
    Peso molecular:284.23
  • U-89843A

    CAS:
    <p>U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents [1].</p>
    Fórmula:C16H24ClN5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:321.85
  • (R)-Baclofen hydrochloride

    CAS:
    <p>Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.</p>
    Fórmula:C10H13Cl2NO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:250.12
  • Lesogaberan

    CAS:
    <p>Lesogaberan: selective GABAB agonist, EC50 8.6 nM, Ki 5.1 nM in rats, weak GABAA affinity (Ki 1.4 μM).</p>
    Fórmula:C3H9FNO2P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:141.08
  • Tracazolate hydrochloride

    CAS:
    <p>Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.</p>
    Fórmula:C16H25ClN4O2
    Pureza:99.52%
    Cor e Forma:Solid
    Peso molecular:340.85
  • RO 4938581

    CAS:
    <p>RO 4938581: potent GABAA α5 inverse agonist (Ki 4.6 nM); lower affinity for α1β3γ2a, α2β3γ2a, α3β3γ2a (Ki: 174, 185, 80 nM).</p>
    Fórmula:C13H8BrF2N5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:352.14
  • AZD 3043

    CAS:
    <p>AZD 3043 (THRX 918661) is a modulator of the gamma-aminobutyric acid type A receptor, a novel sedative-hypnotic, and a potential short-acting anesthetic.</p>
    Fórmula:C19H29NO5
    Pureza:98.19% - 99.55%
    Cor e Forma:Solid
    Peso molecular:351.44
  • Phaclofen

    CAS:
    <p>GABAB antagonist</p>
    Fórmula:C9H13ClNO3P
    Pureza:99.32%
    Cor e Forma:White Solid
    Peso molecular:249.63
  • Panadiplon

    CAS:
    <p>Panadiplon (FG 10571) is a selective gamma-aminobutyric acid receptor agonist and partial agonist of 5GABAA, a benzodiazepine receptor, used in the treatment of</p>
    Fórmula:C18H17N5O2
    Pureza:98.30% - 98.94%
    Cor e Forma:Solid
    Peso molecular:335.36
  • Cirsimaritin

    CAS:
    <p>Cirsimaritin has anti-bacterial, anti-inflammatory, anti-tumor, antioxidant effects, and protects kidneys; it weakly targets GABAA receptors.</p>
    Fórmula:C17H14O6
    Pureza:99.9%
    Cor e Forma:Solid
    Peso molecular:314.29
  • Progabide

    CAS:
    <p>Progabide (SL 76002) is an agonist of the gamma-aminobutyric acid receptor.</p>
    Fórmula:C17H16ClFN2O2
    Pureza:99.68%
    Cor e Forma:Solid
    Peso molecular:334.77
  • Saripidem

    CAS:
    <p>Saripidem (SL-85.0274) is a compound with anxiolytic activity.</p>
    Fórmula:C19H20ClN3O
    Pureza:99.45%
    Cor e Forma:Solid
    Peso molecular:341.83
  • NS-2710

    CAS:
    <p>NS-2710, a GABA receptor agonist, is used potentially for the treatment of anxiety.</p>
    Fórmula:C22H20N4O
    Pureza:99.7% - 99.82%
    Cor e Forma:Solid
    Peso molecular:356.42
  • ELB-139

    CAS:
    <p>ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal cortex of rats.</p>
    Fórmula:C14H16ClN3O
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:277.75
  • Ru-32514

    CAS:
    <p>Ru-32514 is a benzodiazepine receptor agonist.</p>
    Fórmula:C18H17N3O2
    Pureza:99.21%
    Cor e Forma:Solid
    Peso molecular:307.35
  • Fengabine

    CAS:
    <p>Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat depression.</p>
    Fórmula:C17H17Cl2NO
    Pureza:99%
    Cor e Forma:Solid
    Peso molecular:322.23
  • Nerisopam

    CAS:
    <p>Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.</p>
    Fórmula:C18H19N3O2
    Pureza:97.07%
    Cor e Forma:Solid
    Peso molecular:309.36
  • DMCM hydrochloride

    CAS:
    <p>DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.</p>
    Fórmula:C17H19ClN2O4
    Pureza:99.56%
    Cor e Forma:Solid
    Peso molecular:350.8
  • Suriclone

    CAS:
    <p>Suriclone (RP 31264), a cyclic pyrrolidone for anxiety, modulates GABA-A receptors without major sedation.</p>
    Fórmula:C20H20ClN5O3S2
    Pureza:99.21% - 99.73%
    Cor e Forma:Solid
    Peso molecular:477.99
  • NNC 05-711

    CAS:
    <p>NNC 05-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1), exerting anticonvulsant and analgesic effects.</p>
    Fórmula:C21H23ClN2O3
    Pureza:99.92%
    Cor e Forma:Solid
    Peso molecular:386.87
  • Riluzole hydrochloride

    CAS:
    <p>Riluzole hydrochloride, an anticonvulsant Na+ channel blocker, inhibits GABA uptake (IC50: 43 µM).</p>
    Fórmula:C8H6ClF3N2OS
    Pureza:99.76%
    Cor e Forma:Solid
    Peso molecular:270.66
  • BPDBA

    CAS:
    <p>BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 and</p>
    Fórmula:C19H20Cl2N2O
    Pureza:99.37% - 99.95%
    Cor e Forma:Solid
    Peso molecular:363.28
  • RWJ-51204

    CAS:
    <p>RWJ-51204: potent adenosine A2A blocker, GABA(A) partial agonist (IC50: 0.2-2 nM), neuroprotective, may treat Parkinson's.</p>
    Fórmula:C21H19F2N3O3
    Pureza:99.57% - 99.95%
    Cor e Forma:Solid
    Peso molecular:399.39
  • Lirequinil

    CAS:
    <p>Lirequinil (Ro 41-3696) is a small molecule GABAA receptor agonist used to study neurological disorders.</p>
    Fórmula:C26H25ClN2O3
    Pureza:98.54%
    Cor e Forma:Solid
    Peso molecular:448.94
  • L-838417

    CAS:
    <p>L-838417 is a GABAA receptor subtype-selective benzodiazepine site-selective ligand and GABAA receptor-positive modulator used in the study of anxiety disorders</p>
    Fórmula:C19H19F2N7O
    Pureza:98.12% - 99.70%
    Cor e Forma:Solid
    Peso molecular:399.4
  • Divaplon

    CAS:
    <p>Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety.</p>
    Fórmula:C17H17N3O2
    Pureza:97.44% - 98.25%
    Cor e Forma:Solid
    Peso molecular:295.34
  • Alpidem

    CAS:
    <p>Alpidem (Ananxyl), a non-sedative imidazopyridine anxiolytic, treats anxiety with high benzodiazepine receptor affinity.</p>
    Fórmula:C21H23Cl2N3O
    Pureza:99.56% - 99.97%
    Cor e Forma:White To Off-White Solid
    Peso molecular:404.33
  • Sarmazenil

    CAS:
    <p>Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used in the study of chronic hepatic encephalopathy.</p>
    Fórmula:C15H14ClN3O3
    Pureza:99.46%
    Cor e Forma:Solid
    Peso molecular:319.74
  • Golexanolone

    CAS:
    <p>Golexanolone can be used to study neurological diseases.</p>
    Fórmula:C21H31NO2
    Pureza:99.90% - 99.99%
    Cor e Forma:Solid
    Peso molecular:329.48
  • Muscimol HBr

    CAS:
    <p>Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.</p>
    Fórmula:C4H7BrN2O2
    Pureza:98.13%
    Cor e Forma:Off-White Powder
    Peso molecular:195.01
  • DSP-0565

    CAS:
    <p>DSP-0565 is a broad-spectrum anti-epileptic with a high safety margin and effectiveness in several convulsant models.</p>
    Fórmula:C14H12FNO
    Pureza:99.51% - 99.56%
    Cor e Forma:Solid
    Peso molecular:229.25
  • CGP 55845 hydrochloride

    CAS:
    <p>CGP55845 hydrochloride is a potent and selective GABAB receptor antagonist with an IC 50 of 6 nM which can be used in neurological research [1] [2].</p>
    Fórmula:C18H23Cl3NO3P
    Cor e Forma:Solid
    Peso molecular:438.71
  • FGIN-1-27

    CAS:
    <p>FGIN-1-27 is a high-affinity agonist of the translocator protein and a specific peripheral benzodiazepine receptor (PBR) ligand(Ki = 5.0 nM).</p>
    Fórmula:C28H37FN2O
    Pureza:99.86%
    Cor e Forma:Solid
    Peso molecular:436.6
  • GMA-839

    CAS:
    <p>GMA-839 is a selective modulator of gamma-aminobutyric acid(A) receptors.</p>
    Fórmula:C21H31F3O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:388.46
  • NO-711ME

    CAS:
    <p>NO-711ME (N-O711 Methyl ester) is a prodrug of NO-711. It also is a potent and selective GABA uptake inhibitor.</p>
    Fórmula:C22H24N2O3
    Pureza:99.54%
    Cor e Forma:Solid
    Peso molecular:364.44
  • U 89843A

    CAS:
    <p>U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.</p>
    Fórmula:C16H23N5
    Pureza:99.62%
    Cor e Forma:Solid
    Peso molecular:285.39
  • (+)-Bicuculline methiodide

    CAS:
    <p>(+)-Bicuculline methiodide is a GABAA receptor blocker that blocks epileptogens and may be used in the study of neurological disorders.</p>
    Fórmula:C21H20INO6
    Pureza:99.24%
    Cor e Forma:Solid
    Peso molecular:509.29
  • CP-409092

    CAS:
    <p>CP-409092 is a partial GABAA receptor agonist. It has anti-anxiety activity.</p>
    Fórmula:C17H19N3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:297.35
  • mGAT3/4-IN-2

    CAS:
    <p>mGAT3/4-IN-2 are potent inhibitors of mGAT3/mGAT4 with their pIC50 values of 5.44 and 5.25, respectively.</p>
    Fórmula:C26H32ClN3OS2
    Cor e Forma:Solid
    Peso molecular:502.13
  • COR659

    CAS:
    <p>COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.</p>
    Fórmula:C16H16ClNO3S
    Pureza:99.75%
    Cor e Forma:Solid
    Peso molecular:337.82
  • Diproqualone

    CAS:
    <p>Diproqualone, analogous to methaqualone, exhibits sedative, anxiolytic, anti-inflammatory, and analgesic properties [1].</p>
    Fórmula:C12H14N2O3
    Cor e Forma:Solid
    Peso molecular:234.255
  • ADX71441

    CAS:
    <p>ADX71441, a GABAB PAM, lengthens urinary latencies, lessens events &amp; volume, and may aid in alcoholism and bladder pain.</p>
    Fórmula:C19H15ClF2N4O4
    Cor e Forma:Solid
    Peso molecular:436.8
  • Adipiplon

    CAS:
    <p>Adipiplon(NG2-73, NG273) is a novel selective gamma-aminobutyric acid (GABA) partial agonist.</p>
    Fórmula:C18H18FN7
    Cor e Forma:Solid
    Peso molecular:351.38
  • PZ-II-029

    CAS:
    <p>PZ-II-029 is a modulator of α6β3γ2-selective GABAA channel.</p>
    Fórmula:C18H15N3O3
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:321.33
  • CGP 64213

    CAS:
    <p>CGP 64213 is a GABAb receptor agonist.</p>
    Fórmula:C26H36IN2O7P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:646.45
  • (-)-Bicuculline methochloride

    CAS:
    <p>(-)-Bicuculline methochloride is a potent antagonist of GABAA receptor.</p>
    Fórmula:C21H20ClNO6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:417.84
  • GABAA receptor agent 2 TFA

    CAS:
    <p>Potent GABAA antagonist; IC50: 24 nM (α1β2γ2), Ki: 28 nM (rat); inactive on human GABA transporters.</p>
    Fórmula:C22H22F3N3O3
    Cor e Forma:Solid
    Peso molecular:433.42
  • JM-1232

    CAS:
    <p>JM-1232 is a sedative and hypnotic drug being researched as a potential anesthetic.</p>
    Fórmula:C24H27N3O2
    Cor e Forma:Solid
    Peso molecular:389.49
  • CGP-54626 free base

    CAS:
    <p>CGP-54626 is a selective antagonist of the GABAB receptor (IC50 = 4 nM ).</p>
    Fórmula:C18H28Cl2NO3P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:408.3